C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof

Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
12/2002
12/05/2002	WO2002096855A2 Anticholinergic compounds and methods of use
12/05/2002	WO2002096423A2 Combination of a pde4 inhibitor and tiotropium or derivate thereof for treating obstructive airways
12/05/2002	CA2448363A1 Combination of a pde4 inhibitor and tiotropium or derivate thereof for treating obstructive airways
12/05/2002	CA2446532A1 Aryl-8-azabicyclo[3.2.1]octanes for the treatment of depression
12/05/2002	CA2443346A1 Anticholinergic compounds and methods of use
12/04/2002	EP0703791B1 An iodinated neuroprobe for mapping monoamine reuptake sites
11/2002
11/28/2002	WO2002094790A1 Fused heterocyclic compound and medicinal use thereof
11/28/2002	WO2002094273A2 Combination of an adenosine a2a-receptor agonist and tiotropium or a derivative thereof for treating obstructive airways
11/28/2002	US20020177714 Benzoylecgonine, ecgonine and ecgonidine derivatives
11/28/2002	US20020177588 Selectivity
11/28/2002	CA2445789A1 Combination of an adenosine a2a-receptor agonist and tiotropium or a derivative thereof for treating obstructive airways
11/27/2002	EP1259241A1 The use of scopolamine salts
11/26/2002	US6486321 Epoxidation; quaternization
11/21/2002	US20020173659 Indole derivatives for the treatment of osteoporosis
11/20/2002	EP1258480A1 Pharmaceutical use of N-Carbamoylazole derivatives
11/20/2002	EP1258244A1 High affinity ligands for nociceptin receptor ORL-1
11/19/2002	US6482831 Covalently coupled benzoylecgonine, egconine and ecgonidine derivatives
11/19/2002	CA2112061C Alkyl substituted heterocyclic compounds
11/14/2002	WO2002089806A1 Heterobicycles fkbp-ligands
11/14/2002	WO2002081453A8 Thiohydantoins and use thereof for treating diabetes
11/14/2002	WO2002062324A3 A treatment of oesophageal motility disorders and gastro-oesophageal reflux disease
11/14/2002	US20020169321 Crystalline tiotropium bromide monohydrate, processes for the preparation thereof, and pharmaceutical compositions
11/14/2002	US20020169208 Oxybutynin analogs; antichloinergic agents; side effect reduction; short half-life; water-soluble metabolites; incontinence; mydriatic and bronchodilator agents; respiratory system disorders; antiperspirants
11/14/2002	CA2446795A1 Sulfamide, sulfamate, sulfonamide, urea, amide, alpha, alpha-difluoro amide oxalyl diamide, and heterobicycles fkbp-binding ligands
11/12/2002	US6479509 Method of promoting smoking cessation
11/07/2002	US20020165241 Such as 4-((methyl-pyrimidin-2-ylamino)-methyl)-piperidine-1-carboxylic acid benzyl ester; useful for pain relief; treating migraine, depression, anxiety, schizophrenia, Parkinson's disease, and stroke; N-methyl-D-aspartate (NMDA)
11/07/2002	US20020165227 Gramnegative bacteria
11/06/2002	EP1254123A1 2-benzothiazolyl urea derivatives and their use as protein kinase inhibitors
11/06/2002	CN1378544A Substituted azoles compounds
10/2002
10/31/2002	WO2002086427A1 Metering method for particulate material
10/31/2002	WO2002085900A1 8-aza-bicyclo[3.2.1]octan-3-ol derivatives of 2,3-dihydro-1,4-benzodioxan as 5-ht1a antagonists
10/31/2002	US20020161006 1,4-dihydropyridine compounds as bradykinin antagonists
10/31/2002	US20020161005 Nitrogen heterocycle compounds
10/24/2002	WO2002083669A1 Tropane alkaloid multidrug resistance inhibitors from erythroxylum pervillei and use of the same
10/24/2002	CA2443655A1 Tropane alkaloid multidrug resistance inhibitors from erythroxylum pervillei and use of the same
10/22/2002	US6468998 Pyrrolidine compounds and medicinal utilization thereof
10/17/2002	WO2002081453A1 Thiohydantoins and use thereof for treating diabetes
10/17/2002	WO2002081448A1 Benzamidine derivative
10/17/2002	WO2002066468A3 Heterocyclic urea derivatives and their use as dopamine d3 receptor ligands
10/17/2002	US20020150535 Methods for diagnosing and monitoring treatment ADHD by assessing the dopamine transporter level
10/17/2002	CA2444024A1 Thiohydantoins and use thereof for treating diabetes
10/17/2002	CA2442904A1 Benzamidine derivative
10/16/2002	EP1248786A1 Benzofuran derivatives
10/16/2002	EP0934316B1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/15/2002	US6465491 6-phenylpyridyl-2-amine derivatives
10/15/2002	US6465449 Heteroaromatic bicyclic derivatives useful as anticancer agents
10/10/2002	WO2002079190A1 3-substituted indoles as chemokine antagonists
10/10/2002	WO2002079151A1 3-substituted indoels or fused pyrroles as antagonists of the chemokine mcp-1 (ccr2b) receptor
10/10/2002	US20020147212 Azabicyclic amine derivatives and their use as therapeutic agents
10/08/2002	US6462036 Inhibiting signal transduction by modulating activity of receptor and nonreceptor tyrosine and serine/threonine kinases to regulate and modulate abnormal or inappropriate cell proliferation, differentiation, or metabolism
10/02/2002	EP1244450A1 8-aza-bicyclo[3.2.1]octane nmda/nr2b antagonists
10/02/2002	EP0843675B1 Aza-anthracyclinone derivatives
10/01/2002	US6458812 Muscarinic antagonists
10/01/2002	CA2245857C 1,4-dihydropyridine compounds as bradykinin antagonists
10/01/2002	CA2241845C 4,5-dihydronaphth¬1,2-c\|isoxazoles and derivatives thereof having cns activity
10/01/2002	CA2089769C Heterocyclic compounds and their preparation and use
09/2002
09/26/2002	WO2002024636A3 N-acylsulfonamide apoptosis promoters
09/25/2002	EP1243589A1 Heteroaryl-substituted pyrrole derivates, their preparation and their therapeutic uses
09/25/2002	EP1243268A1 Medicinal composition
09/25/2002	EP1242421A1 4-[aryl(8-azabicyclo[3.2.1] octan-3-yl)] aminobenzoic acid derivatives
09/25/2002	EP1242419A1 Azabicyclo 3.2.1]octane derivatives
09/25/2002	EP1242379A1 Curcumin analogues for treating cancer
09/25/2002	EP0923570B1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives
09/19/2002	WO2002072570A2 Non-imidazole compounds as histamine h3 antagonists
09/19/2002	WO2002072095A2 Tiotropium salts for treating inflammatory diseases
09/19/2002	WO2002036106A3 Novel medicament compositions based on anticholinergics and corticosteroids
09/19/2002	US20020133010 Epoxidation; quaternization
09/19/2002	DE10111843A1 Verbindungen zur Behandlung von inflammatorischen Erkrankungen Compounds for the treatment of inflammatory disorders
09/18/2002	EP0858461B1 Fused tropane-derivatives as neurotransmitter reuptake inhibitors
09/18/2002	EP0804427B1 Lta4 hydrolase inhibitors
09/18/2002	CN1370144A Aromatic sulfone hydroxamic acid metalloprotease inhibitor
09/18/2002	CN1370048A Azabicyclo and azacyclo oxime and amine compounds as pesticides
09/17/2002	US6451816 Use of pyridyl alkane, pyridyl alkene and/or pyridyl alkine acid amides in the treatment of tumors or for immunosuppression
09/12/2002	US20020128284 Tropane-derivatives, their preparation and use
09/12/2002	US20020128271 N-benzenesulfonyl l-proline compounds as bradykinin antagonists
09/11/2002	EP1238978A2 Intermediates for the synthesis of radiolabelled tropanes
09/11/2002	EP0828739B1 Bicyclic amines as insecticides
09/10/2002	US6447747 Process for the preparation of radiopharmaceuticals
09/06/2002	WO2002068409A1 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists
09/06/2002	WO2002068388A2 Acylated piperidine derivatives as melanocortin-4 receptor agonists
09/06/2002	WO2002068377A1 Omega-aminoalkylamides of r-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells
09/06/2002	WO2002030405A3 Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance
09/06/2002	CA2438895A1 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists
09/04/2002	EP1236727A1 Azabicyclo compounds as pesticides
09/04/2002	EP1235826A1 Quinuclidine acrylamides
08/2002
08/29/2002	WO2002066469A2 Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands
08/29/2002	WO2002066468A2 Heterocyclic urea derivatives and their use as dopamine d3 receptor ligands
08/29/2002	WO2002066446A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
08/29/2002	US20020119991 Respiratory system disorders; antiallergens
08/29/2002	US20020119961 Bridged piperazine derivatives
08/29/2002	CA2438318A1 Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands
08/29/2002	CA2438316A1 Heterocyclic urea derivatives and their use as dopamine d3 receptor ligands
08/29/2002	CA2438264A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
08/28/2002	EP1233964A1 New use and novel n-azabicyclo-amide derivatives
08/27/2002	US6440996 Monomeric and dimeric heterocycles, and therapeutic uses thereof
08/22/2002	WO2002064128A1 Treatment of diseases characterized by excessive or insufficient cell death
08/22/2002	US20020115680 Anticholinergics which may be used as medicaments as well as processes for preparing them
08/22/2002	US20020115662 Delta-opioid or mu-opioid receptor modulators; useful analgesics, immunosuppressants, antiinflammatory agents, agents for the treatment of respiratory diseases.
08/21/2002	EP0756596B1 Tropane-2-aldoxime derivatives as neurotransmitter reuptake inhibitors
08/15/2002	WO2002062788A1 Sulfonamide compounds, their preparation and use

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