Patents for C07D - Heterocyclic compounds (10,420) |
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12/12/2002 | US20020188133 Producing an isoxazolidinedione compound from beta - methyl L-aspartate via an important intermediate oxazolylethanol derivative |
12/12/2002 | US20020187994 New compounds |
12/11/2002 | EP1263979A1 Method of purifying a fermentation broth |
12/11/2002 | CN1384829A Sodium-hydrogen exchanger type 1 inhibitor crystals |
12/10/2002 | US6492539 Preparation of preparing substituted indanones |
12/10/2002 | US6492402 Anticoagulants; peptide derivatives having high antithrombotic activity and oral bioavailability |
12/10/2002 | US6492390 Treating cyclooxygenase-2 mediated disorders. |
12/10/2002 | US6492374 Benzofuran derivatives, their preparation and use |
12/10/2002 | US6492372 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 |
12/10/2002 | US6492367 Sulfamato hydroxamic acid metalloprotease inhibitor |
12/05/2002 | WO2002096909A1 Optical resolution of (1-benzyl-4-methylpiperidin-3-yl) -methylamine and the use thereof for the preparation of pyrrolo 2,3-pyrimidine derivatives as protein kinases inhibitors |
12/05/2002 | WO2002096896A1 Biologically active methylene blue derivatives |
12/05/2002 | WO2002096879A1 Aminoquinoline and aminopyridine derivatives and their use as adenosine a3 ligands |
12/04/2002 | EP1097139B1 Quinoline derivatives |
12/03/2002 | US6489478 4-amino substituted-2-substituted-1,2,3,4-tetrahydroquinolines |
12/03/2002 | CA2266107C Aralkyl and aralkylidene heterocyclic lactams and imides |
11/28/2002 | US20020177596 2,3,4,4a,5,6-hexahydro-1H-pyrazino(1,2-a)quinoxaline derivatives; treating depression, schizophrenia; (5-hydroxytryptamine=5HT) 5HT2a antagonist or a 5HT2c agonist |
11/28/2002 | US20020176889 And an excipient wherein the pH is within the range of 5.5-7.0; stability; dosage forms |
11/27/2002 | EP1260511A1 Process for the preparation of 5-chloro-1-(4-fluorophenyl)-3-(1,2,3,6-tetrahydropyridin-4-yl)indole and method of manufacturing sertindole |
11/27/2002 | EP1260504A1 Process for the preparation of antihistaminic 4-diphenylmethyl piperidine derivatives |
11/27/2002 | EP1260222A1 Butenyl-substituted taxanes and composition |
11/27/2002 | EP1259240A2 Agents, such as nicotinamide or cadpr for the treatment of skin disorders |
11/27/2002 | EP1000035B1 Substituted 6-phenylphenanthridines |
11/26/2002 | US6486182 Mutual prodrugs of amlodipine and atorvastatin |
11/21/2002 | WO2002092600A1 Retinol derivatives potentiation of active substances by micellar preparation |
11/21/2002 | WO2002092597A1 The citrate salt of 5, 8, 14-triazatetracyclo(10.3.1.0?2,11.04.9¿)-hexadeca-2.(11),3,5,7,9-pentaene and pharmaceutical compositions thereof |
11/21/2002 | WO2002092089A1 Tartrate salts of 5,8,14-triazatetracyclo {10.3.1.0?2,11.04,9¿}-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof |
11/21/2002 | CA2446988A1 The citrate salt of 5, 8, 14-triazatetracyclo(10.3.1.02,11.04.9)-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof |
11/20/2002 | EP1257544A2 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage |
11/20/2002 | EP0920422B1 Crytalline form of 4-[5-methyl-3-phenylisoxazol-4-yl]benzenesulfonamide |
11/20/2002 | CN1380883A Novel derivatives and analogues of galanthamin |
11/20/2002 | CN1380882A C10 ester substituted taxanes as antitumor agents |
11/19/2002 | US6482834 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases |
11/14/2002 | US20020169186 Tetrahydroquinoline derivatives as glycine antagonists |
11/14/2002 | US20020169172 Phenyl or naphthyl-pyrazine compounds useful in the treatment of central nervous system diseases |
11/14/2002 | US20020169170 Arylpiperazines having activity at the serotonin 1A receptor |
11/14/2002 | US20020168427 Plant extract |
11/13/2002 | EP1255751A2 1,3-dihydro-2h-indol-2-one derivatives and their use as ligands for v1b or v1b and v1a arginine-vasopressin receptors |
11/13/2002 | EP1112272B1 Muscarinic agonists and antagonists |
11/13/2002 | EP0843672B1 One pot synthesis of 2-oxazolidinone derivatives |
11/13/2002 | CN1379775A Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
11/13/2002 | CN1379763A Pyrazoloanthrone and derivatives thereof as JNK inhibitors and their compositions |
11/12/2002 | US6479680 Method for reacting an organic compound with a hydroperoxide |
11/12/2002 | US6479663 Intermediates useful for the preparation of antihistaminic piperidine derivatives |
11/12/2002 | US6479492 Compounds which inhibit leukocyte adhesion mediated by VLA-4 |
11/12/2002 | US6479483 3,4,6-substituted pyridine derivatives useful for treating depression and pain, resulting from inflammatory conditions, such as migraine, rheumatoid arthritis, asthma and inflamatory bowel disease; nk1 receptor antagonist |
11/07/2002 | WO2002088094A1 2-iminoimidazole derivatives (1) |
11/07/2002 | WO2002088092A1 2-iminoimidazole derivative (2) |
11/06/2002 | EP1000038B1 Novel pyrimidin derivatives |
11/06/2002 | CN1378547A 5-(2-substituted-5-heterocyclylsulphenylpyrid-3-yl)-dihydropyrazolo [4,3-d] pyrimidin 7-ones as phosphodiesterase inhibitors |
11/06/2002 | CN1093859C Novel indole-2,3-dione-3-oxime derivatives |
11/05/2002 | US6476042 Combination therapy for the treatment of migraine |
11/05/2002 | US6476040 Processes and intermediates for preparing anti-cancer compounds |
10/31/2002 | WO2002085860A1 Pyrazole derivatives for treating hiv |
10/31/2002 | WO2002085855A1 2-iminopyrrolidine derivatives |
10/31/2002 | WO2002085850A1 Cyclic amidine derivative |
10/31/2002 | US20020161000 Treating diseases resulting from tissue breakdown such as heart disease, multiple sclerosis, osteo- and rheumatoid arthritis, atherosclerosis, and osteoporosis |
10/30/2002 | EP1252889A1 Remedies or preventives for pulmonary insufficiency containing diaminotrifluoromethylpyridine derivatives |
10/30/2002 | EP1252145A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis |
10/30/2002 | EP1051425B1 2-(PURIN-9-yl)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES |
10/29/2002 | US6472529 Viricides |
10/29/2002 | US6472388 Psychotherapeutic agents. |
10/29/2002 | CA2342471C Heterocyclecarbonylmethyl amine intermediates |
10/29/2002 | CA2014486C Antitumor and antibacterial substituted disulfide derivatives prepared from compounds possessing a methyltrithio group |
10/24/2002 | WO2002050065A3 Pyrazole compounds useful as protein kinase inhibitors |
10/24/2002 | WO2002030931A3 Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors |
10/24/2002 | US20020156284 Crystalline form of omeprazole |
10/23/2002 | EP1251127A1 Novel sidechain-bearing taxanes and intermediates thereof |
10/23/2002 | EP1250328A1 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
10/23/2002 | CN1093123C Aralkyl and aralkylidene heterocyclic lactams and imides |
10/22/2002 | US6469004 Benzoheterocycles and their uses as MEK inhibitors |
10/17/2002 | US20020151552 Novel compounds |
10/17/2002 | US20020151536 Substituted azetidinone is used as sterol absorption inhibitor and a fibric acid derivative selected from fenofibrate, clofibrate, gemfibrozil, ciprofibrate, bezafibrate, clinofibrate etc |
10/16/2002 | EP1249233A1 Npyy5 antagonists |
10/16/2002 | EP1248785A1 Novel tetrahydropyridines, preparation method and pharmaceutical compositions containing same |
10/16/2002 | EP0991653B1 Novel compounds |
10/16/2002 | EP0948509B1 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives |
10/16/2002 | EP0542136B1 1-[(1,4-benzodioxanyl)alkyl]-4-(heteroaryl) piperidines, piperazines and pyrrolidines as antipsychotic agents |
10/16/2002 | CN1374872A Stabilization of macrolides |
10/16/2002 | CN1374082A Use of glycogen sulphofoenzyme inhibitor |
10/16/2002 | CN1092657C One pot synthesis of 2-oxazolidinone derivatives |
10/15/2002 | US6465481 Exhibit electrophysiological activity; may be more potent and produce fewer side effects including lower incidence of proarrhythmias such as torsades de pointes |
10/10/2002 | WO2002079198A1 Pyridazinone aldose reductase inhibitors |
10/10/2002 | WO2002079143A1 N-phenpropylcyclopentyl-substituted glutaramide derivatives as nep inhibitors for fsad |
10/10/2002 | US20020147341 Kinase inhibitor; benign prostatic hyperplasia |
10/10/2002 | US20020147200 Central nervous system disorders; antiserotonine agents |
10/10/2002 | US20020147194 Psychological disorders; antiserotonin agents; headache therapy |
10/10/2002 | US20020147184 Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions |
10/10/2002 | CA2442476A1 Pyridazinone aldose reductase inhibitors |
10/10/2002 | CA2437113A1 N-phenpropylcyclopentyl-substituted glutaramide derivatives as nep inhibitors for fsad |
10/09/2002 | EP1246804A1 4-carboxyamino-2-ethyl-1,2,3,4-tetrahydroquinoline crystal as cetp inhibitor |
10/09/2002 | EP0996622B1 Novel spiroazabicyclic heterocyclic compounds |
10/09/2002 | EP0679082B1 C10 taxane derivatives and pharmaceutical compositions |
10/09/2002 | CN1373763A Pteridinones and kinase inhibitors |
10/08/2002 | US6462068 Heterocyclylmethyl-substituted pyrazole derivatives |
10/03/2002 | WO2002076953A1 New spirotricyclic derivatives and their use as phosphodiesterase-7 inhibitors |
10/03/2002 | WO2002059127A3 Pyrazinoquinoxaline derivatives as serotonin agonists and antagonists |
10/03/2002 | US20020143017 Pyridazinone aldose reductase inhibitors |
10/03/2002 | US20020142968 For therapeutic and/or prophylactic treatment of idiopathic and adult respiratory distress syndrome, pulmonary fibrosis following treatment with radiation or chemotherapy, septic shock, septicemia, inflammatory responses |
10/03/2002 | US20020142023 Insecticide, miticide |