| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
|---|
| 04/17/2008 | US20080090828 insecticides for soil-borne insects, such as termites and white grubs; less costly and safer to use on crops; N-{4-[(4-{bis[4-(trifluoromethyl)phenyl]methylene}piperidyl)methyl]phenyl}ethoxycarboxamide, N-oxide |
| 04/16/2008 | EP1910354A2 Novel method for producing tiotropium salts |
| 04/16/2008 | EP1910353A1 Tricyclic delta- opioid modulators |
| 04/16/2008 | EP1567526B1 Carbamic acid esters with anticholinergic action |
| 04/16/2008 | CN101163701A Quinolinone compounds as 5-ht4 receptor agonists |
| 04/15/2008 | US7358244 Azabicycloalkane compounds |
| 04/10/2008 | WO2008003702A3 Fused bicyclic compounds interacting with the histamine h4 receptor |
| 04/09/2008 | CN101160307A Benzoxazole carboxamides for treating cinv and ibs-d |
| 04/03/2008 | WO2008019363A3 2-alkylbenzoxazole carboxamides as 5ht3 modulators |
| 04/02/2008 | EP1904492A1 Method for obtaining a pharmaceutically active compound, synthesis intermediates thereof and methods for obtaining them |
| 04/01/2008 | US7351704 Indazole-carboxamide compounds as 5-HT4 receptor agonists |
| 03/27/2008 | WO2008008376A8 Scopine salts and their use in processes for the preparation of n-demethyl-tiotropium and tiotropium bromide |
| 03/27/2008 | US20080076755 4-(Adamantane-1-carbonylamino)-3-oxo-2-aza-bicyclo[2.2.2]octane; 5-(Adamantane-1-carbonylamino)-10-oxo-9-aza-bicyclo[3.3.2]decane for treating autoimmune diseases, vascular disorders, viral infection or replication, asthma, osteoporosis, tumor growth, rheumatoid arthritis, organ transplant rejection |
| 03/26/2008 | EP1902053A2 Benzoimidazolone-carboxamide compounds as 5-ht4 receptor agonists |
| 03/26/2008 | CN101151264A Crystalline form of a quinolinone-carboxamide compound |
| 03/25/2008 | US7348343 N-(N-heteroaryl)1-pyridyl- or -pyrimidyl-hydropyridine-4-carboxamides; e.g., 3'-Chloro-3,6-dihydro-2H-[1,2']bipyridinyl-4-carboxylic acid (6-trifluoromethyl-pyridin-3-yl)-amide and 1-pyrimidin-2-yl-1,2,3,6-tetrahydro-pyridine-4-carboxylic acid (6-trifluoromethyl-pyridin-3-yl)-amide |
| 03/25/2008 | US7348327 (2S)-4,4-difluoro-1-(2-{[1-(2-pyrazinyl)piperidin-4-yl]amino}acetyl)-2-pyrrolidine carbonitrile; enzyme inhibitors; diabetes |
| 03/20/2008 | US20080070948 Including indanones, indolinones and benzoxazolinones containing a piperidine ring, e.g., 1-[3-(4-(Hydroxymethyl)piperidin-1-yl)propyl]-1,3-dihydrobenzoimidazol-2-one; particularly for the M1 and/or M4 receptor subtypes; increase acetylcholine signaling or effect in the brain |
| 03/20/2008 | US20080070880 Specific glucocorticosteroid compound having anti-inflammatory activity |
| 03/19/2008 | EP1532132B1 Novel benzodioxoles |
| 03/18/2008 | US7345056 Bridged N-cyclic sulfonamido inhibitors of gamma secretase |
| 03/18/2008 | US7345037 ipratropium/flutropium/tiotropium derivatives; anticholinergic agent; linked at NO or NO2 group, or group which stimulates endogenous production of NO; beneficial therapeutic effects; asthma, respiratory disorder, cystic fibrosis; synergistic with NO release agent or substrate for nitric oxide synthase |
| 03/12/2008 | EP1896468A1 3 -aryloxy- 8 -aza-bicyclo [3.2.1.] oct- 6- ene derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 03/12/2008 | EP1896467A2 Tricyclic opioid modulators |
| 03/12/2008 | EP1896026A2 Process for preparing tiotropium salts, tiotropium salts as such and pharmaceutical compositions thereof |
| 03/12/2008 | CN101142213A (+) - and (-) -8-alkyl-3-(trifluoralkylsulfonyloxy)-8-azabicycl (3.2.1.)oct-2-ene |
| 03/12/2008 | CN101139346A Benzimidazole-derivatives as factor Xa inhibitors |
| 03/12/2008 | CN101139340A N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines |
| 03/11/2008 | US7342027 1-phenylpiperidin-3-one derivatives and processes for the preparation thereof |
| 03/06/2008 | WO2008026658A1 N-pyridylpiperidine compound, method for producing the same, and pest control agent |
| 03/06/2008 | US20080057074 Nitrogenous Heterocylic Derivative and Medicine Containing the Same as an Active Ingredient |
| 03/06/2008 | CA2661741A1 N-pyridylpiperidine compound, method for producing the same, and pest control agent |
| 03/05/2008 | EP1893610A2 Alpha-(aryl-or heteroaryl-methyl)-beta piperidino propanamide compounds as orl1-receptor antagonists |
| 03/05/2008 | EP1893212A2 Multicyclic compounds and methods of their use |
| 02/28/2008 | US20080051407 These compounds lack a 1,4-bridging group as found in the ecteinascidins; and, have at the C-1 position a substituent selected from an amino or hydroxy group, optionally protected or derivatized; anticarcinogenic agents |
| 02/28/2008 | US20080050795 Mixture Of At Least Two Different Antibodies Specific For Predetermined Antigens And Use Of The Mixture |
| 02/28/2008 | CA2661401A1 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
| 02/27/2008 | EP1891065A1 Novel mchr1 antagonists and their use for the treatment of mchr1 mediated conditions and disorders |
| 02/27/2008 | EP1891064A1 N-amide derivatives of 8-azabicyclo[3.2.1]oct-3-yl as ccr1 antagonists |
| 02/27/2008 | EP1891048A1 Pyrazole-substituted benzimidazole derivatives for use in the treatment of cancer and autoimmune disorders |
| 02/26/2008 | CA2291094C 2-oxoimidazole derivative |
| 02/21/2008 | US20080045569 Cyclic Amine Compound and Pest Control Agent |
| 02/21/2008 | US20080045522 Omega-aminoalkylamides of r-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells |
| 02/20/2008 | EP1888064A1 Benztropinamine analogs as dopamine uptake inhibitors |
| 02/19/2008 | US7332509 Used for controlling animal pests, in particular arthropods, such as insects and acarids, and helminths |
| 02/14/2008 | CA2660349A1 2-aminobenzoxazole carboxamides as 5ht3 modulators |
| 02/13/2008 | CN101124222A Tetrahydroquinoline analogues as muscarinic agonists |
| 02/13/2008 | CN101121713A Method for preparing 2beta-carbonyl-3beta-(4-chlorobenzo)-8-(2-fluoro[18F]ethyl)demethyltropane by one-step method |
| 02/13/2008 | CN100368410C Micronized crystalline tiotropium bromide |
| 02/13/2008 | CN100368409C Novel 8-aza-bicyclo not 3.2.1|octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 02/12/2008 | CA2427583C Inhalable formulation of a solution containing a tiotropium salt |
| 02/06/2008 | CN101119993A Aminophenyl derivatives as selective androgen receptor modulators |
| 02/06/2008 | CN101119992A Tricyclic delta-opioid modulators |
| 01/31/2008 | US20080027094 Tropane Compounds and Pharmaceutical Compositions Comprising the Same as an Active Ingredient |
| 01/30/2008 | EP1881980A2 Novel crystalline forms of tiotropium bromide |
| 01/30/2008 | CN101115751A Tricyclic delta-opioid modulators |
| 01/29/2008 | CA2436540C Pharmaceutical compositions based on anticholinergics and corticosteroids |
| 01/24/2008 | US20080021231 Novel compounds |
| 01/24/2008 | US20080021043 Piperidines and Related Compounds for Treatment of Alzheimer's Disease |
| 01/24/2008 | US20080016674 Method And Installation Means For Installing An Electrical Machine |
| 01/23/2008 | EP1879888A2 Crystalline forms of tiotropium bromide |
| 01/22/2008 | US7321042 Process for preparing N-substituted 3-β-aminonortropanes |
| 01/22/2008 | US7321039 Industrial process for preparing tropenol |
| 01/17/2008 | WO2008008376A2 Scopine salts and their use in processes for the preparation of n-demethyl-tiotropium and tiotropium bromide |
| 01/17/2008 | US20080015360 2,3-Dimethyl-1-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-imidazol-3-ium chloride; intermediate for preparing androstane-type glucocorticoid receptor agonists |
| 01/17/2008 | CA2658165A1 Process for the preparation of tiotropium bromide |
| 01/10/2008 | WO2007116313A3 Pyrrolidine derivatives as modulators of chemokine ccr5 receptors |
| 01/10/2008 | WO2007104652A3 Non-peptidic renin inhibitors nitroderivatives |
| 01/10/2008 | US20080009520 Benzimidazolidinone derivatives as muscarinic agents |
| 01/10/2008 | US20080009489 Androgen receptor modulators and method of treating disease using the same |
| 01/10/2008 | CA2657702A1 Quinazolines and related heterocyclic comp0unds, and their therapeutic use |
| 01/09/2008 | EP1874767A2 Production of dolasetron |
| 01/09/2008 | EP1874766A2 Crystalline form of a quinolinone-carboxamide compound |
| 01/09/2008 | EP1434604A4 4-haloethenylphenyl tropane:serotonin transporter imaging agents |
| 01/02/2008 | EP1871772A1 Quinolinone compounds as 5-ht4 receptor agonists |
| 01/02/2008 | EP1416933B1 Substituted piperidines as modulators of the melanocortin receptor |
| 01/02/2008 | CN101099286A Method and installation means for installing an electrical machine |
| 01/01/2008 | US7314870 Compounds, their preparation and use |
| 12/27/2007 | US20070299260 Method for Preparing Hexahydro-8-Hydroxy-2, 6-Methano-2H-Chinolizin-3 (4H) -One Esters |
| 12/27/2007 | US20070299039 Substituted benz-azoles and methods of their use as inhibitors of Raf kinase |
| 12/26/2007 | EP1869035A2 Novel forms of tiotropium bromide and processes for preparation thereof |
| 12/26/2007 | EP1869034A1 (+) - and (-) -8-alkyl-3-(trifluoralkylsulfonyloxy)-8-azabicycl (3.2.1.)oct-2-ene |
| 12/26/2007 | EP1869033A1 Novel enantiomers and their use as monoamine neurotransmitter re-uptake inhibitors |
| 12/21/2007 | WO2007143847A1 Spirotropane compounds |
| 12/21/2007 | CA2655203A1 Spirotropane compounds |
| 12/20/2007 | US20070293498 used for the treatment of cachexia and other weight loss disorders, such as those resulting from cancer, HIV, old age and anorexia nervosa |
| 12/19/2007 | EP1664031B1 Adamantane and azabicyclo-octane and nonane derivatives process of their preparation and their use as dpp-iv inhibitors |
| 12/19/2007 | CN100355753C Tropan derivatives useful in therapy, method for obtaining thereof and intermediate compounds |
| 12/13/2007 | WO2007141504A1 Fused thiophene derivatives as kinase inhibitors |
| 12/12/2007 | EP1863490A2 Muscarinic modulators |
| 12/11/2007 | US7307087 Antidepressants; analgesics; antiinflammatory agents; side effect reduction |
| 12/11/2007 | US7307075 Tetrahydroquinoline analogues as muscarinic agonists |
| 12/06/2007 | US20070281970 minimal side effects, selectivity, potency, pharmacokinetics, duration of action; CNS disorders like cognitive, behavioral, mood, autonomic functions; 1-isopropyl-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid {(1S,3R,5R)-8-[3-acetylamino-2-hydroxypropyl]-8-azabicyclo[3.2.1]oct-3-yl}amide |
| 12/05/2007 | EP1862457A2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| 12/05/2007 | EP1861397A2 Production of dolasetron |
| 12/05/2007 | EP1860943A2 Novel method |
| 12/05/2007 | EP1399420B1 Pyrrolidines as dipeptidyl peptidase inhibitors |
| 11/29/2007 | CA2647830A1 Central nervous system active fused bicycloheterocycle substituted azabicyclic alkane derivatives |
| 11/28/2007 | CN101080406A Indazole-carboxamide compounds |
| 11/27/2007 | US7300946 For use in controlling insects; controlling tobacco budworm |