| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
|---|
| 10/27/2004 | EP1471068A1 Process for total synthesis of ecteinascidins and intermediates therefor |
| 10/27/2004 | EP1471055A1 6-phenylpyridyl-2-amine derivatives |
| 10/26/2004 | US6809199 (Halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents |
| 10/21/2004 | WO2004089942A2 Benzimidazolidinone derivatives as muscarinic agents |
| 10/21/2004 | WO2004089931A1 Substituted pyrazoles |
| 10/21/2004 | WO2004052888B1 Tropane esters and methods for producing and using them |
| 10/21/2004 | US20040209921 CXCR4 chemokine receptor binding comounds |
| 10/21/2004 | US20040209889 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists |
| 10/21/2004 | US20040209883 Nitrogen-containing heterocyclic compounds and their use as raf inhibitors |
| 10/21/2004 | US20040209876 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
| 10/21/2004 | CA2521201A1 Substituted pyrazoles for use in the prophylaxis or treatment of a disease which can be influenced by the binding of the substitued pyrazoles to 5ht receptors |
| 10/20/2004 | EP1468998A1 Crystalline monohydrate of Tiotropium bromide and process for its preparation |
| 10/20/2004 | EP1467993A1 Method for producing scopine esters |
| 10/20/2004 | CN1538951A Omega-aminoalkylamides of R-2-aryl-propionic acids as inhibitors of chemotaxis of polymorphonucleate and mononucleate cells |
| 10/14/2004 | WO2004087700A1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain |
| 10/14/2004 | WO2004087159A1 Bicyclic piperidine derivatives as melanocortin-4 receptor agonists |
| 10/14/2004 | DE10315572A1 Substituierte Pyrazole Substituted pyrazoles |
| 10/14/2004 | CA2519939A1 Bicyclic piperidine derivatives as melanocortin-4 receptor agonists |
| 10/13/2004 | EP1466913A1 Benzoylecgonine, ecgonine and ecgonidine derivatives |
| 10/13/2004 | EP1465629A1 5-ht3 receptor antagonists and methods of use |
| 10/13/2004 | EP0934928B1 Cyclic amine derivatives |
| 10/06/2004 | EP1037892B1 Piperidine derivatives |
| 10/05/2004 | CA2299200C Process for the preparation of endo-nortropine using 8-benzyl-nortropan-3-one perchlorate as the intermediate, as well as the latter salt |
| 09/30/2004 | US20040192681 N-acylsulfonamide apoptosis promoters |
| 09/29/2004 | EP1461318A2 Tetrahydroquinoline analogues as muscarinic agonists |
| 09/29/2004 | EP1390364B1 Aryl-8-azabicyclo 3.2.1]octanes for the treatment of depression |
| 09/29/2004 | EP1028961B1 Pleuromutilin derivatives as antimicrobials |
| 09/29/2004 | CN1168719C 6-phenylpyridyl-2-amine derivatives and pharmaceutical composition and use |
| 09/23/2004 | US20040186153 Pharmaceutical use of N-carbamoylazole derivatives |
| 09/22/2004 | EP1100781B1 High affinity ligands for nociceptin receptor orl-1 |
| 09/22/2004 | EP0929319B1 Dopamine and serotonin transporter ligands and imaging agents |
| 09/22/2004 | EP0914321B1 Indole derivatives for the treatment of osteoporosis |
| 09/16/2004 | WO2004058712A3 Herbicidally active nicotinoyl derivates |
| 09/16/2004 | WO2003066004A3 Therapeutic compounds |
| 09/16/2004 | US20040180877 Nicotinic acetylcholine receptor cholinergic ligands, monoamine receptor and transporter modulators; such as 1-(2-Benzo[b]thiophenyl-1,1-dioxide)-imidazolidine |
| 09/15/2004 | EP1326862B1 Crystalline monohydrate of tiotropiumbromide, method for producing the same and the use thereof in the production of a medicament |
| 09/15/2004 | EP0990653B1 2-oxoimidazole derivatives |
| 09/14/2004 | US6790857 Benzoylecgonine compositions and methods for producing them |
| 09/14/2004 | US6790856 Fluorenecarboxylic acid esters, process for the manufacture thereof, and use thereof as medicaments |
| 09/10/2004 | WO2004076448A1 Ccr-3 receptor antagonists |
| 09/10/2004 | WO2004076444A2 Novel hydroxycoumaranone derivatives as antitumor and antimetastatic |
| 09/10/2004 | CA2516634A1 Ccr-3 receptor antagonists |
| 09/09/2004 | US20040176416 Bridged bicyclic amine derivatives useful as CCR-3 receptor antagonists |
| 09/09/2004 | US20040176384 inhibit Tissue factor expression and vascular permeability factor expression in cancer cells and in vascular endothelial cells in the tumor microenvironment; low toxicity to normal vascular endothelial cells |
| 09/09/2004 | US20040176361 2H-Isoquinolin-1-one derivatives as poly/ADP-ribose/ polymerase inhibitors |
| 09/08/2004 | EP1453511A1 Tropane derivatives having dopamine reuptake inhibitor activity for the treatment of ischemic diseases |
| 09/08/2004 | EP1345603A4 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents |
| 09/08/2004 | EP1292281B1 Novel tiotropium-containing inhalation powder |
| 09/08/2004 | EP0993456B1 2-substituted 4,5-diaryl imidazoles |
| 09/07/2004 | US6787652 Lowering lipids and serum cholesterol without generating adverse cardiac effects; 4,5-dihydro-3,5-dioxo-1,2,4-triazine derivatives |
| 09/02/2004 | WO2004054974A3 Piperidine derivatives as ccr5 antagonists |
| 09/02/2004 | WO2004035569A3 Novel compounds with antibacterial activity |
| 09/02/2004 | WO2004014851A3 Tyrosine kinase inhibitors |
| 09/02/2004 | US20040171848 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 09/02/2004 | US20040171834 Esterification of tropane with carbonyldiimidazole; then reacting with alkanediol |
| 09/02/2004 | US20040171635 Novel tropane esters and methods for producing and using them |
| 09/02/2004 | US20040168739 Metering method for particulate material |
| 09/01/2004 | EP1452534A1 Pleuromutlin derivatives as antimicrobials |
| 09/01/2004 | EP1452527A1 Azabicyclo compound, matrix metalloprotease inhibitor, and skin preparation |
| 09/01/2004 | CN1525968A Compositions for prevention or treatment of hepatopathy |
| 08/31/2004 | US6784200 Such as n-3-(cis-2,3,3a,4,9,9a-hexahydro-1h-benz(f)isoindol-2-yl)-n-prop-1-yl-n'-3 -acetylphenylurea for prevention of inflammatory diseases (asthma and allergies) |
| 08/26/2004 | WO2004072075A1 Novel 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 08/26/2004 | WO2004072071A1 8-aza-bicyclo (3.2.1) octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 08/26/2004 | WO2004050610A3 Modulators of melanocortin receptor |
| 08/26/2004 | US20040167341 Pyrrolidines as dipeptidyl peptidase inhibitors |
| 08/26/2004 | CA2515732A1 Novel 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 08/26/2004 | CA2515584A1 8-aza-bicyclo (3.2.1) octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 08/25/2004 | EP1448566A2 Chemokine receptor antagonists and methods of use thereof |
| 08/19/2004 | WO2004069285A1 Improved radiometal complex compositions |
| 08/19/2004 | CA2514307A1 Improved radiometal complex compositions |
| 08/17/2004 | US6777423 Crystalline tiotropium bromide monohydrate, processes for the preparation thereof, and pharmaceutical compositions |
| 08/12/2004 | WO2004052888A3 Tropane esters and methods for producing and using them |
| 08/12/2004 | US20040158069 An ester of 3-hydroxy-8-methyl-6,7-(amino-methylenedioxy)-8-azabicyclo(3.2.1)octane; intermediate to tiotropium bromide for example |
| 08/12/2004 | US20040157886 Brain disorders; central nervous system disorders; viricides |
| 08/12/2004 | US20040157844 6-azauracil derivatives as thyroid receptor ligands |
| 08/12/2004 | US20040157832 Fluorenecarboxylic acid esters, process for the manufacture thereof, and use thereof as medicaments |
| 08/11/2004 | EP1444990A1 Improved Radiometal Complex Compositions |
| 08/11/2004 | EP1444230A1 Benzoylecgonine compositions and methods for producing them |
| 08/11/2004 | EP1334092A4 Process for preparation of bicyclic and polycyclic molecules |
| 08/11/2004 | CN1520414A Novel compound, its prepn. and application |
| 08/11/2004 | CN1520413A Technical synthesis method for producing tropenol |
| 08/11/2004 | CN1520294A Crystalline anticholinergic, method for its prodn., and use thereof in prdon of drug |
| 08/05/2004 | WO2004064789A2 Quaternary antimuscarinic compounds for the treatment of bladder diseases |
| 08/05/2004 | US20040152723 Pharmaceutical compositions and methods for use |
| 08/04/2004 | EP1442036A2 Heteroaryl derivatives as superior ligands for nociceptin receptor orl-1 |
| 08/03/2004 | US6770655 2-imidazomethyl- pyrido(4,3-b)indol-1-one or -carbazol-1-one derivatives containing an ester group; especially for treating irritable bowel syndrome. |
| 08/03/2004 | CA2136836C Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension |
| 07/29/2004 | WO2004062610A2 4',4''-SUBSTITUTED 3α-(DIPHENYLMETHOXY)TROPANE ANALOGS FOR TREATMENT OF MENTAL DISORDERS |
| 07/29/2004 | WO2004045533A3 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs |
| 07/29/2004 | WO2003099783A3 Tropane compounds |
| 07/29/2004 | US20040147746 Such as N-{2-[2-(5-Bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-butyl-guanidine; involuntary weight loss disorders |
| 07/29/2004 | US20040147555 Anticoagulants; brain disorders; blood circulation disorders; myocardial infraction |
| 07/28/2004 | EP1440976A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production |
| 07/22/2004 | WO2004060865A2 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines |
| 07/22/2004 | WO2004060371A1 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines |
| 07/22/2004 | US20040142962 Attention defect disorders; alcoholism; drug abuse; Parkinson's disease; anxiolytic agents; antidepressants |
| 07/22/2004 | US20040142922 Benzodioxole derivatives |
| 07/21/2004 | EP1438053A1 Pyrimidine derivatives, pharmaceutical agent containing said compounds, use and method for making same |
| 07/15/2004 | WO2004058712A2 Herbicidally active nicotinoyl derivates |
| 07/15/2004 | WO2004045536A3 Method and compositions for temporarily incapaciting subjets |