Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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08/17/1995 | CA2182568A1 Novel carbamate derivative and medicinal composition containing the same |
08/15/1995 | US5442078 Intermediates for specific 5-HT3 antagonists |
08/15/1995 | CA1336713C Process for the preparation of 1-methylindazole-3-carboxylic acid |
08/08/1995 | US5439666 Iodinated neuroprobe for mapping monoamine reuptake sites |
07/26/1995 | EP0664293A1 2-Phenyl-7-azabicycloheptanes and 6-phenyl-8-azabicyclo |
07/25/1995 | CA1336428C Substituted dibenzocycloheptenimines |
07/18/1995 | US5434161 Imidazopyridines as serotonergic 5-HT3 antagonists |
06/27/1995 | US5428064 N-phenyl-amino-terminated non-peptidyl α-succinamidoacyl aminodiolsas anti-hypertensive agents |
06/27/1995 | US5428054 Renin inhibitor |
06/25/1995 | CA2138745A1 2-phenyl-7-azabicycloheptanes and 6 phenyl-8-azabicyclooctanes |
06/13/1995 | US5424319 Renin inhibitors |
06/13/1995 | US5424307 Renin inhibitors |
05/31/1995 | EP0655056A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension |
05/31/1995 | EP0654997A1 Compositions of substituted azaspiranes and methods of treating psoriasis therewith |
05/30/1995 | US5420127 Morpholino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/24/1995 | EP0654023A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists |
05/23/1995 | US5418249 Renin inhibitors |
05/23/1995 | US5418244 Antiperspirants, mydriatic |
05/16/1995 | US5416111 Cyano-containing n-phenyl-amino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/16/1995 | US5416104 Oxazolidinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/16/1995 | US5416095 Tetrahydro-quinolinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/16/1995 | US5416092 3-azabicyclo[3.2.1]-oct-8-yl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/16/1995 | US5416085 3-oxa-8-azabicyclo[3.2.1]oct-8-yl terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/16/1995 | US5416083 Benzodiazepinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/09/1995 | US5414012 Indalyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/09/1995 | US5413779 Cocaine receptor binding ligands |
05/04/1995 | WO1995011901A1 Substituted 2-carboxyalkyl-3-(fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders |
05/03/1995 | EP0650486A1 New analgesic and nootropic drugs |
05/02/1995 | US5411962 Benzomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/02/1995 | US5411958 Benzothiomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents |
05/02/1995 | US5411957 3-azabicyclo[3.2.1]-nonanyl-terminated non-piptidyl alpha-succinamidoacyl aminodiols as anti-hypertensive agents |
03/29/1995 | EP0645391A2 Aminobenzoic acid derivatives |
03/29/1995 | EP0644775A1 Cocaine receptor binding ligands |
03/28/1995 | US5401750 Derivatives of substituted imidazol-2-one and process for their preparation |
03/23/1995 | WO1995005364A3 Inhibitors of biogenic amine transporters |
03/21/1995 | US5399562 Indolones useful as serotonergic agents |
03/15/1995 | EP0642507A1 Catalytic antibodies against cocaine and methods of using and producing same |
03/14/1995 | US5397800 Gastrointestinal disorders |
03/09/1995 | WO1995006635A1 Carbamate derivative and medicine containing the same |
03/07/1995 | US5395832 Benzamide derivatives |
03/01/1995 | EP0640601A1 Benzamide derivative |
02/23/1995 | WO1995005379A1 Antipsychotic method |
02/23/1995 | WO1995005364A2 Inhibitors of biogenic amine transporters |
02/23/1995 | CA2169287A1 Inhibitors of biogenic amine transporters |
02/21/1995 | US5391761 Preparation of novel amido-alcohol derivatives and their therapeutic uses |
02/21/1995 | US5391744 Cocaine analogs |
02/21/1995 | US5391742 2-(8-Azabicyclo(3.2.1)oct-8-yl)alkanols |
02/21/1995 | US5391549 Cinnoline-3-carboxylic acid derivatives |
02/14/1995 | US5389647 Renin inhibitors |
02/14/1995 | US5389643 Aminobenzoic acid derivatives useful for treating gastro-intestinal conditions |
02/08/1995 | CN1098413A Xanthene derivant |
02/02/1995 | WO1995003301A1 Azalicyclooctane derivatives as anti-arrhythmic agents |
01/31/1995 | US5385898 Hypertensive agents; cardiovascular disorders; renin inhibitors; glaucoma |
01/24/1995 | CA1334095C Aroyl urea and carbamic acid derivatives |
01/12/1995 | WO1995001184A1 An iodinated neuroprobe for mapping monoamine reuptake sites |
01/10/1995 | US5380848 8-azabicyclo(3.2.1)octanes |
01/03/1995 | US5378712 Antithrombosis |
12/28/1994 | EP0630375A1 Biologically active tropane derivatives |
12/27/1994 | US5376667 Derivatives of benzoylecgonine, ecgonine and their multiple pharmacological properties |
12/22/1994 | WO1994029306A1 Cocaine derivatives and their use as anticholinergic agents |
12/21/1994 | EP0629190A1 Compounds as calcium channel antagonists |
12/20/1994 | US5374636 2,3-trans-disubstituted tropane compounds which have useful pharmaceutical utility |
11/30/1994 | CN1095720A Derivatives of benzoylecgonine, ecgonine and ecgonidine and methods for preparing and using same |
11/29/1994 | US5369113 Certain 2,3-diphenyl-2-(1,2,4-oxadiazol-5-yl)tropanes useful as dopamide reuptake inhibitors |
11/24/1994 | WO1994026274A1 Treatment process with biologically active tropane derivatives |
11/24/1994 | CA2163095A1 Treatment process with biologically active tropane derivatives |
11/23/1994 | EP0625507A2 Urea derivatives and their use as acat inhibitors |
11/22/1994 | CA2123728A1 Urea derivatives and their use as acat inhibitors |
11/22/1994 | CA1333174C 2-azabicyclo¬2.2.1|hept-5-ene-2-acetic acid, derivatives thereof and related compounds, process for the preparation of said compounds and the use of said compounds for the manufacture of n-phosphonomethylglycine |
11/15/1994 | US5364863 Treatment of migraine, emesis, schizophrenia, anxiety, gastrointestinal disorders |
11/08/1994 | US5362740 Dihydrobenzofuran carboxamides and process for their preparation |
11/08/1994 | US5362734 Certain benzo-quinolizine compounds and derivatives thereof |
10/25/1994 | US5358954 Benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-HT receptor antagonists |
10/19/1994 | EP0644775A4 Cocaine receptor binding ligands. |
10/18/1994 | US5356912 3-(5-isoxazolyl)-1-methyl-1,2,3,6-tetrahydropyridine useful for treating Alzheimer's disease |
10/18/1994 | US5356905 Neuroprotective 3-piperidino-4-hydroxychroman derivatives and analogs |
10/11/1994 | US5354495 Alkenoylcarbamate compounds as elasticity, adhesion, and dispersibility enhancer |
09/15/1994 | WO1994020496A1 Heterocyclic compounds and their preparation and use |
09/15/1994 | WO1994020464A1 Coupling method using selective amination of maleimide |
09/15/1994 | CA2156704A1 Coupling method using selective amination of maleimide |
09/13/1994 | US5346911 Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment |
09/07/1994 | EP0613899A2 Cocaine derivative, protein conjugate thereof, monoclonal antibody producing cell line, method for preparing the cell line and monoclonal antibody |
08/30/1994 | US5342949 2 step process for preparing biologically active tropane derivatives and starting material therefore |
08/24/1994 | EP0611370A1 Pyridine-3-carboxylic acid esters or amides useful as 5-ht 3? antagonists |
08/23/1994 | US5340936 8-azabicyclo[3.2.1]octane methanone and corresponding oximes |
08/16/1994 | US5338754 Treating stroke or central nervous system disorders |
08/10/1994 | EP0609335A1 Methods for the treatment of hyperlipidemia using azaspiranes |
08/03/1994 | EP0608336A1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment |
08/02/1994 | US5334599 Heteroaryl-8-azabicyclo[3,2,1]octanes as antipsychotic agents, 5-HT3 receptor antagonists and inhibitors of the reuptake of serotonin |
07/21/1994 | WO1994015935A1 Derivatives of benzoylecgonine, ecgonine and ecgonidine as medicines |
07/19/1994 | US5330990 Substituted urea compounds and their preparation and use |
07/05/1994 | US5326768 5-hydroxytryptamine antagonists |
06/29/1994 | EP0604355A2 Akyl Substituted heterocyclic compounds |
06/29/1994 | EP0604354A2 Antidepressant and antiparkinsonian compounds |
06/29/1994 | EP0604352A2 Aryl substituted heterocyclic compounds |
06/29/1994 | CN1025194C 2-azabicyclo |2,2,1¨ hept-5-ene-2-acetic acid derivatives and the prepn. of related compounds |
06/21/1994 | US5322951 Antiserotine agent |
06/09/1994 | WO1994012497A1 Heterocyclic compound |
06/07/1994 | US5319085 Quinoline derivative having serotonin-3 receptor antagonizing activity |
05/10/1994 | US5310912 Ester-substituted nortropane |