Patents for C07D - Heterocyclic compounds (10,420) |
---|
10/08/2008 | EP1606283B1 P38 inhibitors and methods of use thereof |
10/08/2008 | EP1597234B1 Novel compounds |
10/08/2008 | EP1592675B1 Crystalline modifications of triazinylaminostilbenes |
10/08/2008 | CN100424082C 4-(piperidyl- and pyrrolidyl-alkyl-ureido) -quinolines as urotensin ii receptor antagonists |
10/08/2008 | CN100424080C Quinoxaline derivatives as neutrophil elastase inhibitors and their use |
10/08/2008 | CN100424079C Bis-sulfonamides |
10/07/2008 | US7432370 Mixing a racemic mixture of enantiomers of pyrrolo[2,3-d]pyrimidine compounds in a solvent, with a resolving compound having a defined stereospecificity, to form a solution and with resolving agent being capable of binding with enantiomers to form a precipitate collecting precipitate and purifying |
10/01/2008 | CN101274928A 3-substituted-4-pyrimidone derivatives |
10/01/2008 | CN100422160C Novel morpholine derivatives, method for production thereof and pharmaceutical preparations containing said derivatives |
10/01/2008 | CN100422157C Improved production of rosuvastatin calcium salt |
10/01/2008 | CN100422151C Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof |
09/30/2008 | US7429670 antagonists of the GlyR (glycine receptor); diterpene trilactones; cage-like skeleton; neuroprotectant, antioxidant, antiproliferation agent, cognition activator; parallel solution phase synthesis |
09/30/2008 | US7429578 e.g. phenyl-3,4-dihydropyrrolo[4,3,2-de]isoquinolin-5-(1H)-one; anticarcinogenic agent; stroke, head trauma, and neurodegenerative disease; potentiating cytotoxicity of a DNA-damaging cytotoxic agent or ionizing radiation |
09/30/2008 | CA2417417C Method for recovery of copper from sulfidic ore materials using super-fine grinding and medium temperature pressure leaching |
09/30/2008 | CA2355470C Benzoheterocycles and their use as mek inhibitors |
09/25/2008 | US20080234481 Forming salts such as tartrate or mandelate ; chemical intermediate |
09/23/2008 | US7427681 Anticancer agents; antidiabetic agents; Alzheimer's disease |
09/23/2008 | US7427613 7-aryl-3,9-diazabicyclo(3.3.1)non-6-ene derivatives and their use as renin inhibitors in the treatment of hypertension, cardiovascular or renal diseases |
09/23/2008 | CA2432872C Pyrazole compounds useful as protein kinase inhibitors |
09/17/2008 | EP1970374A1 Process for the production of substituted 2-(pyridin-2-ylmethylsulfinyl)-1H-benzimidazoles |
09/17/2008 | EP1968971A1 Dioxolane derivates for the treatment of cancer |
09/17/2008 | EP1409477B1 Piperidine derivatives as nmda receptor antagonists |
09/17/2008 | CN101265262A New oxabispidine compounds useful in the treatment of cardiac arrhythmias |
09/17/2008 | CN101265199A Method for the preparation of escitalopram |
09/17/2008 | CN100418967C Tricyclic inhibitors of poly(ADP-ribose) polymerases |
09/16/2008 | US7425560 Thioxanthine derivatives as myeloperoxidase inhibitors |
09/16/2008 | CA2427221C Process and intermediates for preparing anti-cancer compounds |
09/12/2008 | WO2004078116A9 P38 inhibitors and methods of use thereof |
09/11/2008 | US20080221323 Production of Rosuvastatin Calcium Salt |
09/11/2008 | US20080221178 Benzimidazole Derivatives,Compositions Containing Them, Preparation Thereof and Uses Thereof |
09/11/2008 | US20080221065 Pharmaceutical formulations; epothilone and mannitol or a cyclodextrin parenteral administration in the form of an infusion concentrate or lyophilised composition |
09/11/2008 | US20080220536 Tethering target having reactive thiol contacted with extender forming complex; conjugation; drug screening |
09/11/2008 | US20080220002 Modified transferin-antibody fusion proteins |
09/11/2008 | US20080216606 Grinding to uniform particle size; heating; pressurization;; extraction from ores, concentrates |
09/10/2008 | CN101260072A Novel crystal forms of atorvastatin hemi-calcium and processes for their preparation |
09/09/2008 | US7423049 e.g., 2-(5-fluoro-2-tolyl)-4-(4-aminocarbonylpiperazinylmethyl)-6-[a-aminocarbonyl-2,6-dichlorobenzyl]pyridine; mitogen-activated protein kinase inhibitor; antiinflammatory agent, autoimmune diseases |
09/09/2008 | US7423041 e.g. 3-[2-(4-Aminophenyl)ethyl]-8-benzyl-1-propylxanthine; A1-adenosine receptor antagonist; antiallergen, antiinflammatory agent; AIDS and immune deficiency disorders, asthma; good water solubility |
09/09/2008 | CA2287881C Vitamin d3 analogs with bis c-20 side chains |
09/04/2008 | US20080214824 Process for the Preparation of N-(4-Piperidinyl)-N-Ethyl-Phenylacetamides from N-Boc-4-Oxopiperidine |
09/04/2008 | US20080214812 Trisubstituted triazolopyrimidines for use in platelet aggregation inhibition |
09/04/2008 | US20080214538 Pyridoindolone Derivatives Substituted in the 3-Position by a Phenyl, Their Preparation and Their Application in Therapeutics |
09/03/2008 | EP1603909A4 Linear chain substituted monocyclic and bicyclic derivatives as factor xa inhibitors |
09/03/2008 | CN100415737C Indole derivatives useful for treatment of CNS disorders |
09/03/2008 | CN100415735C Amino alcohol derivatives |
09/03/2008 | CN100415717C Diarylmethylidene piperidine derivatives and their use as delta opioid receptor agonists |
09/02/2008 | US7420079 Intermediates for making 1(alpha-amino-1-(cyclopropyl-fused pyrrolidinylcarbonyl)methyl)-3-hydroxyadamantanes, e.g., methyl 3-hydroxy-<a-oxotricyclo[3.3.1.13,7]decane-1-acetate |
09/02/2008 | US7420061 Process for preparing prodrugs of benzenesulfonamide-containing COX-2 inhibitors |
09/02/2008 | US7419990 e.g. benzyl {1-[2-(1-{[1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl]carbonyl}piperidin-4-yl)-4,5-dimethylphenyl]propyl}carbamate; antidiabetic agent, obesity, sexual disfunctions |
09/02/2008 | CA2426956C Pharmaceutical compositions comprising ascomycin derivatives |
09/02/2008 | CA2283126C Method for preparing 2-thienylethylamine derivatives |
09/02/2008 | CA2273023C Aminoguanidines and alkoxyguanidines as protease inhibitors |
08/28/2008 | US20080207899 N-benzyl-N-{2-[7-(4-cyanobenzyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]ethyl}methane-sulfonamide; trial and ventricular arrhythmias; pharmacokinetics; electrophysiological activity; lowering daily clinical dose, lengthening duration of action; side effect reduction |
08/28/2008 | US20080207612 Analgesics; pain management |
08/28/2008 | US20080206805 Compounds and Related Methods for Mutant p53 Reactivation |
08/27/2008 | EP1622569A4 Aza spiro alkane derivatives as inhibitors of metallproteases |
08/27/2008 | CN100413863C Novel 1,2,3-substituted indolizine derivatives, inhibitors of FGFs, method for making same and pharmaceutical compositions containing same |
08/27/2008 | CN100413860C Piperidine derivative as NMDA receptor antagonist |
08/27/2008 | CN100413849C Benzimidazole derivatives |
08/26/2008 | CA2432129C Pyrazole compounds useful as protein kinase inhibitors |
08/21/2008 | US20080200460 Chemical Compounds |
08/20/2008 | EP1670790B1 Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof |
08/20/2008 | EP1670770B1 Benzimidazole derivatives, compositions containing them, preparation therof and uses thereof |
08/20/2008 | EP1249233B1 Npyy5 antagonists |
08/20/2008 | EP0883404B1 Combination therapy for osteoporosis |
08/20/2008 | CN101245058A Inhibitors of aspartyl protease |
08/20/2008 | CN101245043A Aza-heterocyclic compounds used to treat neurological disorders and hair loss |
08/19/2008 | US7414056 Cytokine inflammatory response suppressors; mitogen activated protein 38 kinases |
08/19/2008 | US7414045 Substituted pyrimido[1,2-a]azepines useful as HIV integrase inhibitors |
08/19/2008 | CA2432799C Pyrazole compounds useful as protein kinase inhibitors |
08/13/2008 | EP1956004A1 Quinoline derivatives and their use as 5-HT6 ligands |
08/13/2008 | EP1678196B1 Sulfonylamino-peptidomimetics active on the somatostatin receptor subtypes 4 (sstr4) and 1 (sstr1) |
08/13/2008 | EP1497290B1 Process for preparing acid salts of gemifloxacin |
08/13/2008 | CN101239973A Substituted aminoquinazolinone (thione) derivative or salts thereof, intermediate compound therefor, pest-controlling agent and using method thereof |
08/13/2008 | CN101239090A Pharmaceutical compositions having appetite suppressant activity |
08/13/2008 | CN101239089A Pharmaceutical compositions having appetite suppressant activity |
08/13/2008 | CN100410245C Arylmethyl-carbonylamino-thiazole derivatives and their use as antitumor agents |
08/12/2008 | US7411070 Form of S-omeprazole |
08/12/2008 | US7410969 Antitumoral analogs of ET-743 |
08/07/2008 | US20080188518 5-Substituted Imidazoles |
08/07/2008 | US20080188371 use as pesticides and/or herbicides and/or microbicides; for the selective control of weeds; synergistic; low application rates and concentrations; in particular in cereals (especially wheat) |
08/06/2008 | EP1953142A1 Process for the preparation of antihistaminic 4-diphenylmethyl piperidine derivatives |
08/06/2008 | CN100408573C Pyrazole compounds useful as protein kinase inhibitors |
08/06/2008 | CN100408564C Pyrazole derivatives for treating HIV |
08/06/2008 | CN100408026C Ceramic based nanoparticles for entrapping therapeutic agents for photodynamic therapy and method of using same |
08/05/2008 | US7408065 P2X7 receptor antagonists and their use |
08/05/2008 | US7407981 e.g., N-butyl-6-chloro-5-phenyl-1H-indazol-3-amine; kinase inhibitor; obesity and stroke; diseases involving phosphorylation of the tau protein such as Alzheimer's disease, Parkinson's disease, frontoparietal dementia |
08/05/2008 | US7407974 e.g. 4-Methoxy-pyrrolidine-1,2-dicarboxylic acid 1-[(4-chloro-phenyl)-amide] 2-{[2-fluoro-4-(2-oxo-2H-pyridin-1-yl)-phenyl]-amide}; anticoagulant, thrombolytic agent; thrombus formation within blood vessels; cardiovascular disease |
08/05/2008 | US7407972 e.g. 4,5-Dihydro-pyrazole-1,5-dicarboxylic acid 1-[(4-chloro-phenyl)-amide] 5-[(3-fluoro-2'-methanesulfonyl-biphenyl-4-yl)-amide]; anticoagulant, thrombolytic agent; thrombus formation within blood vessels; cardiovascular disease |
08/05/2008 | US7407956 Benzamide inhibitors of the P2X7 receptor |
07/31/2008 | US20080183007 Radical initiated coupling reaction between an alkylhalide and a hypophosphorous acid derivative; Bis-(trimethylsilyl)hypophosphite formed with trimethyl silyl chloride/diisopropyl ethylamine |
07/31/2008 | US20080182874 e.g. 1-[6-Chloro-5-[(tricyclo[3.3.1.13,7]dec-1-ylacetyl)amino]-2-quinolinyl]-4piperidinecarboxylic acid; adamantyl-containing purinergic receptor P2X7 antagonists; antiinflammatory agent, immune or cardiovascular diseases; asthma, chronic obstructive pulmonary disease, rheumatoid arthritis |
07/31/2008 | US20080182303 Enzymatic hydrolysis of lovastatin to form the triol acid; lactonization; regioselective acylation to form a 4-acetyl-protecting lactone; enzymatic acylation of the 8'-hydroxyl to form 4-acetyl simvastatin;selectively deprotecting to yield simvastatin; efficiency; nucleic acid-encoded hydrolases; kits |
07/30/2008 | CN101230057A Method for the synthesis of a benzimidazole compound |
07/30/2008 | CN100406459C 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino[4,5-b]indole-1-acetamide derivatives, preparation and use thereof in medicaments |
07/30/2008 | CN100406454C Pyrazole compounds useful as protein kinase inhibitors. |
07/30/2008 | CN100406437C Amino alcohol derivatives or phosphonic acid derivatives and pharmaceutical compositions containing these |
07/29/2008 | US7405306 3-(2-alkoxycarbonyl-3-indolyl)-3-oxo-propionic acid ester or propionamide intermediates: methyl 3-[6-fluoro-2-(methoxycarbonyl)-1-methyl-1H-indol-3-yl]-3-oxopropanoate; peripheral neuropathy, Parkinson's disease, Alzheimer's disease |
07/29/2008 | CA2432222C Pyrazole compounds useful as protein kinase inhibitors |
07/29/2008 | CA2432132C Pyrazole compounds useful as protein kinase inhibitors |
07/29/2008 | CA2333656C A novel vla-4 inhibitor: omepupa-v |