| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
|---|
| 01/27/2005 | US20050020621 Prevent reduced blood flow to brain |
| 01/27/2005 | US20050020578 Oxidoreductase enzyme inhibitors such as (R)-1-[4-(2-methyl-4-phenyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-pyrimidin-2-yl-ethanol, used as antidiabetic agents |
| 01/27/2005 | DE10331350A1 Inhalation powder useful for treating respiratory diseases comprises a 9,9-dimethyl-7-(2,2-diphenylpropionyloxy)-3-oxa-9-azatricyclononane salt and a finely divided excipient |
| 01/26/2005 | EP1500643A1 Benzamide derivatives |
| 01/26/2005 | EP1499619A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and method for the production thereof |
| 01/26/2005 | EP1499311A1 Substituted benzazoles and use thereof as raf kinase inhibitors |
| 01/25/2005 | US6846835 Treating chronic obstructive pulmonary disease, chronic bronchitis, asthma, chronic respiratory tract obstruction, fibroid lung, pulmonary emphysema or rhinitis |
| 01/20/2005 | WO2005005452A1 Specific glucocorticosteroid compound having anti- inflammatory activity |
| 01/20/2005 | WO2005005451A1 Specific glucocorticosteroid compound having anti- inflammatory activity |
| 01/20/2005 | WO2005005425A1 N-(heterobicycloalkanes)-subtituted indoles- or heteroderivatives thereof |
| 01/20/2005 | WO2005005397A1 5-substituted quinazolinone derivatives |
| 01/20/2005 | US20050014782 Novel n-(heterobicycloalkanes)-substituted indoles-or heteroderivatives thereof |
| 01/20/2005 | US20050014757 Serotonin receptor antagonist; psychological disorders; side effect reduction |
| 01/20/2005 | CA2531749A1 N-(heterobicycloalkanes)-subtituted indoles- or heteroderivatives thereof |
| 01/20/2005 | CA2530450A1 5-substituted quinazolinone derivatives |
| 01/19/2005 | EP1497289A1 Medicaments containing betamimetic drugs and a novel anticholinesterase drug |
| 01/19/2005 | EP1497288A1 Novel ester hydroxy-substituted nitrogen heterocycles as antagonists of the muscarinic m3 receptor, methods for the production thereof, and use thereof as a medicament |
| 01/19/2005 | EP1496902A1 Medicaments containing steroids and a novel anticholinesterase drug |
| 01/19/2005 | EP1496858A1 Inhalation kit comprisung inhalable powder of tiotropium |
| 01/18/2005 | US6843979 Radiolabeled compounds useful as imaging agents for visualizing the location and density of serotonin transporter by tomography imaging; as diagnostic and therapeutic agents for diseases associated with serotonin transporter dysfunction |
| 01/13/2005 | WO2005002577A1 Dual nk1/nk3 antagonists for treating schizophrenia |
| 01/13/2005 | US20050009808 Azabicyclo compound matrix metalloprotease inibitor and skin preparation |
| 01/13/2005 | CA2530886A1 Dual nk1/nk3 antagonists for treating schizophrenia |
| 01/12/2005 | EP1496058A1 Novel N-(heterobicycloalkanes)-substituted Indoles or heteroderivatives thereof |
| 01/12/2005 | CN1564811A Acylsulfonamides as inhibitors of steroid sulfatase |
| 01/11/2005 | CA2269128C Piperazino derivatives as neurokinin antagonists |
| 01/06/2005 | US20050004163 opioid receptor modulators; analgesics, cardiovascular agents and respiratory disease medicants, immunosuppressants, antiinflammatories: reduced side effects |
| 01/06/2005 | US20050004148 Human immunodeficiency and hepatitis B infections; high activity, low toxicity |
| 01/05/2005 | EP1493744A1 Tropane analogs and methods for inhibition of monoamine transport |
| 01/05/2005 | EP1492789A1 Tropane derivatives as ccr5 modulators |
| 01/05/2005 | EP0996619B1 Tropane analogs and methods for inhibition of monoamine transport |
| 01/05/2005 | CN1561212A Benzimidazolidinone derivatives as muscarinic agents |
| 12/30/2004 | US20040267010 For therapy of central nervous system disorders |
| 12/29/2004 | WO2004113334A1 Novel 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 12/29/2004 | EP1490336A1 Piperidine or 8-aza-bicyclo(3.2.1)oct-3-yl derivatives useful as modulators of chemokine receptor activity (especially ccr5) |
| 12/29/2004 | CN1558719A Nicotinic acid-heterocyclyl-amides and analogous pyrimidine derivatives serving as pesticides |
| 12/29/2004 | CN1182123C Substituted bicyclic derivatives useful as anticancer agents |
| 12/29/2004 | CA2530023A1 Novel 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 12/28/2004 | US6835733 Tropane linked benzofuran derivatives |
| 12/23/2004 | WO2004091518A3 Cxcr4 chemokine receptor binding compounds |
| 12/23/2004 | CA2528652A1 Nk1 antagonist |
| 12/22/2004 | EP1487832A1 Micronized crystalline tiotropium bromide |
| 12/22/2004 | EP1487831A1 Difurylglycolic acid tropenol esters used as anticholinesterase drugs |
| 12/22/2004 | EP1487822A2 Pyrrole-2,5-dione derivatives and their use as gsk-3 inhibitors |
| 12/22/2004 | EP1487807A2 New compounds |
| 12/22/2004 | CN1556805A Piperidine derivative as NMDA receptor antagonist |
| 12/16/2004 | US20040254190 3-Benzhydrylidene-8-aza-bicyclo[3.2.1]octane derivatives with opioid receptor activity |
| 12/15/2004 | EP0988263B1 Process for the production of radioiodinated neuroreceptor agents |
| 12/09/2004 | WO2004106333A1 Azabicycloalkane compounds as muscarinic receptor antagonists |
| 12/08/2004 | EP1484327A1 Nitrogenous heterocyclic compound and medicine thereof |
| 12/08/2004 | EP1483237A2 Tropane compounds |
| 12/02/2004 | US20040242636 Enzyme inhibitors as antiinflammatory ageents for psoriasis, obesity |
| 12/02/2004 | US20040242622 Azabicycloalkane compounds |
| 12/02/2004 | US20040242572 New carboxamide compounds having melanin concentrating hormone antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture |
| 11/30/2004 | CA2075189C Method and compositions for the synthesis of bch-189 and related compounds |
| 11/25/2004 | WO2004101562A2 Bridged n-arylsulfonylpiperidines as gamma-secretase inhibitors |
| 11/25/2004 | WO2004100946A1 1- (2h-pyrazol -3-yl) -3yl) {4-`1- (benzoyl) -piperidin-4-ylmethyl!-phenyl}-urea derivatives and related compounds as inhbitors of p38 kinase and/or tnf inhibitors for the treatment of imflammations |
| 11/25/2004 | WO2004089942A3 Benzimidazolidinone derivatives as muscarinic agents |
| 11/25/2004 | US20040235906 Substituted amine derivatives and their use as monoamine neurotransmitter re-up-take inhibitors |
| 11/25/2004 | US20040235823 Administering compounds such as N-(2-pyridinylmethyl)-N'-(6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-yl)-1,4-benzenedimethanamine for therapy of disease mediated by a chemokine receptor |
| 11/25/2004 | CA2526065A1 Benzimidazole-derivatives as factor xa inhibitors |
| 11/25/2004 | CA2525124A1 Bridged n-arylsulfonylpiperidines as gamma-secretase inhibitors |
| 11/24/2004 | EP1478356A2 Therapeutic compounds |
| 11/18/2004 | WO2004099178A1 Chemical compounds |
| 11/18/2004 | WO2004087700A8 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain |
| 11/18/2004 | US20040229902 For therapy and prophylaxis of Alzheimer's disease and other diseases relating to the deposition of amyloid protein |
| 11/18/2004 | US20040228806 For use in therapy of chronic obstructive pulmonary disease and asthma; an inhalette capsule contains a mixture of coarser and fine excipient particles |
| 11/18/2004 | CA2521580A1 Chemical compounds |
| 11/17/2004 | EP1476158A1 Nicotinamide derivatives useful as pde4 inhibitors |
| 11/17/2004 | EP1476157A1 Nicotinamide derivatives useful as pde4 inhibitors |
| 11/17/2004 | EP1476151A1 1-arylsulfonyl-3-substitued indole and indoline derivates useful in the treatment of central nervous system disorders |
| 11/17/2004 | CN1546472A Pyridyl alkane acid amides as cytostatics and immunosupressives |
| 11/17/2004 | CN1546470A 6-phenylpyridyl-2-amine derivatives |
| 11/16/2004 | US6818658 Treating obesity, diabetes, sexual dysfunction, including erectile dysfunction and female sexual dysfunction. |
| 11/16/2004 | US6818453 Comprises 8-aza bicyclo(3,2,1) octane bridge structure and maleimide moiety |
| 11/11/2004 | WO2004096799A1 Tropane derivatives and their use as ace inhibitors |
| 11/11/2004 | US20040224975 Nicotinamide derivatives useful as PDE4 inhibitors |
| 11/11/2004 | US20040224925 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs |
| 11/11/2004 | US20040224924 Programming a specific course and rate for a parent drug compound's metabolism that leads to an inactive or weakly active and non-toxic metabolite when the parent drug compound is administered, comprising modifying the parent drug compound by forming one or more of a predetermined chemical arrangement |
| 11/11/2004 | CA2521957A1 Tropane derivatives and their use as ace inhibitors |
| 11/10/2004 | EP1475379A1 Use of scopine ester derivatives for the synthesis of drugs |
| 11/09/2004 | US6815458 Nervous system disorders |
| 11/09/2004 | US6815452 Fluorenecarboxylic acid esters, process for the manufacture thereof, and use thereof as medicaments |
| 11/04/2004 | WO2004060865A3 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines |
| 11/04/2004 | WO2004050681A3 Kinase modulators |
| 11/04/2004 | US20040220246 2-imidazomethyl- pyrido(4,3-b)indol-1-one or -carbazol-1-one derivatives containing an ester group; especially for treating irritable bowel syndrome. |
| 11/04/2004 | US20040220173 central nervous system disorders; psychological disorders; Parkinson's disease; Huntington's disease ; sleep disorders |
| 11/03/2004 | EP1472251A1 Novel fluorene carboxylic acid esters, methods for the production thereof, and use of the same as pharmaceuticals |
| 11/03/2004 | EP1472250A1 Anticholinergic agents, method for producing the same and use thereof as medicaments |
| 11/03/2004 | EP1472249A1 Xanthene-carboxylic acid esters of tropenol and scopine as m3 antagonists, method for producing the same and use thereof as medicaments |
| 11/03/2004 | EP1472248A1 Modulators of acetylcholine receptors |
| 11/03/2004 | EP1212103B1 4-fluoroalkyl-3-halophenyl nortropanes |
| 11/03/2004 | EP1051417B1 Process for the preparation of 8-azabicyclo(3.2.1)octane derivatives |
| 11/02/2004 | CA2296313C 2-aminopyridines containing fused ring substituents as nos inhibitors |
| 10/28/2004 | WO2004092165A1 3-benzhydrylidene-8-aza-bicyclo[3.2.1]octane derivatives with opioid receptor activity |
| 10/28/2004 | WO2004091518A2 Cxcr4 chemokine receptor binding compounds |
| 10/28/2004 | WO2004076444A3 Novel hydroxycoumaranone derivatives as antitumor and antimetastatic |
| 10/28/2004 | WO2004010512A3 Heteroatom-containing diamondoid transistors |
| 10/28/2004 | CA2522199A1 3-benzhydrylidene-8-aza-bicyclo¬3.2.1|octane derivatives with opioid receptor activity |
| 10/28/2004 | CA2520259A1 Cxcr4 chemokine receptor binding compounds |