Patents for C07D - Heterocyclic compounds (10,420) |
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03/26/2003 | CN1406236A Process for the preparation of 5-carboxy-phthalide and its use for the production of CITALOPRAM |
03/25/2003 | CA2379005A1 Low hygroscopic aripiprazole drug substance and processes for the preparation thereof |
03/20/2003 | WO2003022848A2 Process for the preparation of diketopyrrolopyrroles |
03/20/2003 | WO2003022847A2 Process for the direct preparation of pyrrolo[3,4-c]pyrroles |
03/20/2003 | WO2003022824A1 Oxazolidinone and/or isoxazoline as antibacterial agents |
03/20/2003 | WO2003022286A1 Benzothiazepine and benzothiadiazepine derivatives with ileal bile acid transport (ibat) inhibitory activity for the treatment hyperlipidaemia |
03/20/2003 | WO2003022279A1 Inhalation compositions comprising tricyclic 5,6-dihydro-9h-pyrazolo (3,4-c)-1,2,4-triazolo (4,3-alpha) pyridines and a tiotropium salt |
03/20/2003 | WO2003022275A1 Inhalation compositions comprising tricyclic 5,6-dihydro-9h-pyrazolo (3,4-c)-1,2,4-triazolo (4,3-alpha) pyridines |
03/20/2003 | US20030055071 For therapy, prophylaxis or delaying the onset of AIDS and infection by HIV |
03/20/2003 | US20030055068 Pyrazole compounds useful as protein kinase inhibitors |
03/20/2003 | US20030055035 Useful in hyperpolarizing cell membranes, opening potassium channels, relaxing smooth muscle cells, and inhibiting bladder contractions |
03/20/2003 | CA2459766A1 Oxazolidinone and/or isoxazoline as antibacterial agents |
03/20/2003 | CA2457717A1 Use of compounds in a dry powder inhaler |
03/20/2003 | CA2457710A1 Process for the direct preparation of pyrrolo¬3,4-c|pyrroles |
03/19/2003 | EP1292594A1 Quinazoline derivatives for the treatment of tumours |
03/19/2003 | EP1178984B1 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives |
03/19/2003 | EP1177195B1 1-AMINO TRIAZOLO 4,3-a! QUINAZOLINE-5-ONES AND OR -5-THIONES INHIBITING PHOSPHODIESTERASE IV |
03/19/2003 | CN1404479A Novel 1,3-dihydro-2H-indol-2-one derivatives their preparing method and the pharmceutical composition containing the same |
03/19/2003 | CN1404477A 哌嗪和哌啶衍生物 Piperazine and piperidine derivatives |
03/19/2003 | CN1404472A Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
03/19/2003 | CN1403455A Synthesis of 2-oxazolidone derivate by one still process |
03/13/2003 | WO2003020748A1 Anti-cancer cyclopenta[g]quinazoline compounds |
03/13/2003 | US20030050343 Novel potentiating compounds |
03/13/2003 | CA2458399A1 Cyclic indole and heteroindole derivatives, the production and use thereof as medicaments |
03/12/2003 | EP1291346A1 Process for the preparation of trisubstituted imidazole compounds with multiple therapeutic properties |
03/12/2003 | EP1289999A1 Antitumoral analogs of et-743 |
03/12/2003 | EP1036068B1 Process and intermediates for the preparation of a triazoline herbicide |
03/12/2003 | EP0874830B1 A metalloproteinase inhibitor, a pharmaceutical composition containing it and the pharmaceutical use and method useful for the preparation thereof |
03/12/2003 | EP0670835B1 Process for preparing benzopyran compounds |
03/12/2003 | CN1402730A Thiazolo (4,5-D) pyrimidine compounds |
03/12/2003 | CN1402711A 4-carboxyamino-2-ethyl-1,2,3,4-tetrahydroquinoline crystal as CETP inhibitor |
03/12/2003 | CN1402710A Antipicornaviral compound and compositions, their pharmaceutical uses, and material for their synthesis |
03/11/2003 | US6531610 Intermediate acylating carbonate |
03/06/2003 | WO2003018582A1 Novel imidazopyridine compounds with therapeutic effect |
03/06/2003 | WO2002102382A9 A PROCESS FOR PREPARING PAROXETINE HCl WHICH LIMITS FORMATION OF PINK COLORED COMPOUNDS |
03/06/2003 | US20030045721 Process for preparing anhydrous and hydrate forms of antihistaminic piperidine derivatives, polymorphs and pseudomorphs thereof |
03/06/2003 | US20030045479 Novel N-formyl hydroxylamine compounds, compositions and methods of use |
03/06/2003 | CA2456350A1 Novel imidazopyridine compounds with therapeutic effect |
03/05/2003 | EP1288206A1 Substituted benzenesulfonamide derivatives as prodrugs of COX-2 inhibitors |
03/05/2003 | EP1287004A1 Synthetic process for the manufacture of an ecteinascidin compound |
03/05/2003 | EP1286975A1 Biclyclic cyclohexylamines and their use as nmda receptor antagonists |
03/05/2003 | EP1286672A2 S-methyl-dihydro-ziprasidone for treatment of psychiatric and ocular disorders |
03/05/2003 | EP1062214B1 Substituted 2-(2,6-dioxo-3-fluoropiperidin-3-yl)-isoindolines and their use to reduce tnfa levels |
03/05/2003 | EP0991641B1 Crystalline form of omeprazole sodium salt |
03/05/2003 | EP0969819B1 New crystalline form of omeprazole |
03/05/2003 | EP0892791B1 N-[[4-(5-METHYL-3-PHENYLISOXAZOL-4-YL]PHENYL]SULFONYLPROPYLAMIDE and its SODIUMSALT AS PRODRUGS OF COX-2 INHIBITORS |
03/05/2003 | EP0853610B1 Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities |
03/04/2003 | US6528654 Synthesis of histamine dihydrochloride |
03/04/2003 | US6528494 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives |
02/27/2003 | WO2003016306A1 Hiv inhibiting pyrimidines derivatives |
02/27/2003 | WO2003016305A1 Crystals including a malic acid salt of n-[2-(diethylamino) ethyl]-5-[(5-fluoro-2-oxo-3h-indole-3-ylidene) methyl]-2, 4-dimethyl-1h-pyrrole-3-carboxamide, processes for its preparation and compositions thereof |
02/27/2003 | WO2003016302A1 Diamine derivatives |
02/27/2003 | CA2456841A1 Cyclohexyl and piperidine diamine derivatives useful as activated blood coagulation factor x inhibitors |
02/26/2003 | EP1284974A2 Triazolyl tropane derivatives as ccr5 modulators |
02/26/2003 | EP0979034B1 Composition for controlling harmful bio-organisms and method for controlling harmful bio-organisms using the same |
02/26/2003 | CN1399639A New oxabispidine compound useful in treatment of cardiac arrhythmias |
02/25/2003 | US6525204 Oximination reaction of nitro-o-methylphenyl compound with organic nitrite; cyclization with alkene in basic catalyst presence; reduction, bromination, oxidation, carboxylation |
02/25/2003 | US6525060 Triazolo(4,5-d)pyrimidine compounds |
02/25/2003 | US6525048 Aminomethylphenoxymethyl/benzisoxazole substituted azabicyclic compounds; depression, generalized anxiety disorder, obesity, migraine; 2-(5-Fluoro-benzo(d)isoxazol-3-y)-7-(3-morpholin-4-ylmethylphenoxymethyl) -octahydro-pyrido(1,2-a)pyrazine; |
02/20/2003 | WO2002065979A3 (diazolo-pyridinyl)-pyrimidines for use in treatment of cns disorders and diabetes |
02/20/2003 | US20030036554 Oxidizing the corresponding sulfide without sulfone production to product purer omerprazole, lansoprazole, pantoprazole, rabeprazole, etc. |
02/20/2003 | US20030036552 Novel compounds |
02/20/2003 | US20030036543 Especially as inhibitors of Aurora-2 and GSK-3, for treating diseases such as cancer, diabetes and Alzheimer's disease. |
02/19/2003 | EP1283828A1 Novel polymorph v of torasemide |
02/18/2003 | US6521632 Method for the treatment or prevention of a disease mediated by the alpha-2B-adrenoceptor |
02/13/2003 | WO2003011863A1 Novel crystal forms of 9-substituted hypoxanthine derivatives |
02/13/2003 | WO2003011826A1 Crystalline forms vi and vii of atorvastatin calcium |
02/13/2003 | US20030032617 Administering nicotinamide, a nicotinamide agonist, a nicotinamide derivative, a nicotinamide metabolite or prodrugs thereof. |
02/13/2003 | CA2417337A1 Novel crystal forms of 9-substituted hypoxanthine derivatives |
02/12/2003 | EP1283203A1 Crystalline form of 4-(5-methyl-3-phenylisoxazol-4-yl) benzene-sulfonamide |
02/12/2003 | EP1282609A2 Piperazinedione compounds |
02/12/2003 | EP0871623B1 3-azetidinylalkylpiperidines or -pyrrolidines as tachykinin antagonists |
02/12/2003 | CN1396827A Remedies or preventives for pulmonary insufficiency containing diaminotrifluoromethylpyridine derivatives |
02/12/2003 | CN1101384C Process for preparing 1-biphenylmethylmidazole derivatives |
02/11/2003 | US6518310 Non-peptidic; inhibits trypsin-like protease, thrombin and embolus formation; anticoagulant |
02/11/2003 | US6518286 Compounds |
02/11/2003 | US6518277 Disrupting leukocyte function |
02/11/2003 | US6517866 Sertraline salts and sustained-release dosage forms of sertraline |
02/06/2003 | WO2003010159A1 Piperidine derivatives as nmda receptor antagonists |
02/06/2003 | WO2003010141A2 Hepatitis c virus polymerase inhibitors with a heterobicyclic structure |
02/06/2003 | WO2003010140A2 Hepatitis c virus polymerase inhibitors with heterobicyclic structure |
02/06/2003 | WO2002059112A3 Pyrazole compounds useful as protein kinase inhibitors |
02/06/2003 | US20030027831 Arylpiperzine derivatives are useful for treatment of anxiety, depression, hypertension, cognitive disorders, sexual dysfunction, brain trauma, memory loss, eating disorders, obesity, substance abuse, and obsessive-compulsive diseases |
02/06/2003 | US20030027825 Polymorphic form of a tachykinin receptor antagonist |
02/05/2003 | EP1281400A2 Pharmaceutical compositions containing ascomycin derivatives |
02/05/2003 | CN1100771C Phosphononooxymethyl ethers for taxame derivatives |
02/04/2003 | US6514997 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis |
02/04/2003 | US6514976 Arylpiperazines having activity at the serotonin 1A receptor |
02/04/2003 | CA2271566C Substituted phenyl pyrimidines useful in the treatment of cns disorders |
01/30/2003 | WO2003008407A2 Phenylsulfonyl-1,3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use |
01/30/2003 | WO2002012247A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof |
01/30/2003 | US20030022885 Pyrazole compounds useful as protein kinase inhibitors |
01/30/2003 | CA2450437A1 1-phenylsulphonyl-1,3-dihydro-2h-indol-2-one derivatives, their preparation and their therapeutic application |
01/30/2003 | CA2417804A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof |
01/29/2003 | EP1278748A2 Inhibitors of human phosphatidyl-inositol 3-kinase delta |
01/29/2003 | EP1278747A1 Pyrano, piperidino, and thiopyrano compounds and methods of use |
01/29/2003 | EP0641795B9 Carbapenem derivative |
01/28/2003 | US6512116 No drug resistance; intravenous |
01/28/2003 | CA2124375C Compounds containing a fused bicyclic ring and processes therefor |
01/23/2003 | WO2003006449A1 Method for the preparation of escitalopram |