Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
06/2000
06/28/2000CN1258294A 2-oxoimidazole derivs.
06/21/2000CN1257500A 9-azabicyclo (3,3,1) non-2-ene and nonane derivatives as cholinergic ligands at nicotinic ACH receptors
06/21/2000CN1257499A 8-Azabicyclo (3,2,1) oct-2-ene and octane derivatives as cholinergic ligands at nicotinic ACH receptors
06/20/2000US6077848 Benzoylecgonine, ecgonine and ecgonidine derivatives
06/15/2000WO2000034275A1 Process for the production of trifluoromethyltropanone cyanohydrin
06/15/2000CA2351471A1 Process for the production of trifluoromethyltropanone cyanohydrin
06/14/2000EP1007520A1 2-aminopyridines containing fused ring substituents as nos inhibitors
06/08/2000WO2000032600A1 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives
06/08/2000CA2342621A1 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives
06/07/2000EP1006113A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use to inhibit abnormal cell growth
06/07/2000CN1053187C Derivatives of benzoylecgonine, ecgonine and ecgonidine and methods for preparing and using same
06/06/2000US6071900 Heterocyclic compounds and their use
06/02/2000CA2291880A1 Novel derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one, and compositions and methods for inhibiting abnormal cell growth comprising said derivatives
05/2000
05/30/2000US6069152 Nervous system disorders; cardiovascular disorders; gastrointestinal disorders
05/23/2000US6066646 Insecticidal, acaricidal or nematicidal composition
05/17/2000EP1000359A1 Label for making a charge-transfer fluorescent probe
05/17/2000EP1000055A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS
05/11/2000WO2000026186A1 Pyrrolidine compounds and medicinal utilization thereof
05/11/2000CA2348879A1 Pyrrolidine compound and pharmaceutical use thereof
05/03/2000EP0996619A1 Tropane analogs and methods for inhibition of monoamine transport
04/2000
04/26/2000EP0554247B1 Neuroprotective indolone and related derivatives
04/25/2000US6054465 Used to stimulate hematopoiesis and for the treatment of bacterial infectious diseases.
04/25/2000CA2105575C Esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions
04/19/2000EP0993456A1 2-substituted 4,5-diaryl imidazoles
04/19/2000EP0993301A1 Cocaine receptor binding ligands
04/13/2000WO2000020390A1 Monomeric and dimeric heterocycles, and therapeutic uses thereof
04/13/2000CA2346537A1 Monomeric and dimeric heterocycles, and therapeutic uses thereof
04/05/2000EP0990653A1 2-oxoimidazole derivatives
04/04/2000US6046213 Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydroxyphenyl)-2-(piperidinyl-1)-alkanol derivatives
04/04/2000CA1340943C Azacyclic compounds and their preparation and use
03/2000
03/29/2000EP0988263A1 Process for the production of radioiodinated neuroreceptor agents
03/15/2000EP0984966A1 9-AZABICYCLO(3.3.1)NON-2-ENE AND NONANE DERIVATIVES AS CHOLINERGIC LIGANDS AT NICOTINIC ACh RECEPTORS
03/15/2000EP0984965A1 8-azabicyclo(3,2,1)oct-2-ene and octane derivatives as cholinergic ligands at nicotinic ach receptors
03/15/2000CN1050357C Process for preparing pure enantiomers of tropic acid esters
03/02/2000WO1999064043A9 Muscarinic receptor antagonists
02/2000
02/29/2000US6031099 Piperidine derivates having anxiolytic effect
02/29/2000US6030966 Heterocyclic compound and their use
02/23/2000EP0861252B1 Naphthamide derivatives of 3 beta-amino azabicyclo octane or nonane as neuroleptic agents
02/23/2000CN1245499A 8-azabicyclo [3,2,1] octane, 8-azabicyclo [3,2,1] oct-6-ene-,9-azabicyclo [3,2,1] nonane-, 9-aza-3-oxabicyclo [3,3,1] nonane- and 9-aza-3-thiabicyclo[3,3,1] nonane derivatives, their preparation and
02/23/2000CN1245498A 8-azabicyclo [3,2,1] octane derivatives their preparation and their use as insecticides
02/17/2000WO2000007994A1 Novel bi- and tri-cyclic aza compounds and their uses
02/17/2000CA2339122A1 Novel bi- and tri-cyclic aza compounds and their uses
02/15/2000US6025472 N-substituted glycine derivatives as enzyme inhibitors
02/15/2000CA2197739C 1,4-dihydropyridine compounds
02/10/2000WO2000006545A1 High affinity ligands for nociceptin receptor orl-1
02/10/2000WO2000006544A1 Cyclic amine derivatives and process for the preparation thereof
02/08/2000US6022971 Azetidines
02/03/2000WO1999064417A3 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
02/02/2000EP0975631A1 5-aryl-3-(8-azabicyclo(3.2.2)oct-3-yl)-1,3,4-oxadiazol-2(3h)-one derivatives as 5-ht4 receptor ligands
02/02/2000CN1048986C Heterocyclic compounds and their preparation and use
02/01/2000USH1838 Miticides
02/01/2000US6020368 Microbiocides
01/2000
01/27/2000WO2000004017A1 Azabicycle-substituted phenylindole derivatives as ligands for 5-ht2a receptors
01/26/2000EP0973537A1 Cocaethylene immunogens and antibodies
01/19/2000EP0971918A1 Bicyclic amine derivatives
01/12/2000CN1241184A Indole derivs. for treatment of osteoporosis
01/11/2000US6013242 Tropane derivatives with selective binding to the serotonin reuptake transporters for treatment of mental illness and as intermediates in the formation of imaging diagnostic agents for depression
01/05/2000EP0969005A1 Azabicyclic inhibitors of serotonin reuptake
01/05/2000EP0967993A2 Anti-cocaine vaccine
01/05/2000EP0711299B1 AZABICYCLOALKYL DERIVATIVES OF IMIDAZO(1,5-a)INDOL-3-ONE AS 5HT 3 ANTAGONISTS
12/1999
12/28/1999US6008227 Process for blocking 5-HT and dopamine uptake with biologically active tropane derivatives
12/23/1999WO1999065492A1 Inhibition of serotonin reuptake
12/23/1999CA2335336A1 Inhibition of serotonin reuptake
12/22/1999EP0758312B1 Substituted fused and bridged bicyclic compounds as therapeutic agents
12/21/1999US6005110 Process for the production of endotropine
12/21/1999CA2035653C Neuroprotective 3-piperidino-4-hydrosychroman derivatives
12/16/1999WO1999064417A2 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
12/16/1999WO1999064043A1 Muscarinic receptor antagonists
12/16/1999CA2333332A1 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
12/16/1999CA2315883A1 Muscarinic receptor antagonists
12/08/1999CN1237973A Bicyclic amine derivatives
12/08/1999CN1237972A 8-azabicyclo [3,2,1] octane-, 8-azabicyclo [3,2,1] oct-6-ene-, 9-azabicyclo [3,3,1] nonane-, 9-aza-3-oxabicyclo [3,3,1] nonane-, 9-aza-3-thiabicyclo [3,3,1] nonane derivatives
12/07/1999US5998405 Psychological disorders
12/07/1999US5998404 Nervous system disorders
12/07/1999CA2198231C Dihydropyridine derivatives as bradykinin antagonists
12/02/1999WO1999061917A1 Label for making a charge-transfer fluorescent probe
12/02/1999WO1999061023A1 Cocaine receptor binding ligands
12/01/1999EP0655056B1 Azacyclyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
11/1999
11/25/1999WO1999059409A1 Compounds and uses thereof
11/24/1999CN1046722C Heterocyclic compounds and their preparation and use
11/23/1999US5990312 Method for the preparation of esters of anhydroecgonine
11/23/1999US5990285 Catalytic antibodies against cocaine
11/23/1999US5990124 Neuromuscular relaxants
11/17/1999CN1235596A Cyclic amine derivatives
11/17/1999CN1046511C Benzoylecgonine, ecgonine and ecgonidine derivatives
11/16/1999US5985887 Aza-anthracyclinone derivatives
11/16/1999US5985881 Treatment and prevention of respiratory disorders, inflammatory eye diseases, inflammatory skin diseases, intestinal disorders, other inflammatory diseases
11/16/1999US5985878 Angiogenesis inhibiting pyridazinamines
11/09/1999US5981525 Indole derivatives useful in the treatment of osteoporosis
11/09/1999US5980860 Dopamine and serotonin transporter ligands and imaging agents
11/04/1999WO1999055703A1 2-alkyl-3-(hetero)aryl-8-azabicyclo[3.2.1]alkanes as pesticides
11/02/1999US5977314 Catalytic antibodies against cocaine
10/1999
10/28/1999WO1999038866A8 8-azabicyclo[3.2.1]oct-2-ene derivatives in labelled form and use of 8-azabicyclo[3.2.1]oct-2-ene derivatives in labelled and unlabelled form
10/27/1999CN1233245A Oxadiazoles, processes for their preparation and their use as medicaments
10/19/1999US5968947 Bicyclic amine derivatives
10/19/1999US5968926 Schizophrenia treatment with 1,2,5-oxadiazole or 1,2,5-thiadiazole
10/19/1999US5968923 (Azetidin-1-ylalkyl) lactams as tachykinin antagonists
10/13/1999CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/06/1999EP0946553A1 8-azabicyclo 3.2.1]octane derivatives, their preparation and their use as insecticides
10/06/1999EP0946204A1 Process for the preparation of radiopharmaceuticals
1 ... 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 ... 53