| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 08/05/2009 | CN100522976C Novel azacyclic ethynyl derivatives |
| 08/05/2009 | CN100522135C Inhalation kit comprisung inhalable powder of tiotropium |
| 08/04/2009 | US7569582 Aminotropane derivatives, preparation thereof and therapeutic use thereof |
| 08/04/2009 | US7569581 Anticholinergics which may be used as medicaments as well as processes for preparing them |
| 07/30/2009 | WO2009092293A1 Pyrollidine-based compounds |
| 07/30/2009 | WO2009055331A3 Bicyclic heterocycle derivatives and their use as modulators of the activity of gpr119 |
| 07/29/2009 | EP2083007A1 Tiotropium salts, method for creating same and medicinal formulations containing same |
| 07/29/2009 | CN100519558C Crystalline tiotropium bromide monohydrate, processes for the preparation thereof, and the use thereof in the production of a medicament |
| 07/23/2009 | WO2009063061A3 Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
| 07/23/2009 | US20090187021 Indane compounds as ccr5 antagonists |
| 07/23/2009 | US20090186921 Azacyclic compounds |
| 07/23/2009 | US20090186871 Tyrosine kinase inhibitors |
| 07/22/2009 | CN100515419C Substituted benzazoles and its application as inhibitors of Raf kinase |
| 07/21/2009 | US7563803 M3 muscarinic acetylcholine receptor antagonists |
| 07/21/2009 | US7563795 Phenyl-piperazine derivatives as modulators of muscarinic receptors |
| 07/16/2009 | WO2009087419A1 Novel process for the preparation of scopine esters |
| 07/16/2009 | CA2710523A1 Process for the preparation of scopine esters |
| 07/15/2009 | EP2078010A2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors |
| 07/15/2009 | EP1741430B1 Remedy for psychoneurotic diseases |
| 07/14/2009 | US7560546 Tyrosine kinase inhibitors |
| 07/14/2009 | US7560460 2-[(4-Chlorophenyl)methyl]-1-(4- {2-[(cyclopropylmethyl)-(methylsulfonyl)amino]phenyl }-piperazinyl) -4-(2-(1,2,3,4-tetrahydroisoquinolyl))butane-1,4-dione; obesity/dietietics; melanocortin receptor angonists; prophylaxis/treatment of diseases involving activation of the melanocortin recepetors (MCR) |
| 07/10/2009 | WO2008083367A2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors |
| 07/10/2009 | CA2710234A1 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors |
| 07/09/2009 | WO2009055922A8 Labeled iodinated tropane formulation |
| 07/08/2009 | EP2076506A2 Heterocyclic-substituted piperidines as orl-1 ligands |
| 07/08/2009 | EP1626970B1 Azabicycloalkane compounds as muscarinic receptor antagonists |
| 07/08/2009 | CN101475569A Method for preparing granisetron hydrochloride from high tropine alkanamine |
| 07/08/2009 | CN100509809C Novel crystalline anhydride with anticholinergic effect |
| 07/08/2009 | CN100509774C Acylsulfonamides as inhibitors of steroid sulfatase |
| 07/01/2009 | EP2074120A1 Tropane compounds |
| 07/01/2009 | EP1651230B1 Medicaments for inhalation comprising steroids and a novel fluorene carboxylic acid ester |
| 06/25/2009 | US20090163471 Tropane compounds |
| 06/23/2009 | US7550500 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
| 06/23/2009 | US7550469 Heterocyclic amide derivatives and their use as dopamine D3 receptor ligands |
| 06/18/2009 | WO2009075776A1 Process for the preparation of retapamulin and its intermediates |
| 06/11/2009 | US20090149655 Process for the preparation of Retapamulin and its intermediates |
| 06/10/2009 | EP2067779A1 Tiotropium salts, method for their production and medicinal formulas containing them |
| 06/10/2009 | CN100497335C Optical resolution method substituting oxyphosphonate acetate |
| 06/09/2009 | US7544802 Process for the preparation of 2-(ethoxymethyl)-tropane derivatives |
| 06/04/2009 | WO2009070307A1 Amorphous retapamulin and processes for preparation thereof |
| 06/04/2009 | WO2009014610A3 Process for preparing an intermediate to mu opioid receptor antagonists |
| 06/04/2009 | US20090143443 Cyclic amine compound and pest control agent |
| 06/04/2009 | US20090143374 Use of Compounds and Compositions for the Treatment of Amyloid Diseases |
| 06/03/2009 | EP1606288B1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain |
| 06/03/2009 | CN101448825A Fused bicycloheterocycle substituted azabicyclic alkane derivatives |
| 06/03/2009 | CN101445506A 3 alpha-high tropine aliphatic amine salt, crystal formation and preparation method |
| 06/03/2009 | CN101444509A Triple monoamine reuptake inhibitors for the treatment of chronic pain |
| 06/02/2009 | US7541368 Pyrazoles as inhibitors of tumor necrosis factor |
| 05/28/2009 | WO2009067579A1 Biaryl substituted azabicyclic alkane derivatives as nicotinic acetylcholine receptor activity modulators |
| 05/28/2009 | WO2009066735A1 Method for producing 2-azaadamantane |
| 05/28/2009 | US20090137806 Dual nk1/nk3 receptor antagonists |
| 05/28/2009 | US20090137625 Novel Enantiomers and Their Use as Monoamine Neurotransmitter Re-Uptake Inhibitors |
| 05/28/2009 | US20090137585 N-acylsulfonamide apoptosis promoters |
| 05/28/2009 | CA2705296A1 Biaryl substituted azabicyclic alkane derivatives as nicotinic acetylcholine receptor activity modulators |
| 05/27/2009 | EP1833826B1 Tricyclic delta-opioid modulators |
| 05/26/2009 | US7538111 N(2-hydroxyethyl)-4-methoxy-N,2,6-trimethylbenzene- sulphonamide; analgesic, antiinflammatory agent; hyperalgesia and major algesia connected with other pathological conditions such as cancer |
| 05/22/2009 | WO2009064835A1 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors |
| 05/22/2009 | WO2009063061A2 Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
| 05/22/2009 | CA2704628A1 Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
| 05/22/2009 | CA2704599A1 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors |
| 05/21/2009 | US20090130090 N-amide Derivatives of 8-Azabicyclo[3.2.1]OCT-3-YL AS CCR1 Antagonists |
| 05/20/2009 | EP2060557A1 Intermediate compounds useful to prepare dolasetron |
| 05/20/2009 | EP2059515A2 Pyrrolidine derivatives as modulators of chemokine ccr5 receptors |
| 05/20/2009 | EP1807423B1 Quinolinone-carboxamide compounds |
| 05/13/2009 | CN100486973C Novel benzodioxoles |
| 05/12/2009 | US7531661 Such as N-methyl(1-{2-[(1R,5S)-3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-2,3-dihydro-1H-inden-1-yl)methanamine; chemokine receptor antagonists; prevention or treatment of a human T-cell leukemia/lymphoma virus infection |
| 05/07/2009 | WO2009055922A1 Labeled iodinated tropane formulation |
| 05/07/2009 | WO2008077555A3 Substituted isoquinolines and their use as rho-kinase inhibitors |
| 05/07/2009 | US20090118232 Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
| 05/07/2009 | CA2704104A1 Labeled iodinated tropane formulation |
| 05/06/2009 | EP2054368A2 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
| 05/06/2009 | CN100484935C Benzimidazole-derivatives as factor Xa inhibitors |
| 04/30/2009 | WO2009055331A2 Bicyclic heterocycle derivatives and their use as modulators of the activity of gpr119 |
| 04/30/2009 | WO2009055077A1 Tropane compounds |
| 04/30/2009 | CA2703477A1 Tropane compounds |
| 04/30/2009 | CA2703203A1 Bicyclic heterocycle derivatives and methods of use thereof |
| 04/29/2009 | CN100482659C Benzimidazolone compounds having 5-HT4 receptor agonistic activity |
| 04/28/2009 | US7524970 Compounds |
| 04/23/2009 | WO2009027820A3 Substituted-quinoxaline-type-piperidine compounds and the uses thereof |
| 04/22/2009 | EP2050745A1 N-pyridylpiperidine compound, method for producing the same, and pest control agent |
| 04/22/2009 | EP2049120A1 Urotensin ii receptor antagonists |
| 04/22/2009 | EP1689391B1 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylinositol 3 kinase enzymes (pi3) for the treatment of inflammatory airway diseases |
| 04/21/2009 | US7521445 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands |
| 04/16/2009 | WO2009046897A1 Chemical synthesis of i-124beta cit iodine-124 [2-beta-carbomethoxy-3beta- (4. -iodophenyl) -tropane] for pet investigations and for radiotherapy |
| 04/16/2009 | US20090099143 Tetrahydro-indazole cannabinoid modulators |
| 04/15/2009 | CN101407514A Method for producing tiotropium salts, tiotropium salts and pharmaceutical formulations, containing the same |
| 04/09/2009 | WO2009043793A1 Method for producing (1r,5s) anhydroecgonine ester salts |
| 04/09/2009 | US20090093451 IL-8 Receptor Antagonists |
| 04/09/2009 | DE102007046887A1 Verfahren zur Herstellung von (1R,5S)-Anhydroecgoninestersalzen Process for the preparation of (1R, 5S) -Anhydroecgoninestersalzen |
| 04/09/2009 | CA2700932A1 Process for the manufacture of salts of (1r,5s)-anhydroecgonin ester |
| 04/08/2009 | EP2044027A2 Fused bicyclic compounds interacting with the histamine h4 receptor |
| 04/08/2009 | EP1448566B3 Chemokine receptor antagonists and methods of use thereof |
| 04/08/2009 | EP1212299B1 Substituted piperidine compounds useful as modulators of chemokine receptor activity |
| 04/08/2009 | CN101405287A Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 04/08/2009 | CN101405265A Amido compounds and their use as pharmaceuticals |
| 04/07/2009 | US7514583 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes, and parkinson's disease |
| 04/02/2009 | WO2009041567A1 Diaryl ketimine derivative having antagonistic activity on melanin-concentrating hormone receptor |
| 04/02/2009 | WO2008145504A3 Method for producing scopine esters |
| 04/01/2009 | CN101400677A Compounds |
| 04/01/2009 | CN101400676A Tropane prodrugs with central nervous system activity |