| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 01/24/2001 | CN1281459A Piperidine derivatives |
| 01/24/2001 | CN1281456A Process for preparation of 8-azabicyclo (3,2,1) octane derivatives |
| 01/24/2001 | CN1281455A 8-Azabicyclo [3,2,1] octane-3-methanamine derivatives as ligands of D2 and D3 dopamine and 5HT1A and 5HT2 serotonin receptors |
| 01/23/2001 | US6177442 Bicyclic amine derivatives |
| 01/23/2001 | CA2197451C Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkanol derivatives |
| 01/21/2001 | CA2314373A1 Heteroaryl-substituted pyrrole derivatives, their preparation and their thereapeutic uses |
| 01/17/2001 | EP1069124A1 2-Benzimidazolylamine compounds as ORL1-receptor agonists |
| 01/17/2001 | EP1068204A1 8-azabicyclo 3.2.1]oct-2-ene derivatives in labelled and use of 8-azabicyclo 3.2.1]oct-2-ene derivatives in labelled and unlabelled form |
| 01/17/2001 | EP1067903A1 Improved crystal structure |
| 01/17/2001 | CN1280578A Bis-quaternary ammonium derivatives as neuromuscular relaxants |
| 01/17/2001 | CN1060775C Fused troane-derivatives as neurotransmitter reuptake inhibitors |
| 01/17/2001 | CN1060773C Naphthamide derivatives of 3-beta-amino azabicyclo octane or nonane as heuroleptic agents |
| 01/16/2001 | US6174894 As insecticides, pesticides; for controlling acarine or nematode pests |
| 01/16/2001 | US6174723 Cocaine derivative, protein conjugate thereof, monoclonal antibody producing cell line, method for preparing the cell line and monoclonal antibody |
| 01/16/2001 | CA2314008A1 2-benzimidazolylamine compounds as orl1-receptor agonists |
| 01/09/2001 | US6171576 Tropane compound is linked through the n atom at the 8-position to a chelating ligand capable of complexing technetium or rhenium to produce a neutral labeled complex that selectively binds to the dopamine transporter. |
| 01/03/2001 | CN1060168C Xanthene derivant, its preparation method and medicinal composition containing same |
| 12/28/2000 | WO2000078725A1 Synthesis of substituted amidines |
| 12/28/2000 | WO2000078724A2 Imidazolinderivatives their preparation and their pharmaceutical use |
| 12/26/2000 | US6166209 Piperidine derivatives |
| 12/12/2000 | CA2215664C Method for the preparation of esters of anhydroecgonine |
| 12/06/2000 | EP1057819A1 Phthalazine derivatives and remedies for erectile dysfunction |
| 12/05/2000 | US6156752 Optically active 1,4-dihydropyridine compounds as bradykinin antagonists |
| 11/30/2000 | WO2000071519A2 Immunopotentiator agents |
| 11/29/2000 | CN1275124A Phthalazine derivatives and remedies for erectile dysfunction |
| 11/28/2000 | US6153751 Preparing the antiviral b-isomer of a 1,3-oxathiolane nucleoside by reacting in presence of stannic chloride |
| 11/22/2000 | CN1273973A Method of preparing endonortropine by using 9-benzyl-nortropine-3-one-perchlorate as intermediate and salt thereof |
| 11/21/2000 | US6150376 Bi- and tri-cyclic aza compounds and their uses |
| 11/21/2000 | US6150352 Antagonists of gonadotropin releasing hormone |
| 11/21/2000 | CA2187309C Tropane-2-aldoxime derivatives as neurotransmitter reuptake inhibitors |
| 11/15/2000 | EP1051980A2 Dopamine transporter imaging agents |
| 11/15/2000 | EP1051418A1 Process for the preparation of substituted 8-azabicyclo [3.2.1]octanes |
| 11/15/2000 | EP1051417A1 Process for the preparation of 8-azabicyclo(3.2.1)octane derivatives |
| 11/12/2000 | CA2721484A1 Dopamine transporter imaging agents |
| 11/02/2000 | WO2000064491A1 4-fluoroalkyl-3-halophenyl nortropanes |
| 11/02/2000 | WO2000064490A1 Fluoroalkenyl nortropanes |
| 11/02/2000 | CA2369663A1 4-fluoroalkyl-3-halophenyl nortropanes |
| 10/31/2000 | US6140338 For treating acute inflammatory diseases, chronic inflammatory diseases, acquired immune deficiency syndrome, cancer, ischemic reflow disorder and/or arteriosclerosis |
| 10/26/2000 | WO2000063215A2 Indazole derivatives, preparation and therapeutic application thereof |
| 10/26/2000 | WO2000063204A2 Substituted azoles |
| 10/26/2000 | CA2370417A1 Substituted azoles |
| 10/19/2000 | WO2000061569A1 Adamantane derivatives |
| 10/19/2000 | CA2368829A1 Adamantane derivatives |
| 10/18/2000 | EP1043999A1 Novel substituted pyridine compounds useful as modulators of acetylcholine receptors |
| 10/17/2000 | US6131226 1,4-dihydropyridine compounds as bradykinin antagonists |
| 10/12/2000 | WO2000059510A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors |
| 10/12/2000 | CA2366858A1 Sorbitol dehydrogenase inhibitors |
| 10/04/2000 | EP0575581B1 Novel cocaine derivatives and protein and polypeptide cocaine derivative conjugates and labels |
| 09/28/2000 | WO2000056729A1 Chemokine recpetor binding heterocyclic compounds |
| 09/28/2000 | CA2368047A1 Chemokine receptor binding heterocyclic compounds |
| 09/27/2000 | EP1037892A1 Piperidine derivatives |
| 09/27/2000 | EP1037637A1 Use of 5ht1a receptor antagonists for preventing and/or treating temporal lobe epilepsy |
| 09/27/2000 | CN1268133A 2-Aminopyridines containing fused ring substituents as NOS inhibitors |
| 09/27/2000 | CN1056843C Process for producing esters of anhydroecgonine |
| 09/26/2000 | US6124354 Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation |
| 09/26/2000 | US6123917 Useful in biochemical assays, imaging techniques, and in a wide variety of drug treatment methodologies |
| 09/19/2000 | US6121281 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use |
| 09/13/2000 | EP1033914A1 Bicyclic amines and their use as insecticides |
| 09/12/2000 | US6117883 Useful for modulating a muscarinic receptor. |
| 09/12/2000 | US6117882 5-HT4 agonists and antagonists |
| 09/08/2000 | WO2000051608A1 3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity |
| 09/06/2000 | EP1032569A1 Imidazole derivatives, preparation and therapeutic application thereof |
| 09/05/2000 | US6114508 Cocaethylene immunogens and antibodies |
| 09/05/2000 | US6114343 Antiviral activity and resolution of 2-hydroxymethyl-5-(5-flurocytosin-1-yl)-1,3-oxathiolane |
| 09/05/2000 | US6113877 σ-2 receptors as biomarkers of tumor cell proliferation |
| 08/31/2000 | WO2000050396A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor |
| 08/31/2000 | CA2371876A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor |
| 08/24/2000 | WO2000048597A1 Systemic use of 5-ht3 receptor antagonists against rheumatic inflammatory processes |
| 08/23/2000 | EP1029862A1 Process for the preparation of endo-nortropine using 8-benzyl-nortropan-3-one-perchlorate as intermediate, as well as said salt |
| 08/23/2000 | EP1029853A1 Heteroaromatic bicyclic derivatives useful as anticancer agents |
| 08/23/2000 | EP1028961A1 Pleuromutilin derivatives as antimicrobials |
| 08/23/2000 | CN1264377A Substituted pyrazoles as P38 kinase inhabitors |
| 08/22/2000 | US6107307 Psychological disorders |
| 08/17/2000 | WO2000047571A1 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation |
| 08/17/2000 | WO2000047200A1 Combinations of formoterol and a tiotropium salt |
| 08/17/2000 | CA2362389A1 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation |
| 08/09/2000 | EP1025099A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants |
| 08/08/2000 | US6100275 8-azabicyclo[3.2.1.]oct-2-ene derivatives, their preparation and use |
| 08/08/2000 | CA2185512C Treatment of tinnitus using neuroprotective agents |
| 08/08/2000 | CA2027041C Aroyl-ureas |
| 08/03/2000 | WO2000044747A1 Tropane derivatives as serotonin transporter antagonists |
| 08/03/2000 | WO2000044746A1 Novel azabicyclo derivatives and their use |
| 08/03/2000 | WO2000044743A1 Amide derivatives and drug compositions |
| 08/03/2000 | WO2000044728A1 Substituted bicyclic derivatives useful as anticancer agents |
| 08/02/2000 | EP1023289A1 Dopamine transporter imaging ligand |
| 08/02/2000 | CN1261885A 2-substituted 4,5-diaryl imidazoles |
| 08/01/2000 | CA2151618C Derivatives of benzoylecgonine, ecgonine and ecgonidine as medicines |
| 08/01/2000 | CA2066640C Heterocyclic compounds |
| 07/26/2000 | EP1021443A1 Hemoregulatory compounds |
| 07/26/2000 | EP1021442A1 8-azabicyclo 3.2.1] octane-3-methanamine derivatives as ligands of d2 and d3 dopamine and 5ht1a and 5ht2 serotonin receptors |
| 07/26/2000 | EP1021185A1 Didhydropyrimidines and uses thereof |
| 07/25/2000 | US6093726 Bicyclic amine derivatives |
| 07/25/2000 | CA2197086C (azetidin-1-ylalkyl)lactams as tachykinin antagonists |
| 07/19/2000 | CN1260794A 5-aryl-3-(8-azabicyclo (3.2.2) oct-3-yl)-1,3,4-oxadiazol-2(3H)-one derivatives as -5HT4 receptor ligands |
| 07/12/2000 | EP1018513A2 Quinolinecarboxylic acid derivatives |
| 07/12/2000 | EP1018512A1 Novel basic derivatives of benz(e)isoindol-1-ones and pyrrolo(3,4-c)quinolin-1-ones with 5-HT3-antagonistic activity, their preparation and their therapeutic use |
| 07/11/2000 | US6087379 Cyclic amine derivatives |
| 07/06/2000 | WO2000039125A1 Piperidines as ccr5 modulators |
| 07/06/2000 | WO2000038680A1 Azabicycloalkanes as ccr5 modulators |
| 06/28/2000 | EP1013276A1 Aminoazacycloalkanes as CCR5 modulators |