| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
|---|
| 04/24/2003 | WO2003032997A1 Pyrimidine derivatives, pharmaceutical agent containing said compounds, use and method for making same |
| 04/23/2003 | EP1303274A1 Method of promoting smoking cessation |
| 04/22/2003 | US6552036 3-(Diarylmethylene)-8-azabicyclo[3.2.1]octane derivatives |
| 04/22/2003 | US6552015 Azabicycloalkane derivatives and therapeutic uses thereof |
| 04/17/2003 | WO2003031452A2 4-haloethenylphenyl tropane:serotonin transporter imaging agents |
| 04/17/2003 | WO2003031397A1 Acylsulfonamides as inhibitors of steroid sulfatase |
| 04/17/2003 | CA2459727A1 4-haloethenylphenyl tropane: serotonin transporter imaging agents |
| 04/17/2003 | CA2458453A1 Acylsulfonamides as inhibitors of steroid sulfatase |
| 04/16/2003 | EP1302458A1 Ester derivatives |
| 04/15/2003 | US6548041 Diagnosis, therapy of central nervous system disorders |
| 04/11/2003 | WO2002032899A1 Novel anticholinergic agents that can be used as medicaments and method for the production thereof |
| 04/11/2003 | WO2002032898A2 Novel anticholinergics, method for the production thereof and use thereof as medicaments |
| 04/11/2003 | WO2002030928A1 Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament |
| 04/10/2003 | WO2003028650A2 Benzimidazolidinone derivatives as muscarinic agents |
| 04/10/2003 | WO2003028459A1 Nicotinic acid-heterocyclyl-amides and analogous pyrimidine derivatives serving as pesticides |
| 04/10/2003 | WO2003004493A8 Novel compounds, their preparation and use |
| 04/10/2003 | US20030069269 Tropane analogs and methods for inhibition of monoamine |
| 04/10/2003 | CA2457647A1 Benzimidazolidinone derivatives as muscarinic agents |
| 04/09/2003 | EP0993301B1 Cocaine receptor binding ligands |
| 04/09/2003 | CN1104892C Method for curing tinnitus by nerve protecting agent |
| 04/08/2003 | CA2062271C Derivatives of substituted imidazol-2-one and process for their preparation |
| 04/04/2003 | WO2002030390A2 Method for producing powdery formulations |
| 04/03/2003 | WO2003002531A3 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 04/03/2003 | WO2003002530A3 Pyrrolidines as dipeptidyl peptidase inhibitors |
| 04/03/2003 | US20030065179 Diabetic therapy |
| 04/02/2003 | EP0912512B1 Sulphonamide derivatives and their use in the treatment of cns disorders |
| 04/02/2003 | EP0587800B1 Immunomodulatory azaspiranes |
| 04/02/2003 | CN1104430C Angiogenesis inhibiting pyridazinamines |
| 04/01/2003 | US6541481 Substituted bicyclic derivatives useful as anticancer agents |
| 04/01/2003 | US6541004 An immunogen comprising an antigenic protein bonded to at least one molecule of N-methyl tropane substituted at the 2-benzoyloxy group, which is substituted at para position with an aliphatic linking group of form 1-6 carbon atoms |
| 03/27/2003 | WO2003002553A3 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 03/27/2003 | US20030060494 Dipeptidyl peptidase IV inhibiting agent; treatment of gastrointestinal disorders |
| 03/27/2003 | US20030060481 The use of scopolamine salts |
| 03/25/2003 | US6537524 Inflammatory or obstructive airways disease |
| 03/25/2003 | US6537522 Metabolically stable cocaine analogs such as 2-carbometh-oxy-3-(4-iodophenyl)-tropane; chemical intermediates for compounds having high affinities for dopamine and serotonin reuptake sites in brain |
| 03/20/2003 | WO2003022836A1 Nitrogen-containing heterocyclic compounds and their use as raf inhibitors |
| 03/20/2003 | WO2002012245B1 Azabicyclic derivatives and their therapeutic use |
| 03/20/2003 | US20030055049 For therapy of abnormal cell growth, such as cancer, in mammals |
| 03/19/2003 | EP1292281A1 Novel tiotropium-containing inhalation powder |
| 03/19/2003 | EP1037637B1 Use of 5ht1a receptor antagonists for preventing and/or treating temporal lobe epilepsy |
| 03/18/2003 | US6534522 Subtype-selective NMDA receptor ligands and the use thereof |
| 03/13/2003 | WO2002068388A3 Acylated piperidine derivatives as melanocortin-4 receptor agonists |
| 03/13/2003 | WO2002066469A3 Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands |
| 03/12/2003 | EP1289525A2 Tricyclic pyrazole derivatives as protein kinase inhibitors |
| 03/11/2003 | US6531484 Viricides for preventing infection by HIV, treating infection by HIV, delaying of the onset of AIDS, or treating AIDS |
| 03/11/2003 | US6531483 Treating psychostimulant abuse, inhibiting action of psychostimulant, inhibiting neurotransmitter re-uptake, treating Parkinson's Disease, treating depression |
| 03/06/2003 | WO2003017764A1 Substituted propargylamines |
| 03/06/2003 | WO2002072570A3 Non-imidazole compounds as histamine h3 antagonists |
| 03/04/2003 | CA2218913C Substituted oximes, hydrazones and olefins as neurokinin antagonists |
| 02/27/2003 | WO2003015517A1 Agonists and antagonists of 5h3-like receptors of invertebrate s as pesticides |
| 02/27/2003 | CA2456290A1 Agonists and antagonists of 5h3-like receptors of invertebrate s as pesticides |
| 02/26/2003 | EP1284974A2 Triazolyl tropane derivatives as ccr5 modulators |
| 02/26/2003 | EP1284730A1 Aralkyl ester soft drugs |
| 02/20/2003 | WO2003014114A2 Substituted amine derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 02/13/2003 | WO2002096855A3 Anticholinergic compounds and methods of use |
| 02/13/2003 | US20030032648 8-Aza-bicyclo[3.2.1]octan-3-ol derivatives of 2,3-dihydro-1,4-benodioxan as 5-HT1A antagonists |
| 02/13/2003 | US20030032645 Aryl-8-azabicyclo [3.2.1] octanes for the treatment of depression |
| 02/11/2003 | CA2154620C Method of detecting surface contamination by an analyte |
| 02/06/2003 | WO2003010159A1 Piperidine derivatives as nmda receptor antagonists |
| 02/06/2003 | WO2003009847A1 Substituted piperidines as modulators of the melanocortin receptor |
| 02/06/2003 | WO2002096423A3 Combination of a pde4 inhibitor and tiotropium or derivate thereof for treating obstructive airways |
| 02/06/2003 | CA2454903A1 Substituted piperazines as modulators of the melanocortin receptor |
| 02/06/2003 | CA2452328A1 Substituted piperidines as modulators of the melanocortin receptor |
| 02/04/2003 | US6514773 Method of detecting surface contamination by an analyte |
| 01/30/2003 | US20030023090 Used as imaging or pharmaceutical agents, in the diagnosis and therapy of drug addiction, depression, anorexia and neurodegenerative diseases |
| 01/30/2003 | US20030022917 Process for the manufacture of tropenol |
| 01/29/2003 | EP1278745A2 Sigma-2 receptors as biomarkers of tumor cell proliferation |
| 01/29/2003 | EP0984966B1 9-AZABICYCLO(3.3.1)NON-2-ENE AND NONANE DERIVATIVES AS CHOLINERGIC LIGANDS AT NICOTINIC ACh RECEPTORS |
| 01/29/2003 | EP0946553B1 8-azabicyclo 3.2.1]octane derivatives, their preparation and their use as insecticides |
| 01/23/2003 | WO2002051808A3 Muscarinic antagonists |
| 01/22/2003 | EP0901491B1 Tropane derivatives useable in particular for in vivo detection of dopamine transporters |
| 01/22/2003 | CN1392795A Novel tiotropiumonium-containing inhalation powder |
| 01/16/2003 | WO2003004493A1 Novel compounds, their preparation and use |
| 01/16/2003 | US20030013883 Tropane analogs binding to monoamine transporters |
| 01/16/2003 | US20030013675 Combination of an adenosine A2A-receptor agonist and tiotropium or a derivative thereof for treating obstructive airways and other inflammatory diseases |
| 01/16/2003 | CA2448913A1 Sulfone containing bicyclic aromatic ring compounds, their preparation and use as nicotinic acetyl-chloine receptors |
| 01/15/2003 | EP0851756B1 Use of ondansetron in the manufacture of a medicament for the treatment of tremor |
| 01/15/2003 | CN1098850C 3 alpha-alkylacyloxy-6 beta-alkylacyoxy tropene compound and their prepn. |
| 01/09/2003 | WO2003002562A1 Technical synthesis method for producing tropenol |
| 01/09/2003 | WO2003002553A2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 01/09/2003 | WO2003002531A2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 01/09/2003 | WO2003002530A2 Pyrrolidines as dipeptidyl peptidase inhibitors |
| 01/09/2003 | CA2450722A1 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 01/08/2003 | EP1272484A2 Benzoamide piperidine compounds as substance p antagonists |
| 01/07/2003 | US6503926 Nitrogen heterocycle compounds |
| 01/03/2003 | WO2003000265A1 Crystalline anticholinergic, method for its production, and use thereof in the production of a drug |
| 12/27/2002 | WO2002102801A1 Tropane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 12/26/2002 | US20020198178 Viricides for preventing infection by HIV, treating infection by HIV, delaying of the onset of AIDS, or treating AIDS |
| 12/24/2002 | US6498159 Such as 4-((3-chloro-4-methoxybenzyl)amino)-1-((4-hydroxy-4 -hydroxymethyl)piperidino)-6-phthalazine carbonitrile |
| 12/19/2002 | US20020193402 Azabicyclic ether derivatives and their use as therapeutic agents |
| 12/18/2002 | EP1079833A4 Cocaine receptor binding ligands |
| 12/17/2002 | US6495565 For therapy of acute infection, acute phase response, age related macular degeneration, alcoholism, anorexia, asthma, autoimmune disease, autoimmune hepatitis, bechet's disease, cachexia, calcium pyrophosphate dihydrtate deposition |
| 12/12/2002 | WO2002032898A3 Novel anticholinergics, method for the production thereof and use thereof as medicaments |
| 12/12/2002 | US20020188003 Cocaine receptor binding ligands |
| 12/11/2002 | EP1263758A2 3-(diarylmethylene)-8-azabicyclo[3.2.1]octane derivatives |
| 12/11/2002 | EP1263756A2 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha |
| 12/11/2002 | EP1263729A1 Azacyclic compounds for use in the treatment of serotonin related diseases |
| 12/11/2002 | CN1384830A Novel spiroheterocyclic compoundsus reversible inhibitors of cysteine proteases |
| 12/10/2002 | US6492355 Adamantane derivatives |
| 12/05/2002 | WO2002096906A1 Aryl-8-azabicyclo[3.2.1]octanes for the treatment of depression |