Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
12/2009
12/23/2009WO2009153178A2 Aryl ketone as mri
12/23/2009EP1720859B1 Chemokine receptor antagonists
12/23/2009CN101611027A Indol-2-yl-piperazin-1-yl-methanone derivatives
12/23/2009CA2728373A1 Aryl ketone as mri
12/17/2009WO2008117229A4 Muscarinic receptor antagonists
12/16/2009CN101602741A Substituted n-arylsulfonylheterocyclic amines as gamma-secretase inhibitors
12/16/2009CN100569771C Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
12/16/2009CN100569769C Compounds with antibacterial activity
12/15/2009CA2481078C Method and compositions for the synthesis of bch-189 and related compounds
12/09/2009CN100567293C N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists
12/08/2009US7629337 Chemokine receptor binding heterocyclic compounds
12/03/2009WO2009145323A1 Method for oxidizing alcohol by using polycyclic compound
12/03/2009WO2009122034A3 Novel dhsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof
12/03/2009US20090298867 Tricyclic delta-opioid modulators
12/03/2009US20090297446 Labeled iodinated tropane formulation
12/02/2009EP1663220B1 Novel process for the preparation of pleuromutilin derivatives
12/02/2009CN101595100A Heterocyclic-substituted piperidine as ORL-1 ligands
12/01/2009US7626031 5-[(1-Ethylpiperidin-4-yl)amino]-3-[(3-fluorophenyl)(1H-imidazol-2-yl)methylidene]-1,3-dihydro-2H-indol-2-one; antiproliferative agents; modulating cell differentiation,migration, and chemoinvasion; endothelial growth factor-modulated diseases; antiarthritic agents; graft versus host diseases
11/2009
11/25/2009EP2123650A1 Novel form of tiotropium bromide and process for preparation thereof
11/25/2009EP2121676A1 Preperation and utility of ccr5 inhibitors
11/24/2009US7621300 Metering method for particulate material
11/24/2009CA2475712C Nicotinamide derivatives useful as pde4 inhibitors
11/18/2009EP2118089A1 Indol-2-yl-piperazin-1-yl-methanone derivatives
11/18/2009EP1713800B1 Method for producing a 2-(ethoxymethyl)tropane derivative
11/18/2009EP1184379B1 Chromene compound
11/12/2009US20090281072 Diaminopyrimidinecarboxamide Derivative
11/11/2009EP1960396B1 Carbamate compounds as 5-ht4 receptor agonists
11/11/2009EP1594868B1 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
11/11/2009CN101574552A Inhalation kit comprising inhalable powder of tiotropium
11/10/2009US7615555 Piperidine derivatives as modulators of chemokine receptor CCR5
11/10/2009CA2481482C Tropane derivatives as ccr5 modulators
11/05/2009US20090275604 M3 Muscarinic Acetylcholine Receptor Antagonists
11/04/2009EP1499311B1 Substituted benzazoles and use thereof as raf kinase inhibitors
11/04/2009CN101573354A Substituted isoquinolines and their use as Rho-kinase inhibitors
10/2009
10/29/2009US20090270449 Aminophenyl derivatives as selective androgen receptor modulators
10/27/2009US7608714 Production of dolasetron
10/27/2009CA2511664C 4',4''-substituted 3.alpha.-(diphenylmethoxy)tropane analogs for treatment of mental disorders
10/21/2009CN101563344A Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
10/21/2009CN101563343A Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
10/21/2009CN100551924C 8-aza-bicyclo (3.2.1) octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
10/20/2009US7605170 8-azabicyclo[3.2.1]octane derivatives
10/20/2009CA2385130C Novel spiroheterocyclic compounds useful as reversible inhibitors of cysteine proteases
10/15/2009US20090258881 Aryl-substituted polycyclic amines, method for the production thereof, and use thereof as a medicament
10/14/2009CN100549010C Method for producing tiotropium salts, tiotropium salts and pharmaceutical formulations containing the same
10/14/2009CN100548387C Improved radiometal complex compositions
10/08/2009CA2718488A1 Novel dhsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof
10/01/2009WO2009118254A1 Aminopiperidinyl derivatives and uses thereof
10/01/2009WO2009117808A1 Inhibitors of histone deacetylase
10/01/2009US20090247515 11 Beta-HSD1 Modulators
10/01/2009US20090247509 for treating central nervous system disorders such as psychological disorders, drug dependence and abuse, dyskinesia, dementia, anxiety disorders, sleep disorders and mood disorders
10/01/2009CA2712468A1 Aminopiperidinyl derivatives and uses thereof
09/2009
09/24/2009US20090239873 Phenyl-piperazine derivatives as modulators of muscarinic receptors
09/23/2009EP2102157A1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives
09/23/2009CN101541792A Azaadamantane derivatives and methods of use
09/22/2009US7592358 Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds
09/22/2009US7592355 Quinolinone-carboxamide compounds as 5-HT, receptor agonists
09/22/2009CA2333086C Cocaine receptor binding ligands
09/17/2009WO2009114173A1 Azabicyclo [3. 2. i] octyl derivatives as 11 beta-hsdl modulators
09/17/2009US20090234125 Amorphous retapamulin and processes for preparation thereof
09/17/2009CA2718038A1 Azabicyclo [3.2.1] octyl derivatives as 11 beta-hsdl modulators
09/16/2009EP2099795A2 Azaadamantane derivatives and their uses as nicotinic acetylcholine receptors ligands
09/16/2009EP1487807B1 Cyano-pyrrolidines as DPP-IV inhibitors
09/15/2009US7589207 Chemokine receptors; inhibition of HIV replication; acquired immune deficiency syndrome (AIDS); cis N-(4-{2-[3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-4-phenylcyclohexyl)-1H-pyrazole-4-carboxamide
09/15/2009US7589204 Indane compounds as CCR5 antagonists
09/11/2009WO2009110510A1 Alkylaminopyridine derivative
09/11/2009WO2009109477A1 2-aminoquinolines
09/11/2009CA2716122A1 2-aminoquinolines
09/11/2009CA2714617A1 Alkylaminopyridine derivative
09/08/2009US7585877 Aminophenyl derivatives as selective androgen receptor modulators
09/02/2009EP1891064B1 N-amide derivatives of 8-azabicyclo[3.2.1]oct-3-yl as ccr1 antagonists
09/02/2009EP1807422B1 5-ht4 receptor agonist compounds
08/2009
08/27/2009WO2007003934A3 17beta-hydr0xyster0id dehydrogenase type 3 (17beta-hsd3 ) inhibitors
08/27/2009US20090215821 N-Substituted Azacycles
08/26/2009EP1590338B1 Modulators of melanocortin receptor
08/26/2009CN100532382C Novel method for producing tiotropium salts
08/25/2009US7579471 Tropane derivatives useful in therapy
08/25/2009US7579361 Muscle relaxants; respiratory system disorders; asthma; COPD; emphysema; bronchitis
08/20/2009WO2009103032A1 Pyrimidine-2-amine compounds and their use as inhibitors of jak kinases
08/20/2009WO2009101917A1 Bicycloamine derivative
08/20/2009US20090208415 Tropane compounds
08/20/2009CA2715658A1 Pyrimidine-2-amine compounds and their use as inhibitors of jak kinases
08/20/2009CA2714591A1 Bicycloamine derivative
08/19/2009EP2090571A1 Pyrimidine derivates, medicaments comprising them, their use and process of their preparation
08/19/2009CN101511818A N-pyridylpiperidine compound, method for producing the same, and pest control agent
08/18/2009US7576100 Muscarinic agonists
08/18/2009US7576097 Crystalline form of maraviroc
08/18/2009US7576096 Muscarinic acetylcholine receptor antagonists
08/18/2009US7576088 Benzodioxole derivatives
08/18/2009US7576078 Tetrahydroquinoline analogues as muscarinic agonists
08/18/2009US7576074 Receptor-type kinase modulators and methods of use
08/13/2009WO2009098209A1 Novel 9-aza-bicyclo[3.3.1]non-3-yloxy chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
08/13/2009WO2009098208A1 Novel phenylethynyl derivatives of 8-aza-bicyclo[3.2.1]octane and their use as monoamine neurotransmitter re-uptake inhibitors
08/12/2009EP2086958A2 Substituted-quinoxaline-type-piperidine compounds and the uses thereof
08/12/2009EP1343760B1 Muscarinic antagonists
08/06/2009WO2009095634A1 Amorphous forms of retapamulin
08/06/2009US20090198051 Chemical intermediates for sulfiding under mild conditions forming ring compounds for use as marine alkaloids; connecting reaction of 4 components, transforming c22-tert-butyltriphenylsilyl to acety group, cyclization, hydroxy group to methanesulonyl group, reduction of amide, dehydration,Heck reaction
08/06/2009US20090197965 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes, and parkinson's disease
08/06/2009US20090197862 2-aminopyridine kinase inhibitors
08/05/2009EP2085396A2 Novel crystalline forms of tiotropium bromide
08/05/2009EP2084157A1 Crystalline form of tiotropium bromide and urea
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