Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
08/2002
08/15/2002WO2002062324A2 A treatment of oesophageal motility disorders and gastro-oesophageal reflux disease
08/15/2002WO2002044175A3 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit
08/15/2002US20020110529 Inhalable powder containing tiotropium
08/15/2002CA2437380A1 A treatment of oesophageal motility disorders and gastro-oesophageal reflux disease
08/14/2002EP1230219A1 Aromatic sulfons hydroxamic acid metalloprotease inhibitor
08/13/2002US6432976 Analgesics; side effect reduction
08/13/2002CA2060573C N-(aryloxyalkyl)heteroaryl-8-azabicyclo¬3.2.1|octanes, intermediates and a process for the preparation thereof and their use as medicaments
08/08/2002US20020107235 Carbamate and hydroxy groups containing phenanthrene derivatives; useful to treat obesity, diabetes and inflammation
08/08/2002US20020106332 Process for preparing powder formulations
08/07/2002EP1228060A1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof
08/06/2002CA2236707C Fused tropane-derivatives, their preparation and use
08/01/2002WO2002058695A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
08/01/2002US20020102659 Cocaethylene immunogens and antibodies
08/01/2002CA2431904A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
07/2002
07/25/2002WO2002057263A1 8-azabicyclo "3.2.1.! octanes as insecticides
07/25/2002WO2002057262A2 Bicyclic amines as insecticides
07/25/2002WO2002057254A1 Compositions for prevention or treatment of hepatopathy
07/25/2002WO2002036591A3 Inhalative solution formulation containing a tiotropium salt
07/25/2002WO2002032901A3 Bridged piperazine derivatives
07/25/2002WO2001040188A9 Curcumin analogues for treating cancer
07/25/2002US20020099184 Radiolabeled compounds useful as imaging agents for visualizing the location and density of serotonin transporter by tomography imaging; as diagnostic and therapeutic agents for diseases associated with serotonin transporter dysfunction
07/25/2002CA2435141A1 Compositions for prevention or treatment of hepatopathy
07/24/2002EP1224180A2 Substituted azoles
07/24/2002EP0900218B1 Heterocyclic compounds
07/17/2002EP0882044B1 1,4-dihydropyridine compounds as bradykinin antagonists
07/17/2002CN1087737C Dihygropyridine derivatives as bradykinin ant agonists
07/10/2002EP1221441A2 LTA4 Hydrolase inhibitors
07/10/2002EP1220840A2 Bicyclic and tricyclic amines as modulators of chemokine receptor activity
07/09/2002US6417221 Tropane analogs and methods for inhibition of monoamine transport
07/04/2002WO2002051840A1 Method for producing the anticholinergic agent tiotropium bromide
07/04/2002WO2002051808A2 Muscarinic antagonists
07/04/2002US20020086887 N-Acylsulfonamide apoptosis promoters
07/03/2002EP1218372A1 Novel spiroheterocyclic compounds useful as reversible inhibitors of cysteine proteases
07/03/2002EP0831941A4 Iodinated neuroprobes for mapping monoamine reuptake sites
07/02/2002US6414149 Treating diabetes, treating or preventing diabetic complications
07/02/2002US6413978 Basic derivatives of benz[e] isoindol-1-ones and pyrrolo[3,4-c] quinolin-1-ones with 5-HT3-antagonistic activity, their preparation and their therapeutic use
06/2002
06/27/2002WO2002030390A3 Method for producing powdery formulations
06/26/2002CN1086698C Oxadizoles, processes for their preparation and their use as medicaments
06/19/2002EP1214303A1 Heterocyclic compounds and methods of use thereof
06/19/2002EP1067903B1 Improved crystal structure
06/13/2002WO2002012245A3 Azabicyclic derivatives and their therapeutic use
06/13/2002WO2002004442A9 Azabicyclic compounds as inhibitors of nicotinic cholinergic receptors
06/12/2002EP1213289A1 N-benzenesulfonyl L-proline compounds as bradykinin antagonists
06/12/2002EP1212299A1 Substituted piperidine compounds useful as modulators of chemokine receptor activity
06/12/2002EP1212103A1 4-fluoroalkyl-3-halophenyl nortropanes
06/12/2002EP1211940A1 Azabicyclo and azacyclo oxime and amine compounds as pesticides
06/12/2002EP0942909B1 Bicyclic amine derivatives
06/12/2002CN1353702A Adamantane derivatives
06/11/2002CA2169838C Antipsychotic method
06/11/2002CA2112084C Antidepressant and antiparkinsonian compounds
06/06/2002WO2002044175A2 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit
06/04/2002US6399042 4-fluoroalkyl-3-halophenyl nortropanes
05/2002
05/30/2002WO2001080905A3 Sigma-2 receptors as biomarkers of tumor cell proliferation
05/29/2002CN1351601A Heterocyclic compounds binding chemotactic factor receptor
05/29/2002CN1351497A Aminopyrimidines as sorbitol dehydrogenase inhibitors
05/28/2002US6395748 Use treating Alzheimer's disease; monoamine reuptake inhibitor tropanes such as tesofensine (2-methoxymethyl-3-(3,4-dichlorophenyl)-tropane)
05/23/2002WO2000063204A3 Substituted azoles
05/23/2002US20020061913 Bicyclic amine derivatives
05/21/2002US6392045 9-azobicyclo[3.3.1] non-2-ene derivatives as cholinergic ligands at nicotinic ACH receptors
05/21/2002US6391883 Bicyclic amines
05/16/2002WO2002004442A3 Azabicyclic compounds as inhibitors of nicotinic cholinergic receptors
05/15/2002EP1204644A1 Synthesis of substituted amidines
05/10/2002WO2002036106A2 Novel medicament compositions based on anticholinergics and corticosteroids
05/09/2002WO2002036591A2 Inhalative solution formulation containing a tiotropium salt
05/09/2002US20020055631 N-acylsulfonamide apoptosis promoters
05/08/2002EP1202985A2 Chemokine receptor antagonists
05/08/2002DE10152369A1 Stable, propellant-free inhalable liquid medicament for treating asthma or chronic obstructive pulmonary disease, containing tiotropium salt and antiallergic agent, antihistamine, steroid or leukotriene antagonist
05/07/2002US6384042 Systemic use of 5-HT3 receptor antagonists against rheumatic inflammatory processes
05/07/2002US6383490 Drug abuse or dependance
05/02/2002WO2002034736A1 Process for preparation of bicyclic and polycyclic molecules
05/02/2002US20020052355 Inhibition of serotonin reuptake; especially 2-(azabicycloalkyl)alkylenyl)isoquinolin-3-one compounds
05/02/2002EP1201649A1 Glucocorticoid receptor modulators
05/02/2002CA2427021A1 Process for preparation of bicyclic and polycyclic molecules
05/01/2002CN1083840C 8-azabicyclo [3.2.1] oct-2-ene derivs., their preparation and use
04/2002
04/30/2002CA2233541C 8-azabicyclo[3.2.1]oct-2-ene derivatives, their preparation and use
04/25/2002WO2002032901A2 Bridged piperazine derivatives
04/25/2002US20020049220 Substituted azoles
04/25/2002US20020049212 Benzimidazole compounds and salts containing piperidine ring are useful in treatment or prevention or medical conditions selected from pain, and inflammatoy diseases; analgesics
04/25/2002CA2423789A1 Bridged piperazine derivatives
04/23/2002US6376510 Administering a alkoxy- and acyloxy-substituted aralkyl and aralkenyl bis quaternary ammonium derivatives of cyclic alkanol diesters to a human as muscle relaxants
04/18/2002WO2002030405A2 Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance
04/18/2002WO2002030389A1 Novel tiotropium-containing inhalation powder
04/18/2002DE10050995A1 New benzylic acid azabicyclooctane ester quaternary salts useful as anticholinergic agents, especially in treatment of asthma and chronic obstructive pulmonary disease
04/18/2002DE10050994A1 New diphenylalkanoic acid azabicyclooctane ester quaternary salts useful as anticholinergic agents, especially in treatment of asthma and chronic obstructive pulmonary disease
04/17/2002EP0734385B1 Substituted 2-carboxyalkyl-3-(fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders
04/11/2002US20020042426 Novel basic derivatives of benz[e] isoindol-1-ones and pyrrolo[3,4-c] quinolin-1ones with 5-HT3-antagonistic activity, their preparation and their therapeutic use
04/11/2002US20020042421 Antiinflammatory agents
04/10/2002CN1082371C NK-1 receptor antagonist and 5HT3 receptor antagonists for treating emesis
04/04/2002WO2001090717A3 Linker arms for nanocrystals and compounds thereof
04/04/2002WO2001090716A3 Linker arms for nanocrystals and compounds thereof
04/02/2002US6365125 Using organotin compound
03/2002
03/28/2002WO2002024636A2 N-acylsulfonamide apoptosis promoters
03/28/2002WO2001090106A3 Tryasolyl tropane derivatives as ccr5 modulators
03/27/2002EP0782574B1 Bicyclic carboxamides as 5-ht1a receptors ligands
03/21/2002WO2001087846A3 Tricyclic pyrazole derivatives as protein kinase inhibitors
03/21/2002US20020035122 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives
03/19/2002US6358492 Dopamine transporter imaging ligand
03/14/2002WO2001070734A3 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
03/14/2002WO2001066543A3 3-(diarylmethylene)-8-azabicyclo[3.2.1]octane derivatives
03/13/2002EP1185275A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors
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