Patents for C07D - Heterocyclic compounds (10,420) |
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07/29/2008 | CA2218702C Fatty acid esters as bioactive compounds |
07/24/2008 | US20080177094 reducing an alkyl 2,4,9-trithiaadamantane-7-carboxylate to produce 7-hydroxymethyl-2,4,9-trithiaadamantane; andoxidizing 7-hydroxymethyl-2,4,9-trithiaadamantane to produce 7-carbonyl-2,4,9-trithiaadamantane; Molecular wires having 2,4,9-trithiaadamantane surface anchors |
07/24/2008 | US20080176903 Novel Compounds with Analgesic Effect |
07/24/2008 | US20080176880 Activity against strains having acquired resistance nonnucleoside reverse transcriptase inhibitors; human alpha1 acid glycoprotein nonbinding; such as 4-[[(5-bromo-4,6-dichloro)-2-pyrimidinyl]amino]-benzonitrile |
07/24/2008 | US20080176869 e.g. N-(4-fluorobenzyl)-3-hydroxy-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-2-carboxamide; viricide in combination with other HIV/AIDS antivirals, immunomodulators, antibiotics or vaccines; AIDS |
07/23/2008 | EP1671949B1 Substituted Pyridinylamines |
07/23/2008 | EP1615909B1 Piperazine derivatives and their use for the treatment of neurological and psychiatric diseases |
07/23/2008 | EP1080092B1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation |
07/23/2008 | CN100404480C Toluene methylation process |
07/22/2008 | US7402594 isoquinoline ring joined to a phenyl ring by a chemical group that is two bonds long and at least one cation or cationic group selected from sodium, potassium, ammonium, and tetraalkylammonium; Factor Xa inhibitor; anticoagulant; straightforward and economical synthesis |
07/17/2008 | US20080171758 Compounds and methods for the treatment of cancer |
07/16/2008 | EP1943293A1 Light protective additive based on organic/ inorganic hybrid polymer, method for its manufacture and use thereof |
07/16/2008 | EP1165551B1 C10 carbamoyloxy substituted taxanes as antitumor agents |
07/16/2008 | CN101219145A Quinazoline derivatives as VEGF inhibitors |
07/16/2008 | CN100402499C 2-iminopyrrolidine derivatives |
07/15/2008 | US7399577 Halogenated oxime derivatives and the use thereof |
07/10/2008 | US20080167471 comprising 4-[4-[4-(Hydroxydiphenylmethyl)-1-piperidinyl]-1-hydroxybutyl]- alpha , alpha -dimethylbenzeneacetic acid hydrochloride; antiallergic agents and bronchodilators |
07/10/2008 | US20080167469 Preparing anhydrous 4-(4-(4-(Hydroxydiphenylmethyl)-1-piperidinyl)-1-hydroxybutyl)-alpha,alpha -dimethylbenzene acetic acid hydrochloride by azeotropic distillation of the corresponding hydrate |
07/09/2008 | EP1455756B1 Pharmaceutical nanoparticulate composition of a tachykinin receptor antagonist |
07/09/2008 | EP1220842B1 Cyclic amine compound as ccr5 antagonist |
07/08/2008 | US7396935 p38 kinase inhibitors; inflammatory bowel disease, rheumatoid arthritis, psoriasis, multiple sclerosis, endotoxin shock, osteoporosis, Alzheimer's disease, and congestive heart failure |
07/08/2008 | US7396847 Oxazolidinone and/or isoxazoline as antibacterial agents |
07/08/2008 | US7396834 e.g., 3-[(4-[(diethylamino)carbonyl]phenyl)(4-benzyl-piperazin-1-yl)methyl]benzamide; opioid delta rreceptor agonist; analgesic, hypotensive agent; pain, anxiety and functional gastrointestinal disorders, immunomodulatory activities |
07/08/2008 | CA2582172C Preparation of arthropodicidal oxadiazines |
07/08/2008 | CA2432131C Pyrazole compounds useful as protein kinase inhibitors |
07/03/2008 | US20080161334 Macrolides |
07/02/2008 | EP1939203A2 Inhibitors of human phosphatidyl-inositol 3-kinase delta isoform |
07/02/2008 | EP1140857B1 Synthesis of histamine dihydrochloride |
07/01/2008 | US7393846 phosphodiesterase type 4 inhibitors; N-(3,5-dichloropyrid-4-yl)-4-difluoromethoxy-8-methanesulfonamido-dibenzo[b,d]furan-1-carboxamide; antiinflammatory agent, antiallergen; asthma or chronic obstructive pulmonary disease |
06/26/2008 | US20080153893 Pyrazole Carboxamides as Inhibitors of 11-Beta-Hydroxysteroid Dehydrogenase-1 |
06/26/2008 | US20080153864 Spiroazabicyclic Heterocyclic Compounds |
06/26/2008 | US20080153823 a group of aryl ureas in treating raf mediated diseases, and pharmaceutical compositions for use in such therapy |
06/25/2008 | EP1678499B1 Chemical compound and assay |
06/25/2008 | CN100396785C Resoldution method for racemic compound of nucleoside enantiomorph |
06/25/2008 | CN100396680C Vla-4 inhibitors |
06/25/2008 | CN100396276C Compositions containing organic compounds |
06/24/2008 | US7390818 3-(2,4-dimethoxyphenyl)-1,9-dimethyl-2-oxo-2,9-dihydro-1H-pyrido[2,3-b]indole-6-carboxylic acid; gamma-aminobutyric acid modulator; anticarcinogenic, antitumor, antiproliferative agent |
06/24/2008 | US7390810 Pyrazole-amine compounds useful as kinase inhibitors |
06/19/2008 | US20080146812 Novel Oxabispidine Compounds And Their Use In The Treatment Of Cardiac Arrhythmias |
06/18/2008 | EP1932543A2 Combination therapy for osteoporosis consisting of an estrogen agonist/antagonist and a growth hormone secretagogue |
06/18/2008 | CN101200454A Crystalline modifications of triazinylaminostilbenes |
06/18/2008 | CN101200450A 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors |
06/17/2008 | CA2302347C 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocin-10-oles, processes for their preparation and their use for medicaments |
06/12/2008 | US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection |
06/12/2008 | US20080139616 Atherosclerosis; inflammatory diseases, Alzheimer's disease, dyslipidemia, metabolic syndrome; 2-isopropyl-5-phenyl-4-[(4-phenylbutyl)amino]isothiazole-3(2H)-thione 1,1-dioxide for example |
06/11/2008 | EP1556370B1 Method for the synthesis of a benzimidazole compound |
06/11/2008 | EP1497266B1 Quinoline derivatives and their use as 5-ht6 ligands |
06/10/2008 | US7384962 Heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them |
06/10/2008 | US7384955 N-[1-(cyclohexylmethyl)-2-[(4-ethoxyphenyl)methyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]-2,2-dimethyl-propanamide; cannabinoid CB1/CB2 receptor agonists; analgesic; in therapy, in particular in the management of pain |
06/10/2008 | CA2427338C Acyl and sulfonyl derivatives of 6,9-disubstituted 2-(trans-1,4-diaminocyclohexyl)-purines and their use as antiproliferative agents |
06/10/2008 | CA2225896C Process for the production of enantiomerically-pure azetidine-2-carboxylic acid |
06/05/2008 | US20080132502 Phosphatidylinositol (PI) 3-kinase (PI3K); N-[5-(5-Benzylamino-6-chloropyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]acetamide, for example; anticancer agents, cardiovascular disorders, autoimmune disorders, rheumatic diseases |
06/05/2008 | US20080132486 Ligands for Nicotinic Acetylcholine Receptors, and Methods of Making and Using Them |
06/04/2008 | EP1927357A2 Low hygroscopic aripiprazole (crystal E) drug substance and processes for the preparation thereof |
06/04/2008 | EP1927356A1 Low hygroscopic aripiprazole (crystal D) drug substance and processes for the preparation thereof |
06/04/2008 | EP1927355A1 Low hygroscopic aripiprazole (crystal F) drug substance and processes for the preparation thereof |
06/04/2008 | CN100391930C 1, 3-propane diol derivatives as bioactive compounds |
06/03/2008 | US7381828 Forming a salt such as a tartrate or mandelate of 6-amino-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]-dioxol-4-yl]oxy}-1-ethanol, chemical intermediates |
05/28/2008 | EP1925308A1 Low hygroscopic aripiprazole (crystal G) drug substance and processes for the preparation thereof |
05/28/2008 | EP1556382B1 3-phenyl substituted pyridoindolone, preparation and therapeutic use thereof |
05/28/2008 | CN100390153C Intermediate for producing novel pyrazine derivatives |
05/27/2008 | US7378529 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 |
05/21/2008 | EP1603557A4 Synthesis of peloruside a and analogs thereof for use as antitumor agents |
05/21/2008 | EP1599206A4 Aminocyclopentyl fused heterotricylicamide modulators of chemokine receptor activity |
05/21/2008 | CN100389115C Pyridyloxymethyl and benzisoxazole azabicyclic derivatives |
05/20/2008 | US7375227 May be combined with ACE inhibitors, angiotensin or endothelin receptor antagonists, vasopressin antagonists, alpha- and beta-adrenergic antagonists, TNFalpha antagonists, and peroxisome proliferator activator receptor modulators; cardiovascular, renal, metabolic, pulmonary and psychological disorders |
05/20/2008 | CA2432223C Pyrazole compounds useful as protein kinase inhibitors |
05/20/2008 | CA2350801C Hiv replication inhibiting pyrimidines |
05/15/2008 | US20080114041 Benzothiazolesulfonamides |
05/15/2008 | US20080113972 Enzyme inhibitors of cGMP-metabolizing phosphodiesterases, for TREATMENT OF CARDIOVASCULAR DIORDERS, CEREBROVASCULAR DISORDERS, UROGENITAL DISORDERS AND ERECTILE DYSFUNCTION; chemical synthesis |
05/14/2008 | EP1689736A4 Biocidal siloxane coating material containing n-halogenated amine and amide functional groups |
05/14/2008 | EP1606277B1 Imidazol-4-yl-ethynyl-pyridine derivatives |
05/14/2008 | EP1485365B1 Sulfonyl-derivatives as novel inhibitors of histone deacetylase |
05/13/2008 | US7371744 Photosensitizers for photodynamic therapy; killing tissue, cells; anticancer agents |
05/13/2008 | US7371420 Method for producing an avocado unsaponifiable rich in furan lipids |
05/13/2008 | CA2410234C 5-chloro-3-(4-methanesulfonylphenyl)-6'-methyl-[2,3']bipyridinyl in pure crystalline form and process for synthesis |
05/13/2008 | CA2196995C Spiro-azabicyclic compounds useful in therapy |
05/08/2008 | US20080108677 Thioxothiazolidinone Compounds For Use As Pharmaceuticals |
05/08/2008 | US20080108676 Benzothiazolecarboxamides |
05/08/2008 | US20080108626 (5-amino-1-phenyl-1H-pyrazole)-(3-Amino-N-isoxazol-3-yl-4-methyl)-benzamide; p38 mitogen-activated protein kinase inhibitor; reduced levels of TNF- alpha expression; antiinfammatory agent: rheumatoid arthritis, psoriasis, multiple sclerosis, endotoxin shock, osteoporosis, Alzheimer's disease |
05/08/2008 | US20080108619 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
05/08/2008 | US20080108601 anticancer agents; catalytic hydrogenation |
05/08/2008 | US20080108591 2-amino-3,6-dihydro-4-dimethyl-amino-6-ethyl-1,3,5-triazine hydrochloride; advanced glycosylation end-products inhibitor;antidiabetic, insulin resistance, neurodegenerative disorders, renal complications, atherosclerosis, angiopathy |
05/07/2008 | EP1347981B1 Condensed purine derivatives as a 1 adenosine receptor antagonists |
05/06/2008 | US7368574 crystalline hydrate of 5-[4-[2-(N-methyl-N-(2-pyridyl) amino)ethoxy]benzyl]thiazolidine-2,4-dione, maleic acid salt, used as hypoglycemic, antilipemic or antidiabetic agents |
05/06/2008 | US7368566 Process and intermediates for preparing benzazepines |
05/06/2008 | US7368564 Bridged macrocyclic module compositions |
05/01/2008 | US20080103148 Preventing ventilator induced pneumonia; utilizing compounds having longer half life on mucosal surfaces |
05/01/2008 | US20080102031 4-[(4-N,N-diethylaminocarbonyl)phenyl]-spiro[2H,1-benzopyran-2,4'-piperidine; ligands of delta opioid receptor; analgesic, anxiolitic, antidepressant, analgesic; gastrointestinal disorders, neurodegenerative diseases; side effect reduction |
04/30/2008 | CN100384856C Heterocyclic cyclopentyl tetrahydroisoquinoline and tetrahydropyridopyridine modulators of chemokine receptor activity |
04/29/2008 | US7365205 Diamine derivatives |
04/29/2008 | US7364754 Preparing micelles entrapping photosensitive drugs; adding alkoxyorganosilane to the micelles to form complexes of silica and the micelles; subjecting the complexes of silica and micelles to alkaline hydrolysis to precipitate silica nanoparticles; isolating the precipitated nanoparticles by dialysis |
04/24/2008 | US20080097117 chemical intermediates for making antiinflammatory agents treating autoimmune disease; 1-[2-(Fluoren-3-yl)ethyl]-(4-(3-trifluoromethylphenyl)-1,2,3,6-tetrahydropyridine drug |
04/24/2008 | US20080096926 Treatment Of Cognitive Impairment Using A Selective Dopamine D1 Receptor Agonist |
04/23/2008 | CN100383141C Pyrazolo [4,3-d] pyrimidine derivatives |
04/22/2008 | US7361762 Process for preparing acid salts of Gemifloxacin |
04/17/2008 | US20080091024 Processes for the production of substituted 2-(2-pyridylmethyl) sulfinyl-1H-benzimidazoles |
04/16/2008 | EP1911462A2 Compositions comprising a sterol absorption inhibitor |
04/16/2008 | EP1165549B1 C7 carbamoyloxy substituted taxanes as antitumor agents |
04/16/2008 | CN100381423C Novel piperidine derivatives as modulators of chemokine receptor CCR5 |