| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 04/26/2012 | WO2012053606A1 Arylaminoheterocyclic carboxamide compound |
| 04/25/2012 | CN102428083A 色原烯-2-酮衍生物及其作为单胺神经递质再摄取抑制剂的用途 Color-2-one derivatives and original as monoamine neurotransmitter reuptake inhibitor use |
| 04/24/2012 | US8163957 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes and parkinson's disease |
| 04/24/2012 | US8163920 Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
| 04/24/2012 | US8163771 11 β-HSD1 modulators |
| 04/19/2012 | WO2012050315A2 Azetidinium salt as fp-cit precursor, method for selectively preparing same, and fp-cit synthesis |
| 04/18/2012 | EP2018379B1 Scopine salts and their use in processes for the preparation of n-demethyl-tiotropium and tiotropium bromide |
| 04/12/2012 | US20120088789 Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 04/10/2012 | US8153653 Amido-tropane derivatives |
| 04/05/2012 | WO2012043791A1 1,2,4-triazolone derivative |
| 04/05/2012 | CA2811192A1 1,2,4-triazolone derivative |
| 04/04/2012 | EP2435426A1 BENZOXAZEPINES AS INHIBITORS OF PI3K/m TOR AND METHODS OF THEIR USE AND MANUFACTURE |
| 04/04/2012 | EP0831941B1 Iodinated neuroprobes for mapping monoamine reuptake sites |
| 03/28/2012 | EP2433937A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof |
| 03/28/2012 | EP2433936A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof |
| 03/28/2012 | EP2433935A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof |
| 03/28/2012 | EP2432781A1 Salts of tiotropium with 10-camphorsulfonic acid |
| 03/28/2012 | CN102391251A Chemokine receptor antagonists |
| 03/27/2012 | CA2554642C Bicyclic carbonyl amino derivatives as chemokine receptor antagonists |
| 03/22/2012 | WO2012036276A1 Glycine transporter inhibitory substance |
| 03/22/2012 | WO2012035023A1 Triazine-oxadiazoles |
| 03/22/2012 | CA2812081A1 Triazine-oxadiazoles |
| 03/21/2012 | EP2431368A1 CNS active fused bicycloheterocycle substituted azabicyclic alkane derivatives |
| 03/21/2012 | EP2430020A1 Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 03/21/2012 | EP2050745B1 N-pyridylpiperidine compound, method for producing the same, and pest control agent |
| 03/15/2012 | WO2011095800A3 Analytical methods |
| 03/15/2012 | US20120065225 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives and uses thereof |
| 03/14/2012 | CN102372756A Specific glucocorticosteroid compound having anti-inflammatory activity |
| 03/07/2012 | EP2424860A1 Heteroarylthiomethyl pyridine derivative |
| 03/07/2012 | CN102369201A Bicyclic amide derivatives for the treatment of respiratory depression |
| 03/07/2012 | CN102367252A Tropisetron hydrochloride compound |
| 03/07/2012 | CN102367251A More stable tropisetron compound and pharmaceutical composition thereof |
| 03/01/2012 | WO2012026906A1 New tiotropium bromide crystal and its production method |
| 03/01/2012 | WO2012025811A1 Indolylpyrimidines as modulators of gpr119 |
| 03/01/2012 | US20120053348 Method for producing 2-azaadamantane compound from bicyclocarbamate compound |
| 03/01/2012 | US20120053164 Cyclic pyrimidin-4-carboxamides as ccr2 receptor antagonists for treatment of inflammation, asthma and copd |
| 02/29/2012 | CN101759696B Improvement of nortropine synthesizing process |
| 02/21/2012 | US8119627 Heterocyclic compounds as inhibitors of 17beta-HSD3 |
| 02/21/2012 | US8119563 N-substituted azacycles |
| 02/21/2012 | CA2248800C Nitrosated and nitrosylated compounds and compositions and their use for treating respiratory disorders |
| 02/16/2012 | US20120041022 Process for preparing enantiomerically enriched alkaloids |
| 02/16/2012 | US20120040975 Bridged bicyclic heterocycle derivatives and methods of use thereof |
| 02/15/2012 | CN102356075A Compositions and methods for inhibition of the jak pathway |
| 02/15/2012 | CN102351857A Tropiseiron hydrochloride compound |
| 02/15/2012 | CN102351856A Purification method of alpha-tropine |
| 02/09/2012 | WO2012016993A1 Derivatives of pyrazolophenyl-benzenesulfonamide compounds and use thereof as antitumor agents |
| 02/08/2012 | EP2414334A1 Bridged bicyclic heterocycle derivatives and methods of use thereof |
| 02/07/2012 | US8110586 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 02/02/2012 | US20120028970 Heteroarylthiomethyl pyridine derivative |
| 01/31/2012 | CA2463989C Pyrimidine derivatives, pharmaceutical compositions containing these compounds, the use thereof and process for the preparation thereof |
| 01/26/2012 | US20120020881 Triaryl-sulphonium compounds, kit and methods for labeling positron emitting isotopes |
| 01/25/2012 | EP2408763A2 Derivatives of n-ý(2-aza-bicycloý2.1.1¨hex-1-yl)-aryl-methyl¨-heterobenzamide, preparation thereof and application of same in therapeutics |
| 01/24/2012 | US8101768 Cyclic amine compound and pest control agent |
| 01/24/2012 | US8101763 Method for producing scopine esters |
| 01/24/2012 | CA2435687C Omega-aminoalkylamides of r-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells |
| 01/19/2012 | WO2012008435A1 Biaryl amide derivative or pharmaceutically acceptable salt thereof |
| 01/19/2012 | WO2011138751A3 Heterocyclic derivatives as alk inhibitors |
| 01/18/2012 | CN102325752A Carbazole and carboline kinase inhibitors |
| 01/11/2012 | EP2403851A2 New crystal forms |
| 01/11/2012 | CN102317277A C-met protein kinase inhibitors |
| 01/11/2012 | CN101874899B Dopamine transporter imaging medicine and preparation method thereof |
| 01/05/2012 | WO2012000881A1 Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 01/05/2012 | US20120004257 Novel compounds |
| 01/04/2012 | EP1735286B1 Tetrahydro-indazole cannabinoid modulators |
| 01/04/2012 | CN101838266B Citric acid tropisetron raw material medicine and preparation technology of raw material medicine and injection liquid |
| 01/04/2012 | CN101679407B Novel chromen-2-one derivatives |
| 12/29/2011 | WO2011161006A1 Amido-tropane derivatives |
| 12/29/2011 | CA2801458A1 Amido-tropane derivatives |
| 12/28/2011 | EP1664036B1 Benzimidazolone compounds having 5-ht4 receptor agonistic activity |
| 12/28/2011 | CN102300846A 用于标记正电子发射同位素的三芳基锍化合物、药盒和方法 For labeling n triaryl sulfonium compounds, kits and methods of the electron-emitting isotopes |
| 12/22/2011 | US20110313153 5-ht4 inhibitors for treating airway diseases, in particular asthma |
| 12/22/2011 | US20110312993 Amido-tropane derivatives |
| 12/22/2011 | US20110311516 Chemically Programmed Vaccination |
| 12/21/2011 | EP2397477A1 Heterocyclic-substituted piperidine compounds and the uses thereof |
| 12/21/2011 | EP2395992A2 Chemically programmed vaccination |
| 12/20/2011 | CA2733294C Pharmaceutical combination of a tiotropium salt and ciclesonide |
| 12/15/2011 | US20110306597 Nicotinamide Derivatives |
| 12/14/2011 | EP1513529B1 Triple monoamine reuptake inhibitors for the treatment of chronic pain |
| 12/08/2011 | US20110301191 Methods of treatment using selective 5-ht2a inverse agonists |
| 12/07/2011 | EP2391622A1 Process for preparing enantiomerically enriched alkaloids |
| 12/07/2011 | EP2391621A2 Bicyclic amide derivatives for enhancing glutamatergic synaptic responses |
| 12/07/2011 | CN102267993A 一种多羟基去甲基托品烷类化合物及其制备方法与应用 A base plate to a polyhydroxy alkyl compounds product and its preparation method and application |
| 12/07/2011 | CN102267992A 一种截短侧耳素类抗生素的制备方法 A hormone preparation Pleuromutilin antibiotics |
| 12/07/2011 | CN101574552B 含有噻托铵吸入用粉末的吸入用套盒 Tiotropium containing inhalation powder inhalation kit |
| 12/01/2011 | US20110294780 SUBSTITUTED THIAZOLIDINEDIONE INDAZOLES, INDOLES AND BENZOTRIAZOLES AS ESTROGEN-RELATED RECEPTOR-a MODULATORS |
| 12/01/2011 | US20110294749 Diaminopyrimidinecarboxamide derivative |
| 11/30/2011 | EP2389372A1 Compositions and methods for inhibition of the jak pathway |
| 11/30/2011 | CN102264734A 生物碱氨基酯衍生物及其药用组合物 Alkaloid aminoester derivatives and pharmaceutical compositions |
| 11/23/2011 | EP2387565A2 2,4-pyrimidinediamine compounds for treatment of inflammatory disorders |
| 11/22/2011 | US8063045 Fluoropyrrolidines having dipeptidyl peptidase enzyme inhibitory activity |
| 11/22/2011 | CA2484395C Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for the preparation thereof |
| 11/16/2011 | CN101563344B Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 11/16/2011 | CN101010320B Aminotropane derivatives, preparation thereof and therapeutic use thereof |
| 11/10/2011 | WO2011138916A1 Polycyclic compound |
| 11/10/2011 | WO2010093706A3 Chemically programmed vaccination |
| 11/10/2011 | US20110275595 Urea derivatives of substituted nortropanes, medicaments containing such compounds and their use |
| 11/09/2011 | CN101643473B Synthesis method of homatropine hydrobromide |
| 11/03/2011 | WO2011135276A1 3, 3 -disubstituted- ( 8 - aza - bicyclo [3.2.1] oct- 8 - yl) -[5- (1h - pyrazol - 4 -yl) -thiophen-3 -yl] methanones as inhibitors of 11 (beta) -hsd1 |
| 11/03/2011 | US20110270011 Use of opioids or opioid mimetics for the treatment of resistant cancer patients |
| 11/02/2011 | EP2383259A1 New pyridone derivatives with MCH antagonistic activity and medicaments comprising these compounds |