Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
07/1997
07/17/1997WO1997025317A1 4,5-dihydronaphth[1,2-c]isoxazoles and derivatives thereof having cns activity
07/17/1997WO1997025309A1 Carbamoyloxy derivatives of mutiline and their use as antibacterials
07/17/1997CA2240467A1 Carbamoyloxy derivatives of mutiline and their use as antibacterials
07/16/1997CN1154699A (Azetidin-1-ylalkyl) lactams as tachykinin antagonists
07/09/1997EP0782574A1 Bicyclic carboxamides as 5-ht 1a? antagonists
07/08/1997US5646289 Reacting a 3-chloro-1,2,5-thiadiazole with alkali metal bis(trialkyl or arylsilyl)amide; dechlorination; treating nervous system disorders
07/03/1997WO1997023458A1 Subtype-selective nmda receptor ligands and the use thereof
07/02/1997EP0781277A1 Neurokinin antagonists
06/1997
06/24/1997US5641791 Heterocyclic compounds and their preparation and use
06/19/1997WO1997021451A1 Anti-cocaine vaccine
06/19/1997CA2239058A1 Anti-cocaine vaccine
06/12/1997WO1997020840A1 1,2,3-thiadiazole carboxylic acid (thio)esters and the use thereof as a pest control agent or as a microbicide
06/12/1997DE19545637A1 1,2,3-Thiadiazolcarbonsäure(thio)ester 1,2,3-thiadiazolecarboxylic (thio) ester
06/12/1997CA2239580A1 1,2,3-thiadiazole carboxylic acid (thio)esters and the use thereof as a pest control agent or as a microbicide
06/11/1997EP0777653A1 Dihygropyridine derivatives as bradykinin antagonists
06/11/1997EP0777652A1 Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkanol derivatives
06/10/1997US5637601 Antiperspirant, mydriatic, antisecretory agents
06/10/1997US5637596 Reacting aminomethylindole derivative with a carbonyl containing cyclizing agent; 5-ht3 receptor atagonist; useful for treating anxiety, psychosis, gut motility disorder, emesis, migraine and drug addiction
06/05/1997WO1997019944A1 Heterocyclic compounds and their use
06/05/1997WO1997019669A2 Heterocyclic compounds and their use
06/05/1997CA2238555A1 Heterocyclic compounds and their use
06/04/1997EP0776897A1 Heterocyclic compounds and their use
06/04/1997EP0776896A1 Heterocyclic compounds and their use
05/1997
05/28/1997EP0775132A1 (azetidin-1-ylalkyl)lactams as tachykinin antagonists
05/28/1997CN1150802A Benzoylecgonine, ecgonine and ecgonidine derivatives
05/22/1997WO1997018210A1 Hemoregulatory compounds
05/20/1997US5631402 Process for preparing aminobenzoic acid derivatives
05/20/1997US5631255 Affinity for cholinergic receptors, treatment of cognitive and memory disorders, and degenerative syndromes
05/14/1997EP0772613A2 Process for the production of aminoazobicycloalkanes from oximes
05/14/1997CN1149454A Method for curing tinnitus by nerve protecting agent
05/09/1997WO1997016451A1 Fused tropane-derivatives as neurotransmitter reuptake inhibitors
05/09/1997WO1997016210A1 Dopamine transporter imaging agent
05/09/1997WO1997016192A1 Muscarine antagonists
05/07/1997EP0771199A1 Methods
05/07/1997EP0734385A4 Substituted 2-carboxyalkyl-3-(fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders
04/1997
04/30/1997CN1148854A Tropane-z-aldoxine derivatives and preparation process and use thereof
04/29/1997US5625065 Stereoselective process for making endo-tropanamine and like compounds
04/24/1997WO1997014445A1 Dopamine and serotonin transporter ligands and imaging agents
04/17/1997WO1997013770A1 8-azabicyclo[3.2.1]oct-2-ene derivatives, their preparation and use
04/16/1997EP0768086A1 Treatment of tinnitus using neuroprotective agents
04/15/1997US5621010 Urea derivatives and their use as ACAT inhibitors
04/08/1997US5618826 Anticholinergic compounds, compositions and methods of treatment
04/02/1997EP0765326A1 Benzoylecgonine, ecgonine and ecgonidine derivatives
03/1997
03/27/1997WO1997010823A1 5-ht3 receptor antagonists for dyskinesia
03/27/1997CA2231887A1 5-ht3 receptor antagonists for dyskinesia
03/25/1997US5614629 Benzyl quaternary tropinium compound
03/20/1997WO1997010244A1 NAPHTHAMIDE DERIVATIVES OF 3 β-AMINO AZABICYCLO OCTANE OR NONANE AS NEUROLEPTIC AGENTS
03/20/1997CA2232082A1 Naphthamide derivatives of 3 .beta.-amino azabicyclo octane or nonane as neuroleptic agents
03/19/1997CN1145364A Heterocyclic compounds and their preparation and use
03/18/1997US5612351 Azabicyclic derivatives of 1,2,3-oxa(or thia)diazole
03/11/1997US5610188 Mydriatics, antiperspirants
03/11/1997US5610164 (Thiophen-2-yl)-piperidin or tetrahydropyridin azabicyclocarboxamides
03/11/1997US5610163 Esters of thienyl carboxylic acids and amino alcohols and their quaternization products
03/11/1997US5610154 Bicyclic carboxamides
02/1997
02/27/1997WO1997006832A1 Labeled cocaine analogs
02/25/1997US5605908 Treating diseases of central nervous system caused by malfunctioning of muscarinic cholinergic system
02/20/1997WO1997006165A1 Aza-anthracyclinone derivatives
02/19/1997EP0758312A1 Substituted fused and bridged bicyclic compounds as therapeutic agents
02/18/1997US5604239 Imidazopyridines as serotonergic 5-HT3 antagonists
02/13/1997WO1997005136A1 Ipratropium bromide enantiomer with a prolonged duration of action
02/12/1997CN1142498A (Thiophen-2-yl-)-piperidin or tetrahydropyridin azabicyclocarboxamides
02/06/1997DE19528145A1 Neue Arzneimittel und ihre Verwendung New drugs and their use
02/05/1997EP0756596A1 Tropane-2-aldoxime derivatives as neurotransmitter reuptake inhibitors
02/04/1997US5599972 Aminobenzoic acid derivatives
01/1997
01/29/1997EP0755932A1 (Thiophen-2-yl)piperidin or tetrahydropyridin-azabicyclocarboxamides
01/27/1997CA2181759A1 (thiophen-2-yl)-piperidin or tetrahydropyridin azabicyclocarboxamides
01/15/1997CN1140447A Novel carbamate deriv. and medicinal composition contg. the same
01/14/1997US5594007 Method for treating spinal cord trauma with phenolic 2-piperidino-1-alkanols
01/07/1997US5591854 Enantioselective synthesis of seven-membered carbocycles and tropanes
01/07/1997US5591749 Imidazopyridines as serotonergic 5-HT3 -antagonists
01/07/1997US5591748 Immunomodulatory azaspiranes
12/1996
12/19/1996WO1996040672A1 Combinatorial libraries having aminodiol monomer subunits
12/18/1996EP0748808A1 Heterocyclic compound
12/18/1996EP0748321A1 Process for the preparation of an indazole-3-carboxamide derivative
12/17/1996US5585492 LTA4 Hydrolase inhibitors
12/17/1996US5585491 Antibacterial agents
12/12/1996WO1996039198A1 Iodinated neuroprobes for mapping monoamine reuptake sites
12/11/1996EP0747355A1 Novel carbamate derivative and medicinal composition containing the same
12/10/1996US5583221 Antiinflammatory agents, cardiovascular disorders, viricides, fungicides
12/10/1996US5583142 Analgesic and nootropic drugs
12/04/1996EP0640601B1 Benzamide derivative
11/1996
11/28/1996WO1996037494A1 Bicyclic amines as insecticides
11/28/1996CA2217064A1 Bicyclic amines as insecticides
11/26/1996US5578603 Treatment for alzheimer*s disease, gaastrointrestinal disorders
11/26/1996US5578602 Certain 1-azabicyclo[3.3.1]nonene derivatives and their pharmacological uses
11/19/1996US5576321 Compounds having effects on serotonin-related systems
11/19/1996US5576317 NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis
11/13/1996EP0542903B1 Cocaine receptor binding ligands
11/12/1996US5574060 Selective inhibitors of biogenic amine transporters
11/12/1996US5574043 Certain [1,2,5-thiadiazol-4-yl]-1-azabicyclo [3.2.1]octane derivatives and their pharmaceutical uses
11/07/1996WO1996034857A1 Substituted oximes, hydrazones and olefins as neurokinin antagonists
11/05/1996US5571820 Quinoline derivatives, treatment of gastrointestinal disorders caused by decreased motility
10/1996
10/31/1996WO1996033996A1 Process for preparing pure enantiomers of tropic acid esters
10/31/1996DE19515625A1 Verfahren zur Herstellung von enantiomerenreinen Tropasäureestern A process for the preparation of enantiomerically pure Tropasäureestern
10/17/1996WO1996032390A1 PREPARATION OF CHIRAL 5-AMINOCARBONYL-5H-DIBENZO-[a,d]CYCLOHEPTEN-5,10-IMINES BY OPTICAL RESOLUTION
10/17/1996CA2217877A1 Preparation of chiral 5-aminocarbonyl-5h-dibenzo-¬a,d|cyclohepten-5,10-imines by optical resolution
10/10/1996WO1996031508A1 Biphenylamide derivatives as 5ht1d antagonists
10/09/1996EP0636148B1 Visible photosensitizers for photopolymerizable compositions
10/09/1996CN1133044A Antipsychotic method
10/09/1996CN1132625A NK-1 receptor antagonits and 5HT3 receptor antagonists for treatment of emesis
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