Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
07/1986
07/30/1986CN85108556A Process for preparing novel benzoxazol-and benzothiazolamine derivatives and their use
07/08/1986US4599420 Azabicyclic intermediates for pharmaceutical compounds
06/1986
06/11/1986EP0184257A1 Benzoxazol- and benzothiazolamine derivatives
05/1986
05/20/1986US4590270 2,4-diamino-[4-piperidinyl]pyrimidines useful as antibacterial agents, antimalarial agents, antitumors agents
05/06/1986US4587250 Thiazaspirane derivatives, process for their preparation, and medicaments
04/1986
04/29/1986US4585866 Treatment of migraine with substituted tropyl benzoate derivatives
04/29/1986US4585865 Intermediates for anticholinergic agents
04/22/1986US4584378 Mydriatic agents
04/09/1986EP0177122A2 Acrylamide derivatives
03/1986
03/26/1986EP0175440A2 Method of treating migraine headaches
03/18/1986CA1202027A1 Substituted tropyl and pseudotropyl benzoates and their use in migraine treatment
02/1986
02/18/1986US4571396 Antibacterial agents
02/11/1986US4569940 Certain 5-N-mono- or disubstituted sulfamoyl benzamides having use in treatment of emesis, impaired gastro-intestinal motility disorders and central nervous system disorders
01/1986
01/07/1986US4563465 Antiserotonine agents
12/1985
12/24/1985US4560757 9-Azabicyclo(3.3.1) nonane intermediates for compounds useful in the treatment of CNS disorders
12/10/1985US4558054 Spasmolytic endo-8,8-dialkyl-8-azoniabicyclo (3.2.1) octane-6,7-exo-epoxy-3-alkyl-carboxylate salts
12/04/1985EP0163260A1 Novel substituted pyrrolidinones, process for their manufacture and pharmaceutics
11/1985
11/12/1985CA1196641A1 Benzamides
10/1985
10/29/1985US4550115 Certain piperidino-lower-alkylene esters of 3-methylflavone-8-carboxylates possessing smooth muscle relaxant activity
10/23/1985EP0159174A2 Substituted naphthyridine-, quinoline- and benzoxazine- carboxylic acids as antibacterial agents and processes for their production
10/22/1985US4549021 N-(β-Fluoroethyl)-nortropine
10/16/1985EP0158265A2 Benzamide and anilide derivatives
10/08/1985US4546096 Anticholinergic glucuronides and antiperspirant use thereof
10/01/1985US4544660 Dopamine antagonist
09/1985
09/11/1985EP0154446A2 Anti-cholinergic glucuronides and their anti-perspirant use
08/1985
08/20/1985US4536580 4-Amino-5-bromo-2-methoxy-N-[8-(benzyl)]-8-azabicyclo[3.2.1]-3-YL-benzamide or a pharmacologically acceptable acid addition salt thereof
08/07/1985EP0150263A1 Derivatives of cis, endo-2-azabicyclo-[3.3.0]-octane-3-carboxylic acid, process for their preparation, medicaments containing them, and their use
07/1985
07/30/1985US4532244 Method of treating migraine headaches
07/24/1985EP0149088A1 Pyridine-2-ethers respectively pyridine-2-thioethers with a nitrogen containing cycloaliphatic ring and sulfoxides,sulfanes and pyridin-N-oxides thereof
07/17/1985EP0148233A1 Anti-emetic azabicycloalkyl benzamides
07/04/1985WO1985002847A1 Carbocyclic and heterocyclic carbon acid esters and amides of nitrogenous or non nitrogenous bridged or unbridged amines or alcohols
07/03/1985EP0147044A2 Benzofurancarboxamides, process for their preparation and pharmaceutical preparations containing them
06/1985
06/25/1985US4525475 Prevention of thrombolic disorder with imidazole derivatives and salts thereof
06/25/1985CA1189507A1 Substituted dibenzodiazepinones, processes for the preparation thereof and pharmaceutical compositions containing these compounds
05/1985
05/14/1985CA1187087A1 Derivatives of cis, endo-2-azabicyclo-[3.3.0]- octane-3-carboxylic acid, a process for their preparation, agents containing these compounds and their use
04/1985
04/10/1985EP0136945A2 Cinnamoyl compounds, process for their preparation and their therapeutical use
04/03/1985EP0135545A1 Azabicycloalkyl benzamide and anilide derivatives
03/1985
03/14/1985WO1985001048A1 Aromatic esters or amides of carboxylic acid and sulfonic acid
02/1985
02/28/1985EP0083373A4 Motion sickness spray composition and method.
02/26/1985CA1183140A1 Process for preparing carboxylic azo-bicyclo-octane acids
02/20/1985EP0133218A2 Endo-8,8-dialkyl-8-azoniabicyclo (3.2.1) octane-6,7-exo-epoxy-3-alkyl-carboxylate salts, a process for their preparation, and therapeutic compositions which contain them as active principle
02/12/1985US4499099 Nortropane and granatane type compounds useful in treating psychosis
01/1985
01/17/1985WO1985000170A1 Anti-emetic azabicycloalkyl benzamides
01/16/1985EP0131315A2 Nasal preparations comprising anticholinergic quaternary ammonium salts
12/1984
12/19/1984EP0128437A2 Nortropine derivative, process for its preparation and its use
12/05/1984EP0127529A2 Aminocyclic N-oxide derivatives, process for their preparation and their therapeutical use
12/04/1984US4486441 Prophylaxis
12/04/1984US4486430 Melamine derivatives
11/1984
11/28/1984EP0126087A1 Amino-azabicycloalkyl derivatives as dopamine antagonists
10/1984
10/24/1984EP0122580A1 Pyrimidine derivatives, their preparation and pharmaceutical compositions
10/17/1984EP0121614A1 Perfluorotricyclic amine compounds
10/16/1984US4477668 Process for 5-methyl-10,11-dihydro-5H-dibenzo[a,d]-cyclohepten-5,10-imine
09/1984
09/18/1984US4472413 9'-Azabicyclo [3.3.1] nonyl benzamide
09/11/1984US4471120 3-aroylamino-8-benzyl substituted, neuroleptic agents
08/1984
08/30/1984WO1984003281A1 Azabicycloalkyl benzamide and anilide derivatives
08/28/1984CA1173439A1 Process for the dealkylation of tertiary amines by using a-chlorinated chloroformates
08/21/1984US4467095 Anticholinergic compounds
08/14/1984US4465834 Anticholinergic drugs
07/1984
07/10/1984US4459300 Antiemetics, gastrointestinal disorders, central nervous system, psychological disorders
06/1984
06/27/1984EP0112266A2 Substituted tropyl and pseudotropyl benzoates and their use in migraine treatment
06/27/1984EP0111608A1 Pseudotropyl halogeno-benzoates and their use in migraine treatment
06/27/1984EP0111607A1 Tropyl and pseudotropyl alkyl-benzoates and their use in migraine treatment
05/1984
05/15/1984CA1167443A1 Anti-emetic nortropyl(alkyl)benzamides
05/08/1984US4447434 Substituted dibenzodiazepinones
04/1984
04/17/1984US4443452 Antiulcer agents
04/04/1984EP0104984A2 Vinylcarbamic acid esters and their preparation
03/1984
03/29/1984WO1984001151A1 Amino-azabicycloalkyl derivatives as dopamine antagonists
03/07/1984EP0102195A2 Substituted aza bicycloalkyl derivatives with dopamine antagonist activity
02/1984
02/29/1984EP0101641A2 Sulfonylamino-aza-bicyclo-alkyl derivatives
02/28/1984US4434170 Neuroleptic agents, antiemetics, laxatives
02/21/1984US4432983 Conformationally restricted histamine H2 -receptor antagonists containing a tropane ring
01/1984
01/25/1984EP0099194A2 Novel benzamides
01/24/1984CA1161040A1 Salts of endo-8-methyl-8-syn-alkyl-8-azoniabicyclo- ¬3.2.1|-octane-3-alkylcarboxylates, process for their preparation and therapeutic compositions containing them
01/19/1984WO1984000166A1 Benzoic acid piperidyl ester derivatives and method of production and utilization thereof
01/10/1984CA1160227A2 DERIVATIVES OF .beta.-3-AMINO-N-NOR-TROPANES
01/03/1984US4424358 β-3-Amino nor-tropane compounds
12/1983
12/21/1983EP0096524A2 Bicyclic benzamides or anilides, process for their preparation, and pharmaceutical compositions containing them
11/1983
11/30/1983EP0095262A1 Azabicycloalkane derivatives, their preparation and medicaments containing them
11/09/1983EP0093488A2 Nortropyl benzopyrrolinone compounds, process for their preparation and pharmaceutical compositions containing them
11/09/1983EP0093343A1 Process for the preparation of norscopine
11/08/1983US4414154 Anxiolytic, antidepressant, anticonvulsant, muscle relaxants
11/02/1983EP0092814A1 Intermediates for the preparation of N-Alkylnorscopines, their preparation and their application
10/1983
10/18/1983US4410535 Aza-bicyclo-benzamide derivatives and pharmaceutical compositions and use thereof
10/12/1983EP0091071A1 Process for the preparation of 5-methyl-10,11-dihydro-5H-dibenzo(a,d)-cyclohepten-5,10-imine and its salts
10/05/1983EP0090195A1 Quaternised 6,11-dihydro-dibenzo-(b,e)-thiepin-11-N-alkyl-norscopin ethers and process for their preparation
08/1983
08/31/1983EP0086980A1 Substituted dibenzodiazepinones, process for their preparation and medicines containing these compounds
08/24/1983EP0086453A2 Thiazaspiro derivatives, process for their preparation and pharmaceutical composition
08/17/1983EP0085892A1 Substituted benzodiazepinones, process for their preparation and medicines containing them
08/16/1983US4399141 5-Alkyl or hydroxyalkyl substituted-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imines and anticonvulsant use thereof
08/16/1983CA1152077A1 Indolizine derivatives and process for preparing the same
08/09/1983US4397857 Enzyme inhibitors
07/1983
07/20/1983EP0083737A1 N-azabicycloalkane benzamides, process for their preparation and pharmaceutical compositions containing them
07/13/1983EP0083373A1 Motion sickness spray composition and method
07/12/1983US4393069 8-Arylalkyl-3-phenyl-3-nortropanols and salts thereof
06/1983
06/15/1983EP0081054A2 Azabicyclo alkyl derivatives
05/1983
05/18/1983EP0079022A2 Derivatives of cis, endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid, process for their preparation, medicines containing them and their use
04/1983
04/13/1983EP0076592A2 Azabicyclo-(3,3,1)-nonylbenzamide derivatives, processes for their preparation, and pharmaceutical compositions containing them
04/12/1983US4379936 Analgesics
04/06/1983EP0076089A2 Azabicycloalkane derivatives, process for their preparation, and a pharmaceutical composition containing them
03/1983
03/29/1983CA1143734A1 8-arylalkyl-3-phenyl-3-nortropanols, their acid addition salts, medicaments containing the same and processes for the preparation thereof
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