Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
08/1995
08/17/1995CA2182568A1 Novel carbamate derivative and medicinal composition containing the same
08/15/1995US5442078 Intermediates for specific 5-HT3 antagonists
08/15/1995CA1336713C Process for the preparation of 1-methylindazole-3-carboxylic acid
08/08/1995US5439666 Iodinated neuroprobe for mapping monoamine reuptake sites
07/1995
07/26/1995EP0664293A1 2-Phenyl-7-azabicycloheptanes and 6-phenyl-8-azabicyclo
07/25/1995CA1336428C Substituted dibenzocycloheptenimines
07/18/1995US5434161 Imidazopyridines as serotonergic 5-HT3 antagonists
06/1995
06/27/1995US5428064 N-phenyl-amino-terminated non-peptidyl α-succinamidoacyl aminodiolsas anti-hypertensive agents
06/27/1995US5428054 Renin inhibitor
06/25/1995CA2138745A1 2-phenyl-7-azabicycloheptanes and 6 phenyl-8-azabicyclooctanes
06/13/1995US5424319 Renin inhibitors
06/13/1995US5424307 Renin inhibitors
05/1995
05/31/1995EP0655056A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
05/31/1995EP0654997A1 Compositions of substituted azaspiranes and methods of treating psoriasis therewith
05/30/1995US5420127 Morpholino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/24/1995EP0654023A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists
05/23/1995US5418249 Renin inhibitors
05/23/1995US5418244 Antiperspirants, mydriatic
05/16/1995US5416111 Cyano-containing n-phenyl-amino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416104 Oxazolidinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416095 Tetrahydro-quinolinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416092 3-azabicyclo[3.2.1]-oct-8-yl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416085 3-oxa-8-azabicyclo[3.2.1]oct-8-yl terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416083 Benzodiazepinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/09/1995US5414012 Indalyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/09/1995US5413779 Cocaine receptor binding ligands
05/04/1995WO1995011901A1 Substituted 2-carboxyalkyl-3-(fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders
05/03/1995EP0650486A1 New analgesic and nootropic drugs
05/02/1995US5411962 Benzomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411958 Benzothiomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411957 3-azabicyclo[3.2.1]-nonanyl-terminated non-piptidyl alpha-succinamidoacyl aminodiols as anti-hypertensive agents
03/1995
03/29/1995EP0645391A2 Aminobenzoic acid derivatives
03/29/1995EP0644775A1 Cocaine receptor binding ligands
03/28/1995US5401750 Derivatives of substituted imidazol-2-one and process for their preparation
03/23/1995WO1995005364A3 Inhibitors of biogenic amine transporters
03/21/1995US5399562 Indolones useful as serotonergic agents
03/15/1995EP0642507A1 Catalytic antibodies against cocaine and methods of using and producing same
03/14/1995US5397800 Gastrointestinal disorders
03/09/1995WO1995006635A1 Carbamate derivative and medicine containing the same
03/07/1995US5395832 Benzamide derivatives
03/01/1995EP0640601A1 Benzamide derivative
02/1995
02/23/1995WO1995005379A1 Antipsychotic method
02/23/1995WO1995005364A2 Inhibitors of biogenic amine transporters
02/23/1995CA2169287A1 Inhibitors of biogenic amine transporters
02/21/1995US5391761 Preparation of novel amido-alcohol derivatives and their therapeutic uses
02/21/1995US5391744 Cocaine analogs
02/21/1995US5391742 2-(8-Azabicyclo(3.2.1)oct-8-yl)alkanols
02/21/1995US5391549 Cinnoline-3-carboxylic acid derivatives
02/14/1995US5389647 Renin inhibitors
02/14/1995US5389643 Aminobenzoic acid derivatives useful for treating gastro-intestinal conditions
02/08/1995CN1098413A Xanthene derivant
02/02/1995WO1995003301A1 Azalicyclooctane derivatives as anti-arrhythmic agents
01/1995
01/31/1995US5385898 Hypertensive agents; cardiovascular disorders; renin inhibitors; glaucoma
01/24/1995CA1334095C Aroyl urea and carbamic acid derivatives
01/12/1995WO1995001184A1 An iodinated neuroprobe for mapping monoamine reuptake sites
01/10/1995US5380848 8-azabicyclo(3.2.1)octanes
01/03/1995US5378712 Antithrombosis
12/1994
12/28/1994EP0630375A1 Biologically active tropane derivatives
12/27/1994US5376667 Derivatives of benzoylecgonine, ecgonine and their multiple pharmacological properties
12/22/1994WO1994029306A1 Cocaine derivatives and their use as anticholinergic agents
12/21/1994EP0629190A1 Compounds as calcium channel antagonists
12/20/1994US5374636 2,3-trans-disubstituted tropane compounds which have useful pharmaceutical utility
11/1994
11/30/1994CN1095720A Derivatives of benzoylecgonine, ecgonine and ecgonidine and methods for preparing and using same
11/29/1994US5369113 Certain 2,3-diphenyl-2-(1,2,4-oxadiazol-5-yl)tropanes useful as dopamide reuptake inhibitors
11/24/1994WO1994026274A1 Treatment process with biologically active tropane derivatives
11/24/1994CA2163095A1 Treatment process with biologically active tropane derivatives
11/23/1994EP0625507A2 Urea derivatives and their use as acat inhibitors
11/22/1994CA2123728A1 Urea derivatives and their use as acat inhibitors
11/22/1994CA1333174C 2-azabicyclo¬2.2.1|hept-5-ene-2-acetic acid, derivatives thereof and related compounds, process for the preparation of said compounds and the use of said compounds for the manufacture of n-phosphonomethylglycine
11/15/1994US5364863 Treatment of migraine, emesis, schizophrenia, anxiety, gastrointestinal disorders
11/08/1994US5362740 Dihydrobenzofuran carboxamides and process for their preparation
11/08/1994US5362734 Certain benzo-quinolizine compounds and derivatives thereof
10/1994
10/25/1994US5358954 Benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-HT receptor antagonists
10/19/1994EP0644775A4 Cocaine receptor binding ligands.
10/18/1994US5356912 3-(5-isoxazolyl)-1-methyl-1,2,3,6-tetrahydropyridine useful for treating Alzheimer's disease
10/18/1994US5356905 Neuroprotective 3-piperidino-4-hydroxychroman derivatives and analogs
10/11/1994US5354495 Alkenoylcarbamate compounds as elasticity, adhesion, and dispersibility enhancer
09/1994
09/15/1994WO1994020496A1 Heterocyclic compounds and their preparation and use
09/15/1994WO1994020464A1 Coupling method using selective amination of maleimide
09/15/1994CA2156704A1 Coupling method using selective amination of maleimide
09/13/1994US5346911 Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
09/07/1994EP0613899A2 Cocaine derivative, protein conjugate thereof, monoclonal antibody producing cell line, method for preparing the cell line and monoclonal antibody
08/1994
08/30/1994US5342949 2 step process for preparing biologically active tropane derivatives and starting material therefore
08/24/1994EP0611370A1 Pyridine-3-carboxylic acid esters or amides useful as 5-ht 3? antagonists
08/23/1994US5340936 8-azabicyclo[3.2.1]octane methanone and corresponding oximes
08/16/1994US5338754 Treating stroke or central nervous system disorders
08/10/1994EP0609335A1 Methods for the treatment of hyperlipidemia using azaspiranes
08/03/1994EP0608336A1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment
08/02/1994US5334599 Heteroaryl-8-azabicyclo[3,2,1]octanes as antipsychotic agents, 5-HT3 receptor antagonists and inhibitors of the reuptake of serotonin
07/1994
07/21/1994WO1994015935A1 Derivatives of benzoylecgonine, ecgonine and ecgonidine as medicines
07/19/1994US5330990 Substituted urea compounds and their preparation and use
07/05/1994US5326768 5-hydroxytryptamine antagonists
06/1994
06/29/1994EP0604355A2 Akyl Substituted heterocyclic compounds
06/29/1994EP0604354A2 Antidepressant and antiparkinsonian compounds
06/29/1994EP0604352A2 Aryl substituted heterocyclic compounds
06/29/1994CN1025194C 2-azabicyclo |2,2,1¨ hept-5-ene-2-acetic acid derivatives and the prepn. of related compounds
06/21/1994US5322951 Antiserotine agent
06/09/1994WO1994012497A1 Heterocyclic compound
06/07/1994US5319085 Quinoline derivative having serotonin-3 receptor antagonizing activity
05/1994
05/10/1994US5310912 Ester-substituted nortropane
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