Patents for C07D - Heterocyclic compounds (10,420) |
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12/25/2008 | US20080319198 N-benzyl-N-{2-[7-(4-cyanobenzyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]ethyl}methane-sulfonamide; trial and ventricular arrhythmias; pharmacokinetics; electrophysiological activity; lowering daily clinical dose, lengthening duration of action; side effect reduction |
12/25/2008 | US20080319017 Non-Anilinic Derivatives of Isothiazol-3(2H)-Thione 1,1-Dioxides As Liver X Receptor Modulators |
12/24/2008 | CN101328151A Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof |
12/24/2008 | CN101328150A 新的苯并咪唑衍生物 New benzimidazole derivatives |
12/24/2008 | CN100445276C Sulfonylamino-derivatives as novel inhibitors of histone deacetylase |
12/18/2008 | US20080312449 New Compounds |
12/18/2008 | US20080312434 Process for imidazo [4,5-c] pyridin-4-amines |
12/18/2008 | US20080312242 7-aryl-3, 9-diazabicyclo(3.3.1)non-6-ene derivatives and their use as renin inhibitors in the treatment of hypertension, cardiovascular or renal diseases |
12/18/2008 | US20080312219 Biologically active methylene blue derivatives |
12/18/2008 | DE60224400T2 Hepatitis c virus polymerase inhibitoren mit heterobicylischer struktur Hepatitis C virus polymerase inhibitors with heterobicylischer structure |
12/17/2008 | EP1753736B1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
12/17/2008 | EP1282609B1 Piperazinedione compounds |
12/17/2008 | EP1077943B1 Heterocyclic inhibitors of p38 |
12/17/2008 | CN101326217A Light protective additive based on organic/ inorganic hybrid polymer, method for its manufacture and use thereof |
12/17/2008 | CN101323622A 4-biphenylsubstituted pyrazolidin-3,5-dione derivatives |
12/17/2008 | CN100443469C 病毒聚合酶抑制剂 Viral polymerase inhibitors |
12/11/2008 | US20080306107 Compounds |
12/11/2008 | US20080306103 Methods and compositions for treatment of central and peripheral nervous system disorders and novel compounds useful therefor |
12/10/2008 | CN101318957A Substituted thiazolidinedione derivative, process for its preparation and its pharmaceutical use |
12/10/2008 | CN101318956A Substituted thiazolidinedione derivative, process for its preparation and its pharmaceutical use |
12/09/2008 | US7462614 7-(2-Bromophenyl)-5-methyl-N-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine; to treat neoplasms; polo like kinases inhibitors; antineoplastic/antiproliferative agents; cyclization of 1,2,4-triazine derivatives; coupling if imidazo[5,1-f][1,2,4]triazines with amine or halogen derivatives |
12/09/2008 | CA2352054C New amidino derivatives and their use as thrombin inhibitors |
12/09/2008 | CA2294059C New amidino derivatives and their use as thrombin inhibitors |
12/03/2008 | EP1997811A2 Indazole, benzoxazole and pyrazolopyridine derivatives as P38 kinase inhibitors |
12/03/2008 | EP1997810A2 Indazole, benzoxazole and pyrazolopyridine derivatives for medical use |
12/03/2008 | EP1997809A2 Indazole, benzoxazole and pyrazolopyridine derivatives for medical use |
12/03/2008 | CN100439360C Crystals including a malic acid salt of a 3-pyrrole substituted 2-indolinone, and compositions thereof |
12/03/2008 | CN100439333C Process for producing of enantiomerically-pure azetidein-2-carboxylic acid |
12/03/2008 | CN100439320C Intermediates for preparation of arthropodicidal oxadiazines |
12/02/2008 | US7459463 Crystalline forms of 2,3-dimethyl-8-(2,6-dimethylbenzylamino)-N-hydroxyethyl-imidazo[1,2-a] pyridine-6-carboxamide mesylate salt |
12/02/2008 | US7459460 Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators |
12/02/2008 | CA2469315C Pharmaceutical nanoparticulate composition of a tachykinin receptor antagonist |
12/02/2008 | CA2305548C Prostaglandin agonists and their use to treat bone disorders |
11/27/2008 | US20080293748 Thioxanthine Derivatives as Myeloperoxidase Inhibitors |
11/27/2008 | US20080293743 (5S)-5-({[6-(2-cyclopropylpyrimidin-5-yl)-3,4-dihydroisoquinolin-2(1H)-yl]sulfonyl}methyl)-5-methylimidazolidine-2,4-dione; asthma, chronic obstructive pulmonary disease |
11/27/2008 | US20080293705 A1 adenosine receptor antagonists |
11/27/2008 | US20080290034 Bridged macrocyclic module compositions |
11/26/2008 | CN100436452C Pyrazole compounds useful as protein kinase inhibitors |
11/25/2008 | US7456182 Phenylpiperazines |
11/25/2008 | CA2385728C Novel photochromic naphthopyrans |
11/25/2008 | CA2320182C Compositions containing organic compounds |
11/20/2008 | US20080287685 Detomidine Hydrochloride Crystallization Method |
11/20/2008 | US20080287674 Inhibitors of Factor XA and Other Serine Proteases Involved in the Coagulation Cascade |
11/20/2008 | US20080287444 Pyrazole compounds useful as protein kinase inhibitors |
11/18/2008 | US7452913 Patterns of enzyme inhibitors formed by dissolving compounds and isolation by precipitation |
11/18/2008 | US7452888 Quinoline and aza indole compounds having pharmacological activity, for example, 8-(4-Methyl-piperazin-1-yl)-3-phenylsulfonylquinoline; use in the treatment of CNS and other disorders |
11/18/2008 | US7452883 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
11/18/2008 | CA2516557C Triazole compounds useful in therapy |
11/18/2008 | CA2434682C Combinations of peroxisome proliferator-activated receptor (ppar) activator(s) and sterol absorption inhibitor(s) and treatments for vascular indications |
11/12/2008 | EP1990341A1 Triazolyl tropane derivatives as CCR5 modulators |
11/12/2008 | CN101302204A Quinazolone compound, composition and application including the same |
11/12/2008 | CN101302182A Virus polymerase inhibitors |
11/12/2008 | CN101302180A 8-azaprostaglandin derivative compound and agent comprising the compound as active ingredient |
11/11/2008 | US7450293 Electrochromic salts, solutions, and devices |
11/11/2008 | US7449478 Treatment of peroxisome proliferation activated receptor diseases such as diabetes, skin disorders or high blood pressure |
11/11/2008 | US7449475 e.g. 2-{[(2S)-3-(5-Chloro-1'H,3H-spiro[1-benzofuran-2,4'-piperidin]-1'-yl)-2-hydroxypropyl]oxy}-N-cyclopropylbenzamide; macrophage inflammatory protein (MIP)-1 alpha chemokine receptor modulator; antiinflammatory, antiproliferative agent, autoimmune diseases |
11/06/2008 | US20080275252 Atipamezole Hydrochloride Crystallization Method |
11/06/2008 | US20080275092 Aryl-substituted pyrazole-amide compounds useful as kinase inhibitors |
11/06/2008 | US20080275059 Novel physiologically active substances |
11/06/2008 | US20080275041 3-[5-({4-[2-(Dipropylamino)ethyl]piperazin-1-yl}sulfonyl)pyridin-2-yl]-2-hydroxy-1H-indole-6-carbonitrile hydrochloride; Alzheimer's Disease, Parkinson's Disease, depression, schizophrenia, HIV, Down syndrome, bone disorders, alopecia |
11/06/2008 | US20080275033 Administering Diamino-substituted phenothiazinium compound; antimicrobial photosensitisers effective against Gram negative bacteria, Gram positive bacteria; photodynamic therapy |
11/05/2008 | EP1200424B1 C7 heterosubstituted acetate taxanes as antitumor agents |
11/05/2008 | CN101298433A 2-, 3-, 4-, or 5-substituted-n1-(benzensulfonyl)indoles and their use in therapy |
11/05/2008 | CN100430396C 2-phenyl-substituted imidazo-triazone used as phosphodiesterase inhibitor |
11/05/2008 | CN100430379C Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof |
11/04/2008 | CA2443449C Pyrazole derivatives for treating hiv |
10/30/2008 | US20080269216 Gastrointestinal disorders; irritable bowel syndrome |
10/30/2008 | US20080269197 antipsychotic agents; phenylsulfonyl compounds; 7-Methoxy-8-(3-phenoxy-benzenesulfonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine; schizophrenia |
10/30/2008 | US20080269176 New Salts |
10/30/2008 | US20080268033 Biologically active methylene blue derivatives |
10/30/2008 | US20080267867 Imidazole, pyridine derivative silver complexes; nanofiber with radioactive transition metal, lanthanide, actinide; radiopharmaceutical peptide, polyamine, imaging and tumor treatment |
10/29/2008 | CN101293869A Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p561lck tyrosine kinases |
10/29/2008 | CN101293867A Phenylalanine enamide derivatives possessing a cyclobutene group, for use as integrin inhibitors |
10/29/2008 | CN100429208C Process for prepn. of racemic citalopram and/or S-or R-citalopram by separation of mixture of R-and S-citalopram |
10/29/2008 | CN100429201C Heterocyclic compounds and methods of use thereof |
10/28/2008 | US7442708 Inhibitors of basic fibroblast growth factors (FGFs); treating cancer, rheumatoid arthritis, inflammatory bowel disease, cardiovascular disorders, diabetic retinopathy, achondroplasia, hypochondoplasia, or thanathophoric dysplasia |
10/28/2008 | US7442705 HIV replication inhibiting pyrimidines and triazines |
10/28/2008 | US7442702 Prostaglandin agonists |
10/28/2008 | CA2342102C Tan-1057 derivatives |
10/28/2008 | CA2262791C Amino acid ester containing azole antifungals |
10/23/2008 | US20080262037 Piperidine Derivatives for the Treatment of Chemokine Mediated Disease |
10/23/2008 | US20080261997 Use of aminoindazole derivatives for the inhibition of tau phosphorylation |
10/23/2008 | US20080261960 Photosensitizers for photodynamic therapy; killing tissue, cells; anticancer agents |
10/22/2008 | EP1603562A4 Sulfonyl-amidino containing and tetrahydropyrimidino containing compounds as factor xa inhibitors |
10/21/2008 | US7439251 Methods and compositions for treatment of central and peripheral nervous system disorders and novel compounds useful therefor |
10/21/2008 | CA2296732C Polyhydroxyalkylpyrazine derivatives, their preparation and medicines containing them |
10/16/2008 | US20080255363 Novel Form of S-Omeprazole |
10/16/2008 | US20080255207 5-Thioxo-1,5-Dihydro-2H-Pyrrol-2-One Derivatives As Liver X Receptor Modulators |
10/16/2008 | US20080255199 Using 2-(((4-x-3,5-dimethyl(or1-oxo)pyridin-2-yl)methylthio)5-methoxy-1H-benzimidazole where x is a leaving group; oxidation; using titanium complex catalyst and a base |
10/16/2008 | US20080255146 Macrolide compounds comprising 18,19-epoxytricosa-8,12,14-trien-11-olide derivatives; angiogenesis inhibitors; anticarcinogenic, antimetastasis, antiinflammatory, and antitumor agents; antihypoxic agents; endothelial growth factor suppressors; retinal neovascularization, diabetic retinopathy |
10/16/2008 | US20080255129 3-Heteroaryl-3,5-dihydro-4-oxo-4H-pyridazino[4,5-b]indole-1-acetamide derivatives, their preparation and their application in therapeutics |
10/15/2008 | CN101284819A Fused pyridazine derivative compounds and drugs containing these compounds as the active ingredient |
10/15/2008 | CN100425609C N-heteroarylnicotinamide derivatives |
10/14/2008 | US7436570 Electrochromic salts, solutions, and devices |
10/14/2008 | US7435832 Preparing an anhydrous crystal of a malic acid salt of N-[2-(diethylamino)ethyl]-5-[(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide by reacting the acid and amine in a solvent and crystallizing under various process conditions |
10/14/2008 | US7435744 Brain disorders; central nervous system disorders; viricides |
10/09/2008 | US20080249319 Process for the preparation of 5-Carboxyphthalide |
10/09/2008 | US20080249110 Novel Substituted 3-Sulfur Indoles |
10/09/2008 | US20080249086 N-benzyl-N-{2-[7-(4-cyanobenzyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]ethyl}methane-sulfonamide; trial and ventricular arrhythmias; pharmacokinetics; electrophysiological activity; lowering daily clinical dose, lengthening duration of action; side effect reduction; arrhythmia |
10/08/2008 | EP1977749A1 Use of cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia |