Patents for C07D - Heterocyclic compounds (10,420) |
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03/23/2010 | US7683178 Method for the synthesis of a benzimidazole compound |
03/23/2010 | US7683067 3-heterocyclyl-indole derivatives as inhibitors of glycogen synthase kinase-3 (GSK-3) |
03/23/2010 | CA2389767C Quinazoline derivatives as vegf inhibitors |
03/18/2010 | US20100069408 Trisubstituted triazolopyrimidines for use in platelet aggregation inhibition |
03/18/2010 | US20100069375 Indolone-Acetamide Derivatives, Processes for Preparing Them and Their Uses |
03/17/2010 | EP2163546A1 Quinazoline derivatives |
03/16/2010 | US7678802 Voltage gated sodium and calcium channel inhibitors |
03/16/2010 | CA2510519C Condensed furan compounds |
03/11/2010 | US20100062996 Dioxolane derivates for the treatment of cancer |
03/10/2010 | EP2161258A2 4-oxoquinoline compound and use thereof as hiv integrase inhibitor |
03/04/2010 | US20100056632 CRYSTALLINE FORM OF y-AMINOBUTYRIC ACID ANALOG |
03/04/2010 | US20100056551 Anti-cancer cyclopenta [G] quinazoline compounds |
03/02/2010 | US7671053 such as 2-chloro-N-(1-hydroxy-cycloheptylmethyl)-5-[4-(2-hydroxy-3-methoxy-propyl)-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl]-benzamide for treatment of asthma and COPD; purinergic receptors (P2X7) |
03/02/2010 | US7671051 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 |
02/25/2010 | WO2004092124A8 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |
02/24/2010 | CN100591676C 2- and 2,5-substituted phenylketo-enols |
02/24/2010 | CN100591657C Indane acetic acid compound |
02/23/2010 | US7666881 4-(4-(4-(Hydroxydiphenylmethyl)-1-piperidinyl)-1-hydroxybutyl)-alpha,alpha -dimethylbenzene acetic acid hydrochloride formed by azeotropic distillation |
02/16/2010 | US7663001 Preparation of isoxazolin-3-ylacylbenzene |
02/16/2010 | US7662835 Methods of treating allergic reactions using an anhydrous form of antihistaminic piperidine derivatives |
02/16/2010 | CA2406095C Synthetic process for the manufacture of an ecteinaschidin compound |
02/16/2010 | CA2385938C Cyclic amine compounds as ccr5 antagonists |
02/11/2010 | US20100035891 Pharmaceutically Active Compounds |
02/11/2010 | US20100035842 Amino alcohol compounds or phosphonic acid derivatives thereof |
02/09/2010 | US7659408 Especially in which the amide nitrogen is substituted with an adamantyl group, e.g., N-adamantyl-4-chloro-5-(o-fluorophenyl)-1-methyl-3-pyrazolecarboxamide; treating hyperglycemia, diabetes or insulin resistance |
02/09/2010 | US7659276 1-{[1-(2,6-dimethylphenyl)-1H-tetrazol-5-yl]phenylmethyl}-4-(3-phenylallyl)piperazine; G-protein coupled receptor antagonist; antidepressant, anxiolitic agent, obesity |
02/09/2010 | CA2484954C 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors |
02/09/2010 | CA2407112C Method for treating cancer, visualizing cell structures, and isolating organelles using organelle crystallizing agents |
02/09/2010 | CA2274201C Di-or triaza-spiro[4,5]decane derivatives |
02/04/2010 | US20100029639 Ion channel modulating compounds and uses thereof |
02/02/2010 | US7655664 Hydantoin derivatives as metalloproteinase inhibitors |
02/02/2010 | US7655650 Oxadiazine derivatives |
02/02/2010 | CA2516682C Imidazol-4-yl-ethynyl-pyridine derivatives |
02/02/2010 | CA2507923C Tetracyclic 3-substituted indoles having serotonin receptor affinity |
02/02/2010 | CA2294809C Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same |
01/28/2010 | US20100021388 Benzothiazole derivative compounds, compositions and uses |
01/27/2010 | CN101633655A Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof |
01/21/2010 | US20100016323 2-phenyl substituted imidazotriazinones as phosphodiesterase inhibitors |
01/21/2010 | US20100016320 Aryl-substituted pyrazole-amide compounds useful as kinase inhibitors |
01/20/2010 | EP2145888A1 Deazapurine derivatives as HSP90-Inhibitors |
01/19/2010 | US7649008 Crystal of 4-(1-((4-methylbenzothiophen-3-yl)methyl)benzimidazol-2-ylthio)butanoic acid; has chymase inhibitory activity in living body and can be used as a preventive and/or remedy for inflammatory diseases, allergic diseases, respiratory tract diseases, circulatory diseases, or bone metabolic diseases |
01/19/2010 | US7648992 Metalloproteinase 9 and/or 12 inhibitors; such as 5-({[4-[(2-cyclopropylpyrimidin-5-yl)ethynyl]-3,6-dihydropyridin-1(2H1)-yl]sulfonyl}methyl)-5-methylimidazolidine-2,4-dione; synthesis; asthma, chronic obstructive pulmonary disease |
01/19/2010 | US7648985 Oxabispidine compounds and their use in the treatment of cardiac arrhythmias |
01/14/2010 | US20100009999 Alkyl substituted indoloquinoxalines |
01/14/2010 | US20100009900 2-{3-[2-(2,3-Dihydro-benzofuran-5-yl)-ethyl]-1H-indol-4-yloxy} beta -D-glucopyranoside; sodium glucose transporter inhibitor; antidiabetic agent; Syndrome X, obesity, nephropathy, neuropathy, retinopathy, atherosclerosis, hypertension, ischemia, stroke, heart disease, irritable bowel disorder, cataracts |
01/13/2010 | EP1144388B1 Acyl derivatives which treat vla-4 related disorders |
01/13/2010 | CN100579976C P38 inhibitors and methods of use thereof |
01/12/2010 | US7645887 Indolone-acetamide derivatives, processes for preparing them and their uses |
01/12/2010 | US7645784 Benzimidazole derivatives |
01/12/2010 | US7645761 Indoline derivatives |
01/12/2010 | CA2560489C Pyranone compounds useful to treat retroviral infections |
01/12/2010 | CA2481461C Derivatives of n-[phenyl(piperidin-2-yl) methyl] benzamide, the preparation method thereof and application of same in therapeutics |
01/12/2010 | CA2407838C Pyrano, piperidino, and thiopyrano compounds and methods of use |
01/07/2010 | US20100004444 Novel Triazolo pyrimidine compounds |
01/07/2010 | US20100004285 POLYMORPH OF 4-[2-[4-[1-(2-ETHOXYETHYL)-1H-BENZIMIDAZOLE-2-YL]-1-PIPERIDINYL]ETHYL]-alpha alpha-DIMETHYL-BENZENEACETIC ACID |
01/07/2010 | US20100004188 Substituted benzimidazole-, benztriazole-, and benzimidazolone-o-glucosides |
01/06/2010 | EP2140864A2 Use of GAL3 receptor antagonists for the treatment of depression and / or anxiety and compounds useful in such methods |
01/06/2010 | EP2140862A2 Use of GAL 3 receptor antagonists for the treatment of depression and /or anxiety and compounds useful in such methods |
01/06/2010 | CN100577680C Inhibition of SyK kinase expression |
01/06/2010 | CN100577643C Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists |
01/05/2010 | US7642279 Atipamezole hydrochloride crystallization method |
12/31/2009 | US20090326233 4-phenylpiperidine compounds |
12/31/2009 | US20090326221 New oxabispidine compunds useful in the treatment of cardiac arrhythmias |
12/31/2009 | US20090326038 Method for treating a immunology-related disease |
12/31/2009 | US20090325968 Compositions Useful as Inhibitors of Protein Kinases |
12/30/2009 | EP1608632B1 Quinazolines useful as modulators of ion channels |
12/29/2009 | US7638635 Using alkylmetal reagents for directed metalation of azaaromatics |
12/29/2009 | US7638630 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors |
12/29/2009 | US7638623 Galactoside inhibitors of galectins |
12/29/2009 | US7638551 Amino alcohol compounds or phosphonic acid derivatives thereof |
12/29/2009 | US7638527 4-[(4-N,N-diethylaminocarbonyl)phenyl]-spiro[2H,1-benzopyran-2,4'-piperidine; ligands of delta opioid receptor; analgesic, anxiolitic, antidepressant, analgesic; gastrointestinal disorders, neurodegenerative diseases; side effect reduction |
12/29/2009 | CA2408914C Novel triazolo pyrimidine compounds |
12/23/2009 | EP2135952A2 Cripto antagonism of activin and TGF-beta signaling |
12/23/2009 | EP1608654B1 8-SUBSTITUTED-6, 7, 8,9-TETRAHY9DROPYRIMIDO (1,2- a) PYRIMIDIN-4-ONE DERIVATIVES |
12/23/2009 | CN100572364C HIV replication inhibiting pyrimidines and triazines |
12/17/2009 | US20090312543 Pyrazole compounds useful as protein kinase inhibitors |
12/16/2009 | EP2133348A1 Aryl-substituted pyrazole-amide compounds useful as kinase inhibitors |
12/15/2009 | US7632970 Such as (R,R)-trans-1-[3,5-bis(trifluoromethyl)phenyl]-3-[2-(N,N-dimethylamino)cyclohexyl]thiourea |
12/15/2009 | CA2481078C Method and compositions for the synthesis of bch-189 and related compounds |
12/10/2009 | US20090306141 Novel Compounds |
12/08/2009 | US7629467 Diphenyl substituted cycloalkanes, compositions containing such compounds and methods of use |
12/08/2009 | US7629374 Use of aminoindazole derivatives for the inhibition of tau phosphorylation |
12/03/2009 | US20090299066 Triazolone derivatives as mmp inhibitors for the treatment of asthma and copd |
12/03/2009 | US20090299065 Process for the manufacture of organic compounds |
12/03/2009 | US20090298841 serotonin receptor modulators such as 8-(4-Methyl-piperazin-1-yl)-3-phenylsulfonylquinoline, used for treating obesity, nervous system disorders such as dementia, schizophrenia and Alzheimer's disease, and as cognition activators |
12/02/2009 | EP1551802B1 Indole-3-sulphur derivatives |
12/02/2009 | CN100564358C Method for making 4-(3,4-dichlorophenoxy)piperidine |
12/02/2009 | CN100564344C 2- and 2,5-substituted phenylketo-enols |
12/01/2009 | US7625913 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease |
11/24/2009 | US7622489 Kinesin spindle protein inhibitor; antiproliferative agents; anticancer agents; 4-(2,5-difluorophenyl)-N-3-fluoropyrrolidin-3-yl)-2-hydroxymethyl-2-phenyl-2,5-dihydro-1N-pyrrol-1-carboxamide |
11/24/2009 | CA2451124C Method for the preparation of escitalopram |
11/19/2009 | US20090286876 Neuroprotective benzoate and benzamide compounds |
11/18/2009 | EP1765779B1 New substituted piperidines as modulators of dopamine neurotransmission |
11/18/2009 | EP1218354B1 Quinazoline derivatives and their use as pharmaceuticals |
11/18/2009 | CN101579344A Low hygroscopic aripiprazole drug substance and processes for the preparation thereof |
11/18/2009 | CN101579343A Low hygroscopic aripiprazole drug substance and processes for the preparation thereof |
11/17/2009 | US7619100 Physiologically active substances |
11/17/2009 | CA2521950C Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |
11/17/2009 | CA2432181C Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists |
11/17/2009 | CA2398992C Therapeutic or preventive agent for pulmonary insufficiency containing a diaminotrifluoromethylpyridine derivative |