| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 03/07/2002 | WO2001077100A3 Benzoamide piperidine compounds as substance p antagonists |
| 03/06/2002 | CN1338928A Combinations of formoterol and a tiotropium salt |
| 03/05/2002 | US6353106 Process for the production of trifluoromethyltropanone cyanohydrin |
| 03/05/2002 | US6353105 Inhibitors of 5-hydroxy-tryptamine reuptake of a monoamine transporter; analogs of cocaine; |
| 02/28/2002 | WO2002016340A1 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same |
| 02/28/2002 | WO2002016339A1 Aminoalkylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same |
| 02/28/2002 | CA2415852A1 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same |
| 02/27/2002 | CN1337960A Piperdine and piperazine derivatives as inhibitors of the ABETA fibril formation |
| 02/26/2002 | US6350758 Tropane derivatives and method for their synthesis |
| 02/21/2002 | WO2002014273A1 Indoline derivatives as 5ht2c antagonists |
| 02/19/2002 | CA2112083C Aryl substituted heterocyclic compounds |
| 02/14/2002 | WO2002012245A2 Azabicyclic derivatives and their therapeutic use |
| 02/14/2002 | WO2002012235A1 1,4-dihydropyridines as bradykinin antagonists |
| 02/14/2002 | US20020019382 Curcumin analogs with anti-tumor and anti-angiogenic properties |
| 02/14/2002 | CA2417967A1 Azabicyclic derivatives and their therapeutic use |
| 02/06/2002 | EP1178048A1 Azabicycloalkane derivatives for use as serotonin reuptake inhibitors and 5HT2a antagonists |
| 02/05/2002 | US6344449 Headache and morphine dependence |
| 02/05/2002 | US6344179 Bind to dopamine transporter with high affinity and selectivity; useful as diagnostic and therapeutic agents; containing radioactive isomers f18 or 19; pet scanning |
| 01/31/2002 | US20020013341 For therapy of acute infection, acute phase response, age related macular degeneration, alcoholism, anorexia, asthma, autoimmune disease, autoimmune hepatitis, Bechet's disease, cachexia, calcium pyrophosphate dihydrtate deposition |
| 01/31/2002 | US20020013337 For therapy of respiratory disorder including adult respiratory distress syndrome (ARDS), bronchitis, chronic bronchitis, chronic obstructive pulmonary disease, cystic fibrosis, asthma, emphysema, rhinitis or chronic sinusitis |
| 01/30/2002 | EP1021442B1 8-azabicyclo 3.2.1] octane-3-methanamine derivatives as ligands of d2 and d3 dopamine and 5ht1a and 5ht2 serotonin receptors |
| 01/30/2002 | CN1333758A Substituted bicyclic derivatives useful as anticancer agents |
| 01/24/2002 | WO2001029000A3 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
| 01/24/2002 | US20020010207 Tropane analogs and methods for inhibition of monoamine transport |
| 01/24/2002 | US20020010186 Dihydropyrimidines and uses thereof |
| 01/23/2002 | CN1332726A Pyrrolidine compounds and medicinal utilizaion thereof |
| 01/22/2002 | US6340681 Useful as analgesics in mammals |
| 01/17/2002 | WO2002004442A2 Azabicyclic compounds as inhibitors of nicotinic cholinergic receptors |
| 01/17/2002 | WO2002004402A1 Ester derivatives |
| 01/17/2002 | WO2001025236A3 A stereoselective process for the preparation of endo-3-aminoazabicycloalkanes |
| 01/17/2002 | CA2415468A1 Ester derivatives |
| 01/16/2002 | EP1171432A1 Adamantane derivatives |
| 01/16/2002 | CN1331691A Piperidines as CCR5 modulators |
| 01/16/2002 | CN1331591A Piperidines as CCR5 modulators |
| 01/10/2002 | US20020004513 Azacyclic compounds |
| 01/09/2002 | CN1077574C Tropane derivatives, their preparation and use |
| 01/03/2002 | US20020002170 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation |
| 01/02/2002 | CN1329612A Process for production of trifluoromethyltropanone cyanohydrin |
| 12/27/2001 | US20010056110 Systemic use of 5-HT3 receptor antagonists against rheumatic inflammatory processes |
| 12/19/2001 | EP1163238A1 Chemokine recpetor binding heterocyclic compounds |
| 12/13/2001 | US20010051633 E.g.,N-((4-amino-3-nitrophenoxy)ethyl)-1,2,3,4-tetrahydro -isoquinoline; stroke; antiischemic agents; CNS trauma, hyperglycemic agents; surgery; neurodegenerative diseases including Alzheimer's disease, amyotrophic lateral sclerosis |
| 12/12/2001 | CN1326456A 8-Azabicyclo [3.,2.1] Oct-2-Ene and-Octane derivatives |
| 12/11/2001 | US6329520 Used as imaging or pharmaceutical agents, in the diagnosis and treatment of drug addiction, depression, anorexia and neurodegenerative diseases or in determining doses of therapeutic agents that occupy many receptors |
| 12/06/2001 | US20010049379 Nitric oxide synthase inhibitors; treatment and prevention of central nervous system and other disorders. |
| 12/05/2001 | EP1158970A1 Combinations of formoterol and a tiotropium salt |
| 11/29/2001 | WO2001090717A2 Linker arms for nanocrystals and compounds thereof |
| 11/29/2001 | WO2001090716A2 Linker arms for nanocrystals and compounds thereof |
| 11/29/2001 | WO2001090106A2 Tryasolyl tropane derivatives as ccr5 modulators |
| 11/29/2001 | WO2001089524A1 Method of promoting smoking cessation |
| 11/29/2001 | US20010047028 8-azabicyclo(3.2.1)oct-2-ene and 9-azabicyclo(3.3.1)non-2-ene derivatives; monoamine neurotransmitter and serotonine reuptake inhibitors; radionuclide-labeled derivatives for diagnosis and detection |
| 11/29/2001 | CA2410530A1 Method of promoting smoking cessation |
| 11/28/2001 | EP0677051B1 Derivatives of benzoylecgonine, ecgonine and ecgonidine as medicines |
| 11/28/2001 | CN1323798A 3 alpha-alkylacyloxy-6 beta-alkylacyoxy tropane compounds and their prepn. |
| 11/27/2001 | US6323343 Process for the preparation of 8-azabicyclo(3.2.1)octane derivatives |
| 11/27/2001 | US6323216 Selective antagonists of the 5-ht.sub.3 serotonin-like receptor and can therefore be used, as anti-emetics as well as in various pathological conditions of the central nervous system, and as antitussives. |
| 11/22/2001 | WO2001087846A2 Tricyclic pyrazole derivatives as protein kinase inhibitors |
| 11/22/2001 | WO2001087299A1 Aralkyl ester soft drugs |
| 11/22/2001 | CA2409225A1 Tricyclic pyrazole derivatives |
| 11/22/2001 | CA2407099A1 Aralkyl ester soft drugs |
| 11/21/2001 | EP1156045A1 Amide derivatives and drug compositions |
| 11/21/2001 | EP0772613B1 Process for the production of aminoazobicycloalkanes from oximes |
| 11/13/2001 | US6316624 Process for the preparation of substituted 8-azabicyclo[3,2,1]octanes |
| 11/08/2001 | US20010039287 Aromatic sulfone hydroxamic acid metalloprotease inhibitor |
| 11/07/2001 | EP1150971A1 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation |
| 11/07/2001 | EP0843676B1 Preparations containing ipratropium bromide enantiomer with a prolonged duration of action |
| 11/07/2001 | EP0822935B1 Process for preparing pure enantiomers of tropic acid esters |
| 11/01/2001 | WO2001080905A2 Sigma-2 receptors as biomarkers of tumor cell proliferation |
| 11/01/2001 | US20010036946 Antiinflammatory agents |
| 11/01/2001 | US20010036474 Antiemitic agent |
| 10/31/2001 | EP1149095A1 Novel azabicyclo derivatives and their use |
| 10/25/2001 | US20010034351 A quinazoline compound |
| 10/25/2001 | US20010034348 Nitric oxide synthase inhibitor; nervous system disorders |
| 10/24/2001 | EP1147093A1 Substituted bicyclic derivatives useful as anticancer agents |
| 10/23/2001 | US6306876 4-[aryl(8-azabicyclo[3.2.1]octan-3-yl)]aminobenzoic acid derivatives |
| 10/18/2001 | WO2001077100A2 Benzoamide piperidine compounds as substance p antagonists |
| 10/18/2001 | CA2405089A1 Benzoamide piperidine containing compounds and related compounds |
| 10/16/2001 | US6303593 For therapy human immunodeficiency virus infection, aquired immunodeficiency syndrome (aids), inflammatory and immunoregulatory disorder or disease, asthma, allergic rhinitis, dermatitis, conjunctivitis, atherosclerosis |
| 10/11/2001 | WO2001014374A3 Processes for the prepration of exo- and endo-indolotropanes |
| 10/10/2001 | EP1140920A1 Piperidines as ccr5 modulators |
| 10/10/2001 | EP1140085A1 Azabicycloalkanes as ccr5 modulators |
| 10/10/2001 | CN1072666C (Azetidin-1-ylalkyl) lactams as tachykinin antagonists |
| 10/09/2001 | US6300347 For therapy of tumor necrosis factor and interleukin-1 mediated diseases such as rheumatoid arthritis and diseases of bone metabolism, e.g. osteoporosis |
| 10/09/2001 | US6299861 Administering aerosol of inhalable ipratropium bromide for inhibiting acetylcholine induced bronchospasm in humans |
| 10/04/2001 | WO2001072303A1 Selective ligands for the delta opioid receptor |
| 10/04/2001 | EP1137648A1 Process for the production of trifluoromethyltropanone cyanohydrin |
| 10/04/2001 | EP0975631B1 5-aryl-3-(8-azabicyclo[3.2.1]oct-3-yl)-1,3,4-oxadiazol-2(3h)-one derivatives as 5-ht4 receptor ligands |
| 10/02/2001 | CA2037541C Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment |
| 09/27/2001 | WO2001070734A2 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha |
| 09/27/2001 | CA2400168A1 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha |
| 09/25/2001 | US6294545 Bicyclic amines and their use as insecticides |
| 09/19/2001 | EP1133494A1 8-azabicyclo 3.2.1]oct-2-ene and -octane derivatives |
| 09/18/2001 | US6291474 Bicyclic amine derivatives |
| 09/13/2001 | WO2001066543A2 3-(diarylmethylene)-8-azabicyclo[3.2.1]octane derivatives |
| 09/13/2001 | WO2001066521A1 Azacyclic compounds for use in the treatment of serotonin related diseases |
| 09/13/2001 | CA2402039A1 3-(diarylmethylene)-8-azabicyclo[3.2.1]octane derivatives |
| 09/11/2001 | US6288079 Tropane-derivatives, their preparation and use |
| 09/06/2001 | US20010020096 Reacting a cycloheptatriene derivative with a primary amine or ammonia in the presence of a base |
| 09/05/2001 | EP1130020A1 Tropane-derivatives, their preparation and use |
| 09/05/2001 | CN1311787A Oxazolidinone derivatives, process for their prepn. and pharmaceutical compositions contg. same |
| 09/05/2001 | CN1311777A High affinity ligands for nociceptin receptor ORL-1 |