Patents for C07D - Heterocyclic compounds (10,420) |
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07/21/2010 | EP1399445B9 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists |
07/21/2010 | CN1751031B HIV replication inhibiting pyrimidines |
07/20/2010 | US7759486 2,4,5-Trisubstituted pyrimidine compounds |
07/20/2010 | US7759361 treating a cancer, autoimmune diseases and cardiovscular disorders comprising administering drugs such as Isobutyric acid 2-isobutyryloxymethyl-3-oxo-1-aza-bicyclo[2.2.2]oct-ylmethyl ester; antiproliferative agents |
07/20/2010 | US7759346 [[2-(amino-3,4-dioxo-1-cyclobuten-1-yl)amino]alkyl]-acid derivatives for the treatment of pain |
07/13/2010 | CA2448303C Biologically active methylene blue derivatives |
07/08/2010 | US20100172834 Method for automated, large-scale measurement of the molecular flux rates of the proteome or the organeome using mass spectrometry |
07/07/2010 | CN1615166B Device for mini-invasive ultrasound treatment of an object by a heat-isolated transducer |
07/06/2010 | US7749999 Alpha-ketoamides and derivatives thereof |
07/06/2010 | CA2397497C Process for the preparation of 5-carboxyphthalide and its use for the production of citalopram |
06/30/2010 | EP1841763B1 5-heteroaryl thiazoles and their use as pi3k inhibitors |
06/30/2010 | CN101759645A P38 inhibitors and methods of use thereof |
06/29/2010 | US7745481 Methods and compositions for the treatment and prevention of tumors, tumor-related disorders and cachexia |
06/29/2010 | US7745466 Magnesium salt of S-omeprazole trihydrate of crystal form and another drug such as NSAID, antibiotic, antacid, alginates or prokinetic agents; gastric acid secretion inhibitor, and is useful as an antiulcer agent |
06/29/2010 | US7745465 Antiischemic agents; antiinflammatory agents; antiallergens; autoimmune disease |
06/29/2010 | US7745426 vitamin B6-based component selected from pyridoxal, pyridoxamine or pyridoxine chemically linked to antiepileptic agents, neuroprotectants, neurotransmitters or nootropic agents, used for the treatment of epilepsy |
06/29/2010 | CA2442881C New process for the industrial synthesis of the tetraesters of 5-[bis(carboxymethyl)amino]-3-carboxymethyl-4-cyano-2-thiophenecarboxylic acid, and application to the synthesis ofbivalent salts of ranelic acid and their hydrates |
06/24/2010 | US20100160343 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by vla-4 |
06/24/2010 | US20100160341 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by vla-4 |
06/23/2010 | CN1821236B Therapeutic heterocyclic compounds |
06/22/2010 | US7741362 4-amino-(S)-2-N-(4-methyl-1-naphthalenesulfonyl)amino-N'-(1,2,3,4-tetrahydro-1-naphthyl)butanamide, arylsulfonylamino based peptidomimetics used for imaging tissues and/or organs such as brain, blood vessels or tumors; medical diagnosis |
06/22/2010 | US7741338 mixtures comprising a polyene macrolide antibiotic and an antioxidant such as 2,6-di-tert.-butyl-4-methylphenol, that improves the stability of the polyene macrolide to oxidation |
06/22/2010 | US7741328 Treating inflammatory diseases such as rheumatoid arthritis, multiple sclerosis or Crohn's disease; Very Late Antigen-4 (VLA-4), also called alpha 4 beta 1 integrin; N-(sulfonamido-substituted pyrimidyl, pyridyl or pyrazyl)-L-4-(N,N-dimethylcarbamyloxy)phenylalanine compounds |
06/17/2010 | US20100152185 Diphenyl substituted cycloalkanes, compositions containing such compounds and methods of use |
06/16/2010 | CN1982308B Substituted pyrazoles |
06/16/2010 | CN1863806B 4-biphenylsubstituted pyrazolidin-3,5-dione derivatives |
06/16/2010 | CN1829711B Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders, process for their preparation and pharmaceutical compositions containing them |
06/16/2010 | CN1694871B Imidazolopyridines and methods of making and using the same |
06/16/2010 | CN101735131A New salts |
06/16/2010 | CN101099462B Composition for controlling harmful bio-organisms and method for controlling harmful bio-organisms using the same |
06/15/2010 | US7737161 such as 5-amino-N-(5-chloropyridin-2-yl)-3-{[(trans-4-pyrrolidin-1-ylcyclohexyl)carbonyl]amino}furo[3,2-b]pyridine-2-carboxamide, used as activated blood coagulation factor X inhibitors |
06/15/2010 | CA2379103C Novel spiro compounds |
06/15/2010 | CA2299495C Process for preparing growth hormone secretagogues |
06/10/2010 | US20100144771 Novel Hydantoin Derivatives for the Treatment of Obstructive Airway Diseases |
06/09/2010 | CN1926108B Non-nucleotide reverse transcriptase inhibitors |
06/09/2010 | CN1780835B Novel fused heterocycles and uses thereof |
06/09/2010 | CN101723948A C-6 modified indazolylpyrrolotriazines |
06/08/2010 | US7732439 Diamino-substituted phenothiazinium compound; antimicrobial photosensitisers effective against Gram negative bacteria, Gram positive bacteria; photodynamic therapy |
06/03/2010 | US20100137243 Oxazolidinone And/Or Isoxazoline As Antibacterial Agents |
06/02/2010 | EP2191832A1 Quinazoline derivatives which promote the release of parathyroid hormone |
06/01/2010 | US7728147 catalytic hydrogenation in aqueous solution comprising hydrochloric acid, concentrating, distilling; avoids use of isopropanol and ethylacetate solvents; animal sedation |
06/01/2010 | US7727997 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives |
06/01/2010 | CA2481217C Process for preparing acid salts of gemifloxacin |
05/26/2010 | CN1839116B Asymmetric urea compound and process for producing asymmetric compound by asymmetric conjugate addition reaction with the same as catalyst |
05/26/2010 | CN1713907B N-substituted pyrrolidin derivatives as dipeptidyl peptidase IV inhibitors |
05/26/2010 | CN1391469B Npyy5拮抗剂 Npyy5 antagonist |
05/25/2010 | US7723373 3-(Aryl or heteroaryl)sulfonyl- or sulfinyl-1-indoleacetic acid derivatives, e.g., 3 -[(4-chlorophenyl)sulfonyl]-2,5-dimethyl-1H-indol-1-acetic acid; treating asthma, rhinitis and other diseases in which raised levels of PGD2 or its metabolites |
05/25/2010 | US7723349 N-hydroxy-5-methyl-6-{[4-(3-methylphenyl)piperazin-1-yl]carbonyl}-5-azaspiro[2.5]octane-7-carboxamide for example; treating arthritis, cancer, cardiovascular disorders, skin disorders, inflammation and allergic conditions |
05/25/2010 | US7723333 used in treating and/or preventing cardiovascular disorders, inflammatory diseases, Alzheimer's disease, dyslipidemia and metabolic syndrome |
05/18/2010 | US7718690 e.g. [2-(1-(Benzenesulfonyl)-1H-indol-3-yloxy)ethyl]dimethylamine; serotonin, melatonin receptor ligand; antidepressant, anxiolytic agent; cognition activator; psychosis, schizophrenia, migraine headache, drug addiction, convulsions, osteoporosis, ischemic stroke, Alzheimer's, Parkinson's diseases |
05/18/2010 | US7718686 Gastrointestinal disorders; irritable bowel syndrome |
05/18/2010 | CA2430508C Condensed purine derivatives as a1 adenosine receptor antagonists |
05/13/2010 | US20100120808 Spirocyclic heterocyclic derivatives and methods of their use |
05/12/2010 | EP1564210B9 4-oxoquinoline compounds and utilization thereof as hiv integrase inhibitors |
05/12/2010 | CN1762957B 2,3-dihydro-1-indene compound and preparation method thereof |
05/11/2010 | US7714009 Nitrogen-containing fused heterocyclic compounds |
05/11/2010 | CA2318696C Triazepinones, process for their preparation and their therapeutic application |
05/05/2010 | CN1832925B New P2X7 receptor avtagonists and their use |
05/04/2010 | US7709506 Kinase inhibitors to mediate disease and as antiinflammatory agents |
05/04/2010 | US7709487 Sulfonyl-derivatives as novel inhibitors of histone deacetylase |
05/04/2010 | US7709479 Quinazoline derivatives and their use as pharmaceuticals |
04/29/2010 | US20100105920 Preparation of isoxazolin-3-ylacylbenzenes |
04/29/2010 | US20100105712 Chemical compounds |
04/29/2010 | US20100105681 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors |
04/27/2010 | US7705033 Methods and compounds for producing dipeptidyl peptidase IV inhibitors and intermediates thereof |
04/27/2010 | US7705006 Anti-cancer cyclopenta[g]quinazoline compounds |
04/27/2010 | US7704999 2-phenyl substituted imidazotriazinones as phosphodiesterase inhibitors |
04/27/2010 | US7704998 Sulfonyl-derivatives as novel inhibitors or histone deacetylase |
04/27/2010 | CA2449180C Viral polymerase inhibitors |
04/21/2010 | EP2177520A1 1,5-Di(aryl or heteroaryl)-3-halo-2(1H)-pyridones as intermediates for the preparation of AMPA receptor inhibitors |
04/21/2010 | EP1761494B1 Chemical compounds i |
04/21/2010 | EP1610780B1 Cyclic protein tyrosine kinase inhibitors |
04/21/2010 | EP1250328B2 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
04/20/2010 | US7700783 Synthesis of discodermolide and variants thereof |
04/20/2010 | US7700763 3-triazolyl-galactoside inhibitors of galectins |
04/20/2010 | US7700617 Salt of naphthyridine carboxylic acid derivative |
04/20/2010 | US7700604 (5S)-5-methyl-5-({[6-[2-(trifluoromethyl)pyrimidin-5-yl]-3,4-dihydroisoquinolin-2(1H)-yl]sulfonyl}methyl)imidazolidine-2,4-dione; asthma, rhinitis, chronic obstructive pulmonary diseases (COPD), arthritis (such as rheumatoid arthritis and osteoarthritis), atherosclerosis, cancer |
04/20/2010 | US7700591 to prevent or treat inflammatory and immunoregulatory disorders and diseases, allergic diseases, atopic conditions including allergic rhinitis, dermatitis, conjunctivitis, and asthma, as well as autoimmune pathologies such as rheumatoid arthritis and atherosclerosis |
04/20/2010 | US7700329 Methods for making simvastatin and intermediates |
04/15/2010 | US20100094017 Using alkylmetal reagents for directed metalation of azaaromatics |
04/15/2010 | US20100093785 Diamine derivatives |
04/15/2010 | US20100093735 Cytokine inhibitors |
04/15/2010 | US20100093734 Cytokine inhibitors |
04/14/2010 | EP1633727B1 Improved production of the rosuvastatin calcium salt |
04/14/2010 | EP1294922B1 Treating cancer using organelle crystallizing agents |
04/14/2010 | CN101692832A Composition for controlling harmful bio-organisms and method for controlling harmful bio-organisms using the same |
04/13/2010 | US7696217 N-(pyridin-2-ylmethyl)-4-methyl-3-oxo-4-aza-5 alpha -androst-1-en-17 beta -acetamide; enhancement of weakened muscle tone; osteoporosis, bone disorders; ; periodontal disease, frailty, aging skin, male hypogonadism, postmenopausal symptoms, inflammatory arthritis, cachexia, Alzheimer's disease |
04/13/2010 | US7696214 Confining solid tumors; administering a tyrosine kinase inhibitor as antitumor agents; 4-(6-chloro-2,3-methylenedioxyanilino)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-tetrahydropyran-4-yloxyquinazoline |
04/13/2010 | US7696206 2-phenyl substituted imidazotriazinones as phosphodiesterase inhibitors |
04/13/2010 | CA2432303C Pyrazole compounds useful as protein kinase inhibitors |
04/13/2010 | CA2425440C Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors |
04/06/2010 | US7691875 Imidazopyridine compounds, processes for their preparation and therapeutic uses thereof |
04/06/2010 | CA2453383C Piperidine derivatives as nmda receptor antagonists |
04/06/2010 | CA2397636C Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
04/06/2010 | CA2351709C Novel triazolo(4,5-d)pyrimidine compounds |
03/31/2010 | EP1756111B1 Alkyl substituted indoloquinoxalines |
03/30/2010 | US7687535 Substituted 3-sulfur indoles |
03/30/2010 | CA2572508C One pot synthesis of 2-oxazolidinone derivatives |
03/25/2010 | US20100077497 Ip-10 antibodies and their uses |
03/24/2010 | EP1615699B1 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |