Patents for C07D - Heterocyclic compounds (10,420) |
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08/07/2002 | CN1362959A C10 carbamoyloxy substituted taxanes as antitumor agents |
08/07/2002 | CN1362958A C7 carbonate substituted taxanes as antitumor agents |
08/07/2002 | CN1362957A C17 heterosubustituted acetate taxanes as antitumor agents |
08/07/2002 | CN1362956A C7 carbamoyloxy substituted taxanes as antitumor agents |
08/07/2002 | CN1362954A Sulfamato hydroxamic acid metalloprotease inhibitor |
08/06/2002 | US6429210 Orthorombic polymorph of clopidogrel hydrogen sulfate with improved stability and lower solubility; antithrombotic agent; specific crystal structure and thermodynamic properties |
08/01/2002 | WO2002059127A2 Pyrazinoquinoxaline derivatives as serotonin agonists and antagonists |
08/01/2002 | WO2002059124A2 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists |
08/01/2002 | WO2002059112A2 Pyrazole compounds useful as protein kinase inhibitors |
08/01/2002 | WO2002059111A2 Pyrazole compounds useful as protein kinase inhibitors |
08/01/2002 | WO2002059110A1 Pyrimidineamines as angiogenesis modulators |
08/01/2002 | WO2002059083A2 Novel compounds |
08/01/2002 | WO2002058734A2 Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions |
08/01/2002 | WO2002058732A2 Combinations of peroxisome proliferator-activated receptor (ppar) activator(s) and sterol absorption inhibitor(s) and treatments for vascular indications |
08/01/2002 | US20020103209 Serotonergic modulators; for treatment of disorders of the central nervous system including psychotic disorders, hypertension and vascular disorders, migraine |
08/01/2002 | US20020103204 Piperazinyl)-3-(2-(3-(4-morpholinylmethyl)phenoxy)ethoxy) pyrazine derivatives; for prophylaxis or treatment of serotonin-related diseases |
08/01/2002 | CA2563051A1 Combinations of peroxisome proliferator-activated receptor (ppar) activator(s) and sterol absorption inhibitor(s) and treatments for vascular indications |
08/01/2002 | CA2434504A1 Combinations of sterol absorption inhibitor(s) with blood modifiers for treating vascular conditions |
08/01/2002 | CA2431970A1 Substituted pyrazinoquinoxaline derivatives as serotonin receptor agonists and antagonists |
07/31/2002 | EP1227095A2 A process for the purification of (S)-4-((3-(dimethylamino)ethyl)-1H-indol-5yl)-methyl)-2-oxazolidinone |
07/31/2002 | EP1227092A2 Isonitrile intermediates for the preparation of tri-substituted imidazole compounds with multiple therapeutic properties |
07/31/2002 | EP1227091A2 Formamide intermediates for the preparation of tri-substituted imidazole compounds with multiple therapeutic properties |
07/31/2002 | EP1227088A1 Crystalline base of citalopram and hydrochoride or hydrobromide salt thereof |
07/31/2002 | EP1226137A1 Phenyl- and pyridyl-tetrahydro-pyridines having tnf inhibiting activity |
07/31/2002 | EP0854867B1 Tetrahydroquinolines as nmda antagonists |
07/31/2002 | EP0527801B1 Thiophene sulfonamides useful as carbonic anhydrase inhibitors |
07/31/2002 | CN1361765A Inhibitors of aspartyl protease |
07/31/2002 | CN1360890A Use of active retiene derivative with negative hormone and/or antagonist |
07/30/2002 | US6426337 Antiinflammatory agents |
07/25/2002 | WO2002057267A1 Compounds specific to adenosine a1, a2a, and a3 receptor and uses thereof |
07/25/2002 | WO2002057259A2 Pyrazole compounds useful as protein kinase inhibitors |
07/25/2002 | WO2002042268A3 Ep4 receptor selective agonists in the treatment of osteoporosis |
07/25/2002 | WO2002032901A3 Bridged piperazine derivatives |
07/25/2002 | US20020099217 Process for preparing azacycloalkanoylaminothiazoles |
07/25/2002 | US20020099212 Sulfonamide compounds and pharmaceutical use thereof |
07/25/2002 | US20020099068 I kappa B kinase inhibitors for treating various disorders including arthritis |
07/25/2002 | CA2430577A1 Compounds specific to adenosine a1, a2a, and a3 receptor and uses thereof |
07/24/2002 | EP1224179A2 Sodium-hydrogen exchanger type 1 inhibitor crystals |
07/24/2002 | EP1224172A1 Drugs for the treatment of malignant tumours |
07/24/2002 | EP0741716B1 Delta 12,13 -iso-taxol analogs, antineoplastic use and pharmaceutical compositions containing them |
07/24/2002 | CN1360588A Hemisynthetic method and intermediate thereof |
07/23/2002 | US6423842 Act preferentially on m4 receptors; side effect reduction; used to treat nervous system disorders, psychological disorders and as an analgesic; alzheimer's disease; cognition activators. |
07/23/2002 | US6423722 Antiinflammatory agents |
07/23/2002 | CA2041594C Pyrido[2,3-f][1,4]thiazepines and pyrido[3,2-b][1,5]benzothiazepines |
07/18/2002 | US20020094999 Highly selective butyrylcholinesterase inhibitors for the treatment and diagnosis of Alzheimer's disease and dementias |
07/17/2002 | EP1222927A2 Pharmaceutical compositions having appetite suppressant activity |
07/17/2002 | EP1222195A1 Novel thiazolo(4,5-d)pyrimidine compounds |
07/17/2002 | EP1222190A1 5-(2-substituted-5-heterocyclylsulphonylpyrid-3-yl)-dihydropyrazolo[4,3-d]pyrimidin-7-ones as phosphodiesterase inhibitors |
07/17/2002 | EP1222173A1 Process for preparing 4-trifluoromethylsulphinylpyrazole derivative |
07/17/2002 | EP0888340B1 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives as endothelin antagonists |
07/17/2002 | EP0766668B1 Processes for preparing anhydrous and hydrate forms of antihistaminic piperidine derivatives, polymorphs and pseudormophs thereof |
07/16/2002 | US6420359 5,11-Dihydro-11-ethyl-5-methyl-8-(2-((1-oxido-4-quinolinyl)oxy)ethyl)-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one for example; antiviral agents for HIV infection |
07/11/2002 | WO2002053558A1 Quinazolone derivatives as alpha 1a/b adrenergic receptor antagonists |
07/11/2002 | WO2002053542A1 Process for making amlodipine maleate |
07/11/2002 | WO2002053134A1 Pharmaceutical compositions comprising amlodipine maleate |
07/11/2002 | US20020091265 4-phenyl-pyridine derivatives |
07/11/2002 | US20020091262 Armoatic or heteroarmoatic compound containing substituted amides or thioamides |
07/11/2002 | US20020091119 Aralkyl and aralkylidene heterocyclic lactams and imides |
07/11/2002 | US20020091118 Psychotherapeutic agents. |
07/11/2002 | US20020091117 Psychotherapeutic agents. |
07/10/2002 | EP1221314A1 New crystalline form of omeprazole |
07/10/2002 | EP1220856A2 Pyrazolo[4,3-d]pyrimidine derivatives |
07/10/2002 | EP1220842A1 Cyclic amine compounds as ccr5 antagonists |
07/10/2002 | CN1087288C Crystalline [R-(R+,R+)]-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(5-methylethyl)-3-phenyl-4-(phenylamino) carbonyl]-1H-pyrole-1-heptanoic acid hemi-calcium salt (atorvastatin) |
07/09/2002 | CA2041224C Azatetracycle compounds |
07/04/2002 | US20020086888 Substantially free from amlodipine aspartate side products, by reacting amlodipine or an acid addition salt thereof with excess maleic acid under acidic environment |
07/04/2002 | US20020086874 Substituted indoline derivative compounds which are antagonists of the progesterone receptor; contraceptives; antineoplastic agents |
07/04/2002 | US20020086850 Antiinflammatory agents |
07/03/2002 | EP1218354A1 Quinazoline derivatives and their use as pharmaceuticals |
07/03/2002 | EP1218347A1 Pyrazoloanthrone and derivatives thereof as jnk inhibitors and their compositions |
07/03/2002 | EP0563345B1 Novel 4-arylpiperazines and 4-arylpiperidines |
07/03/2002 | CN1356991A Quinoline and quinoxaline compounds as PDGF-R and/or LCD tyrosine kinase inhibitors |
07/03/2002 | CN1356323A Benzothiazolone derivative |
07/02/2002 | US6414156 Efficent, notoxic process of making new key intermediate quaternary ammonium salts and 2-oxazolylalkyl sulfide derivatives and avoids the reaction of a-haloketones with an azide followed by reducing the resulting a-aminoketone |
07/02/2002 | US6414009 Cardiovascular disorders; anticoagulants |
07/02/2002 | US6413985 Selective antagonists for the strychnine insensitive glycine binding site associated with the nmda receptor complex. |
07/02/2002 | US6413980 Nitrogen containing heterobicycles as factor Xa inhibitors |
06/27/2002 | WO2002050066A2 Pyrazole compounds useful as protein kinase inhibitors |
06/27/2002 | WO2002050065A2 Pyrazole compounds useful as protein kinase inhibitors |
06/27/2002 | WO2001051051A3 Agents, such as nicotinamide or cadpr for the treatment of skin disorders |
06/26/2002 | CN1355799A 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives |
06/26/2002 | CN1086700C Benzothiophene compounds, intermediates, composition, and methods |
06/26/2002 | CN1086569C Dehydration plant |
06/25/2002 | US6410747 Highly selective butyrylcholinesterase inhibitors for the treatment and diagnosis of alzheimer's disease and dementias |
06/25/2002 | US6410740 Heterocyclylmethyl-substituted pyrazol derivatives |
06/25/2002 | US6410480 Plant safening agents and growth regulators for controlling weeds and grasses; post/preemergence herbicides |
06/20/2002 | US20020077482 Novel intermediates useful for the preparation of antihistaminic piperidine derivatives |
06/20/2002 | US20020077341 C10 carbamoyloxy substituted taxanes |
06/19/2002 | EP1214310A1 Novel photochromic naphthopyrans |
06/19/2002 | EP0980354B1 Vitamin d3 analogs with bis c-20 side chains |
06/18/2002 | US6407237 Crystal forms of 9-substituted hypoxanthine derivatives |
06/18/2002 | US6407104 Pyrrolo[1,2-a]pyrazine spla2 inhibitor |
06/13/2002 | US20020072616 3-azabicyclo[3.1.0]hexane derivatives useful in therapy |
06/13/2002 | US20020072519 Useful as psychotherapeutic agents |
06/13/2002 | DE10041671C1 Verfahren zur Herstellung von Imidazo[1,2-c][2,3]benzodiazepinen sowie Phenylessigsäureester und Oxazol-Derivate als Zwischenprodukte bei deren Herstellung Benzodiazepines process for the preparation of imidazo [1,2-c] [2,3] oxazole and phenylacetic acid esters and derivatives, as intermediates in the preparation thereof |
06/12/2002 | EP1213291A1 Spiro [1-azabicyclo[2.2.2]octane-3,2'(3'H)-furo[2,3-b]pyridine for use in the treatment of psychotic and intellectual impairment disorders |
06/12/2002 | EP1213020A2 Pharmaceutical compositions having appetite suppressant activity |
06/12/2002 | EP1212320A2 Phenylpiperazines as serotonin reuptake inhibitors |
06/12/2002 | EP1032571B1 Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance p antagonists |
06/12/2002 | EP0885221B1 Azabicyclic esters of carbamic acids useful in therapy |