| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 04/06/2006 | CA2582297A1 Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 04/05/2006 | EP1641801A2 Bridged n-arylsulfonylpiperidines as gamma-secretase inhibitors |
| 04/04/2006 | US7022706 Central nervous system disorders |
| 04/04/2006 | CA2233173C Dopamine and serotonin transporter ligands and imaging agents |
| 03/30/2006 | US20060069077 Receptor-type kinase modulators and methods of use |
| 03/29/2006 | EP1638965A1 Novel 8-aza-bicyclo¬3.2.1|octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 03/29/2006 | CN1753891A Ccr-3 receptor antagonists |
| 03/28/2006 | CA2219533C Process for preparing enantiomerically pure tropic acid esters |
| 03/23/2006 | US20060063796 Pyrazoles as inhibitors of tumor necrosis factor |
| 03/23/2006 | CA2580292A1 Process for preparing substituted 8-azabicyclo[3.2.1] octan-3-ols |
| 03/22/2006 | CN1246315C Amino alkoxybenzoyl-benzofuran or benzothiophene derivatives, methods for preparing same and compositions containing same |
| 03/21/2006 | CA2263983C Cyclic amine derivatives for inhibiting blood platelet aggregation |
| 03/16/2006 | WO2005115361A3 Androgen receptor modulators and method of treating disease using the same |
| 03/16/2006 | US20060058344 Esters of hydroxyl-substituted nitrogen heterocycles, processes for the preparation thereof as well as the use thereof as pharmaceutical compositions |
| 03/16/2006 | US20060058343 Process for preparing substituted 8-azabicyclo[3.2.1]octan-3-ols |
| 03/16/2006 | US20060058335 Fluorenecarboxylic acid esters, process for the manufacture thereof, and use thereof as medicaments |
| 03/15/2006 | EP1448566B1 Chemokine receptor antagonists and methods of use thereof |
| 03/14/2006 | US7012142 Sultam compounds |
| 03/14/2006 | US7012078 For therapy and prophylaxis of migraine, inflammatory diseases, stroke, acute and chronic pain, hypovolemic shock, traumatic shock, reperfusion injury, Crohn's disease, ulcerative colitis, septic shock, multiple sclerosis, etc. |
| 03/14/2006 | US7011813 Cocaine receptor binding ligands |
| 03/09/2006 | WO2006025324A1 Tropan compound |
| 03/09/2006 | WO2005105770A3 Arylphenylamino-, arylphenylamide-, and arylphenylether-sulfide derivatives |
| 03/09/2006 | US20060052595 Heterocyclic compounds as ccr5 antagonists |
| 03/09/2006 | US20060052413 Novel piperidine derivatives as modulators of chemokine receptor ccr5 |
| 03/09/2006 | US20060052247 Novel herbicides |
| 03/08/2006 | EP1632483A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands |
| 03/08/2006 | EP1326585B1 Method for producing powdery formulations |
| 03/08/2006 | CN1744899A Piperidine derivatives as CCR5 antagonists |
| 03/08/2006 | CN1744895A N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines |
| 03/08/2006 | CN1244581C Method for producing anticholinergic agent substitute bromide |
| 03/02/2006 | WO2006021657A1 Amino-tropane derivatives, preparation thereof and therapeutic use thereof |
| 03/02/2006 | WO2006021656A2 Aminopiperidine derivatives, preparation thereof and use thereof as melanocortin receptor agonists |
| 03/02/2006 | WO2006021655A2 Oxopiperidine derivatives, preparation and therapeutic use thereof |
| 03/02/2006 | US20060047116 Such as N-methyl(1-{2-[(1R,5S)-3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-2,3-dihydro-1H-inden-1-yl)methanamine; chemokine receptor antagonists; prevention or treatment of a human T-cell leukemia/lymphoma virus infection |
| 03/02/2006 | US20060046995 anti-bacterial agents; staphylococci; coliform bacteria; 7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide; bridged bicyclic ureas or carbamates having bridgehead nitrogen |
| 03/02/2006 | DE102004041253A1 Neues Verfahren zur Herstellung von Tiotropiumsalzen New method for the preparation of tiotropium |
| 03/02/2006 | DE102004039789A1 Arylsubstituierte polycyclische Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Aryl-substituted polycyclic amines, process for their preparation and their use as medicaments |
| 03/02/2006 | CA2577177A1 Oxopiperidine derivatives, preparation and therapeutic use thereof |
| 03/02/2006 | CA2574517A1 Amino-tropane derivatives, preparation thereof and therapeutic use thereof |
| 03/02/2006 | CA2574454A1 Aminopiperidine derivatives, preparation thereof and use thereof as melanocortin receptor agonists |
| 03/02/2006 | CA2573373A1 Method for producing tiotropium salts and silicon derivatives as intermediates |
| 03/01/2006 | CN1742011A 8-aza-bicyclo (3.2.1) octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 02/23/2006 | WO2006018609A2 Anti-inflammatory agents |
| 02/23/2006 | US20060040949 Treating antibiotic resistant bacterial infections; compounds based on quinoline rings; (3S)-2-(3-{[(Benzo[1,2,5]thiadiazol-5-ylmethyl)-amino]-methyl}-piperidin-1-yl)-(1RS)-(6-methoxy-quinolin-4-yl)-ethanol for example |
| 02/23/2006 | US20060039868 For use in therapy of chronic obstructive pulmonary disease and asthma; an inhalette capsule contains a mixture of coarser and fine excipient particles |
| 02/23/2006 | CA2577274A1 Anti-inflammatory agents |
| 02/22/2006 | EP1626970A1 Azabicycloalkane compounds as muscarinic receptor antagonists |
| 02/22/2006 | EP1626967A1 Substituted pyrazoles |
| 02/15/2006 | EP1625120A1 Chemical compounds |
| 02/15/2006 | EP1624845A2 4',4''-substituted 3alpha-(diphenylmethoxy)tropane analogs for treatment of mental disorders |
| 02/15/2006 | CN1733761A Crystalline tiotropium bromide monohydrate, processes for the preparation thereof, and the use thereof in the production of a medicament |
| 02/14/2006 | US6998406 Fluorenecarboxylic acid esters, process for the manufacture thereof, and use thereof as medicaments |
| 02/14/2006 | CA2189567C Substituted fused and bridged bicyclic compounds as therapeutic agents |
| 02/09/2006 | US20060030585 N-(2-[9-(8-Azabicyclo[3.2.1]oct-3-ylidene)-9H-xanthen-3-yl]-phenyl)-acetamide; veterinary medicine; side effect reduction; analgesics; antagonist; antiinflammatory agents; psychhological/nervous system/urogenital disorders; drug abuse; diarrhea; gastritis; cardiovascular/respiratory disorders; kits |
| 02/08/2006 | EP1622901A1 Tropane derivatives and their use as ace inhibitors |
| 02/08/2006 | EP1622610A1 1-(2h-pyrazol-3-yl)-3- 4-[1-(benzoyl)-piperidin-4-ylmethyl]-phenyl -urea derivatives and related compounds as inhibitors of p38 kinase and/or tnf inhibitors for the treatment of inflammations |
| 02/08/2006 | EP1318978B1 N-acylsulfonamide apoptosis promoters |
| 02/08/2006 | CN1732166A Novel herbicides |
| 02/07/2006 | CA2360308C Glucocorticoid receptor modulators |
| 02/05/2006 | WO2007030089A1 Tricyclic delta- opioid modulators |
| 02/05/2006 | CA2574768A1 Tricyclic delta-opioid modulators |
| 02/02/2006 | WO2005103002A3 Novel alkyne compounds with an mch-antagonistic action and medicaments comprising said compounds |
| 02/02/2006 | US20060025402 Benzimidazolidinone derivatives as muscarinic agents |
| 02/01/2006 | EP1621197A2 Composition comprising a steroid and an anticholinergic agent |
| 02/01/2006 | CN1729178A N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines |
| 01/26/2006 | US20060019962 Modulators of muscarinic receptors |
| 01/26/2006 | US20060019960 Antitumoral analogs of ET-743 |
| 01/25/2006 | CN1237970C Inhalant containing tiotropium salt solution |
| 01/24/2006 | US6989396 Anticancer agents; modulating glycoprotein |
| 01/24/2006 | CA2292984C Ccr5 modulators |
| 01/19/2006 | US20060014964 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
| 01/19/2006 | US20060014780 Nicotinamide derivatives useful as PDE4 inhibitors |
| 01/19/2006 | US20060014739 Androgen receptor modulators and method of treating disease using the same |
| 01/18/2006 | EP1615920A1 3-benzhydrylidene-8-aza-bicyclo [3.2.1] octane derivatives with opioid receptor activity |
| 01/18/2006 | CN1723196A Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 01/11/2006 | EP1613613A2 Cxcr4 chemokine receptor binding compounds |
| 01/11/2006 | EP1442036B1 Heteroaryl derivatives as superior ligands for nociceptin receptor orl-1 |
| 01/10/2006 | CA2485556C Pyrrolopyrimidine and pyrrolopyridine derivatives substituted with cyclic amino group |
| 01/10/2006 | CA2364178C N-benzenesulfonyl l-proline compounds as bradykinin antagonists |
| 01/05/2006 | WO2006001894A1 Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
| 01/05/2006 | WO2005100352A8 Selected cgrp-antagonists, their preparation processes and their use as medicaments |
| 01/05/2006 | US20060004004 Novel gamma secretase inhibitors |
| 01/05/2006 | DE102004004965B4 Verfahren zur Herstellung eines 2-(Ethoxymethyl)-tropanderivates A process for preparing a 2- (ethoxymethyl) -tropanderivates |
| 01/05/2006 | CA2570893A1 Novel piperidine/8-azabicyclo [3.2.1] octan derivatives as moduilators of chemokine receptor ccr5 |
| 01/05/2006 | CA2568804A1 Pyrrolopyrimidine and pyrrolopyridine derivatives substituted with a cyclic amino group as crf antagonists |
| 01/05/2006 | CA2567977A1 Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
| 01/04/2006 | EP1610789A1 Bicyclic piperidine derivatives as melanocortin-4 receptor agonists |
| 01/04/2006 | EP0934288B1 Oxadiazoles, processes for their preparation and their use as medicaments |
| 01/04/2006 | CN1717408A Carbamic acid esters with anticholinergic activity |
| 01/03/2006 | CA2244773C Tropane-derivatives, their preparation and use |
| 12/29/2005 | WO2005123728A1 Novel 9-aza-bicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 12/29/2005 | US20050288321 Alzheimer's disease ; 3-(2,3-dihydro-5,6-difluorobenzofur-7-yl)-4-[1-(piperidin-4-yl)-1H-indol-3-yl]pyrrole-2,5-dione; stimulating bone deposition |
| 12/28/2005 | EP1497288B1 Novel ester hydroxy-substituted nitrogen heterocycles as antagonists of the muscarinic m3 receptor, methods for the production thereof, and use thereof as a medicament |
| 12/28/2005 | EP1461318B9 Tetrahydroquinoline analogues as muscarinic agonists |
| 12/22/2005 | US20050283006 Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses |
| 12/22/2005 | US20050282857 e.g. 1-(4-amino-3-chloro-5-trifluoromethyl-benzyl)-2-oxo-2-[4-(2-piperidin-1-yl-ethyl)-piperidin-1-yl]-ethyl 4-(2-oxo-1 ,2,4,5-tetrahydro-benzo[d][1,3]diazepin-3-yl)-piperidine-1-carboxylate; calcitonin gene related peptide antagonist; migraine or cluster headaches, non-insulin-dependent diabetes |
| 12/21/2005 | EP1606288A1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain |
| 12/21/2005 | EP1362039B1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands |
| 12/20/2005 | US6977264 For therapy and prophylaxis of obesity, diabetes |
| 12/20/2005 | CA2338206C High affinity ligands for nociceptin receptor orl-1 |