Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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01/30/2007 | CA2302411C Improved method for preventing crystal formation in a scopolamine transdermal device |
01/25/2007 | US20070020177 Radiometal complex compositions |
01/24/2007 | CN1902197A Improved aza-bridged-bicyclic amino acid derivatives as alpha4 integrin antagonists |
01/18/2007 | US20070015788 N-(3-Aryl-3-substitutedphenylpropyl) piperidines or 8-azabicyclo[3.2.1]octanes that are additionally substituted with an optionally fused 5-member N-heterocycle; the compounds are modulators of CCR5 receptor activity and are used in treating diseases such as rheumatoid arthritis |
01/17/2007 | EP1742944A1 Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
01/17/2007 | CN1897947A Muscarinic acetylcholine receptor antagonists field of the invention |
01/16/2007 | US7164027 Aralkyl ester soft drugs |
01/11/2007 | WO2007003934A2 17beta-hydr0xyster0id dehydrogenase type 3 (17beta-hsd3 ) inhibitors |
01/11/2007 | WO2007003522A1 Method for obtaining a pharmaceutically active compound, synthesis intermediates thereof and methods for obtaining them |
01/11/2007 | US20070010557 Novel amides useful for treating pain |
01/11/2007 | US20070009432 Boat tropanes |
01/10/2007 | EP1741703A1 Pyridone derivative |
01/10/2007 | EP1741430A1 Remedy for psychoneurotic diseases |
01/10/2007 | EP1740570A2 Novel gamma secretase inhibitors |
01/10/2007 | EP1740565A2 Arylphenylamino-, arylphenylamide-, and arylphenylether-sufide derivatives |
01/10/2007 | EP1740177A2 Muscarinic acetylcholine receptor antagonists |
01/10/2007 | CN1893948A Muscarinic acetylcholine receptor antagonists |
01/09/2007 | US7160920 Nitrosated and nitrosylated compounds and compositions and their use for treating respiratory disorders |
01/09/2007 | CA2236578C Dopamine transporter imaging agent |
01/04/2007 | WO2006108127A3 Crystalline form of a quinolinone-carboxamide compound |
01/03/2007 | EP1737863A2 2-cyanopyrrolidinecarboxamides as dipeptidyl peptidase-iv inhibitors |
01/03/2007 | EP1737860A1 Selected cgrp-antagonists, their preparation processes and their use as medicaments |
01/03/2007 | EP1737853A1 3-(diheteroarylmethylene)-8-azabicyclo¬3.2.1|octane and 3-((aryl)(heteroaryl)methylene)-8-azabicyclo¬3.2.1|octane derivatives |
01/03/2007 | EP1737842A1 Selected cgrp antagonists, method for producing the same and the use thereof as drugs |
01/03/2007 | EP1737840A1 1-amino-phthalazine derivatives, the preparation and the therapeutic use thereof |
01/03/2007 | EP1737823A2 Novel alkyne compounds with an mch-antagonistic action and medicaments comprising said compounds |
01/03/2007 | CN1890239A Azabicyclooctene and other tetrahydropyridine derivatives with a new side-chain |
01/03/2007 | CN1890237A Method for producing n-substituted 3beta-aminonortropanes |
12/28/2006 | WO2006117299A9 Novel crystalline forms of tiotropium bromide |
12/28/2006 | WO2006117299A2 Novel crystalline forms of tiotropium bromide |
12/28/2006 | CA2612491A1 Tricyclic opioid modulators |
12/27/2006 | EP1736467A1 Novel sulfonamide derivative |
12/27/2006 | EP1736156A1 STABILIZED 4-AMINO-5-CHLORO-N-¬(1R,3r,5S)-8-METHYL-8- AZABICYCLO¬3.2.1|OCT-3-YL|-2-¬1-METHYLBUT-2-YNYLOXY|-BENZAMIDE CONTAINING COMPOSITION |
12/27/2006 | EP1735304A1 Quinolinone-carboxamide compounds as 5-ht4 receptor agonists |
12/27/2006 | EP1735286A1 Tetrahydro-indazole cannabinoid modulators |
12/27/2006 | EP1534282B1 Pharmaceutical compositions of anticholinergics and p38 kinase inhibitors in the treatment of respiratory diseases |
12/27/2006 | CN1886135A Phenyl-piperazine derivatives as modulators of muscarinic receptors |
12/27/2006 | CN1291986C Anticholinergics, processes for the preparation thereof, and pharmaceutical compositions |
12/21/2006 | WO2006135715A1 Benztropinamine analogs as dopamine uptake inhibitors |
12/21/2006 | WO2006134486A2 Alpha-(aryl-or heteroaryl-methyl)-beta piperidino propanamide compounds as orl1-receptor antagonists |
12/21/2006 | WO2006134318A1 Pyrazole-substituted benzimidazole derivatives for use in the treatment of cancer and autoimmune disorders |
12/21/2006 | WO2006134021A2 Process for preparing tiotropium salts, tiotropium salts as such and pharmaceutical compositions thereof |
12/21/2006 | WO2006133802A1 N-amide derivatives of 8-azabicyclo[3.2.1]oct-3-yl as ccr1 antagonists |
12/21/2006 | US20060286099 Hapten-carrier conjugates for use in drug-abuse therapy and methods for preparation of same |
12/21/2006 | US20060286098 Derived from cocaine linked to cholera B toxin; antibodies; for treatment of cocaine addiction; immunization |
12/21/2006 | US20060286097 Hapten-carrier conjugates for use in drug-abuse therapy and methods for preparation of same |
12/21/2006 | US20060286096 Hapten-carrier conjugates for use in drug-abuse therapy and methods for preparation of same |
12/21/2006 | US20060286095 Hapten-carrier conjugates for use in drug-abuse therapy and methods for preparation of same |
12/21/2006 | US20060286094 Hapten-carrier conjugates for use in drug-abuse therapy and methods for preparation of same |
12/21/2006 | CA2612299A1 Alpha-(aryl-or heteroaryl-methyl)-beta piperidino propanamide compounds as orl1-receptor antagonists |
12/21/2006 | CA2609577A1 Benztropinamine analogs as dopamine uptake inhibitors |
12/20/2006 | EP1732923A2 Muscarinic acetylcholine receptor antagonists |
12/20/2006 | EP1732552A2 2,6-disubstituted piperidines as modulators of chemokine receptor activity |
12/20/2006 | EP1622610B1 1-(2h-pyrazol-3-yl)-3-{4-[1-(benzoyl)-piperidin-4-ylmethyl]-phenyl}-urea derivatives and related compounds as inhibitors of p38 kinase and/or tnf inhibitors for the treatment of inflammations |
12/20/2006 | EP1263729B1 Azacyclic compounds for use in the treatment of serotonin related diseases |
12/20/2006 | CN1882582A Method for producing tiotropium salts, tiotropium salts and pharmaceutical formulations, containing the same |
12/20/2006 | CN1880319A Tropane derivatives as CCR5 modulators |
12/14/2006 | WO2006131525A1 3 -aryloxy- 8 -aza-bicyclo [3.2.1.] oct- 6- ene derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
12/14/2006 | US20060280736 Hapten-carrier conjugates for use in drug-abuse therapy and methods for preparation of same |
12/14/2006 | CA2620986A1 3 -aryloxy- 8 -aza-bicyclo [3.2.1.] oct- 6- ene derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
12/13/2006 | EP1731518A1 Cyclic amine compound and pest control agent |
12/13/2006 | EP1392676B1 Heterocyclic urea derivatives and their use as dopamine d3 receptor ligands |
12/12/2006 | US7148240 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same |
12/12/2006 | US7148236 Modulate neurotransmission by promoting the release of neurotransmitters such as acetylcholine, dopamine and norepinephrine; thio-bridged aryl derivatives; treats central and autonomic nervous system disorders |
12/07/2006 | WO2006130075A1 Novel mchr1 antagonists and their use for the treatment of mchr1 mediated conditions and disorders |
12/07/2006 | WO2005100350A8 Quinolinone-carboxamide compounds as 5-ht4 receptor agonists |
12/07/2006 | US20060276503 Novel process salts compositions and use |
12/07/2006 | US20060276487 New compounds useful for DPP-IV enzyme inhibition |
12/07/2006 | US20060276482 Benzoimidazolone-carboxamide compounds as 5-HT4 receptors agonists |
12/07/2006 | CA2610671A1 Novel mchr1 antagonists and their use for the treatment of mchr1 mediated conditions and disorders |
12/06/2006 | EP1727812A1 Novel cycloalkyl-containing 5-acylindolinones, their preparation and their use as pharmaceutical products |
12/06/2006 | EP1572668A4 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines |
12/06/2006 | EP1397135B1 Combination of a pde4 inhibitor and tiotropium or derivative thereof for treating obstructive airways |
12/06/2006 | CN1875020A Novel tiotropium salts, methods for the production thereof, and pharmaceutical formulations containing the same |
12/06/2006 | CN1875019A Novel crystalline anhydride with anticholinergic effect |
12/06/2006 | CN1874775A 4-fluoro-4-(pyridin-2-yl)-piperidine-1-carboxamide derivatives and related compounds which modulate the function of the vanilloid-1 receptor (VR1) for the treatment of pain |
12/06/2006 | CN1288154C Technical synthesis method for producing tropenol |
11/29/2006 | EP1726590A1 Cycloalkanopyridine derivative |
11/29/2006 | EP1572207A4 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines |
11/23/2006 | WO2006076317A3 Aminophenyl derivatives as selective androgen receptor modulators |
11/23/2006 | US20060264434 Chemokine receptor binding heterocyclic compounds |
11/23/2006 | US20060264419 Substituted pyrazoles |
11/23/2006 | CA2608240A1 Multicyclic compounds and methods of their use |
11/22/2006 | CN1867330A N-substituted azacycles |
11/16/2006 | WO2006105035A3 Muscarinic modulators |
11/16/2006 | WO2006021559A8 Method for producing tiotropium salts and silicon derivatives as intermediates |
11/16/2006 | US20060258707 Benzimidazolidinone derivatives as muscarinic agents |
11/15/2006 | EP1720859A2 Chemokine receptor antagonists |
11/15/2006 | EP1453511B1 Tropane derivatives having dopamine reuptake inhibitor activity for the treatment of ischemic diseases |
11/15/2006 | CN1861598A Preparation process of thiatro bromoaminium anhydrous compound |
11/14/2006 | CA2128493C Aminobenzoic acid derivatives |
11/09/2006 | WO2006117300A2 Crystalline forms of tiotropium bromide |
11/09/2006 | CA2606552A1 Crystalline forms of tiotropium bromide |
11/09/2006 | CA2606549A1 Crystalline forms of tiotropium bromide |
11/08/2006 | EP1718643A1 Indazole-carboxamide compounds as 5-ht4 receptor agonists |
11/07/2006 | US7132541 Microbiocides |
11/07/2006 | US7132443 Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
11/02/2006 | US20060247219 Specific glucocorticosteriod compound having anti-inflamatory activity |
11/01/2006 | CN1856485A Benzimidazolone and quinazolinone derivatives as agonists on human ORL1 receptors |
10/31/2006 | US7129235 Amides useful for treating pain |