| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 09/30/1999 | WO1999048475A1 Improved crystal structure |
| 09/30/1999 | CA2325551A1 Improved crystal structure |
| 09/29/1999 | EP0944627A1 8-azabicyclo 3.2.1]octane-, 8-azabicyclo 3.2.1]oct-6-ene-, 9-azabicyclo 3.3.1]nonane-, 9-aza-3-oxabicyclo 3.3.1]nonane- and 9-aza-3-thiabicyclo 3.3.1]nonane derivatives, their preparation and their use as insecticides |
| 09/29/1999 | EP0944626A1 Tropane derivatives and method for their synthesis |
| 09/29/1999 | EP0944625A1 8-azabicyclo 3.2.1]octane-, 8-azabicyclo 3.2.1]oct-6-ene-, 9-azabicyclo 3.3.1]nonane-, 9-aza-3-oxabicyclo 3.3.1]nonane-, 9-aza-3-thiabicyclo 3.3.1]nonane derivatives, their preparation and their use as insecticides |
| 09/29/1999 | CN1230196A Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn. |
| 09/28/1999 | US5958945 Psychological disorders |
| 09/22/1999 | EP0942909A1 Bicyclic amine derivatives |
| 09/15/1999 | CN1228777A Pyridyl alkene- and pyridyl alkine-acid amides as cytostatics and immunosuppressives |
| 09/14/1999 | US5952505 Acetylating a tropic acid with acetychloride to form an acetylated tropic acid, reacting the acetylated tropic acid chloride in an inert solvent with the methanesulphonate of an amino alcohol, deacetylating |
| 09/07/1999 | US5948933 Tropane analogs and methods for inhibition of monoamine transport |
| 08/26/1999 | WO1999042452A1 Phthalazine derivatives and remedies for erectile dysfunction |
| 08/25/1999 | EP0937069A1 Piperazino derivatives as neurokinin antagonists |
| 08/25/1999 | CN1226886A Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation |
| 08/11/1999 | EP0934928A1 Cyclic amine derivatives |
| 08/11/1999 | EP0934316A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use |
| 08/11/1999 | EP0934288A1 Oxadiazoles, processes for their preparation and their use as medicaments |
| 08/10/1999 | US5935953 Methods for controlling invertebrate pests using cocaine receptor binding ligands |
| 08/10/1999 | CA1340695C Antibacterial agents |
| 08/05/1999 | WO1999038866A1 8-azabicyclo[3.2.1]oct-2-ene derivatives in labelled form and use of 8-azabicyclo[3.2.1]oct-2-ene derivatives in labelled and unlabelled form |
| 08/05/1999 | WO1999038865A1 8-azabicyclo(3.2.1)oct-2-ene derivatives as pesticides |
| 08/04/1999 | EP0644775B1 Cocaine Receptor Binding Ligands |
| 07/27/1999 | US5929247 Heterocyclic compounds and their preparation and use |
| 07/21/1999 | EP0929319A1 Dopamine and serotonin transporter ligands and imaging agents |
| 07/13/1999 | US5922732 Bicyclic amines |
| 07/07/1999 | EP0927192A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production |
| 07/06/1999 | US5919932 Biphenylamide derivatives as 5HT1D antagonists |
| 07/06/1999 | US5919802 Methods of preventing and/or treating temporal lobe epilepsy |
| 07/01/1999 | WO1999032117A1 Novel substituted pyridine compounds useful as modulators of acetylcholine receptors |
| 07/01/1999 | CA2315941A1 Novel substituted pyridine compounds useful as modulators of acetylcholine receptors |
| 06/30/1999 | EP0526540B1 Use of 5-ht4-receptor antagonists in the treatment of atrial fibrillation, including the prevention of stroke |
| 06/23/1999 | EP0923570A1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives |
| 06/23/1999 | EP0923536A1 Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation |
| 06/23/1999 | CN1043764C Bicycle carboxamides as 5-HT1A antagonists |
| 06/23/1999 | CN1043763C Tropane-aldoxine derivatives and preparation process and use thereof |
| 06/22/1999 | US5914400 Method and compositions for the synthesis of BCH-189 and related compounds |
| 06/17/1999 | WO1999029696A1 Piperidine derivatives |
| 06/17/1999 | WO1999029691A1 Process for the preparation of substituted 8-azabicyclo[3.2.1]octanes |
| 06/17/1999 | WO1999029690A1 Process for the preparation of 8-azabicyclo(3.2.1)octane derivatives |
| 06/17/1999 | WO1999029323A1 Use of 5ht1a receptor antagonists for preventing and/or treating temporal lobe epilepsy |
| 06/17/1999 | CA2312760A1 Use of 5ht1a receptor antagonists for preventing and/or treating temporal lobe epilepsy |
| 06/17/1999 | CA2309685A1 Process for the preparation of 8-azabicyclo(3.2.1)octane derivatives |
| 06/15/1999 | US5912254 Bicycle amine derivatives |
| 06/09/1999 | EP0748321B1 Process for the preparation of an indazole-3-carboxamide derivative |
| 06/03/1999 | WO1999026478A1 Bicyclic amines and their use as insecticides |
| 06/02/1999 | CN1218470A Bicycle amines as insecticides |
| 06/01/1999 | CA2103590C Benzamide derivative |
| 05/27/1999 | WO1999025710A1 Imidazole derivatives, preparation and therapeutic application thereof |
| 05/26/1999 | EP0859641A4 Dopamine transporter imaging agent |
| 05/19/1999 | EP0916668A1 Chemokine receptor antagonists |
| 05/12/1999 | EP0914321A1 Indole derivatives for the treatment of osteoporosis |
| 05/06/1999 | WO1999021855A1 Pleuromutilin derivatives as antimicrobials |
| 05/06/1999 | WO1999021854A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants |
| 05/06/1999 | EP0912512A1 Sulphonamide derivatives and their use in the treatment of cns disorders |
| 05/06/1999 | CA2306878A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants |
| 05/05/1999 | CN1216046A 3-[(1,2,3,4-tetrahydroisoquinoline-2-yl) methyl]-8-azabicyclo [3.2.1] octane derivs, their preparation and their use in therapeutics |
| 04/28/1999 | CN1215391A 6-phenylpyridyl-2-amine derivatives |
| 04/22/1999 | WO1999019325A1 8-azabicyclo [3.2.1] octane-3-methanamine derivatives as ligands of d2 and d3 dopamine and 5ht1a and 5ht2 serotonin receptors |
| 04/15/1999 | WO1999018103A1 Dopamine transporter imaging ligand |
| 04/15/1999 | WO1999017772A1 5ht4 agonists and antagonists |
| 04/15/1999 | CA2305754A1 Dopamine transporter imaging ligand |
| 04/15/1999 | CA2304826A1 5ht4 agonists and antagonists |
| 04/14/1999 | EP0908459A1 5-HT4 Agonists and antagonists |
| 04/14/1999 | CN1214046A 4,5-dihydronaphth [1,2-C] isoxazoles and derivatives thereof having CNS activity |
| 04/14/1999 | CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials |
| 04/13/1999 | CA1340492C Novel naphthyridine-and quinoline-carboxylic acids as bacterial agents |
| 03/31/1999 | EP0905135A2 Cocaine receptor binding ligands |
| 03/31/1999 | EP0904266A1 Nitrosated and nitrosylated compounds and compositions and their use for treating respiratory disorders |
| 03/30/1999 | US5889019 Heterocyclic compounds and their use |
| 03/30/1999 | US5888475 Labeled cocaine analogs |
| 03/24/1999 | CN1211982A Tropane derivatives, their preparation and use |
| 03/17/1999 | EP0901491A1 Tropane derivatives useable in particular for in vivo detection of dopamine transporters |
| 03/17/1999 | EP0901490A1 Bicyclic amines as insecticides |
| 03/17/1999 | EP0901489A1 Antagonists of gonadotropin releasing hormone |
| 03/17/1999 | CN1211251A 1,4-dihydropyridine compounds as bradykinin antagonists |
| 03/17/1999 | CN1042534C Aroyl urea derivatives or preparing method for additive salts of medicinal acid |
| 03/16/1999 | CA2164689C Nk-1 receptor antagonists and 5ht3 receptor antagonists for the treatment of emesis |
| 03/16/1999 | CA2058264C Dihydrobenzofuran carboxamides and process for their preparation |
| 03/10/1999 | EP0900218A1 Heterocyclic compounds |
| 03/04/1999 | WO1999010339A1 2-aminopyridines containing fused ring substituents as nos inhibitors |
| 03/03/1999 | EP0899261A1 Optical active 1,4-dihydropyridine compounds as bradykinin antagonists |
| 02/24/1999 | EP0897922A2 Cocaine receptor binding ligands |
| 02/18/1999 | CA2245041A1 Optical active 1,4-dihydropyridine compounds as bradykinin antagonists |
| 02/17/1999 | CN1208415A Angiogenesis inhibiting pyridazinamines |
| 02/10/1999 | CN1207739A 1,2,3-thiadiazole carboxylic acid (thio) esters and use thereof as pest control agent or as microbicide |
| 01/27/1999 | EP0892800A1 3- (1,2,3,4-tetrahydroisoquinoline-2-yl)methyl]-8-azabicyclo 3.2.1]octane derivatives, their preparation and their application in therapeutics |
| 01/26/1999 | US5864038 Fluorine or iodine labels for imaging |
| 01/21/1999 | WO1999002526A1 Tropane analogs and methods for inhibition of monoamine transport |
| 01/21/1999 | CA2297187A1 Tropane analogs and methods for inhibition of monoamine transport |
| 01/20/1999 | EP0891332A1 6-phenylpyridyl-2-amine derivatives |
| 01/19/1999 | US5861418 Aminobenzoic acid derivatives |
| 01/19/1999 | US5861402 1,4-dihydropyridine compounds |
| 01/19/1999 | CA2165294C An iodinated neuroprobe for mapping monoamine reuptake sites |
| 01/14/1999 | WO1999001449A1 2-substituted 4,5-diaryl imidazoles |
| 01/14/1999 | WO1998051311A3 Dihydropyrimidines and uses thereof |
| 01/14/1999 | CA2291758A1 2-substituted 4,5-diaryl imidazoles |
| 01/12/1999 | US5859024 Pesticides |
| 01/12/1999 | US5859011 Dihydropyridine derivatives as bradykinin antagonist |
| 01/07/1999 | EP0888345A1 Sigma-2 receptors as biomarkers of tumor cell proliferation |
| 01/05/1999 | US5856489 Catalytic hydrogenation |