| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
|---|
| 09/28/2010 | CA2383524C Thiazolyl alkynyl compounds and methods of use thereof |
| 09/23/2010 | WO2010106269A2 Derivatives of n-[(2-aza-bicyclo[2.1.1]hex-1-yl)-aryl-methyl]-heterobenzamide, preparation thereof and application of same in therapeutics |
| 09/23/2010 | CA2755526A1 Derivatives of n-[(2-aza-bicyclo[2.1.1]hex-1-yl)-aryl-methyl]-heterobenzamide, preparation thereof and application of same in therapeutics |
| 09/22/2010 | EP2076506B1 Heterocyclic-substituted piperidines as orl-1 ligands |
| 09/22/2010 | CN101838266A Citric acid tropisetron raw material medicine and preparation technology of raw material medicine and injection liquid |
| 09/21/2010 | CA2451573C Technical process for the manufacture of tropenol |
| 09/21/2010 | CA2440559C Novel non-imidazole compounds |
| 09/21/2010 | CA2405002C Antitumoral analogs of et-743 |
| 09/16/2010 | WO2010048526A3 Modulators of cystic fibrosis transmembrane conductance regulator |
| 09/16/2010 | US20100234395 Ureide derivative and pharmaceutical application thereof |
| 09/16/2010 | US20100234392 4-sulfonylpiperidine derivatives |
| 09/16/2010 | US20100234354 Pyridazinone derivatives |
| 09/15/2010 | EP2228364A1 Acylsulfonamides as inhibitors of steroid sulfatase |
| 09/10/2010 | WO2010101538A2 New crystal forms |
| 09/09/2010 | US20100227883 Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 09/08/2010 | CN101824033A Stereoisomeric compounds and methods for the treatment of gastrointestinal and central nervous system disorders |
| 09/07/2010 | US7790719 used for the treatment of cachexia and other weight loss disorders, such as those resulting from cancer, HIV, old age and anorexia nervosa |
| 09/02/2010 | US20100221181 Method of differentially diagnosing different types of dementia |
| 09/01/2010 | EP1874766B1 Crystalline form of a quinolinone-carboxamide compound |
| 09/01/2010 | CN101821265A Substituted bicyclic piperidinyl-and piperazinyl- sulfonamides useful to inhibit 11ss-hydroxysteroid dehydrogenase type-1 |
| 09/01/2010 | CN101817815A Compounds with antibacterial activity |
| 08/26/2010 | US20100217002 Novel chromen-2-one derivatives |
| 08/26/2010 | US20100216988 Regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles |
| 08/26/2010 | US20100216840 Benzimidazolidinone derivatives as muscarinic agents |
| 08/26/2010 | US20100216726 Substituted-Quinoxaline-Type Piperidine Compounds and the Uses Thereof |
| 08/25/2010 | EP2221306A1 Method for producing 2-azaadamantane |
| 08/25/2010 | EP2220068A1 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors |
| 08/25/2010 | EP2220048A2 Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
| 08/24/2010 | US7781455 (4R)-3-(2-{[8-(2-Pyrimidinyl)-8-azabicyclo[3.2.1]oct-3-yl]exo-amino}acetyl)thiazolidine-4-carbonitrile; dipeptidylpeptidase-IV enzyme inhibitors; diabetes |
| 08/24/2010 | CA2423103C N-acylsulfonamide apoptosis promoters |
| 08/19/2010 | WO2010093706A2 Chemically programmed vaccination |
| 08/19/2010 | WO2009122034A8 Novel hsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof |
| 08/19/2010 | US20100210838 Fluoropyrrolidines having dipeptidyl peptidase enzyme inhibitory activity |
| 08/18/2010 | EP2217596A2 Bicyclic heterocycle derivatives and their use as modulators of the activity of gpr119 |
| 08/18/2010 | EP1737842B1 Selected cgrp antagonists, method for producing the same and the use thereof as drugs |
| 08/18/2010 | EP1682543B1 Methods for the production of novel tiotropium salts |
| 08/17/2010 | US7776888 such as 3-[2-(2-methoxy-ethoxymethyl)-6-trifluoromethyl-pyridine-3-carbonyl]-1,5-dimethyl-8-oxa-bicyclo[3.2.1]oct-6-ene-2,4-dione, used for controlling undesired plant growth or weeds |
| 08/17/2010 | US7776885 Benzimidazolone compounds having 5-HT4 receptor agonistic activity |
| 08/12/2010 | US20100204264 Polymorphic form of granisetron base, methods for obtaining it and formulation containing it |
| 08/11/2010 | CN101801378A Novel combination of therapeutic agents |
| 08/11/2010 | CN101798257A Automatic synthesis method of methylation reagent [11C] CH3Br |
| 08/10/2010 | US7772252 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands |
| 08/05/2010 | WO2010086612A1 Process for preparing enantiomerically enriched alkaloids |
| 08/05/2010 | US20100197922 Azabicycloalkane compounds |
| 08/05/2010 | US20100196368 Substituted benz-azoles and methods of their use as inhibitors of raf kinase |
| 08/05/2010 | CA2751285A1 Bicyclic amide derivatives for enhancing glutamatergic synaptic responses |
| 08/04/2010 | EP2212320A1 Chemical synthesis of i-124beta cit iodine-124 [2-beta-carbomethoxy-3beta- (4. -iodophenyl) -tropane] for pet investigations and for radiotherapy |
| 08/04/2010 | EP2212319A1 Labeled iodinated tropane formulation |
| 08/03/2010 | US7767814 2-benzyl-3-[4a-(3-hydroxy-phenyl)-10a-methyl-3,4,4a,5,10,10a-hexahydro-1H-benzo[g]isoquinolin-2-yl]-propionic acid, used for prevention or treatment of gastrointestinal disorders, obesity, pain and reducing side effects associated with an opioid such as constipation, nausea and vomiting |
| 07/29/2010 | WO2010085684A1 Compositions and methods for inhibition of the jak pathway |
| 07/29/2010 | US20100191475 Method for identification and functional characterization of agents which modulate ion channel activity |
| 07/29/2010 | US20100190821 3,8-substituted 8-aza-bicyclo[3.2.1]octane derivatives and their use as monomine neurotransmitter re-uptake inhibitors |
| 07/29/2010 | CA2749217A1 Compositions and methods for inhibition of the jak pathway |
| 07/28/2010 | CN101790529A 8-azabicyclo[3.2.1]octyl-2-hydroxybenzamide compounds as mu opioid receptor antagonists |
| 07/28/2010 | CN101787021A High-purified tropisetron hydrochloride compound |
| 07/27/2010 | US7763747 Bis- and tris-dihydroxyaryl compounds and their methylenedioxy analogs; Alzheimer's disease; diabetes; A beta amyloidosis |
| 07/27/2010 | US7763637 Gastrointestinal disorders; selectivity, potency, pharmacokinetics, duration of action; minimal side effects |
| 07/27/2010 | CA2373559C Serotonin transport inhibitors |
| 07/22/2010 | US20100184987 Preparation of Retapamulin via its Pleuromutilin-thiol precursor |
| 07/21/2010 | EP1610789B1 Bicyclic piperidine derivatives as melanocortin-4 receptor agonists |
| 07/15/2010 | WO2010080474A1 Carbazole and carboline kinase inhibitors |
| 07/15/2010 | US20100179164 2,4-pyrimidinediamine compounds for treatment of inflammatory disorders |
| 07/14/2010 | EP2206712A1 "Alkaloid aminoester derivatives and medicinal composition thereof" |
| 07/14/2010 | EP2205597A1 Method for producing (1r,5s) anhydroecgonine ester salts |
| 07/13/2010 | US7754886 N-acylsulfonamide apoptosis promoters |
| 07/08/2010 | US20100173935 Muscarinic Receptor Agonists that are Effective in the Treatment of Pain, Alzheimer's Disease and Schizophrenia |
| 07/07/2010 | EP2204368A1 4-sulfonylpiperidine derivatives |
| 07/07/2010 | CN101768158A Tiotropium bromide anhydride and preparation method thereof |
| 07/01/2010 | WO2010075273A1 Bicyclic heterocycle derivatives and methods of use thereof |
| 07/01/2010 | WO2010074387A1 Aza-bicyclo[2.2.1] heptene derivatives, preparation method thereof, and method for preparing oseltamivir intermediates using the same |
| 07/01/2010 | WO2010072338A1 Alkaloid aminoester derivatives and medicinal composition thereof |
| 07/01/2010 | WO2010046445A3 Urea derivatives of substituted nortropanes, medicaments containing such compounds and their use |
| 07/01/2010 | US20100168083 Adamantane derivatives for the treatment of the metabolic syndrome |
| 07/01/2010 | CA2748100A1 Alkaloid aminoester derivatives and medicinal composition thereof |
| 06/30/2010 | CN101765599A Tropane derivatives useful as pesticides |
| 06/30/2010 | CN101759696A Improvement of nortropine synthesizing process |
| 06/29/2010 | US7745628 Method for obtaining a pharmaceutically active compound, synthesis intermediates thereof and methods for obtaining them |
| 06/24/2010 | US20100160328 New compounds useful for dpp-iv enzyme inhibition |
| 06/22/2010 | CA2389553C Heteroaryl-diazabicycloalkanes |
| 06/17/2010 | WO2010066380A1 Triaryl-sulphonium compounds, kit and methods for labeling positron emitting isotopes |
| 06/17/2010 | US20100152167 Pyrimidine derivatives |
| 06/17/2010 | US20100152148 Novel compounds |
| 06/17/2010 | CA2748691A1 Triaryl-sulphonium compounds, kit and methods for labeling positron emitting isotopes |
| 06/16/2010 | EP2195315A1 Substituted bicyclic piperidinyl-and piperazinyl- sulfonamides useful to inhibit 11 -hydroxysteroid dehydrogenase type-1 |
| 06/16/2010 | EP2195314A1 Disubstituted alkyl-8-azabicyclo [3.2.1.]octane compounds as mu opioid receptor antagonists |
| 06/16/2010 | EP2195313A1 Heteroarylalkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists |
| 06/16/2010 | CN101743245A Process for preparing an intermediate to mu opioid receptor antagonists |
| 06/16/2010 | CN101099286B Method and installation means for installing an electrical machine |
| 06/15/2010 | CA2383340C Thienoisoxazolyl- and thienylpyrrazolyl-phenoxy substituted propyl derivatives useful as d4 antagonists |
| 06/10/2010 | WO2010031517A8 Radioactively marked cyclopropane derivatives of dat affine tropanes |
| 06/09/2010 | EP2194053A1 Stereoisomeric compounds and methods for the treatment of gastrointestinal and central nervous system disorders |
| 06/09/2010 | CN1982309B Industrial synthesis method for producing tropenol |
| 06/09/2010 | CN1880319B Tropane derivatives as CCR5 modulators |
| 06/09/2010 | CN1852712B Dual NK1/NK3 antagonists for treating schizophrenia |
| 06/08/2010 | US7732456 such as 4-benzyloxy-1-{4-[2-(dimethylamino)ethoxy]phenyl}-1H-pyridin-2-one, that as antagonists to melanin concentrating hormone receptors, used for treating cardiovascular, nervous system, metabolic, reproductive system, respiratory system and gatrointestinal disorders |
| 06/08/2010 | US7732441 Azabicycloalkane compounds |
| 06/03/2010 | WO2010028213A3 N-sulfonamido polycyclic pyrazolyl compounds |
| 06/03/2010 | WO2010014257A3 Tetrahydropyridinyl and dihydropyrrolyl compounds and the use thereof |
| 06/02/2010 | EP2190831A2 Method for the production of 1,3-dioxolane-2-ones and carboxylic acid esters by means of transacylation in basic reaction conditions |
| 06/02/2010 | EP2190824A1 Naphthylpyrimidine, naphthylpyrazine and naphthylpyridazine analogs and their use as agonists of the wnt-beta-catenin cellular messaging system |