Patents
Patents for C07D 419 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms (1,431)
02/2015
02/04/2015CN104327843A 一种汞离子荧光探针及制备方法和用途 One kind of mercury ion fluorescent probe and preparation and use
02/03/2015US8946434 Dihydropyridin-2(1H)-one compound as S-nirtosoglutathione reductase inhibitors and neurokinin-3 receptor antagonists
01/2015
01/28/2015CN104321320A 制备他汀的方便方法 A convenient method for preparing statins
01/27/2015US8940899 Process for the preparation of 5-substituted 1-alkyltetrazolyl oxime derivatives
01/13/2015US8933102 Pyrrolidine derived β3 adrenergic receptor agonists
01/13/2015US8933083 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
12/2014
12/30/2014US8921349 Compounds and methods for treating AIDS and HIV infections
12/18/2014US20140371205 Substituted pyrimidines for the treatment of diseases such as cancer
12/16/2014US8912326 Process of making gyrase and topoisomerase inhibitors
12/16/2014US8912324 Optically active pyrazolylaminoquinazoline, and pharmaceutical compositions and methods of use thereof
12/10/2014CN101835377B 用于防治无脊椎动物害虫的吡唑化合物 For controlling invertebrate pests pyrazole compounds
12/02/2014US8901143 Pyrimidine derivatives
12/02/2014US8901114 Oxathiazine derivatives substituted with carbocycles or heterocycles, method for producing same, drugs containing said compounds, and use thereof
11/2014
11/25/2014US8895547 Substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
11/11/2014US8883794 Pharmaceutical composition
10/2014
10/28/2014US8871930 Preparation method of alpha-imatinib mesylate
10/28/2014US8871758 Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
10/21/2014US8865900 Methyltetrazole sulfides and sulfones
10/21/2014US8865723 Selective PDE4 B inhibition and improvement in cognition in subjects with brain injury
10/07/2014US8853219 Compounds and compositions for cognition-enhancement, methods of making, and methods of treating
09/2014
09/30/2014US8846930 Derivatives of heteroarylsulfonamides, their preparation and their application in human therapy
09/30/2014US8846666 Oxathiazine derivatives which are substituted with benzyl or heteromethylene groups, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
09/30/2014US8846654 Therapeutic applications in the cardiovascular field of quinazolinedione derivatives
09/25/2014WO2014152588A1 Covalent inhibitors of kras g12c
09/16/2014CA2653666C Aryl-substituted heterocycles and their use
08/2014
08/28/2014WO2014128022A1 Convenient process for the preparation of statins
08/27/2014EP2769979A1 Process for the preparation of key intermediates for the synthesis of Statins
08/19/2014US8809372 Pyridine derivatives
08/19/2014US8809324 Substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
08/12/2014US8802675 Neuroprotective multifunctional compounds and pharmaceutical compositions comprising them
08/07/2014US20140221352 Compositions and methods for inhibition of the jak pathway
07/2014
07/29/2014CA2621137C Biocompatible n,n-disubstituted sulfonamide-containing fluorescent dye labels
07/22/2014US8785459 Quinazoline compounds as kinase inhibitors
07/16/2014CN1890221B 1-n-苯基-氨基-1h-咪唑衍生物和含有它们的医药组合物 1-n- phenyl - amino -1h- imidazole derivatives and pharmaceutical compositions containing them
07/15/2014US8779133 Compound, novel ligand, novel transition metal complex, and catalyst including novel transition metal complex
07/15/2014US8778950 Cannabinoid receptor modulators
07/08/2014US8772493 Compounds having auditory protective effect
07/08/2014US8772285 Benzothiazoles having histamine H3 receptor activity
07/01/2014US8765774 3-arylquinazolin-4-one compounds for combating invertebrate pests
07/01/2014US8765767 Positive allosteric modulators of mGluR2
07/01/2014US8765732 Aryl- or heteroaryl-substituted benzene compounds
06/2014
06/17/2014US8754226 Piperidinyl-substituted lactams as GPR119 modulators
06/12/2014WO2014086712A1 New indanyloxydihydrobenzofuranylacetic acids
06/11/2014CN103857659A Fused benzoxazepinones as ion channel modulators
06/10/2014US8748442 sGC stimulators
05/2014
05/27/2014US8735362 Insecticidal compounds based on isoxazoline derivatives
05/20/2014US8729271 Glycine transporter inhibiting substances
05/20/2014US8729085 Pharmaceutical composition
05/08/2014US20140128410 Tyrosine kinase inhibitors containing a zinc binding moiety
05/07/2014EP2726466A1 Fused benzoxazepinones as ion channel modulators
05/01/2014WO2014063929A1 Substituted pesticidal pyrazole compounds
04/2014
04/29/2014US8710231 Inhibitor of casein kinase 1delta and casein kinase 1E
04/29/2014US8710050 Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
04/23/2014EP2721016A1 Trpv4 antagonists
04/22/2014US8703941 IRAK inhibitors and uses thereof
04/22/2014US8703763 Bridged piperidine derivatives
04/22/2014CA2752131C Novel derivatives of dihydrobenzoxathiazepines, their preparation process and pharmaceutical compositions containing them
04/17/2014WO2014057435A1 Orexin receptor antagonists which are [ortho bi (hetero )aryl]-[2-(meta bi (hetero )aryl)-pyrrolidin-1-yl]-methanone derivatives
04/15/2014US8697721 Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
04/10/2014US20140100223 Compounds and methods for the treatment of isocitrate dehydrogenase related diseases
04/08/2014US8691821 Oxazolidinones as modulators of mGluR5
04/03/2014WO2014047707A1 Heteroaromatic compounds, method for preparing the compounds, pharmaceutical compositions, uses and method for treating acute and chronic pain
03/2014
03/06/2014US20140066437 Oxathiazine derivatives which are substituted with benzyl or heteromethylene groups, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
02/2014
02/25/2014US8658656 Methods and compositions utilizing quinazolinones
02/25/2014US8658650 Substituted 1,1,3,1-tetraoxidobenzo[D][1,3,2]dithiazoles as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
02/25/2014CA2593439C Thiazole-4-carboxamide derivatives as mglur5 antagonists
02/11/2014US8648189 Method for the preparation of rivoraxaban
02/05/2014EP2691391A2 Compounds and methods for the treatment of isocitrate dehydrognase related diseases
02/04/2014US8642611 Alkynylpyrimidines and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same
01/2014
01/23/2014US20140024584 Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
01/21/2014US8633210 Triazole compounds useful as protein kinase inhibitors
01/21/2014US8633208 6-1H-imidazo-quinazoline and quinolines derivatives, new MAO inhibitors and imidazoline receptor ligands
01/21/2014CA2609288C Heteroaryl-carboxylic acid (sulfamoyl alkyl) amide - derivatives as factor xa inhibitors
01/15/2014EP2683713A1 Isoxazole derivatives
01/15/2014EP2683703A1 Novel substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
01/15/2014EP2683702A1 Novel substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
01/15/2014EP2683701A1 Oxathiazine derivatives which are substituted with benzyl or heteromethylene groups, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
01/15/2014EP2683700A1 Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
01/15/2014EP2683699A1 Di- and tri-substituted oxathiazine derivates, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
01/09/2014US20140011770 Compositions and methods for inhibition of the jak pathway
01/08/2014CN103502246A Isoxazole derivatives
12/2013
12/26/2013US20130345128 Oxathiazine derivatives substituted with carbocycles or heterocycles, method for producing same, drugs containing said compounds, and use thereof
12/26/2013US20130345127 Novel substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
12/24/2013US8614231 Immunosuppressor based on the blockage of TCR-Nck interaction
12/19/2013US20130338150 Di and tri - substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
12/19/2013US20130338066 Novel substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
12/17/2013US8609686 Substituted azabicyclic compounds and the use thereof
12/10/2013US8604042 Bi-aryl meta-pyrimidine inhibitors of kinases
12/10/2013US8604032 Chemical compounds, compositions and methods for kinase modulation
12/04/2013EP2669272A1 Indole derivative and pharmacologically acceptable salt of same
12/03/2013US8598206 Trypsin-like serine protease inhibitors, and their preparation and use
11/2013
11/27/2013EP2665723A1 Process for the preparation of statins in the presence of base
11/27/2013EP2665722A1 Process for the preparation of diol sulfones
11/27/2013EP2665721A1 Methyltetrazole sulfides and sulfones
11/27/2013CN101765591B Pyrimidine derivatives useful for treatment of inflammatory or allergic conditions
11/21/2013US20130310364 Compositions and methods for inhibition of the jak pathway
11/14/2013US20130303525 Kappa opioid receptor agonists
11/12/2013US8580820 Tubulysin compounds with high cytotoxicity, pharmaceutical compositions thereof, and method of use thereof
10/2013
10/29/2013US8569302 Inhibitors of flaviviridae viruses
10/29/2013US8569285 Dihydrobenzoxathiazepine compounds, a process for their preparation and pharmaceutical compositions containing them
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