Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
02/1992
02/16/1992CA2089268A1 Renin inhibitors
02/11/1992CA1295613C 4-benzyl-1-(2h)-phthalazinone derivatives
02/05/1992EP0469992A1 6-Alkylpyridazine derivatives, process for their preparation and compositions containing them
02/05/1992EP0338010B1 Pharmaceutical compositions for treatment of hyperproliferate skin disease
02/04/1992US5086179 Process for the preparation of optically pure amides
02/01/1992CA2048162A1 6-alkylpyridazine derivatives, method of preparation and pharmaceutical compositions in which they are present
01/1992
01/22/1992EP0467365A2 Use of a 5-hydroxytryptamine-3(5-HT3) receptor antagonist for the preparation of a pharmaceutical composition for treating urinary incontinence
01/21/1992US5082843 Pyrazinyl and pyridazinyl ethers
01/20/1992CA2044854A1 Method for preventing or treating urinary incontinence
01/14/1992CA1294281C Specific 5-ht--antagonists
12/1991
12/26/1991WO1991016045A3 Use of 5-ht4 receptor antagonists in the treatment of arrythmias and stroke
12/17/1991CA1293256C2 Substituted benzoic acid alkylene bridged pyridil derivatives
12/10/1991US5071854 Hydroxytryptamine antagonists
12/03/1991US5070094 N-benzyltropaneamides
11/1991
11/27/1991EP0458636A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them
11/27/1991CN1056497A Neuroprotective indolone and related derivatives
11/21/1991EP0457243A1 Novel tricyclic compounds
11/20/1991CN1014790B Process for preparing novel benzoxazol-and benzothiazolamine derivatives and their use
11/15/1991CA2042443A1 Tricyclic compounds
11/14/1991WO1991017156A1 Neuroprotective indolone and related derivatives
11/05/1991US5063231 Gastrointestinal
10/1991
10/31/1991WO1991016045A2 Use of 5-ht4 receptor antagonists in the treatment of arrythmias and stroke
10/31/1991WO1991016024A1 Cationic lipids for intracellular delivery of biologically active molecules
10/29/1991US5061722 Hypotensive agents; e.g. ramipril
10/28/1991WO1991017161A1 Isoquinoline amides and esters as 5 ht3 receptor antagonists
10/28/1991CA2081350A1 Isoquinoline amides and esters as 5 ht3 receptor antagonists
10/24/1991WO1991016888A1 Spiro[benzofurancycloalkane]carboxamides as 5ht3 antagonists
10/24/1991CA2081011A1 Spiro[benzofurancycloalkane]carboxamides as 5ht3 antagonists
10/09/1991EP0450757A2 Use of 5-hydroxytryptamine-antagonists in the treatment of mental disorders originating in childhood
10/01/1991US5053519 Hypotensive agents; diuretics; vasodilation
09/1991
09/17/1991US5049556 Certain N-azabicyclo-2,3-dihydro-indole-1-carboxamides having anti-emetic properties, further found useful in treating headaches, neuralgia and anxiety
09/11/1991EP0445731A1 Azabicyclo and azacyclo oxime and amine cholinergic agents and pharmaceutically acceptable salts thereof
09/10/1991US5047410 Indolyl derivatives and their use as 5-HT3, receptor antagonists
09/05/1991WO1991009593A3 5-ht3 antagonists for treatment of nausea, bradycardia of hypotension associated with myocardial instability
09/03/1991US5045546 8-azabicyclo[3.2.1]octylalkylthiazolidines
08/1991
08/22/1991WO1991012005A1 Neuroprotective 3-piperidino-4-hydroxychroman derivatives and analogs
08/21/1991CN1053923A Neuroprotective 3-piperidino-4-hydroxychroman derivatives
08/20/1991US5041456 Pharmaceutically useful 3-(indol-3-yl)-1,2,4-oxa- and thiadiazoles substituted in the 5-position by an amino containing group
08/17/1991WO1991012254A1 Substituted urea compounds and their preparation and use
08/17/1991CA2074803A1 Substituted urea compounds and their preparation and use
08/14/1991EP0441506A2 Neuroprotective 3-piperidino-4-hydrosychroman derivatives
08/08/1991WO1991011186A1 Method and compositions for the synthesis of bch-189 and related compounds
08/08/1991CA2678778A1 Method and compositions for the synthesis of bch-189 and related compounds
07/1991
07/23/1991US5034398 1H-indazole-3-carboxamide-N-2-azabicyclo[2.2.2]octanes useful for treating anxiety, psychosis, neuralgia, migraine and cluster headaches
07/11/1991WO1991009593A2 5-ht3 antagonists for treatment of nausea, bradycardia of hypotension associated with myocardial instability
07/10/1991EP0436245A1 Substituted 3,4-annelated benzimidazol-2(1H)-ones
07/10/1991CN1052857A Antipicornaviral pyridazinamines
07/03/1991EP0435381A1 Antipicornaviral pyridazinamines
06/1991
06/28/1991CA2032885A1 Substituted 3,4-annelated benzimidazol-2(1h)-ones
06/27/1991CA2031889A1 Antipicornaviral pyridazinamines
06/22/1991CA2071994A1 Pharmaceuticals
06/05/1991EP0430190A2 New tricyclic compounds
05/1991
05/29/1991EP0429344A1 Pyridazine derivatives, process for their preparation and pharmaceutical compositions containing them
05/21/1991US5017582 Method of inducing a serotonin M receptor antagonist effect with N-quinuclidinyl-benzamides
05/18/1991CA2030133A1 Pyridazine derivatives, process for their preparation and pharmaceutical compositions containing them
05/16/1991DE4037686A1 Quantitative determn. of cocaine and its main metabolites - by thin layer chromatography followed by conversion to a fluorescing prod. by heating
04/1991
04/30/1991CA1283658C Process for quinoline-3-carboxylic acid antibacterial agents
04/24/1991CN1050875A Aroyl-urres
04/23/1991US5010198 Intermediates for the synthesis of benzoxazol- and benzothiazolamine derivatives, useful as anti-anoxic agents
04/18/1991WO1991004738A1 Dibenzofurancarboxamides
04/17/1991EP0422846A2 Aroyl-ureas
04/15/1991WO1991005783A1 Heterocyclic compounds
04/09/1991US5006533 Neuroleptic agents, side effect reduction
03/1991
03/27/1991EP0419397A1 Substituted urea compounds and their preparation and use
03/27/1991EP0418716A1 Thienylcarboxylic acid ester of aminoalcohols, their quaternary products, their preparation and use of the compounds
03/19/1991US5001133 Benzoic acid derivatives
03/17/1991WO1991004252A1 New esters of thienyl carboxylic acids and amino alcohols, their quaternization products, and manufacture and use of said compounds
03/13/1991EP0416521A1 N-Benzyltropaneamides
03/13/1991EP0416097A1 Process for producing tropane alkaloids
03/09/1991WO1991003475A1 Substituted urea compounds and their preparation and use
03/09/1991CA2066696A1 Substituted urea compounds and their preparation and use
03/06/1991CA2024579A1 N-benzyltropaneamides
03/05/1991US4997956 Certain 2,3-dihydro-2;2-dimethyl-benzothiophene carboxylic acids which are intermediates
03/05/1991US4997839 2-quinolyl ethers
02/1991
02/26/1991US4996211 Anticonvulsants, treating neurodegenerative diseases
02/13/1991EP0412797A2 The therapeutic use of substituted benzenes, formulations thereof and novel substituted benzenes
02/12/1991US4992546 Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives
02/12/1991US4992436 Spiro-azabicyclic muscarinic agonists
02/12/1991US4992433 Novel pyridazinamine derivatives
02/07/1991WO1991001316A1 New 9-azabicyclo[3.3.1]nonane-derivate
01/1991
01/29/1991US4988691 Analgesics, cardiovascular disorders, nervous system disorders
01/15/1991US4985437 Medicaments
01/09/1991EP0407137A2 Benzazine compounds and pharmaceutical uses thereof
01/08/1991US4983600 Heterocyclic compounds useful as 5-HT3 antagonists
01/04/1991CA2020315A1 Benzazine compounds and pharmaceutical uses thereof
01/02/1991EP0405617A2 Medicaments for the treatment of anxiety
12/1990
12/27/1990EP0403882A2 Indole derivatives and processes for preparation thereof
12/23/1990CA2017621A1 Indole derivatives and processes for preparation thereof
12/11/1990US4977141 Renin inhibitors
12/04/1990US4975436 Treatment of anxiety
11/1990
11/29/1990WO1990014088A1 2-piperidino-1-alkanol derivatives as antiischemic agents
11/29/1990WO1990014087A1 2-piperidino-1-alkanol derivatives as antiischemic agents
11/28/1990EP0398967A1 Antibacterial agents
11/28/1990CN1047291A 2-piperidino-1-alkanol derivatives as antiischemic agents
11/27/1990US4973594 Treatment of depression
11/22/1990EP0398578A2 2-piperidino-1-alkanol derivatives as antiischemic agents
11/10/1990WO1990013297A1 5-AMINOCARBONYL-5H-DIBENZO[a,d]CYCLOHEPTEN-5,10-IMINES FOR TREATMENT OF EPILEPSY AND COCAINE ADDICTION
11/06/1990US4968799 Antibacterial agents
11/06/1990US4968691 Heterocyclo-substituted azabicyclo muscannic agonists
10/1990
10/22/1990WO1990012569A1 Therapeutic use of 5-ht3 receptor antagonists
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