Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
12/1998
12/30/1998CN1203233A Process for production of endotropine
12/29/1998US5853696 Substituted 2-carboxyalkyl-3(fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders
12/23/1998WO1998057909A1 Process for the production of radioiodinated neuroreceptor agents
12/23/1998EP0885220A1 Tropane-derivatives, their preparation and use
12/23/1998CA2293317A1 Process for the production of radioiodinated neuroreceptor agents
12/15/1998US5849754 Bicyclic amine derivatives
12/09/1998EP0882045A1 Process for the preparation of granisetron
12/09/1998EP0882044A1 1,4-dihydropyridine compounds as bradykinin antagonists
12/09/1998CN1201461A Fused tropane-derivatives as neurotransmitter reuptake inhibitors
12/09/1998CN1201390A 5-HT3 receptor antagonists for treating dyskinesia
12/03/1998WO1998054182A1 9-AZABICYCLO(3.3.1)NON-2-ENE AND NONANE DERIVATIVES AS CHOLINERGIC LIGANDS AT NICOTINIC ACh RECEPTORS
12/03/1998WO1998054181A1 8-azabicyclo(3,2,1)oct-2-ene and octane derivatives as cholinergic ligands at nicotinic ach receptors
12/03/1998WO1998054168A1 2-oxoimidazole derivatives
12/02/1998EP0544779B1 Heterocyclic compounds and their preparation and use
12/02/1998CN1040979C Antipsychotic method
11/1998
11/26/1998WO1998052940A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS
11/26/1998CA2291115A1 Substituted pyrazoles as p38 kinase inhibitors
11/24/1998US5840725 Substituted oximes, hydrazones and olefins as neurokinin antagonists
11/19/1998WO1998051311A2 Dihydropyrimidines and uses thereof
11/18/1998CN1199400A 8-azabicycle [3.2.1]oct-2-ene derivs, their preparation and use
11/18/1998CN1199399A Naphthamide derivs, of 3-beta-amino azabicyclo octane or nonane as neuroleptic agents
11/18/1998CN1040756C Heterocyclic compounds preparation process
11/11/1998EP0876366A2 Angiogenesis inhibiting pyridazinamines
11/11/1998EP0687266B1 Heterocyclic compounds and their preparation and use
11/10/1998US5834484 Used to treat human patient suffering from cocaine addiction or overdose
11/04/1998EP0874833A1 4,5-dihydronaphth 1,2-c]isoxazoles and derivatives thereof having cns activity
11/04/1998EP0874809A1 Carbamoyloxy derivatives of mutiline and their use as antibacterials
11/03/1998US5831095 Synthesis of 5-aminocarbonyl-5H-dibenzo a,d!cyclohepten-5,10-imine
11/03/1998CA2131789C Biologically active tropane derivatives
10/1998
10/29/1998WO1998047898A1 5-aryl-3-(8-azabicyclo(3.2.2)oct-3-yl)-1,3,4-oxadiazol-2(3h)-one derivatives as 5-ht4 receptor ligands
10/29/1998CA2286106A1 5-aryl-3-(8-azabicyclo(3.2.1)oct-3-yl)-1,3,4-oxadiazol-2(3h)-one derivatives as 5-ht4 receptor ligands
10/22/1998WO1998046600A1 Bicyclic amine derivatives
10/21/1998EP0872237A1 Method and compositions for the synthesis of BCH-189 and related compounds
10/20/1998US5824669 Treating asthma
10/13/1998US5821371 Heterocyclic compounds and their preparation and use
10/13/1998US5821370 Muscarinic cholinergic drugs
10/13/1998US5821249 Anhydroecogonine compounds and their use as anticholinergic agents
10/07/1998EP0866067B1 Process of preparation of endo-tropine
10/06/1998US5817770 N-methyltropane, 2-carboxyethyl- or n-ethylcarboxamide, 3-benzoyloxy- or benzamido-
10/01/1998WO1998042359A1 Cocaethylene immunogens and antibodies
10/01/1998CA2284613A1 Cocaethylene immunogens and antibodies
09/1998
09/30/1998CN1194646A Aza-Anthracyclinone derivatives
09/29/1998US5814639 Treating aids
09/24/1998WO1998041523A1 Process for preparing dibenzo-1-carboxamido-1,4-azabicyclo(3.2.1.) octanes
09/23/1998EP0866067A1 Process of preparation of endo-tropine
09/23/1998EP0865441A1 1,2,3-thiadiazole carboxylic acid (thio)esters and the use thereof as a pest control agent or as a microbicide
09/23/1998EP0865439A1 Combinatorial libraries having aminodiol monomer subunits
09/23/1998CN1039909C Aminobenzoic acid derivatives
09/16/1998EP0654023B1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists
09/15/1998US5808074 Benzoylecgonine conjugate diagnostic reagents
09/15/1998US5807871 Psychological disorders, alzheimer or parkinson disease
09/09/1998EP0513200B1 Method and compositions for the synthesis of bch-189 and related compounds
09/02/1998EP0861252A1 NAPHTHAMIDE DERIVATIVES OF 3 $g(b)-AMINO AZABICYCLO OCTANE OR NONANE AS NEUROLEPTIC AGENTS
09/02/1998EP0593511B1 Piperidine derivates having anxiolytic effect
08/1998
08/26/1998EP0859777A1 8-azabicyclo 3.2.1]oct-2-ene derivatives, their preparation and use
08/26/1998EP0859641A1 Dopamine transporter imaging agent
08/26/1998CN1191535A Medicine composition and use thereof
08/19/1998EP0859004A1 Piperidine derivatives having anxiolytic effect
08/19/1998EP0858461A1 Fused tropane-derivatives as neurotransmitter reuptake inhibitors
08/11/1998US5792775 High affinity for dopamine transporter; inhibit dopamine uptake; do not have a cocaine-like behavorial profile; used to image binding sites; diagnosis and monitoring of neurodegenerative diseases, e.g parkinson's
08/05/1998CN1189821A Substituted oximes, hydrazones and olefins as neurokinin antagonists
08/04/1998CA2066248C Esters of thienyl carboxylic acids and amino alcohols, their quaternization products, and manufacture and use of said compounds
07/1998
07/28/1998CA2016860C 2-piperidino-1-alkanol derivatives as antiischemic agents
07/15/1998EP0853085A1 Piperidine derivatives having anxiolytic effect
07/14/1998US5780494 Piperidinyl-terminated alkylamino ethynl alanine amino diol compounds for treatment of hypertension
07/08/1998EP0851756A1 5-ht 3? receptor antagonists for dyskinesia
06/1998
06/23/1998US5770738 Esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions
06/23/1998US5770180 Bridge-substituted tropanes for methods of imaging and therapy
06/18/1998WO1998025924A1 8-azabicyclo[3.2.1]octane-, 8-azabicyclo[3.2.1]oct-6-ene-, 9-azabicyclo[3.3.1]nonane-, 9-aza-3-oxabicyclo[3.3.1]nonane- and 9-aza-3-thiabicyclo[3.3.1]nonane derivatives, their preparation and their use as insecticides
06/18/1998WO1998025923A1 8-azabicyclo[3.2.1]octane derivatives, their preparation and their use as insecticides
06/18/1998CA2272076A1 8-azabicyclo¬3.2.1|octane derivatives, their preparation and their use as insecticides
06/18/1998CA2271749A1 8-azabicyclo¬3.2.1|octane-, 8-azabicyclo¬3.2.1|oct-6-ene-, 9-azabicyclo¬3.3.1|nonane-, 9-aza-3-oxabicyclo¬3.3.1|nonane- and 9-aza-3-thiabicyclo¬3.3.1|nonane derivatives, their preparation and their use as insecticides
06/17/1998CN1185154A Bicyclic amines as insecticides
06/11/1998WO1998024788A1 Tropane derivatives and method for their synthesis
06/09/1998US5763456 Benzoylecgonine, ecgonine and ecgonidine derivatives
06/09/1998US5763455 Biologically active tropane derivatives
06/02/1998US5760055 Biologically active tropane derivatives
05/1998
05/28/1998WO1998022463A1 Bicyclic amine derivatives
05/28/1998WO1998022462A1 8-azabicyclo[3.2.1]octane-, 8-azabicyclo[3.2.1]oct-6-ene-, 9-azabicyclo[3.3.1]nonane-, 9-aza-3-oxabicyclo[3.3.1]nonane-, 9-aza-3-thiabicyclo[3.3.1]nonane derivatives, their preparation and their use as insecticides
05/28/1998CA2271726A1 8-azabicyclo¬3.2.1|octane-, 8-azabicyclo¬3.2.1|oct-6-ene-, 9-azabicyclo¬3.3.1|nonane-, 9-aza-3-oxabicyclo¬3.3.1|nonane-, 9-aza-3-thiabicyclo¬3.3.1|nonane derivatives, their preparation and their use as insecticides
05/28/1998CA2269917A1 Bicyclic amine derivatives
05/27/1998EP0843676A1 Ipratropium bromide enantiomer with a prolonged duration of action
05/27/1998EP0843675A1 Aza-anthracyclinone derivatives
05/27/1998CN1183098A Process for preparing pure enantiomers of tropic acid esters
05/26/1998US5756508 Muscarine antagonists
05/20/1998EP0608336B1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment
05/19/1998US5753673 Quinolinecarboxylic acid derivatives
05/12/1998US5750089 Halogenated neuroprobe for mapping monoamine reuptake sites
05/12/1998CA2030718C Tricyclic compounds
05/07/1998WO1998018788A1 Piperazino derivatives as neurokinin antagonists
05/07/1998WO1998018499A1 Process for the preparation of radiopharmaceuticals
05/07/1998CA2270242A1 Process for the preparation of radiopharmaceuticals
05/05/1998US5747522 Anticoagulants; antiinflammatory agents; antitumor agents
05/05/1998US5747503 Indeno(1,2b)pyroles
04/1998
04/30/1998WO1998017652A1 Oxadiazoles, processes for their preparation and their use as medicaments
04/23/1998DE19643037A1 Neue Oxadiazole, Verfahren zu ihrer Herstellung sowie deren Verwendung als Arzneimittel New oxadiazoles, processes for their preparation and their use as medicaments
04/22/1998EP0697871A4 Treatment process with biologically active tropane derivatives
04/21/1998US5741790 Tachykinin antagonist and intermediates for nervous system disorders, antiinflammatory agents, antiarthritic agents, antidepressants and gastrointestinal disorders
04/15/1998CN1179157A Method for preparation of esters of anhydroecgonine
04/14/1998US5739337 Process for preparing dibenzo-1-carboxamido-1,4-azabicyclo 3.2.1!octanes
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