Patents for C07D - Heterocyclic compounds (10,420) |
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08/08/2001 | EP1121345A1 Esters of (+)-alpha-( 2,3- dimethoxyphenyl) -1- 2-(4- fluorophenyl) ethyl]-4- piperidinemethanol and their use as prodrugs of the 5ht2a receptor antagonist mdl 110,907 |
08/08/2001 | CN1307561A Novel VLA-4 inhibitor: oMePUPA-V |
08/08/2001 | CN1069321C New inhibitors of platelet aggregation |
08/07/2001 | US6271376 Process for the preparation of N-(amino-4,6-dihalo-pyrimidine) formamides |
08/07/2001 | US6271253 Cyclooxygenase inhibitors |
08/07/2001 | CA2104782C 1-substituted, 2-substituted 1h-imidazo-[4,5-c]quinolin-4- amines |
08/02/2001 | WO2001055130A2 Novel 1,3-dihydro-2h-indol-2-one derivatives and their use as ligands for v1b and v1a arginine-vasopressin receptors |
08/02/2001 | WO2001055122A1 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
08/02/2001 | WO2001055082A2 Intermediates for biologically active compounds |
08/02/2001 | WO2001054481A2 Enhanced propertied pharmaceuticals |
08/02/2001 | WO2001014330A3 Phenylpiperazines as serotonin reuptake inhibitors |
08/02/2001 | US20010011136 Anticancer agents |
08/02/2001 | US20010011135 Anticancer agents |
08/02/2001 | US20010011091 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists |
08/02/2001 | CA2397831A1 Enhanced propertied pharmaceuticals |
08/01/2001 | CN1306520A Non-yellowing para-tertiary-alkyl phenyl substituted triazine and pyrimidine ultraviolet light absorbers |
08/01/2001 | CN1306512A Heterocyclic inhibitors of P38 |
08/01/2001 | CN1306511A Novel heterocyclic compounds |
07/31/2001 | US6268506 Process for the preparation of a triazolinone herbicide |
07/31/2001 | US6268369 5-(heterocyclic alkyl)-6-aryl-dihydropyrimidines |
07/31/2001 | CA2282890C Therapeutic heterocyclic compounds |
07/26/2001 | WO2001053284A1 Process for the preparation of 5-carboxyphthalide and its use for the production of citalopram |
07/26/2001 | US20010009962 One pot process for preparing sildenafil (drug for erectile dysfunction) and derivatives by reacting for example 4-(2-methoxy-5-(4-methyl-1-piperazinylsulfonyl)benzamido)-1-methyl-3-propyl -1H-pyrazole-5-carboxamide with ethanol |
07/26/2001 | US20010009921 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists |
07/26/2001 | US20010009920 Combination therapy for osteoporosis |
07/25/2001 | EP1118614A2 Process for the preparation of 5-carboxyphthalide |
07/25/2001 | EP1117652A1 Tan-1057 derivatives |
07/25/2001 | EP1117648A1 Tetrahydroquinoline derivatives having selective activity for retinoid x receptors |
07/25/2001 | CN1305483A Polymorphic clopidogrel hydrogenesulphate form |
07/25/2001 | CN1305478A Pyrazolopyrimidinone cGMP PDE 5 inhibitors for treatment of sexual dysfunction |
07/25/2001 | CN1305477A Azablicyclic 5-HT, receptor ligands |
07/25/2001 | CN1305378A Therapeutic combinations of (selective) estrogen receptor modulators (SERM) and growth hormone secretagogues (GHS) for treating musculoskeletal fragility |
07/25/2001 | CN1305373A Therapeutic combinations comprising selective estrofen receptor modulator and parathyroid hormone |
07/25/2001 | CN1304930A Arylsulfurylisooximino acid derivative |
07/25/2001 | CN1068880C N-substituted piperidingl bicyclic benzoate derivatives |
07/24/2001 | US6265397 Amidino derivatives and their use as thrombin inhibitors |
07/24/2001 | CA2218503C Arylsulfonyl hydroxamic acid derivatives |
07/24/2001 | CA2111974C Carbapenem derivatives |
07/19/2001 | WO2001051051A2 AGENTS, SUCH AS NICOTINAMIDE OR cADPR FOR THE TREATMENT OF SKIN DISORDERS |
07/19/2001 | US20010008890 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists |
07/18/2001 | EP1115708A1 Aminoalkyl-3,4-dihydroquinoline derivates as no-synthase inhibitors |
07/18/2001 | EP1115704A1 Novel substituted indolinones with an inhibitory effect on various kinases and cyclin/cdk complexes |
07/18/2001 | CN1304307A 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective NMDA receptor antagonists |
07/17/2001 | US6262067 Polymorphs of a crystalline azo-bicyclo 2,2,2 OCT-3-yl amine dihydrochloride and their pharmaceutical compositions |
07/17/2001 | US6262052 Amino acid ester containing azole antifungals |
07/17/2001 | US6262028 CONTAINING OXY-SUBSTITUTED AMIDINOBENZYL DERIVATIVES OF DIPEPTIDES FROM CYCLOHEXYLGLYCINE AND AZETIDINE-2-CARBOXYLIC ACID; ximelagatran |
07/17/2001 | CA2223023C N-hydroxyureas as antiinflammatory agents |
07/12/2001 | WO2001049684A1 Novel tetrahydropyridines, preparation method and pharmaceutical compositions containing same |
07/11/2001 | EP1114817A1 Substituted benzylamino piperidine compounds |
07/11/2001 | EP1114032A1 4-amino substituted-2-substituted-1,2,3,4-tetrahydroquinolines as cetp inhibitors |
07/11/2001 | EP1114031A1 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinolines as cetp inhibitors |
07/11/2001 | CN1303384A Pyrrolo [1,2-a] pyrazine sPLA2 inhibitor |
07/11/2001 | CN1303379A 2-Aminopyridines containing fused ring substituents as nitric oxide synthase inhibitors |
07/11/2001 | CN1303378A 3-(Amino-or aminoalkyl) pyridinone derivatives and their use for treatment of HIV related diseases |
07/11/2001 | CN1303364A Aminocyclohexyl ether compounds and uses thereof |
07/11/2001 | CN1302800A Method for preparing 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinoline |
07/11/2001 | CN1068313C 2[(dihydro)pyrazolyl-3'-oxymethyene]-anilides, prepn. method and use thereof |
07/10/2001 | US6258824 Treatment of hyperproliferative diseases, such as cancers, in mammals. this invention also relates to a pharmaceutical compositions containing such compounds. |
07/10/2001 | US6258809 6-aryloxy and arylthiopurines |
07/10/2001 | US6258804 Triazepinones, process for their preparation and their therapeutic application |
07/10/2001 | CA2139653C Optically pure salts of pyridinylmethyl sulfinyl-ih- benzimidazole compounds |
07/05/2001 | WO2001047926A1 Compounds and methods for the treatment of pain |
07/05/2001 | WO2001047893A1 New azabicyclooctane derivatives useful in the treatment of cardiac arrhythmias |
07/05/2001 | US20010006976 Efficent, notoxic process of making new key intermediate quaternary ammonium salts and 2-oxazolylalkyl sulfide derivatives and avoids the reaction of a-haloketones with an azide followed by reducing the resulting a-aminoketone |
07/05/2001 | CA2394097A1 New azabicyclooctane derivatives useful in the treatment of cardiac arrhythmias |
07/04/2001 | EP1113013A1 Benzothiophene compounds, intermediates, compositions and methods |
07/04/2001 | EP1112272A1 Muscarinic agonists and antagonists |
07/04/2001 | EP1112255A1 4,4-biarylpiperidine derivatives with opioid receptor activity |
07/04/2001 | CN1302301A Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidine sas inhibitors of cellular proliferation |
07/04/2001 | CN1302184A Composition for keeping away vermin |
07/04/2001 | CN1067989C New compound with analgesic and local anaesthetic effect |
07/03/2001 | US6255307 Pyrazine compounds |
07/03/2001 | US6255305 Substituted triazolo-pyridazine derivatives as ligands for GABA receptors |
06/28/2001 | WO2001046263A1 Novel compounds |
06/28/2001 | WO2001046140A1 Ep4 receptor selective agonists in the treatment of osteoporosis |
06/28/2001 | CA2394864A1 Novel compounds |
06/27/2001 | EP1110954A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics |
06/27/2001 | EP1110953A1 Quinazoline derivatives |
06/27/2001 | EP1110949A1 EP4 receptor selective agonists in the treatment of osteoporosis |
06/27/2001 | EP1109787A1 Arylpiperazines and their use as metalloproteinase inhibiting agents (mmp) |
06/27/2001 | CN1301253A Carboxy substituted carboxamide derivatives as tachykinin receptor antagonists |
06/26/2001 | US6251916 For therapy of pain |
06/26/2001 | US6251904 Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction |
06/26/2001 | US6251894 1-(1,2-disubstituted piperidinyl)-4 (fused imidazole)-piperidine derivatives |
06/22/2001 | CA2329678A1 Ep4 receptor selective agonists in the treatment of osteoporosis |
06/21/2001 | WO2001044242A1 N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl]carboxamide inhibitors of cyclin dependent kinases |
06/21/2001 | CA2394552A1 N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl]carboxamideinhibitors of cyclin dependent kinases |
06/20/2001 | EP0920438B1 N6 heterocyclic substituted adenosine derivatives |
06/20/2001 | CN1300291A Modulators of protein tyrosine phosphatases |
06/20/2001 | CN1300284A Method for producing isoxazoline-3-yl-acyl benzene |
06/19/2001 | US6248897 From beta-methyl l-aspartate |
06/19/2001 | US6248747 5-(heterocyclic alkyl)-6-aryl-dihydropyrimidines |
06/19/2001 | US6248735 Ophthalmic compositions comprising combinations of a carbonic anhydrase inhibitor and a β-adrenergic antagonist |
06/19/2001 | CA2191129C Drugs containing metronidazole or a synergistic mixture of metronidazole and clindamycin |
06/19/2001 | CA2029838C Process for the preparation of aminotriazine derivatives |
06/14/2001 | US20010003752 Crystalline form of 4- [ 5-methyl-3-phenylisoxazol-4-yl ] benzenesulfonamide |
06/14/2001 | US20010003749 Arylpiperazines having activity at the serotonin 1A receptor |
06/14/2001 | US20010003646 Composition for keeping away vermin |
06/13/2001 | EP1106606A2 N-(3-piperidinylcarbonyl)-beta-alanine derivatives as paf antagonists |
06/13/2001 | CN1299367A 2''-deoxy hygromycin derivatives |