Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
10/1996
10/08/1996US5563148 Specific 5-HT3 antagonists
10/03/1996WO1996030371A1 Method for the preparation of esters of anhydroecgonine
10/02/1996EP0734385A1 Substituted 2-carboxyalkyl-3-(fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders
10/01/1996US5561149 For nasal administration
09/1996
09/24/1996US5559123 Derivatives of benzoylecgonine, ecgonine and ecgonidine and methods for preparing and using same
09/17/1996US5556851 Treatment of nausea or emesis from anticancer drugs or x-ray treatment
09/10/1996US5554626 Substituted heterocyclic compounds as dopamine-reuptake inhibitors
09/03/1996US5552408 Benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-ht receptor antagonists
09/03/1996US5552407 Bronchodilator agents
08/1996
08/28/1996EP0727993A1 (non descriptive)-a method for delaying hiv individual aids by administration of substituted azaspirane compounds
08/13/1996US5545658 Amino acid derivatives
08/06/1996US5543426 Use of certain 3,7-disubstituted indole compounds for treating depression or cognitive disorders
07/1996
07/25/1996WO1996022290A1 Compounds having effects on serotonin-related systems
07/25/1996CA2210220A1 Compounds having effects on serotonin-related systems
07/24/1996EP0722941A2 Compounds having effects on serotonin-related systems
07/23/1996US5539116 Method and compositions for the synthesis of BCH-189 and related compounds
07/18/1996WO1996021644A1 Indole derivatives useful in the treatment of osteoporosis
07/18/1996CA2209936A1 Indole derivatives useful in the treatment of osteoporosis
07/11/1996WO1996020940A1 A novel radioisotope labelled compound, a mixture comprising said compound and a method for its preparation
07/11/1996CA2206954A1 A novel radioisotope labelled compound, a mixture comprising said compound and a method for its preparation
07/04/1996WO1996003401A3 Process for the production of aminoazobicycloalkanes from oximes
07/03/1996CN1032209C Process for preparing 2-piperidino-1-alkanol derivatives as antiischemic agents
06/1996
06/27/1996WO1996019493A1 N-SUBSTITUTED GLYCINE DERIVATIVES AS INHIBITORS OF FACTOR Xa
06/18/1996US5527912 Useful intreatment of central nervous system disorders
06/18/1996US5527813 Heterocyclic compounds and their preparation and use
06/12/1996EP0715855A2 NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis
06/11/1996US5525613 Covalently coupled benzoylecgonine ecgonine and ecgonidine
06/05/1996EP0714394A1 Antipsychotic method
06/04/1996US5523299 Administering in treatment of psychotic disorders
05/1996
05/29/1996EP0713484A1 Inhibitors of biogenic amine transporters
05/22/1996EP0703791A4 An iodinated neuroprobe for mapping monoamine reuptake sites
05/17/1996WO1996014316A1 A method of treating urinary bladder dysfunctions
05/15/1996EP0711299A1 AZABICYCLOALKYL DERIVATIVES OF IMIDAZO(1,5-a)INDOL-3-ONE AS 5HT 3 ANTAGONISTS
05/08/1996EP0710662A1 Quinolinecarboxylic acid derivative
05/08/1996EP0710236A1 Azalicyclooctane derivatives as anti-arrhythmic agents
05/08/1996EP0472526B1 5-AMINOCARBONYL-5H-DIBENZO a,d]CYCLOHEPTEN-5,10-IMINES FOR TREATMENT OF EPILEPSY AND COCAINE ADDICTION
05/02/1996WO1996012711A1 Heterocyclic compounds and their use
05/02/1996CA2203426A1 Heterocyclic compounds and their use
05/01/1996EP0709381A1 Heterocyclic compounds and their preparation and use
04/1996
04/30/1996US5512579 Aminobenzoic acid derivatives
04/25/1996WO1996011928A1 Enantioselective synthesis of seven-membered carbocycles and tropanes
04/25/1996CA2202615A1 Enantioselective synthesis of seven-membered carbocycles and tropanes
04/25/1996CA2161176A1 Heterocyclic compounds and their preparation and use
04/24/1996CN1121349A Heterocyclic compounds and their preparation and use
04/18/1996WO1996011192A1 Lta4 hydrolase inhibitors
04/18/1996CA2202371A1 Lta4 hydrolase inhibitors
04/10/1996EP0688316A4 Coupling method using selective amination of maleimide
04/09/1996US5506359 Cocaine analogues and their use as cocaine drug therapies and therapeutic and imaging agents for neurodegenerative disorders
04/03/1996EP0703791A1 An iodinated neuroprobe for mapping monoamine reuptake sites
03/1996
03/28/1996WO1996009302A1 Bicyclic carboxamides as 5-ht1a antagonists
03/28/1996CA2200443A1 Bicyclic carboxamides as 5-ht1a antagonists
03/21/1996WO1996008480A1 Neurokinin antagonists
03/21/1996CA2200083A1 Neurokinin antagonists
03/19/1996US5500422 Benzamide derivative
03/12/1996US5498610 Blocking agent for n-methyl aspartic acid receptor sites
03/06/1996EP0699906A2 Method for detecting the contamination of a surface with an analyte
03/05/1996US5496953 Dopamine transporter sites, radioactive, diagnosis, imaging, nortropane derivatives
02/1996
02/29/1996WO1996006083A1 2-(piperazinyl-1-carbonylmethyl)-1,4-dihydropyridines as bradykinin antagonists
02/29/1996WO1996006082A1 Dihydropyridine derivatives as bradykinin antagonists
02/29/1996WO1996006081A1 Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkanol derivatives
02/28/1996EP0697871A1 Treatment process with biologically active tropane derivatives
02/28/1996EP0494978B1 Heterocyclic compounds
02/22/1996WO1996005193A1 (azetidin-1-ylalkyl)lactams as tachykinin antagonists
02/20/1996US5493026 Labeled with radioactive isotopes for tomography
02/13/1996US5491148 Treating gastrointestinal, cardiovascular, central nervous system disorders, emesis, pain
02/08/1996WO1996003401A2 Process for the production of aminoazobicycloalkanes from oximes
02/08/1996WO1996003123A1 Methods
01/1996
01/09/1996US5482938 Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
01/03/1996EP0690055A1 Stereoselective process for making endo-tropanamine and like compounds
01/02/1996CA2053247C 5-aminocarbonyl-5h-dibenzo(a,d)cyclohepten-5, 10-imines for treatment of epilepsy and cocaine addiction
12/1995
12/28/1995CA2152312A1 Stereoselective process for making endo-tropanamine and like compounds
12/27/1995EP0688316A1 Coupling method using selective amination of maleimide
12/21/1995WO1995034561A1 Benzoylecgonine, ecgonine and ecgonidine derivatives
12/21/1995CA2190611A1 Covalently coupled benzoylecgonine, ecgonine and ecgonidine derivatives
12/20/1995EP0687266A1 Heterocyclic compounds and their preparation and use
11/1995
11/30/1995WO1995032209A1 AZABICYCLOALKYL DERIVATIVES OF IMIDAZO(1,5-a)INDOL-3-ONE AS 5HT3 ANTAGONISTS
11/30/1995CA2166621A1 Azabicycloalkyl derivatives of imidazo(1,5-a)indol-3-one and process for their preparation
11/23/1995WO1995031455A1 Quinolinecarboxylic acid derivative
11/23/1995CA2167055A1 Quinolinecarboxylic acid derivative
11/21/1995US5468758 5-HT antagonists
11/16/1995WO1995030640A1 Substituted fused and bridged bicyclic compounds as therapeutic agents
10/1995
10/31/1995US5463028 Compound comprising a methyl ecgonine group chemically attached to a phenylphosphonic group which is an analog to an intermediate of the hydrolysis transition-state of a cocaine benzoyl ester group
10/26/1995WO1995028401A1 Tropane-2-aldoxine derivatives as neurotransmitter reuptake inhibitors
10/24/1995US5461053 Pyridazine derivatives
10/24/1995CA1337415C Indole derivatives
10/18/1995EP0677051A1 Derivatives of benzoylecgonine, ecgonine and ecgonidine as medicines
10/17/1995US5459161 Cognition activators
10/17/1995US5459127 Cationic lipids for intracellular delivery of biologically active molecules
10/17/1995CA1337347C Benzimidazoline-2-one-1-carboxylic acid derivatives useful as 5-ht receptor antagonists
10/11/1995CN1029960C Neuroprotective 3-piperidino-4-hydroxychroman derivatives
10/10/1995US5457273 Processing Waste solidification
10/03/1995US5455250 Treating central nervous system disorders
10/03/1995CA1337199C Five-membered ring systems with bonded azacyclic ring substituents
09/1995
09/20/1995EP0564650B1 Quinoline derivative
09/08/1995WO1995023799A1 Process for the preparation of an indazole-3-carboxamide derivative
09/06/1995EP0670319A1 Heterocyclic compound
08/1995
08/31/1995WO1995023147A1 Heterocyclic compound
08/31/1995CA2184366A1 Heterocyclic compound
08/22/1995US5444070 Treating a disease or disorder which is responsive to the inhibition of dopamine reuptake by administering a tropane derivative
08/17/1995WO1995021820A1 Novel carbamate derivative and medicinal composition containing the same
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