Patents
Patents for C07D 475 - Heterocyclic compounds containing pteridine ring systems (2,718)
03/2015
03/05/2015WO2015028927A1 Compositions and methods for the treatment of metabolic diseases
03/05/2015US20150065708 Compound jk12a and preparation thereof
02/2015
02/19/2015WO2015022407A1 Hemisulfate salt of 5,10-methylene-(6r)-tetrahydrofolic acid
02/18/2015EP2837631A1 New stable salt of 5,10-methylene-(6R)-tetrahydrofolic acid
02/18/2015EP2837630A1 Method for synthesizing sapropterin dihydrochloride
02/18/2015EP2837629A1 Method for synthesizing sapropterin dihydrochloride
02/04/2015CN104327082A 一种从结晶母液中高效环保回收核黄素的方法 An efficient method for the mother liquor from the crystallization of riboflavin recycling
02/03/2015US8946450 Composition, synthesis, and use of new substituted pyran and pterin compounds
01/2015
01/29/2015US20150030669 Targeting aminoacid lipids
01/29/2015DE112013002484T5 Pteridinketon-Derivat und Anwendungen desselben als EGFR-, BLK- und FLT3-Inhibitor Pteridinketon derivative and applications thereof as EGFR, PFC and FLT3 inhibitor
01/22/2015US20150025039 Antiviral phosphonate analogs
01/21/2015EP2825156A1 Targeting aminoacid lipids
01/21/2015CN103274943B 4-[1-(2-丙炔基)-3,4-二氧代正丁基]苯甲酸酯及其制备方法 4- [1- (2-propynyl) -3,4-dioxo-n-butyl] benzoate and its preparation method
01/20/2015CA2670371C 18f-labelled folates
01/15/2015US20150018357 Crystal form of (6s)-5-methyltetrahydrofolate salt and method for preparing same
01/15/2015US20150017189 Methods of making and using nanostructures
01/14/2015CN104277044A 一种高效制备低钙含量亚叶酸的方法 A low calcium content and efficient method for the preparation of leucovorin
01/13/2015US8933228 Respiratory formulations and compounds for use therein
01/13/2015US8932638 Polyamine derivatives
12/2014
12/11/2014US20140364437 Optically Pure Diastereomers of 10-Propargyl-10-Deazaaminopterin and Methods of Using Same
12/02/2014US8900621 Polyamine derivatives
11/2014
11/25/2014US8895568 Compositions comprising substituted pteridines as agrochemicals
11/04/2014US8877756 Substituted pteridines
10/2014
10/28/2014US8871785 Antiviral phosphonate analogs
10/23/2014US20140316132 Modulators of toll-like receptors
10/23/2014US20140315911 Dihydropteridinones
10/21/2014US8865716 Dihydropteridinones II
09/2014
09/23/2014CA2675246C Compositions and methods of reducing side effects and toxicity of methotrexate when given as orotate derivatives
09/18/2014WO2014144737A1 Heteroaryl compounds and uses thereof
09/18/2014US20140275024 Dna-pk inhibitors
09/16/2014US8835451 Compounds
09/16/2014US8835433 Optically pure diastereomers of 10-Propargyl-10-deazaaminopterin and methods of using same for the treatment of cancer
09/10/2014EP2773355A1 Methods, formulations, and kits for rapidly repleting folate levels in women
09/09/2014CA2652840C 2-piperazino-6-chloro-pteridines as pde4-inhibitors for the treatment of inflammatory diseases
08/2014
08/28/2014WO2014127816A1 Dihydropteridinones ii
08/28/2014WO2014127815A1 Dihydropteridinones i
08/26/2014US8815860 Methods for preventing oxidative stress injury of a tissue by a Folate-TEMPOL conjugate
08/20/2014EP2766364A1 Folate conjugates of albumin-binding entities
08/19/2014US8809553 Process for the preparation of pteridine derivatives
08/19/2014US8809527 Modulators of toll-like receptors
08/13/2014CN103980277A 一种叶酸巯基化衍生物的制备方法 A method for preparing folic acid thiolated derivatives
08/12/2014US8802697 Inhibitors of the fibroblast growth factor receptor
08/07/2014US20140221646 Novel immune system modulators
08/06/2014CN102516246B 一种从蚕体中提取纯化高纯度墨蝶呤的方法 An extraction and purification methods methotrexate ink from silkworm body
07/2014
07/31/2014US20140212459 10h-benzo[g]pteridine-2,4-dione derivatives, method for the production thereof, and use thereof
07/30/2014CN103951668A 叶酸衍生物的正电子核素标记物及其应用 Folic acid derivative positron marker and its Application
07/17/2014US20140200329 Bisaminoethanethiol-targeting ligand conjugates and compositions
07/08/2014CA2523083C Antiviral phosphonate analogs
07/03/2014WO2014102511A1 Folate derivatives, useful in particular in the context of the folate assay
07/03/2014WO2014101134A1 Folic acid derivative, and preparing method and application thereof
07/03/2014WO2013135359A8 Targeting aminoacid lipids
07/02/2014CN203678382U 一种生产核黄素的乳化磨料罐 A method for producing riboflavin emulsifying abrasive tank
07/02/2014CN103896945A 一种简便的叶酸环保生产方法 A simple and environmentally friendly production methods folate
07/02/2014CN103333169B 一种巯基化叶酸及其制备方法 An SH group of folic acid and its preparation method
06/2014
06/25/2014CN102633799B 一种从消旋体中间体拆分路线合成二盐酸沙丙蝶呤的方法 A synthetic sapropterin dihydrochloride from racemic intermediate split line method
06/19/2014WO2013018103A3 Extraction of b-vitamins from plant matter
06/17/2014US8754212 Process for the preparation of stable, amorphous calcium salt of (6S)-N(5)-methyl-5,6,7,8-tetrahydrofolic acid
05/2014
05/29/2014US20140148433 Bicyclic aza heterocycles, and use thereof
05/15/2014US20140135315 Pyrido-, Pyrazo- and Pyrimido-Pyrimidine Derivatives as mTOR Inhibitors
05/15/2014US20140134157 Antibodies to opgl
05/08/2014WO2014041446A3 Compositions and methods for treatment of metabolic diseases
05/08/2014US20140128403 Use of 10h-benzo[g]pteridine-2,4-dione derivatives
05/07/2014CN102093361B 稠合的哌嗪-2-酮衍生物的制备方法 The method for preparing a fused piperazin-2-one derivatives
05/01/2014WO2014066772A1 Processes and reagents for making diaryliodonium salts
05/01/2014US20140121371 Processes and reagents for making diaryliodonium salts
05/01/2014US20140121361 Novel n3s1 chelator-folate derivatives, preparation method thereof and composition for diagnosis or treatment of cancer containing the same as an active ingredient
04/2014
04/30/2014EP2723743A1 10h-benzo[g]pteridine-2,4-dione derivatives, method for the production thereof, and use thereof
04/30/2014EP2723742A1 10h-benzo[g]pteridine-2,4-dione derivatives, method for the production thereof, and use thereof
04/30/2014CN103755706A Environment-friendly preparation method of synthetic folic acid
04/23/2014CN103739604A Preparation method of Pralatrexate suitable for industrial large scale production
04/16/2014CN103732595A Folate conjugates of albumin-binding entities
04/16/2014CN102627644B Method for preparing sapropterin dihydrochloride through direct chiral synthesis method
04/08/2014US8691822 Dihydropteridinone derivatives, preparation process and pharmaceutical use thereof
04/02/2014CN103694239A Crystal form A of 5-methyl-(6S)-tetrahydrofolic acid and preparation method thereof
03/2014
03/27/2014US20140088100 Inhibitors of the fibroblast growth factor receptor
03/26/2014CN103664945A Preparation method of L-5-methyl tetrahydrofolate amino acid salt
03/26/2014CN102399223B Preparation method of medicinal calcium folinate
03/25/2014CA2577982C Dihydropteridinone derivatives, methods for the production thereof and their use as medicaments
03/20/2014WO2014016740A3 Improved process for the preparation of pralatrexate
03/20/2014US20140081022 Modulators of toll-like receptors
03/20/2014US20140079724 Novel immune system modulators
03/19/2014CN103113372B High-yield preparation method of calcium levofolinate
03/04/2014US8664222 Specific salt, anhydrous and crystalline form of a dihydropteridione derivative
02/2014
02/27/2014WO2014011900A3 Inhibitors of the fibroblast growth factor receptor
02/20/2014US20140050775 Polyamine Derivatives
02/19/2014CN103588775A Pralatrexate degradation impurity and preparation method thereof
02/06/2014WO2014020553A1 Salts of pralatrexate
01/2014
01/30/2014WO2014016740A2 Improved process for the preparation of pralatrexate
01/30/2014US20140031546 Hydrodeoxygenation catalyst
01/22/2014CN103524506A Preparation method and application of radioiodine labeled biomolecules
01/21/2014US8633210 Triazole compounds useful as protein kinase inhibitors
01/21/2014US8633202 Crystalline levofolinic acid and process for its preparation
01/14/2014US8629142 Modulators of toll-like receptors
01/09/2014WO2014005194A1 Immunological reagents and uses therefor
01/08/2014CN103497192A Modulators of TOLL-like receptors
12/2013
12/31/2013US8618106 Protein kinase inhibitors
12/25/2013CN103467447A Novel organic electroluminescent (EL) material and application thereof in devices
12/18/2013CN103450202A Method for reacting L-5-methyltetrahydrofolic acid with organic base to form salt
12/12/2013US20130331376 Inhibitors of polo-like kinase
12/11/2013CN101360746B Pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors
1 2 3 4 5 6 7 8 9 10 11 ... 28