| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 09/04/2001 | US6284764 Antiproliferative agent |
| 08/30/2001 | US20010018444 Tropane-derivatives, their preparation and use |
| 08/29/2001 | EP1127887A1 Process for synthesizing anhydroecgonine derivative |
| 08/29/2001 | EP0815109B1 Method for the preparation of esters of anhydroecgonine |
| 08/28/2001 | US6281233 Method of treating gastrointestinal motility disorders |
| 08/28/2001 | US6281232 Azabicyclic ring-substituted thia- or oxadiazoles |
| 08/28/2001 | US6281226 Pleuromutilin derivatives as antimicrobials |
| 08/22/2001 | EP1125922A1 Pyrrolidine compounds and medicinal utilization thereof |
| 08/22/2001 | EP0777653B1 Dihygropyridine derivatives as bradykinin antagonists |
| 08/21/2001 | US6277872 Antiischemic agents; brain disorders |
| 08/16/2001 | WO2001009119A3 Chemokine receptor antagonists |
| 08/14/2001 | US6274757 Neuromuscular relaxants |
| 08/14/2001 | US6274623 Neuromuscular relaxants |
| 08/09/2001 | WO2001057008A1 2-benzothiazolyl urea derivatives and their use as protein kinase inhibitors |
| 08/09/2001 | CA2398754A1 2-benzothiazolyl urea derivatives and their use as protein kinase inhibitors |
| 08/08/2001 | EP1122257A1 Benzimidazole compounds as ORL1-receptor agonists |
| 08/07/2001 | US6271381 Cocaine derivative, protein conjugate thereof, monoclonal antibody producing cell line, method for preparing the cell line and monoclonal antibody |
| 08/07/2001 | US6271229 Method of treating gastrointestinal motility disorders |
| 08/02/2001 | CA2331029A1 Process for synthesizing anhydroecgonine derivative |
| 08/01/2001 | EP1119553A1 Monomeric and dimeric heterocycles, and therapeutic uses thereof |
| 07/31/2001 | US6268498 Process for the preparation of granisetron |
| 07/25/2001 | EP0876366B1 Angiogenesis inhibiting pyridazinamines |
| 07/24/2001 | US6265408 Sulphonamide derivatives and their use in the treatment of CNS disorders |
| 07/11/2001 | EP0885220B1 Tropane-derivatives, their preparation and use |
| 07/11/2001 | EP0823896B1 Substituted oximes, hydrazones and olefins as neurokinin antagonists |
| 07/10/2001 | US6258825 Analgesic, a reliever against tolerance to a narcotic analgesic represented by morphine, remedy for parkinsonism, a remedy for chorea, an antidepressant, a remedy for diabetes insipidus, a remedy for polyuria, or hypotension |
| 07/04/2001 | EP0579615B1 New bi- and tricyclic aminoalcohol esters, their preparation and their use in medicaments |
| 07/03/2001 | US6255319 5-aryl-3-(8-azabicyclo[3.2.1]oct-3-yl)-1,3,4-oxadiazol-2(3H)-one derivatives as 5-ht4 receptor ligands |
| 06/28/2001 | WO2001046191A1 4-[aryl(8-azabicyclo[3.2.1]octan-3-yl)]aminobenzoic acid derivatives |
| 06/28/2001 | WO2001046187A1 Azabicyclo[3.2.1]octane derivatives |
| 06/28/2001 | WO2001046186A1 Benzofuran derivatives |
| 06/28/2001 | US20010005722 endo-N-(9-methyl-9-azabicyclo[3.3.1]non-3-yl)-1-methyl-1h-indazole-3-carboxamide hydrochloride |
| 06/28/2001 | CA2395471A1 4-[aryl(8-azabicyclo[3.2.1]octan-3-yl)]aminobenzoic acid derivatives |
| 06/21/2001 | WO2001043746A1 Medicinal composition |
| 06/21/2001 | WO2001043745A1 The use of scopolamine salts |
| 06/20/2001 | EP0714394B1 Antipsychotic method with thiadiazole and oxadiazole derivatives |
| 06/13/2001 | EP1106615A1 Substituted 1,4-dihydropyridine compounds as bradykinin antagonists |
| 06/13/2001 | CN1067069C Bicycle amines as insecticides |
| 06/12/2001 | US6245773 Benign prostatic hyperplamia; reduction of intraocular pressure |
| 06/10/2001 | CA2327946A1 Substituted 1,4-dihydropyridine compounds as bradykinin antagonists |
| 06/07/2001 | WO2001040188A1 Curcumin analogues for treating cancer |
| 06/07/2001 | DE19952146A1 Arylalkane, Arylalkene und Aryl-azaalkane, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung Arylalkanes, aryl alkenes and aryl azaalkane, pharmaceutical compositions containing them and methods for their preparation |
| 06/07/2001 | CA2393440A1 Curcumin analogs with anti-tumor and anti-angiogenic properties |
| 06/06/2001 | CN1066730C Bicycle amines as insecticides |
| 06/05/2001 | US6241963 Dopamine and serotonin transporter ligands and imaging agents |
| 05/30/2001 | EP1102751A1 Novel bi- and tri-cyclic aza compounds and their uses |
| 05/29/2001 | US6239175 Carbamoyloxy derivatives of mutiline and their use as antibacterials |
| 05/29/2001 | CA2195923C Azetidines |
| 05/25/2001 | WO2001036417A1 New use and novel n-azabicyclo-amide derivatives |
| 05/25/2001 | CA2389604A1 New use and novel n-azabicyclo-amide derivatives |
| 05/23/2001 | EP1100781A1 High affinity ligands for nociceptin receptor orl-1 |
| 05/23/2001 | EP0900218A4 Heterocyclic compounds |
| 05/22/2001 | US6235747 6-phenyl-pyridin-2-ylamine derivatives |
| 05/22/2001 | US6235732 Neurokinin antagonists |
| 05/10/2001 | WO2001032649A1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof |
| 05/10/2001 | WO2001032179A1 8-aza-bicyclo[3.2.1]octane nmda/nr2b antagonists |
| 05/10/2001 | CA2388171A1 8-aza-bicyclo[3.2.1]octane nmda/nr2b antagonists |
| 05/10/2001 | CA2387613A1 Arylalkanes, arylalkenes and aryl-azaalkanes, pharmaceutical compositions containing these compounds and processes for preparing them |
| 04/26/2001 | WO2001029034A1 Quinuclidine acrylamides |
| 04/26/2001 | WO2001029000A2 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
| 04/26/2001 | WO2000071519A3 Immunopotentiator agents |
| 04/26/2001 | CA2386049A1 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
| 04/24/2001 | US6221879 8-azabicyclo[3.2.1] octane-3-methanamine derivatives as ligands of D2 and D3 dopamine and 5HT1A and 5HT2 serotonin receptors |
| 04/17/2001 | US6218404 Therapy and prophylaxis of neuronal loss associated with stroke, ischemia, cns trauma, hypoglycemia and surgery, neuro-degenerative diseases including alzheimer's disease, amyotrophic lateral sclerosis, huntington's disease |
| 04/17/2001 | CA2097815C Quinoline derivative |
| 04/17/2001 | CA2080475C Neuroprotective indolone and related derivatives |
| 04/12/2001 | WO2001025236A2 A stereoselective process for the preparation of endo-3-aminoazabicycloalkanes |
| 04/04/2001 | EP1088819A2 6-azauracil derivatives as thyroid receptor ligands |
| 04/04/2001 | EP0710662B1 Quinolinecarboxylic acid derivative |
| 03/28/2001 | EP1086066A1 Muscarinic receptor antagonists |
| 03/28/2001 | EP0775132B1 (azetidin-1-ylalkyl)lactams as tachykinin antagonists |
| 03/27/2001 | USRE37116 Nitrosated and nitrosylated compounds, and compositions and their use for treating respiratory disorders |
| 03/27/2001 | US6207677 Adminisering sigma receptor binding piperidine derivative for treating anxiety, epilepsy, convulsion, movement disorder, amnesia |
| 03/27/2001 | US6207676 Bicyclic amines |
| 03/22/2001 | WO2001019816A1 Novel spiroheterocyclic compounds useful as reversible inhibitors of cysteine proteases |
| 03/14/2001 | EP1082323A2 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them |
| 03/14/2001 | CN1063178C Aza-anthracyclinone derivatives |
| 03/13/2001 | US6200991 Imidazole derivatives, preparation and therapeutic application thereof |
| 03/08/2001 | WO2001016121A1 Heterocyclic compounds and methods of use thereof |
| 03/08/2001 | WO2001015532A1 Azabicyclo and azacyclo oxime and amine compounds as pesticides |
| 03/07/2001 | EP1081147A2 Substituted nortropanes and their use as imaging agents for neurodegenerative disorders |
| 03/07/2001 | EP1079833A1 Cocaine receptor binding ligands |
| 03/06/2001 | US6197762 Nitrosated and nitrosylated steroids compositions, and methods for treating respiratory disorders |
| 03/01/2001 | WO2001014374A2 Processes for the prepration of exo- and endo-indolotropanes |
| 03/01/2001 | WO2001014333A1 Substituted piperidine compounds useful as modulators of chemokine receptor activity |
| 02/27/2001 | US6194438 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one, and compositions and methods for inhibiting abnormal cell growth comprising said derivatives |
| 02/27/2001 | US6194416 Central nervous system disorders; alzheimer's disease |
| 02/27/2001 | CA2111204C Piperidine derivatives having anxiolytic effect |
| 02/22/2001 | WO2000078724A3 Imidazolinderivatives their preparation and their pharmaceutical use |
| 02/20/2001 | US6191272 Catalytic hydrogenation of the perchlorate in aqueous suspension with palladium, recovering catalyst by filtration, passing filtrate over anion exchange, and hydrogenating product to endo-nortropine intermediate to spasmolytics |
| 02/20/2001 | US6191135 Respiratory system disorders, antiinflammatory agents; analgesics |
| 02/14/2001 | EP0865441B1 1,2,3-thiadiazole carboxylic acid (thio)esters and the use thereof as a pest control agent or as a microbicide |
| 02/13/2001 | US6187776 Heterocyclic compounds and their use |
| 02/08/2001 | WO2001009119A2 Chemokine receptor antagonists |
| 02/07/2001 | CN1283197A Pleuromutilin derivatives as antimicrobials |
| 02/06/2001 | US6184389 Feature a plurality of functional groups attached to backbone and phosphoramidate sites |
| 02/06/2001 | US6184013 Antibody for reducing concentration of drug in patient |
| 02/01/2001 | WO2000063215A3 Indazole derivatives, preparation and therapeutic application thereof |
| 01/30/2001 | US6180083 Tropane derivatives useable in particular for in vivo detection of dopamine transporters |
| 01/24/2001 | EP1070711A2 Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses |