Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
---|
06/14/2011 | CA2494962C Tyrosine kinase inhibitors |
06/09/2011 | US20110136854 Novel 9-aza-bicyclo[3.3.1]non-3-yloxy chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
06/09/2011 | US20110136833 Tetrahydropyridinyl and Dihydropyrrolyl Compounds and the Use Thereof |
06/09/2011 | US20110135958 Schiff base type compound and coloring material containing the same |
06/08/2011 | EP2328880A2 6-substituted benzoxazines as 5-ht-5a receptor antagonists |
06/01/2011 | CN101166738B Novel crystalline forms of tiotropium bromide |
05/26/2011 | WO2011061590A1 Novel carboxamide derivatives as hiv inhibitors |
05/26/2011 | WO2010138720A3 Compounds and methods for chelating metals in aqueous solutions |
05/26/2011 | US20110124693 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylinositol 3 kinase enzymes (pi3) for the treatment of inflammatory diseases |
05/26/2011 | US20110124676 Biaryl substituted azabicyclic alkane derivatives |
05/26/2011 | US20110124624 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylinositol 3 kinase enzymes (pi3) for the treatment of inflammatory diseases |
05/25/2011 | EP2323654A1 Polymorphic form of granisetron hydrochloride and methods of making the same |
05/25/2011 | CN1849330B Specific glucocorticosteroid compound having anti-inflammatory activity |
05/25/2011 | CN102070630A New tiotropium salts, pharmaceutical compositions containing the same and use thereof |
05/24/2011 | US7947838 Radiolabelled benzamide analogues, their synthesis and use in diagnostic imaging |
05/24/2011 | US7947710 Disubstituted alkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists |
05/24/2011 | CA2490888C Diaminopyrimidinecarboxamide derivative |
05/19/2011 | WO2011059048A1 Novel amide derivative |
05/19/2011 | WO2011059021A1 8-azabicyclo[3.2.1]octane-8-carboxamide derivative |
05/19/2011 | US20110118305 Compounds |
05/19/2011 | CA2778175A1 8-azabicyclo[3.2.1]octane-8-carboxamide derivative |
05/18/2011 | EP2322522A1 New tiotropium salts, processes for their preparation and drug formulations containing them |
05/18/2011 | EP2001876B1 8-azabicycloý3.2.1¨octane compounds as mu opioid receptor antagonists |
05/18/2011 | CN102066320A Aryl ketone as MRI |
05/18/2011 | CN102060853A Method for separating alkaloid by reversely two-way eluted pH-zone-refining counter-current chromatography |
05/18/2011 | CN101475569B Method for preparing granisetron hydrochloride from high tropine alkanamine |
05/18/2011 | CN101405287B Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
05/12/2011 | US20110112139 Novel 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
05/11/2011 | EP2319844A1 Tiotropium salts, method for creating same and medicinal formulations containing same |
05/11/2011 | EP2318404A1 Bicyclic heterocycle derivatives and use thereof as gpr119 modulators |
05/11/2011 | EP2318403A1 Aryl- and heteroarylcarbonyl derivatives of substituted nortropanes, medicaments containing such compounds and their use |
05/11/2011 | EP1984362B1 Process for preparing intermediates to 5-ht4 receptor agonist compounds |
05/10/2011 | US7939533 Dual NK1/NK3 receptor antagonists |
05/05/2011 | WO2011053706A1 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators |
05/05/2011 | US20110105546 Spirotropane compounds |
05/05/2011 | CA2779108A1 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators |
05/05/2011 | CA2778684A1 Bridged bicyclic piperidine derivatives and methods of use thereof |
04/26/2011 | US7932235 Triazolyl tropane derivatives |
04/26/2011 | CA2509892C Herbicidally active nicotinoyl derivates |
04/21/2011 | US20110092535 Novel Epilepsy Treatment |
04/20/2011 | EP2311835A1 Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
04/20/2011 | EP2311807A1 Compounds and composition as protein kinase inhibitors |
04/20/2011 | CN1830445B Composition of tropane derivatives having therapy use and polymorph thereof |
04/20/2011 | CN102026992A Novel HSP inhibitory carbazole derivatives, compositions containing same, and use thereof |
04/13/2011 | EP1888064B1 Benztropinamine analogs as dopamine uptake inhibitors |
04/13/2011 | EP1140085B1 Azabicycloalkanes as ccr5 modulators |
04/07/2011 | WO2010138720A9 Compounds and methods for chelating metals in aqueous solutions |
04/06/2011 | CN102007124A Pyrimidine-2-amine compounds and their use as inhibitors of jak kinases |
04/05/2011 | CA2537127C Benzimidazolone compounds having 5-ht4 receptor agonistic activity |
04/05/2011 | CA2425638C Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance |
03/30/2011 | CN101993443A Novel crystal form of benzilic acid nortropine easter and preparation method thereof |
03/30/2011 | CN101993442A Novel crystal forms of benzilic acid nortropinyl hydrochloride and preparation method thereof |
03/29/2011 | US7915260 Urotensin II receptor antagonists |
03/24/2011 | WO2011033255A1 (4-phenyl-piperidin-1-yl)-[5-1h-pyrazol-4yl)-thiophen-3-yl]-methanone compounds and their use |
03/24/2011 | WO2011032214A1 A method for the n-demethylation of n-methyl heterocycles |
03/24/2011 | WO2010087981A3 Bicyclic amide derivatives for enhancing glutamatergic synaptic responses |
03/24/2011 | CA2772504A1 (4-phenyl-piperidin-1-yl)-[5-(1h-pyrazol-4-yl)-thiophen-3-yl]-methanone compounds and their use |
03/23/2011 | EP2298415A1 Micronisation method |
03/23/2011 | EP2297096A2 Aryl ketone as mri |
03/23/2011 | EP2195314B1 Disubstituted alkyl-8-azabicyclo [3.2.1.]octane compounds as mu opioid receptor antagonists |
03/23/2011 | CN101990536A Pyrollidine-based compounds |
03/22/2011 | US7908735 Method and installation means for installing an electrical machine |
03/16/2011 | EP2132194B1 Substituted isoquinolines and their use as rho-kinase inhibitors |
03/15/2011 | US7906531 M3 muscarinic acetylcholine receptor antagonists |
03/10/2011 | WO2011027865A1 Novel 2-aza-adamantane compound and method for producing the same |
03/10/2011 | US20110059937 Il-8 receptor antagonists |
03/10/2011 | US20110059929 SUBSTITUTED BICYCLIC PIPERIDINYL-AND PIPERAZINYL- SULFONAMIDES USEFUL TO INHIBIT 11beta-HYDROXYSTEROID DEHYDROGENASE TYPE-1 |
03/09/2011 | EP1624845B1 4',4''-substituted 3alpha-(diphenylmethoxy)tropane analogs for the treatment of adhd |
03/08/2011 | US7902375 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylin ositol 3 kinase enzymes (PI13) for treatment of inflammatory diseases |
03/08/2011 | US7902222 Biaryl substituted azabicyclic alkane derivatives |
03/08/2011 | US7902220 8-azabicyclo[3.2.1]octyl-2-hydroxybenzamide compounds as mu opioid receptor antagonists |
03/08/2011 | US7902217 Indoles, 1H-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
03/03/2011 | US20110053162 Reactive cyanine compounds |
03/01/2011 | CA2542657C Muscarinic acetylcholine receptor antagonists |
02/24/2011 | WO2011021645A1 Bicyclic urea derivative or pharmacologically permitted salt thereof |
02/23/2011 | EP2286811A1 Chemokine receptor antagonists and methods of use thereof |
02/23/2011 | CN101979391A Method for preparing tiotropium bromide |
02/22/2011 | US7893256 Azabicycloalkane compounds |
02/22/2011 | CA2624558C Cross-linked cyclic amine compounds and agents for pest control |
02/17/2011 | WO2011018796A1 An improved process for the synthesis of alkyl/aralkyl (2s)-2-(tert-butoxycarbonyl)-amino-2-[-8-azabicyclo[3.2.1]oct-3-yl]-exo-acetate and analogs thereof: key intermediates for the preparation of dppiv inhibitors |
02/16/2011 | EP2284170A1 Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
02/16/2011 | CN101977904A Aminopiperidinyl derivatives and uses thereof |
02/15/2011 | US7888358 Serotonine, dopamine and norendrenaline receptors; antidepressants, anxiolytic agents, eating disorders; obesity; bipolar; drug abuse; neurodegenerative diseases |
02/15/2011 | CA2558272C Pyridone derivative |
02/10/2011 | WO2011015884A1 Process to prepare scopine esters |
02/10/2011 | WO2011015883A1 Dichloromethane solvate of tiotropium bromide and its use |
02/10/2011 | WO2011015882A2 Novel anhydrate |
02/10/2011 | CA2768553A1 Anhydrate of tiotropium bromide |
02/09/2011 | EP2280966A1 Azabicyclo [3.2.1]octyl derivatives as 11 beta-hsd1 modulators |
02/08/2011 | CA2471755C Process for preparing scopine esters |
02/02/2011 | EP2280010A2 Biaryl substituted azabicyclic alkane derivatives as nicotinic acetylcholine receptor activity modulators |
02/02/2011 | EP2280008A2 Heterocyclic-substituted piperidines as ORL-1 ligands |
02/02/2011 | EP2280003A2 Process for preparing receptor-type kinase modulators |
02/02/2011 | CN1838953B 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylinositol 3 kinase enzymes (pi3) for the treatment of inflammatory airway diseases |
02/01/2011 | US7879871 Crystalline forms of tiotropium bromide |
02/01/2011 | CA2481468C Medicaments containing betamimetic drugs and a novel anticholinesterase drug |
01/27/2011 | WO2010101538A3 New crystalline forms of tiotropium bromide |
01/26/2011 | EP2277869A1 Cycloalkylamidbenzoxa(thia)zoles as fungicides |
01/26/2011 | EP2277867A2 Compounds, pharmaceutical compositions thereof and their use in treating cancer |
01/26/2011 | CN101959876A 2-aminoquinolines |