| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 10/26/2006 | WO2006075004A3 3, 8 - substituted 8-aza-bicyclo[3.2.1] octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 10/25/2006 | EP1713800A2 Method for producing a 2-(ethoxymethyl)tropane derivative |
| 10/25/2006 | CN1852712A Dual NK1/NK3 antagonists for treating schizophrenia |
| 10/24/2006 | US7125886 2-imidazomethyl- pyrido(4,3-b)indol-1-one or -carbazol-1-one derivatives containing an ester group; especially for treating irritable bowel syndrome. |
| 10/24/2006 | CA2167584C Aza spiro compounds acting on the cholinergic system with muscarinic agonist activity |
| 10/19/2006 | WO2006108790A1 (+) - and (-) -8-alkyl-3-(trifluoralkylsulfonyloxy)-8-azabicycl (3.2.1.)oct-2-ene |
| 10/19/2006 | WO2006108789A1 Novel enantiomers and their use as monoamine neurotransmitter re-uptake inhibitors |
| 10/19/2006 | US20060235044 Azabicyclononene derivatives |
| 10/19/2006 | CA2603923A1 (+)- and(-)-8-alkyl-3-(trifluoralkylsulfonyloxy)-8-azabicyclo(3.2.1.) oct-2-ene |
| 10/18/2006 | EP1711463A2 Amino-substituted tricyclic derivatives and methods of use |
| 10/18/2006 | EP1711183A2 Muscarinic acetylcholine receptor antagonists |
| 10/18/2006 | CN1849330A Specific glucocorticosteroid compound having anti-inflammatory activity |
| 10/17/2006 | US7122666 Antiinflammatory agents; autoimmune disease; antiarthritic agents |
| 10/12/2006 | US20060229336 HIV, acquired immune deficiency syndrome (AIDS); 1-(8-{2-[1-(2,2-Dimethylpropanoyl)-4-phenylpiperidin-4-yl]ethyl}-8-azabicyclo[3.2.1]oct-3-yl)-2-methyl-1H-benzimidazole |
| 10/12/2006 | US20060229332 crystalline hydrochloride salt of 1-isopropyl-2-oxo-1,2-dihydroquinoline-3-carboxylic acid {(1S,3R,5R)-8-[(R)-2-hydroxy-3-(methanesulfonyl-methyl-amino)propyl]-8-azabicyclo[3.2.1]oct-3-yl}amide or solvate thereof; treating disease associated with 5-HT4 receptor activity; gastrointestinal tract disorder |
| 10/11/2006 | CN1845933A Specific glucocorticosteriod compound having anti-inflamatory activity |
| 10/11/2006 | CN1845922A Benzimidazolone compounds having 5-HT4 receptor agonistic activity |
| 10/11/2006 | CN1845921A Adamantane and azabicyclo-octane and nonane derivatives, process of their preparation and their use as DPP-IV inhibitors |
| 10/11/2006 | CN1845908A 5-substituted quinazolinone derivatives |
| 10/11/2006 | CN1279040C Tryasolyl tropane derivatives for therapy |
| 10/05/2006 | WO2006105035A2 Muscarinic modulators |
| 10/05/2006 | US20060223840 Substituted piperidine compounds and methods of their use |
| 10/05/2006 | US20060223784 Method and compositions for temporarily incapacitating subjects |
| 10/04/2006 | EP1707205A2 Pharmaceutical compositions of anticholinergics and p38 kinase inhibitors in the treatment of respiratory diseases |
| 10/04/2006 | EP1487831B1 Difurylglycolic acid tropenol esters used as anticholinesterase drugs |
| 10/04/2006 | EP1406900B1 Novel compounds, their preparation and use |
| 10/04/2006 | CN1840529A Process for preparing an anticholinergic |
| 10/03/2006 | US7115607 Substituted piperazinyl amides and methods of use |
| 09/28/2006 | WO2006005057A3 Muscarinic acetylcholine receptor antagonists |
| 09/28/2006 | US20060217534 Bis (amino acid) molecular scaffolds |
| 09/27/2006 | EP1704146A1 Stereoisomeric compounds and methods for the treatment of gastrointestinal and central nervous system disorders |
| 09/27/2006 | CN1838953A 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylinositol 3 kinase enzymes (pi3) for the treatment of inflammatory airway diseases |
| 09/27/2006 | CN1837204A Process for preparing N-2-fluoro ethyl-2 beta-carbomethoxy-3 beta-(4-chlorphenyl) nor tropane |
| 09/20/2006 | EP1158970B1 Combinations of formoterol and a tiotropium salt |
| 09/20/2006 | CN1275962C Novel anticholinergic agents that can be used as medicaments and method for the production thereof |
| 09/14/2006 | WO2006031788A3 Process for preparing substituted 8-azabicyclo[3.2.1] octan-3-ols |
| 09/14/2006 | US20060205785 Fused ring compounds substituted with a 8-azabicyclo[3.2.1]octane(cyclo)alkylene group, including benzothiazolones, e.g., 3-[3-(3-Propyl-8-aza-bicyclo[3.2.1]oct-8-yl)-propyl]-3H-benzothiazol-2-one; highly selective muscarinic agonists, particularly for the M1 and/or M4 receptor subtypes |
| 09/14/2006 | US20060205769 Piperidine or 8-aza-bicyclo[3.2.1]oct-3-yl derivatives useful as modulators of chemokine receptor activity |
| 09/14/2006 | US20060205768 Tropane derivatives and their use as ace inhibitors |
| 09/13/2006 | CN1830445A Tropane derivatives having therapy using, compounds and polymorph thereof |
| 09/12/2006 | US7105678 Boat tropanes |
| 09/08/2006 | WO2006094063A1 Quinolinone compounds as 5-ht4 receptor agonists |
| 09/08/2006 | WO2006092334A1 Novel polymorph of mutilin |
| 09/08/2006 | WO2006092268A1 Bicyclic five-membered heteroaryl derivatives and their use as renin inhibitors |
| 09/08/2006 | WO2006064340A3 Process for the preparation of n-acyl beta-aminoaldehydes |
| 09/08/2006 | CA2599404A1 Quinolinone compounds as 5-ht4 receptor agonists |
| 09/07/2006 | US20060199813 Neurodegenerative diseases, psychological disorders; e.g. 1-[3-(4-Butyl-piperidin-1-yl)-propyl]-1,2,3,4-tetrahydroquinoline |
| 09/07/2006 | US20060199810 Neurodegenerative diseases, psychological disorders; e.g. 1-[3-(4-Butyl-piperidin-1-yl)-propyl]-1,2,3,4-tetrahydro-quinoline |
| 09/07/2006 | US20060199799 Benzimidazolidinone derivatives as muscarinic agents |
| 09/06/2006 | EP1259241B8 The use of scopolamine salts |
| 08/31/2006 | US20060194834 Serotonin receptor antagonist; psychological disorders; Alzheimer's disease |
| 08/31/2006 | US20060194790 Bridged bicyclic amine derivatives useful as CCR-3 receptor antagonists |
| 08/31/2006 | US20060194780 N-Azacycloalkylcarbonyl-substituted bicyclic piperidines, e.g., N-tert-butyl)-8-{[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl]carbonyl}-3-cyclohexyl-8-azabicyclo[3.2.1]octane-3-carboxamide; useful for treating obesity, diabetes, and sexual dysfunction |
| 08/31/2006 | US20060194778 Serotonin receptor antagonist; psychological disorders; side effect reduction |
| 08/30/2006 | EP1385519B1 Compounds for treating inflammatory diseases |
| 08/30/2006 | CN1826339A 2-acylamino-4-phenylthiazole derivatives, preparation thereof and therapeutic application thereof |
| 08/24/2006 | WO2006089100A1 Benzoxazole carboxamides for treating cinv and ibs-d |
| 08/24/2006 | WO2006088988A1 Crystalline form of an indazole-carboxamide compound |
| 08/24/2006 | US20060189596 Bridged bicyclic amine derivatives useful as CCR-3 receptor antagonists |
| 08/24/2006 | CA2597962A1 Benzoxazole carboxamides for treating cinv and ibs-d |
| 08/23/2006 | EP1401445B1 Crystalline anticholinergic, method for its production, and use thereof in the production of a drug |
| 08/23/2006 | CN1822840A Muscarinic acetylcholine receptor antagonists |
| 08/23/2006 | CN1822839A Muscarinic acetylcholine receptor antagonists |
| 08/23/2006 | CN1822838A Muscarinic acetylcholine receptor antagonists |
| 08/23/2006 | CN1822837A 2-methoxymethyl-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octane tartrate salts |
| 08/22/2006 | US7094788 A tropane ester derivative for treating asthma, chronic obstractive pulmonary disease, vagally induced sinus bradycardia, heart rhythm disorders, spasms in the gastrointestinal or urinary tracts, and menstrual pain |
| 08/16/2006 | EP1690539A2 Salts of tiotropium for treating inflammatory disorders |
| 08/16/2006 | EP1689391A2 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylinositol 3 kinase enzymes (pi3) for the treatment of inflammatory airway diseases |
| 08/16/2006 | EP1432702B1 Nitrogen-containing heterocyclic compounds and their use as raf inhibitors |
| 08/16/2006 | CN1820010A Bridged n-arylsulfonylpiperidines as gamma-secretase inhibitors |
| 08/16/2006 | CN1269470C Method for producing powdery formulations |
| 08/15/2006 | US7091227 Serine/threonine and tyrosine kinases inhibitors |
| 08/10/2006 | WO2006069276A3 TRICYCLIC ō-OPIOID MODULATORS |
| 08/10/2006 | US20060178396 e.g. (3-endo)-3-(2-Hydroxy-2,2-di-2-thienylethyl)-8,8-dimethyl-8-azoniabicyclo[3.2.1]octane bromide; muscle relaxants, respiratory system disorders; asthma, emphysema, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis |
| 08/10/2006 | US20060178395 3-(2-Benzyl-2-hydroxy-3-phenyl-propylidene)-8,8-dimethyl-8-azonia-bicyclo[3.2.1]octane iodide; muscle relaxants, respiratory system disorders; asthma, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis |
| 08/10/2006 | US20060178360 N(2-hydroxyethyl)-4-methoxy-N,2,6-trimethylbenzene- sulphonamide; analgesic, antiinflammatory agent; hyperalgesia and major algesia connected with other pathological conditions such as cancer |
| 08/09/2006 | EP1688418A2 Chemokine receptor antagonists and methods of use thereof |
| 08/09/2006 | EP1688412A2 Novel heterocyclic amide derivatives and their use as dopamine D3 receptor ligands |
| 08/09/2006 | EP1472249B1 Xanthene-carboxylic acid esters of tropenol and scopine as m3 antagonists, method for producing the same and use thereof as medicaments |
| 08/08/2006 | US7087749 Substituted piperidine compounds and methods of their use |
| 08/08/2006 | US7087593 Psychological disorder treatments that increase the activity of cholinergic receptors |
| 08/03/2006 | US20060173044 Substituted propargylamines |
| 08/03/2006 | US20060173037 Aminophenyl derivatives as selective androgen receptor modulators |
| 08/02/2006 | EP1358177B1 Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance |
| 08/01/2006 | US7084158 Substituted propargylamines |
| 07/27/2006 | US20060166962 2-{4-[(4-{bis[4-(trifluoromethyl)phenyl]methyl}1-oxypiperazinyl)methyl]phenoxy}pyrimidine; insecticide, controlling tobacco budworm, wheat, corn, soybeans, potatoes, and cotton; for soil-borne insects, such as termites and white grubs |
| 07/26/2006 | EP1682543A1 Novel tiotropium salts, methods for the production thereof, and pharmaceutical formulations containing the same |
| 07/26/2006 | EP1682542A1 Novel crystalline anhydride with anticholinergic effect |
| 07/26/2006 | EP1682541A1 Method for producing tiotropium salts, tiotropium salts and pharmaceutical formulations, containing the same |
| 07/26/2006 | EP1682142A2 M3 muscarinic acetylcholine receptor antagonists |
| 07/26/2006 | EP1682141A1 4-fluoro-4-(pyridin-2-yl)-piperidine-1-carboxamide derivatives and related compounds which modulate the function of the vanilloid-1 receptor (vr1) for the treatment of pain |
| 07/26/2006 | EP1513838B1 Technical method for producing tropenol |
| 07/25/2006 | US7081531 Bridged bicyclic amine derivatives useful as CCR-3 receptor antagonists |
| 07/20/2006 | WO2006076317A2 Aminophenyl derivatives as selective androgen receptor modulators |
| 07/20/2006 | WO2006075004A2 3, 8 - substituted 8-aza-bicyclo[3.2.1] octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 07/20/2006 | WO2006044174A9 Aryl substituted 8-azabicyclo[3.2.1]octane compounds as ligands of the melanin concentrating hormone receptor |
| 07/20/2006 | US20060160845 Aminophenyl derivatives as selective androgen receptor modulators |
| 07/20/2006 | US20060160844 3-(2-Benzyl-2-hydroxy-3-phenyl-propylidene)-8,8-dimethyl-8-azonia-bicyclo[3.2.1]octane iodide; muscle relaxants, respiratory system disorders; asthma, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis |
| 07/20/2006 | CA2594340A1 Aminophenyl derivatives as selective androgen receptor modulators |
| 07/19/2006 | EP1680419A1 Improved aza-bridged-bicyclic amino acid derivatives as a4 integrin antagonists |