| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 04/27/1994 | EP0593511A1 Piperidine derivates having anxiolytic effect |
| 04/26/1994 | US5306723 A racemic optical compound for treating central nervous system is also an antihypertensive agent |
| 04/26/1994 | US5306718 Analgesics, cognition activators |
| 04/19/1994 | US5304552 Renin inhibitors |
| 04/13/1994 | EP0591426A1 Sigma receptor ligands and the use thereof |
| 03/30/1994 | CN1084516A Azacyclic and azabicyclic alkyliden hydroxylamines |
| 03/29/1994 | US5298510 Medicaments |
| 03/29/1994 | CA1328106C Anticholinergic compounds, pharmaceutical compositions and method of treatment |
| 03/23/1994 | EP0587800A1 Immunomodulatory azaspiranes |
| 03/23/1994 | CN1084169A Compounds |
| 03/23/1994 | CA2086403A1 Cocaine analogs |
| 03/15/1994 | CA1327750C Therapeutic use of serotonin-antagonists |
| 03/08/1994 | CA1327573C Pyridazinamine derivatives |
| 03/03/1994 | WO1994004495A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension |
| 03/03/1994 | WO1994004151A1 Compositions of substituted azaspiranes and methods of treating psoriasis therewith |
| 03/03/1994 | WO1994004146A1 Cocaine analogues and their use as cocaine drug therapies and therapeutic and imaging agents for neurodegenerative disorders |
| 03/02/1994 | EP0584192A1 Prodrug esters of phenolic 2-piperidino-1-alkanols |
| 03/01/1994 | US5290795 Substituted urea compound and use |
| 02/22/1994 | US5288872 A tropane ring cholinergic agents for alzheimer's, parkinson's diseases |
| 02/22/1994 | US5288731 2,6-methano-2H-1-benzoxocincarboxylic acids, esters and amides |
| 02/17/1994 | WO1994003426A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists |
| 02/17/1994 | CA2141791A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists |
| 02/02/1994 | EP0581165A2 Acrylamide derivatives as antirussive agent |
| 02/01/1994 | US5283344 Coupling method using selective amination of maleimide |
| 01/26/1994 | EP0579615A1 New bi- and tricyclic aminoalcohol esters, their preparation and their use in medicaments |
| 01/20/1994 | WO1994001435A1 New analgesic and nootropic drugs |
| 01/20/1994 | CA2139739A1 New analgesic and nootropic drugs |
| 01/12/1994 | EP0578560A2 Amido-alcohol derivatives as psychotropic agents |
| 01/09/1994 | CA2100007A1 Preparation of new amido-alcohol derivatives and their therapeutical applications |
| 01/06/1994 | WO1994000448A1 Azacyclic and azabicyclic hydroxylamines as muscarinic receptor agonists |
| 01/04/1994 | US5276036 Central nervous system |
| 12/29/1993 | EP0575581A1 Novel cocaine derivatives and protein and polypeptide cocaine derivative conjugates and labels |
| 12/21/1993 | US5272160 2-piperidino-1-alkanol derivatives as antiischemic agents |
| 12/21/1993 | US5272154 3,7 substituted indole and indazole compounds and pharmaceutical compositions containing them |
| 12/07/1993 | US5268480 Cocaine analogs |
| 12/01/1993 | EP0422154B1 Therapeutic use of 5-ht3 receptor antagonists |
| 11/23/1993 | US5264618 For transport of biological active agents into cells for viral agents or polynucleotides or immunogenic peptides |
| 11/16/1993 | US5262428 Biologically active tropane derivatives |
| 11/16/1993 | US5262427 3-substituted and optionally 1-substituted azacyclic or azabicyclic compounds, pharmaceutical compositions, thereof and their use as stimulants of cognitive functions |
| 11/09/1993 | US5260314 Certain 3-(1,2,5-oxa- or thiadiazol-4-yl)-1-azabicyclo [2.2.2]octanes having pharmaceutical properties |
| 11/09/1993 | US5260303 Imidazopyridines as serotonergic 5-HT3 antagonists |
| 11/09/1993 | US5260293 Simulate central muscarinic acetlycholine receptors |
| 11/03/1993 | EP0567767A1 Crystalline forms of endo-2,3-dihydro-N-(8-methyl-8-azabicyclo 3.2.1 oct-3-yl)-2-oxo-1H-benzimidazole-1-carboxamide hydrochloride monohydrate and of endo-3-ethyl-2,3-dihydro-N-(8-methyl-8-azabicyclo 3.2.1 oct-3-yl)-2-oxo-1H-benzimidazole-1-carboxamide hydrochloride monohydrate as 5-HT antagonists |
| 11/02/1993 | US5258388 Antisecretory agents, mydriatic agents and antiperspirants |
| 10/28/1993 | WO1993021236A1 Visible photosensitizers for photopolymerizable compositions |
| 10/27/1993 | EP0566609A1 Azabicydic and azatricydic derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them |
| 10/14/1993 | WO1993020076A1 Catalytic antibodies against cocaine and methods of using and producing same |
| 10/13/1993 | EP0564650A1 Quinoline derivative |
| 10/12/1993 | US5252570 Amidino and guanidino derivatives |
| 10/06/1993 | EP0563087A1 Azabicyclic amides or esters of halogenated benzoic acids |
| 09/29/1993 | EP0561910A1 Pharmaceuticals |
| 09/28/1993 | US5248684 Certain 2-oxo-quinoline carboxylates or corresponding carboxamides useful as anti-emetics and suppressants of migraine |
| 09/21/1993 | US5246942 Pharmaceutically useful dibenzofurancarboxamides of specific stereo-configuration |
| 09/16/1993 | WO1993018033A1 Biologically active tropane derivatives |
| 09/15/1993 | EP0560633A1 Use of tropane derivatives for the manufacture of a medicament for the treatment of neurodegenerative diseases |
| 09/15/1993 | EP0560604A1 Cinnoline-3-carboxylic acid derivatives as 5-HT3 antagonists |
| 09/14/1993 | US5244910 Renin inhibitors |
| 09/13/1993 | CA2091375A1 Cinnoline-3-carboxylic acid derivatives |
| 09/08/1993 | EP0559297A1 Use of heterocyclic derivatives for the manufacture of medicaments |
| 09/07/1993 | US5242929 Derivatives of substituted imidazol-2-one and process for their preparation |
| 08/19/1993 | WO1993015735A1 (non descriptive)-a method for delaying hiv individual aids by administration of substituted azaspirane compounds |
| 08/17/1993 | US5236808 Visible photosensitizers for photopolymerizable compositions |
| 08/11/1993 | EP0554794A1 Aminobenzoic acid derivatives |
| 08/11/1993 | EP0554247A1 Neuroprotective indolone and related derivatives |
| 08/11/1993 | CN1075145A Aminobenzoic acid derivatives |
| 08/10/1993 | US5234931 Heteroaryl-8-azabicyclo[3.2.1]octanes as antipsychotic agents, 5-HT3 receptor antagonists and inhibitors of the reuptake of serotonin |
| 08/05/1993 | WO1993015052A1 Compounds as calcium channel antagonists |
| 08/03/1993 | US5233042 Cocaine derivatives |
| 07/27/1993 | US5231184 Viricide intermediate |
| 07/21/1993 | EP0551963A2 Use of heterocyclic derivatives for the manufacture of medicaments |
| 07/14/1993 | EP0550587A1 Stereoselective preparation of acid sensitive amides and intermediates useful in said preparation |
| 07/13/1993 | US5227385 Method for treatment of neurodegenerative diseases |
| 07/06/1993 | US5225419 Certain 1,8-ethano or propano-1,4-dihydro-4-oxo-quinoline-3-carboxamides and derivatives thereof |
| 06/29/1993 | US5223528 Anticholinergic compounds, composititons and methods of treatment |
| 06/29/1993 | US5223511 Benzimidazoline-2-oxo-1-carboxylic acid compounds useful as 5-HT receptor antagonists |
| 06/23/1993 | CN1021328C Process for preparing pyridazinamine derivatives |
| 06/17/1993 | WO1993012111A1 Novel cocaine derivatives and protein and polypeptide cocaine derivative conjugates and labels |
| 06/17/1993 | DE4140861A1 Enantiomers of quaternary tropaic acid alkaloid derivs. - sepd. from racemates and enantiomer mixts using chiral polysaccharide phases and certain organic and aq. eluants and anionic modifiers |
| 06/09/1993 | EP0544779A1 Heterocyclic compounds and their preparation and use |
| 06/02/1993 | EP0543936A1 Renin inhibitors |
| 05/27/1993 | WO1993009814A1 Cocaine receptor binding ligands |
| 05/18/1993 | US5212185 Piperidinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension |
| 05/11/1993 | US5210085 Method for the synthesis, compositions and use of 2'-deoxy-5-fluoro-3'-thiacytidine and related compounds |
| 04/29/1993 | WO1993008192A1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment |
| 04/29/1993 | WO1993008186A1 Pyridine-3-carboxylic acid esters or amides useful as 5-ht3 antagonists |
| 04/29/1993 | WO1993008185A1 N-aryl-n1-azabicyclo-ureas as 5-ht3 antagonists |
| 04/29/1993 | WO1993007871A1 Methods for the treatment of hyperlipidemia using azaspiranes |
| 04/20/1993 | US5204470 Azabicyclic derivatives |
| 04/20/1993 | US5204466 Stereoselective preparation of biologically active isomer |
| 04/14/1993 | EP0536512A1 A method and intermediates for the preparation of 6-fluorobenzisothiazoles |
| 04/13/1993 | US5202333 Tricyclic 5-HT3 receptor antagonists |
| 04/13/1993 | US5202318 Tricyclic compounds acting at serotonin receptor subtypes |
| 04/07/1993 | EP0513200A4 Method and compositions for the synthesis of bch-189 and related compounds |
| 04/06/1993 | US5200413 Indolyl carboxamides useful treating migraine, cluster headache, trigeminal neuralgia or emesis |
| 04/01/1993 | WO1993006092A1 Piperazinyl (sulfonyl)amide derivatives of camphor as oxytocin antagonists |
| 03/31/1993 | CN1070399A Substituted amide derivatives of piperizinylcamphorsulfonyl oxytocin antagonists |
| 03/23/1993 | US5196535 Viricides |
| 03/23/1993 | US5196415 5-aminocarbonyl-5H-dibenzo[a.d]cyclohepten-5,10-imines for treatment of epilepsy and cocaine addiction |
| 03/17/1993 | EP0532097A1 Piperazinyl(sulfon)amide derivatives of camphor as oxytocin antagonists |
| 03/17/1993 | CN1020102C Preparation for bicyclic carboxylic ether and bicyclic carboxylic amide |