Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
03/1993
03/14/1993CA2077922A1 Substituted amide derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
03/10/1993EP0530353A1 New imidazopyridines as serotonergic 5-ht 3? antagonists
03/09/1993US5192770 Serotonergic alpha-oxoacetamides
03/04/1993WO1993000313A3 Sigma receptor ligands and the use thereof
03/03/1993EP0529484A1 Antitussive and expectorant composition
02/1993
02/28/1993CA2076114A1 Antitussive and expectorant composition
02/23/1993CA2076556A1 A method and intermediates for the preparation of 6-fluorobenzisothiazoles
02/16/1993US5187164 Psychological disorders, antiemetics
02/10/1993EP0526545A1 Isoquinoline amides and esters as 5 ht3 receptor antagonists
02/10/1993EP0526540A1 Use of 5-ht 4? receptor antagonists in the treatment of arrythmias and stroke
02/09/1993US5185343 Nortropyl-1-alkanol derivatives as antiischemic agents
02/09/1993US5185333 Benzazine compounds and pharmaceutical uses thereof
02/02/1993US5183822 Substituted 3,4-annelated benzimidazol-2(1h)-ones
01/1993
01/20/1993EP0523189A1 Cationic lipids for intracellular delivery of biologically active molecules
01/13/1993EP0523013A2 Use of benzimidazoline-2-oxo-1-carboxylic acid derivatives in the treatment of organic mental diseases
01/07/1993WO1993000313A2 Sigma receptor ligands and the use thereof
01/07/1993CA2111957A1 Sigma receptor ligands and the use thereof
01/05/1993CA2072911A1 Use of benzimidazoline-2-oxo-1-carboxylic acid derivatives
12/1992
12/29/1992US5175173 Reduced side effects
12/23/1992WO1992022554A1 Piperidine derivates having anxiolytic effect
12/23/1992WO1992022294A1 Immunomodulatory azaspiranes
12/23/1992CA2110577A1 Immunomodulatory azaspiranes
12/16/1992EP0518805A1 Piperidine derivatives
12/10/1992WO1992021673A1 Novel azabicyclobenzisoquinolines
12/01/1992CA1310958C Physical property-improving reagent
11/1992
11/19/1992EP0514277A1 3-Aminopyridazine derivatives active on the central nervous system
11/19/1992EP0513200A1 Method and compositions for the synthesis of bch-189 and related compounds
11/17/1992CA2068770A1 3-aminopyridazine derivatives active on the central nervous system, method of preparation and pharmaceutical compositions in which they are present
11/04/1992CN1065866A Prodrug esters of phenolic 2-piperidino-1-alkanols
11/03/1992CA1309658C Pharmaceutical compositions for treatment of hyperproliferate skin disease
10/1992
10/28/1992EP0510129A1 Muscarinic receptor antagonists
10/28/1992CN1065661A Heterocyclic compounds
10/19/1992WO1992018502A1 Prodrug esters of phenolic 2-piperidino-1-alkanols
10/19/1992CA2108557A1 Prodrug esters of phenolic 2-piperidino-1-alkanols
10/07/1992EP0507637A2 Use of benzobicyclic carboxamides for the manufacture of a medicament for use as analgesic
10/07/1992EP0506813A1 5-ht 3? antagonists for treatment of nausea, bradycardia of hypotension associated with myocardial instability
10/06/1992CA2063912A1 Analgesic use of benzobicyclic carboxamides
09/1992
09/30/1992EP0505868A2 N-Acyl-alpha-aminoacids derivatives
09/30/1992EP0505778A1 Derivatives of substituted imidazol-2-one and process for their preparation
09/27/1992CA2061661A1 N-acyl-.alpha.-amino derivatives
09/23/1992EP0504679A1 New imidazopyridines as serotonergic 5-HT3 antagonists
09/22/1992CA1307790C Ethers
09/17/1992DE4108393A1 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln New bi- and tricyclic ester amino alcohols, their production and their use in medicinal products
09/16/1992WO1992016528A1 New bi- and tricyclic aminoalcohol esters, their preparation and their use in medicaments
09/08/1992WO1992015593A1 New imidazopyridines as serotonergic 5-ht3 antagonists
09/08/1992CA2082414A1 Imidazopyridines as serotonergic 5-ht3 antagonists
09/03/1992WO1992014733A1 Pharmaceuticals
08/1992
08/16/1992WO1992014705A1 Benzamide derivative
08/12/1992EP0498466A1 Indazole-3-carboxamide and -3-carboxylic acid derivatives
08/12/1992EP0498331A1 N-(aryloxyalkyl)heteroaryl-8-azabicyclo(3.2.1)octanes, intermediates and a process for the preparation thereof and their use as medicaments
07/1992
07/29/1992EP0496064A1 Process for the preparation of substituted benzofuran derivatives
07/23/1992WO1992012150A1 Quinoline derivative
07/23/1992WO1992012149A1 Azabicydic and azatricydic derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them
07/15/1992EP0494140A1 Dibenzofurancarboxamides
07/15/1992EP0340270B1 5-ht 3? receptor antagonists for treatment of cough and bronchoconstriction
07/07/1992US5128118 Cocaine receptor binding ligands
07/01/1992EP0493041A2 Use of benzobicyclic carboxamides for the treatment of anxiety and migraine
07/01/1992EP0493031A1 Dihydrobenzofuran carboxamides and process for their preparation
07/01/1992EP0491770A1 Substituted urea compounds and their preparation and use
06/1992
06/30/1992US5126364 Antiemetics, antipsychotics
06/30/1992CA1304369C Azoniaspironortropanol esters and processes for the preparation thereof
06/28/1992WO1992012147A1 Process for the preparation of substituted benzofuran derivatives
06/28/1992CA2099107A1 Process for the preparation of substituted benzofuran derivatives
06/28/1992CA2057973A1 Method for alleviating anxiety using benzobicyclic carboxamides
06/24/1992EP0491664A1 Serotonin antagonists
06/23/1992CA1304082C Benzoxazine compounds and pharmaceutical use thereof
06/20/1992WO1992011259A1 Azabicyclic amides or esters of halogenated benzoic acids
06/20/1992CA2098729A1 Azabicyclic amides or esters of halogenated benzoic acids
06/19/1992CA2057391A1 Serotonin antagonists
06/17/1992EP0490263A1 Alpha-oxoacetamide derivatives
06/16/1992US5122528 Analgesic use of benzobicyclic carboxamides
06/14/1992WO1992010494A1 Pharmaceuticals
06/14/1992CA2098309A1 Pharmaceuticals
06/09/1992CA1303043C Esters of n-alkyl-nortropines and their quaternary derivatives having anti-bronchospastic activity, process for their preparation and pharmaceutical compositions containing them
06/08/1992CA2057181A1 Scrotonergic .alpha.-oxoacetamide
05/1992
05/29/1992WO1992005172A3 Muscarinic receptor antagonists
05/19/1992US5114947 Benzofuran-7-carboxamides as anxiolytic agents
05/19/1992CA1301170C Benzofuran 7-carboxamides useful as antiemetic or antipsyschotic agents
05/12/1992CA1300606C Derivatives of 5-methyl-10,11-dihydro-5h-dibenzo ¬a,d| cyclohepten-5,10-imine
05/06/1992EP0483633A1 8-Azabicyclo[3.2.1]octylalkylthiazolidinones, a process for their preparation and their use as medicaments
04/1992
04/28/1992USRE33907 Anti-spasmodic agents having a heterocyclic ring
04/28/1992CA1299564C Cephalosporin derivative
04/27/1992CA2054225A1 8-azabicyclo[3.2.1] octylalkylthiazolidinones, a process for their preparation and their use as medicaments
04/21/1992US5106973 Pyridzainamine derivatives
04/21/1992US5106851 Benzofused-n-containing heterocycle derivatives
04/21/1992US5106843 Treatment of migraine, emesis, anxiety, gastrointestinal disorders, psychological disorders
03/1992
03/31/1992US5100893 Viricides, effective against picorna virus, durability
03/25/1992WO1992005146A1 Stereoselective preparation of acid sensitive amides and intermediates useful in said preparation
03/25/1992CN1059724A Tricyclic compounds
03/25/1992CA2092179A1 Stereoselective preparation of acid sensitive amides and intermediates useful in said preparation
03/24/1992US5098909 5-ht3 receptor antagonists for treatment of cough and bronchoconstriction
03/24/1992CA1297877C Benzofurancarboxamides useful as antiemetic or antipsychotic agents
03/17/1992US5096901 Pharmacologically active amides and esters containing an azabicycloalkane moiety
03/14/1992WO1992005172A2 Muscarinic receptor antagonists
03/14/1992CA2068527A1 Muscarinic receptor antagonists
03/05/1992WO1992003433A1 Heterocyclic compounds and their preparation and use
02/1992
02/20/1992WO1992002260A1 Cocaine receptor binding ligands
02/18/1992US5089471 Renin inhibitors
02/18/1992CA1296004C Aza-indole derivatives
02/16/1992WO1992003429A1 Renin inhibitors
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