Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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08/15/2002 | WO2002062324A2 A treatment of oesophageal motility disorders and gastro-oesophageal reflux disease |
08/15/2002 | WO2002044175A3 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit |
08/15/2002 | US20020110529 Inhalable powder containing tiotropium |
08/15/2002 | CA2437380A1 A treatment of oesophageal motility disorders and gastro-oesophageal reflux disease |
08/14/2002 | EP1230219A1 Aromatic sulfons hydroxamic acid metalloprotease inhibitor |
08/13/2002 | US6432976 Analgesics; side effect reduction |
08/13/2002 | CA2060573C N-(aryloxyalkyl)heteroaryl-8-azabicyclo¬3.2.1|octanes, intermediates and a process for the preparation thereof and their use as medicaments |
08/08/2002 | US20020107235 Carbamate and hydroxy groups containing phenanthrene derivatives; useful to treat obesity, diabetes and inflammation |
08/08/2002 | US20020106332 Process for preparing powder formulations |
08/07/2002 | EP1228060A1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof |
08/06/2002 | CA2236707C Fused tropane-derivatives, their preparation and use |
08/01/2002 | WO2002058695A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents |
08/01/2002 | US20020102659 Cocaethylene immunogens and antibodies |
08/01/2002 | CA2431904A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents |
07/25/2002 | WO2002057263A1 8-azabicyclo "3.2.1.! octanes as insecticides |
07/25/2002 | WO2002057262A2 Bicyclic amines as insecticides |
07/25/2002 | WO2002057254A1 Compositions for prevention or treatment of hepatopathy |
07/25/2002 | WO2002036591A3 Inhalative solution formulation containing a tiotropium salt |
07/25/2002 | WO2002032901A3 Bridged piperazine derivatives |
07/25/2002 | WO2001040188A9 Curcumin analogues for treating cancer |
07/25/2002 | US20020099184 Radiolabeled compounds useful as imaging agents for visualizing the location and density of serotonin transporter by tomography imaging; as diagnostic and therapeutic agents for diseases associated with serotonin transporter dysfunction |
07/25/2002 | CA2435141A1 Compositions for prevention or treatment of hepatopathy |
07/24/2002 | EP1224180A2 Substituted azoles |
07/24/2002 | EP0900218B1 Heterocyclic compounds |
07/17/2002 | EP0882044B1 1,4-dihydropyridine compounds as bradykinin antagonists |
07/17/2002 | CN1087737C Dihygropyridine derivatives as bradykinin ant agonists |
07/10/2002 | EP1221441A2 LTA4 Hydrolase inhibitors |
07/10/2002 | EP1220840A2 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
07/09/2002 | US6417221 Tropane analogs and methods for inhibition of monoamine transport |
07/04/2002 | WO2002051840A1 Method for producing the anticholinergic agent tiotropium bromide |
07/04/2002 | WO2002051808A2 Muscarinic antagonists |
07/04/2002 | US20020086887 N-Acylsulfonamide apoptosis promoters |
07/03/2002 | EP1218372A1 Novel spiroheterocyclic compounds useful as reversible inhibitors of cysteine proteases |
07/03/2002 | EP0831941A4 Iodinated neuroprobes for mapping monoamine reuptake sites |
07/02/2002 | US6414149 Treating diabetes, treating or preventing diabetic complications |
07/02/2002 | US6413978 Basic derivatives of benz[e] isoindol-1-ones and pyrrolo[3,4-c] quinolin-1-ones with 5-HT3-antagonistic activity, their preparation and their therapeutic use |
06/27/2002 | WO2002030390A3 Method for producing powdery formulations |
06/26/2002 | CN1086698C Oxadizoles, processes for their preparation and their use as medicaments |
06/19/2002 | EP1214303A1 Heterocyclic compounds and methods of use thereof |
06/19/2002 | EP1067903B1 Improved crystal structure |
06/13/2002 | WO2002012245A3 Azabicyclic derivatives and their therapeutic use |
06/13/2002 | WO2002004442A9 Azabicyclic compounds as inhibitors of nicotinic cholinergic receptors |
06/12/2002 | EP1213289A1 N-benzenesulfonyl L-proline compounds as bradykinin antagonists |
06/12/2002 | EP1212299A1 Substituted piperidine compounds useful as modulators of chemokine receptor activity |
06/12/2002 | EP1212103A1 4-fluoroalkyl-3-halophenyl nortropanes |
06/12/2002 | EP1211940A1 Azabicyclo and azacyclo oxime and amine compounds as pesticides |
06/12/2002 | EP0942909B1 Bicyclic amine derivatives |
06/12/2002 | CN1353702A Adamantane derivatives |
06/11/2002 | CA2169838C Antipsychotic method |
06/11/2002 | CA2112084C Antidepressant and antiparkinsonian compounds |
06/06/2002 | WO2002044175A2 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit |
06/04/2002 | US6399042 4-fluoroalkyl-3-halophenyl nortropanes |
05/30/2002 | WO2001080905A3 Sigma-2 receptors as biomarkers of tumor cell proliferation |
05/29/2002 | CN1351601A Heterocyclic compounds binding chemotactic factor receptor |
05/29/2002 | CN1351497A Aminopyrimidines as sorbitol dehydrogenase inhibitors |
05/28/2002 | US6395748 Use treating Alzheimer's disease; monoamine reuptake inhibitor tropanes such as tesofensine (2-methoxymethyl-3-(3,4-dichlorophenyl)-tropane) |
05/23/2002 | WO2000063204A3 Substituted azoles |
05/23/2002 | US20020061913 Bicyclic amine derivatives |
05/21/2002 | US6392045 9-azobicyclo[3.3.1] non-2-ene derivatives as cholinergic ligands at nicotinic ACH receptors |
05/21/2002 | US6391883 Bicyclic amines |
05/16/2002 | WO2002004442A3 Azabicyclic compounds as inhibitors of nicotinic cholinergic receptors |
05/15/2002 | EP1204644A1 Synthesis of substituted amidines |
05/10/2002 | WO2002036106A2 Novel medicament compositions based on anticholinergics and corticosteroids |
05/09/2002 | WO2002036591A2 Inhalative solution formulation containing a tiotropium salt |
05/09/2002 | US20020055631 N-acylsulfonamide apoptosis promoters |
05/08/2002 | EP1202985A2 Chemokine receptor antagonists |
05/08/2002 | DE10152369A1 Stable, propellant-free inhalable liquid medicament for treating asthma or chronic obstructive pulmonary disease, containing tiotropium salt and antiallergic agent, antihistamine, steroid or leukotriene antagonist |
05/07/2002 | US6384042 Systemic use of 5-HT3 receptor antagonists against rheumatic inflammatory processes |
05/07/2002 | US6383490 Drug abuse or dependance |
05/02/2002 | WO2002034736A1 Process for preparation of bicyclic and polycyclic molecules |
05/02/2002 | US20020052355 Inhibition of serotonin reuptake; especially 2-(azabicycloalkyl)alkylenyl)isoquinolin-3-one compounds |
05/02/2002 | EP1201649A1 Glucocorticoid receptor modulators |
05/02/2002 | CA2427021A1 Process for preparation of bicyclic and polycyclic molecules |
05/01/2002 | CN1083840C 8-azabicyclo [3.2.1] oct-2-ene derivs., their preparation and use |
04/30/2002 | CA2233541C 8-azabicyclo[3.2.1]oct-2-ene derivatives, their preparation and use |
04/25/2002 | WO2002032901A2 Bridged piperazine derivatives |
04/25/2002 | US20020049220 Substituted azoles |
04/25/2002 | US20020049212 Benzimidazole compounds and salts containing piperidine ring are useful in treatment or prevention or medical conditions selected from pain, and inflammatoy diseases; analgesics |
04/25/2002 | CA2423789A1 Bridged piperazine derivatives |
04/23/2002 | US6376510 Administering a alkoxy- and acyloxy-substituted aralkyl and aralkenyl bis quaternary ammonium derivatives of cyclic alkanol diesters to a human as muscle relaxants |
04/18/2002 | WO2002030405A2 Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance |
04/18/2002 | WO2002030389A1 Novel tiotropium-containing inhalation powder |
04/18/2002 | DE10050995A1 New benzylic acid azabicyclooctane ester quaternary salts useful as anticholinergic agents, especially in treatment of asthma and chronic obstructive pulmonary disease |
04/18/2002 | DE10050994A1 New diphenylalkanoic acid azabicyclooctane ester quaternary salts useful as anticholinergic agents, especially in treatment of asthma and chronic obstructive pulmonary disease |
04/17/2002 | EP0734385B1 Substituted 2-carboxyalkyl-3-(fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders |
04/11/2002 | US20020042426 Novel basic derivatives of benz[e] isoindol-1-ones and pyrrolo[3,4-c] quinolin-1ones with 5-HT3-antagonistic activity, their preparation and their therapeutic use |
04/11/2002 | US20020042421 Antiinflammatory agents |
04/10/2002 | CN1082371C NK-1 receptor antagonist and 5HT3 receptor antagonists for treating emesis |
04/04/2002 | WO2001090717A3 Linker arms for nanocrystals and compounds thereof |
04/04/2002 | WO2001090716A3 Linker arms for nanocrystals and compounds thereof |
04/02/2002 | US6365125 Using organotin compound |
03/28/2002 | WO2002024636A2 N-acylsulfonamide apoptosis promoters |
03/28/2002 | WO2001090106A3 Tryasolyl tropane derivatives as ccr5 modulators |
03/27/2002 | EP0782574B1 Bicyclic carboxamides as 5-ht1a receptors ligands |
03/21/2002 | WO2001087846A3 Tricyclic pyrazole derivatives as protein kinase inhibitors |
03/21/2002 | US20020035122 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives |
03/19/2002 | US6358492 Dopamine transporter imaging ligand |
03/14/2002 | WO2001070734A3 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha |
03/14/2002 | WO2001066543A3 3-(diarylmethylene)-8-azabicyclo[3.2.1]octane derivatives |
03/13/2002 | EP1185275A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors |