Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
04/1998
04/07/1998US5736556 Parkinson*s disease; antidepressants; antiobesity; antinarcolepsy; drug abruse
04/07/1998US5736123 Cocaine receptor binding ligands
04/01/1998EP0831941A1 Iodinated neuroprobes for mapping monoamine reuptake sites
04/01/1998CN1177957A Indole derivatives useful in the treatment of osteoporosis
03/1998
03/31/1998US5733917 Gastrointestinal disorders
03/24/1998US5731317 Bridged piperidines promote release of growth hormone
03/19/1998WO1998011128A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production
03/19/1998CA2262818A1 Modified amino acids, pharmaceuticals containing these compounds and methods for their production
03/18/1998EP0828739A1 Bicyclic amines as insecticides
03/10/1998US5726172 Benzoxazinone derivatives; treatment of preterm labor, dysmenorrhea
03/05/1998WO1998008811A1 Cyclic amine derivatives
03/03/1998US5723472 Aminobenzoic acid derivatives
02/1998
02/26/1998WO1998007427A1 Cocaine receptor binding ligands
02/24/1998CA2043071C Heterocyclic compounds
02/18/1998EP0823896A1 Substituted oximes, hydrazones and olefins as neurokinin antagonists
02/18/1998CN1037439C Method for prepn. fo neuroprotective indolone and related derivatives
02/17/1998US5719306 LTA4 hydrolase inhibitors
02/12/1998WO1998005659A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
02/12/1998CA2262460A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
02/11/1998EP0822935A1 Process for preparing pure enantiomers of tropic acid esters
02/10/1998US5716961 Treatment of tinnitus using neuroprotective agents
02/05/1998WO1998004554A1 Chemokine receptor antagonists
02/05/1998WO1998004517A1 Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation
02/05/1998CA2261692A1 Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation
02/05/1998CA2261633A1 Chemokine receptor antagonists
02/04/1998CN1037268C Method for preparation of antipicornaviral phridazinamines
01/1998
01/27/1998US5712287 Method of treating urinary bladder dysfunctions
01/27/1998US5712284 Azalicyclooctane derivatives as anti-arrhythmic agents
01/27/1998US5712271 Method of treating urinary bladder dysfunctions
01/21/1998EP0819126A1 Biphenylamide derivatives as 5ht 1d? antagonists
01/21/1998CN1171116A N-substituted glycine derivatives as inhibotors of factor Xa
01/20/1998US5710168 2-piperidino-1-alkanol derivatives as neuroprotective agents
01/20/1998US5710151 Method of treating urinary bladder dysfunctions
01/15/1998WO1998001443A1 Indole derivatives for the treatment of osteoporosis
01/15/1998CA2259598A1 Indole derivatives for the treatment of osteoporosis
01/13/1998US5708006 Neurokinin antagonists
01/08/1998DE19624659A1 Neue Pyridylalken- und Pyridylalkinsäureamide New pyridylalkene and pyridylalkine acid
01/07/1998EP0815109A1 Method for the preparation of esters of anhydroecgonine
12/1997
12/29/1997EP0813532A1 PREPARATION OF CHIRAL 5-AMINOCARBONYL-5H-DIBENZO- a,d]CYCLOHEPTEN-5,10-IMINES BY OPTICAL RESOLUTION
12/24/1997WO1997048696A1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives
12/24/1997WO1997048681A1 Sulphonamide derivatives and their use in the treatment of cns disorders
12/24/1997CA2258247A1 Sulphonamide derivatives and their use in the treatment of cns disorders
12/16/1997US5698179 Iodinated neuroprobe for mapping monoamine reuptake sites
12/09/1997US5696267 Substituted oximes, hydrazones and olefins as neurokinin antagonists
12/09/1997US5696231 N-substituted glycine derivatives as enzyme inhibitors
12/09/1997US5696126 Prodrug esters of phenolic 2-piperidino-1-alkanols
12/09/1997US5696123 Neurokinin antagonists
11/1997
11/27/1997WO1997044339A1 Antagonists of gonadotropin releasing hormone
11/27/1997CA2254769A1 Antagonists of gonadotropin releasing hormone
11/25/1997CA2106563C Cocaine derivatives and protein and polypeptide cocaine derivative conjugates and labels
11/20/1997WO1997043286A1 Bicyclic amines as insecticides
11/20/1997WO1997043285A1 Tropane derivatives useable in particular for in vivo detection of dopamine transporters
11/20/1997WO1997042956A1 Didhydropyrimidines and uses thereof
11/20/1997CA2254089A1 Tropane derivatives useable in particular for in vivo detection of dopamine transporters
11/20/1997CA2253862A1 Dihydropyrimidines and uses thereof
11/20/1997CA2251851A1 Bicyclic amines as insecticides
11/11/1997US5686614 Preparation of chiral 5-aminocarbonyl-5H-dibenzo a,d!cyclohepten-5,10-imines by optical resolution
11/11/1997US5686463 Oxadiazoles useful in the treatment of senile dementia
11/06/1997WO1997040859A1 Bridge-substituted tropanes and uses
11/05/1997EP0804427A1 Lta4 hydrolase inhibitors
10/1997
10/30/1997WO1997040044A1 Heterocyclic compounds
10/30/1997CA2250873A1 Heterocyclic compounds
10/29/1997EP0802902A1 Indole derivatives useful in the treatment of osteoporosis
10/23/1997WO1997038998A1 3-[(1,2,3,4-tetrahydroisoquinoline-2-yl)methyl]-8-azabicyclo[3.2.1]octane derivatives, their preparation and their application in therapeutics
10/23/1997CA2251335A1 3-[(1,2,3,4-tetrahydroisoquinoline-2-yl)methyl]-8-azabicyclo[3.2.1]octane derivatives, their preparation and their application in therapeutics
10/22/1997EP0801654A1 N-SUBSTITUTED GLYCINE DERIVATIVES AS INHIBITORS OF FACTOR Xa
10/21/1997US5679686 Antipsychotic method
10/15/1997EP0800523A1 A novel radioisotope labelled compound, a mixture comprising said compound and a method for its preparation
10/14/1997US5677313 Antipsychotic method
10/14/1997US5677311 Serotonin antagonism and acetylcholine release accelerating action; antiemetic and oxiolytic agent
10/09/1997WO1997036871A1 6-phenylpyridyl-2-amine derivatives
10/02/1997WO1997035860A1 Novel benzimidazol derivatives having an affinity for the serotoninergic 5-ht3/5 ht4 receptors
09/1997
09/30/1997US5672709 Heterocyclic compounds and their preparation and use
09/25/1997WO1997034892A1 Sigma-2 receptors as biomarkers of tumor cell proliferation
09/25/1997WO1997034871A1 Nitrosated and nitrosylated compounds and compositions and their use for treating respiratory disorders
09/23/1997US5670515 Amino acid derivatives
09/12/1997WO1997032877A1 Process for preparing dibenzo-1-carboxamido-1,4-azabicyclo[3.2.1]octanes
09/09/1997US5665745 1,2,5-thiadiazole derivatives for treating diseases of central nervous system
09/09/1997US5665725 Piperidine derivatives having anxiolytic effect
09/03/1997CN1158615A Bicyclic carboxamides as 5-ht1A antagonists
09/02/1997US5663345 Immunoregulatory, neuromuscular, joint and connective tissue disorders
09/02/1997US5663182 Administering an azabicyclic ring substituted thiadiazole or oxadiazole to a mammal
08/1997
08/28/1997WO1997030997A1 Tropane-derivatives, their preparation and use
08/28/1997WO1997019669A3 Heterocyclic compounds and their use
08/27/1997EP0791592A2 Azetidines
08/27/1997EP0790995A1 A method of treating urinary bladder dysfunctions
08/21/1997WO1997030049A1 Process for the preparation of granisetron
08/21/1997WO1997030048A1 1,4-dihydropyridine compounds as bradykinin antagonists
08/20/1997EP0790250A2 Inhibitors of biogenic amine transporters
08/20/1997EP0790239A1 Novel 4-phenyl-2-(piperazinyl/perhydrodiazepinyl/aminoalkyl)carbonylmethyl)-1,4-dihydropyridine-3,5-dicarboxylic acid derivatives as bradykinin receptor antagonists
08/19/1997US5658928 Anticoagulants, antiinflammatory agents, antitumor agents,wound healing agents, osteoporosis
08/19/1997US5658925 Aminobenzoic acid derivatives
08/13/1997EP0788489A1 Heterocyclic compounds and their use
08/12/1997US5656631 Pyridazine derivatives
08/06/1997CN1156449A Dihygropyridine derivatives as bradykinin antagonists
08/05/1997US5654314 Respiratory system disorders
08/05/1997US5654302 Nervous system disorders; brain disorders
07/1997
07/30/1997EP0515537B1 Substituted urea compounds and their preparation and use
07/24/1997WO1997026258A1 Angiogenesis inhibiting pyridazinamines
07/23/1997CN1155279A Neuroprotective 3-(piperidinyl-1)-chroman-4,7,-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkane alcohol
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