Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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07/13/2006 | US20060154951 Quaternary antimuscarinic compounds for the treatment of bladder diseases |
07/12/2006 | EP1677796A2 Muscarinic acetylcholine receptor antagonists field of the invention |
07/12/2006 | EP1677795A1 Muscarinic acetycholine receptor antagonists |
07/11/2006 | CA2227984C Aza-anthracyclinone derivatives |
07/06/2006 | US20060148847 Novel 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
07/06/2006 | US20060148840 Pyrrolodihydroisoquinolines as pde10 inhibitors |
07/06/2006 | US20060148838 Novel pyrrolodihydroisoquinolines useful in the treatment of cancer |
07/05/2006 | EP1675851A1 Method for producing n-substituted 3beta-aminonortropanes |
07/05/2006 | EP1259241B1 The use of scopolamine salts |
07/05/2006 | CN1798745A Novel 8-aza-bicyclo not 3.2.1|octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
07/04/2006 | US7071216 Anticancer agents |
07/04/2006 | US7070800 Inhalable powder containing tiotropium |
06/29/2006 | WO2006069277A1 TRICYCLIC δ-OPIOID MODULATORS |
06/29/2006 | WO2006069276A2 TRICYCLIC ō-OPIOID MODULATORS |
06/29/2006 | WO2006069125A1 Indazole-carboxamide compounds |
06/29/2006 | WO2006068904A1 Tetrahydroquinoline analogues as muscarinic agonists |
06/29/2006 | WO2006067584A1 8-aza-bicyclo (3.2.1) octane derivatives with an activity on chemokine ccr5 receptors |
06/29/2006 | WO2006052889A3 Quinolinone-carboxamide compounds |
06/29/2006 | US20060142331 of serotonin, dopamine and noradrenaline receptors; e.g. 2-(2,3-Dichlorophenoxymethyl)-8-methyl-3-(3-chlorophenyl)-8-aza-bicyclo[3.2.1]octane; antidepressant. anxiolytic agent; eating, bipolar disorders, obesity; drug, tobacco, alcohol abuse; neurodegenerative diseases |
06/29/2006 | CA2594602A1 8-aza-bicyclo (3.2.1) octane derivatives with an activity on chemokine ccr5 receptors |
06/29/2006 | CA2592464A1 Tricyclic .delta.-opioid modulators |
06/29/2006 | CA2591963A1 Tricyclic o-opioid modulators |
06/29/2006 | CA2591766A1 Tetrahydroquinoline analogues as muscarinic agonists |
06/29/2006 | CA2588037A1 Indazole-carboxamide compounds |
06/28/2006 | EP1673089A2 Phenyl-piperazine derivatives as modulators of muscarinic receptors |
06/28/2006 | EP1673083A2 N-substituted azacycles |
06/27/2006 | CA2408909C Azabicyclo[3.2.1]octane triazolyl tropane derivatives as ccrs5 modulators |
06/22/2006 | WO2006064340A2 Process for the preparation of n-acyl beta-aminoaldehydes |
06/22/2006 | US20060135764 Indazole-carboxamide compounds |
06/22/2006 | US20060135504 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines |
06/22/2006 | DE102004061008A1 3-Arylalkyl- und 3-Heteroarylalkyl-substituierte 1,2,4-Triazin-5(2H)-one 3-arylalkyl and heteroarylalkyl 3-substituted-1,2,4-triazine-5 (2H) -ones |
06/22/2006 | DE102004061006A1 3-Benzylthio-1,2,4-triazin-5(2H)-one 3-benzylthio-1,2,4-triazin-5 (2H) -ones |
06/21/2006 | EP1366049B1 Pirazino¬1'2':1,6|pyrido¬3,4-b|indole derivatives |
06/21/2006 | CN1791598A Benzimidazole-derivatives as factor Xa inhibitors |
06/15/2006 | WO2005007134A8 Powdery formulations for inhalation, containing a novel anticholinergic agent |
06/15/2006 | US20060128756 Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses |
06/15/2006 | US20060128637 Phenolic acid complexes of hyoscyamine and process for preparing the same |
06/13/2006 | USRE39128 Antibacteria drug; respiratory system disorders; otitis |
06/13/2006 | US7060717 Phosphodiesterase inhibitor; antiinflammatory agents; antiallergens; respiratory system disorders; wound healing agents |
06/13/2006 | CA2268954C Oxadiazoles, processes for their preparation and their use as medicaments |
06/08/2006 | WO2006044174A3 Aryl substituted 8-azabicyclo[3.2.1]octane compounds as ligands of the melanin concentrating hormone receptor |
06/08/2006 | WO2006021656A3 Aminopiperidine derivatives, preparation thereof and use thereof as melanocortin receptor agonists |
06/08/2006 | US20060122218 e.g. (2R,3S)-2-(2,3-Dichlorophenoxymethyl)-8-methyl-3-(2-thienyl-8-aza-bicyclo[3.2.1]octane; antidepressants; anxiolytic agents |
06/08/2006 | US20060122171 5-[(1-Ethylpiperidin-4-yl)amino]-3-[(3-fluorophenyl)(1H-imidazol-2-yl)methylidene]-1,3-dihydro-2H-indol-2-one; antiproliferative agents; modulating cell differentiation,migration, and chemoinvasion; endothelial growth factor-modulated diseases; antiarthritic agents; graft versus host diseases |
06/08/2006 | US20060122166 Chemokine receptors; inhibition of HIV replication; acquired immune deficiency syndrome (AIDS); cis N-(4-{2-[3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-4-phenylcyclohexyl)-1H-pyrazole-4-carboxamide |
06/07/2006 | EP1664036A1 Benzimidazolone compounds having 5-ht4 receptor agonistic activity |
06/07/2006 | EP1664031A2 Adamantane and azabicyclo-octane and nonane derivatives process of their preparation and their use as dpp-iv inhibitors |
06/07/2006 | EP1664017A1 Benzimidazolone and quinazolinone derivatives as agonists on human orl1 receptors |
06/07/2006 | EP1663220A1 Novel process, salts, compositions and use |
06/07/2006 | EP1492789B1 Tropane derivatives as ccr5 modulators |
06/07/2006 | CN1784393A Chemical compounds |
06/01/2006 | WO2006056081A1 Method for preparing hexahydro-8-hydroxy-2,6-methano-2h-chinolizin-3(4h)-one esters |
06/01/2006 | US20060116393 Substituted pyrido [2,1-a] isoquinoline derivatives |
05/31/2006 | EP1420644B1 Substituted propargylamines |
05/31/2006 | EP1163238B1 Chemokine recpetor binding heterocyclic compounds |
05/31/2006 | CN1780833A Tropane derivatives and their use as ace inhibitors |
05/30/2006 | US7053089 Such as 4-((methyl-pyrimidin-2-ylamino)-methyl)-piperidine-1-carboxylic acid benzyl ester; useful for pain relief; treating migraine, depression, anxiety, schizophrenia, Parkinson's disease, and stroke; N-methyl-D-aspartate (NMDA) |
05/30/2006 | CA2321380C 6-azauracil derivatives as thyroid receptor ligands |
05/23/2006 | US7049326 Altering a drug's distribution, metabolism and elimination properties, especially by modifying with aralkyl ester moieties to increase rate of metabolism to inactive and nontoxic metabolites when exposure is halted; surgery, riots |
05/18/2006 | WO2006052640A1 5-ht4 receptor agonist compounds |
05/18/2006 | WO2005067537A3 Muscarinic acetylcholine receptor antagonists |
05/18/2006 | US20060106219 making a fluoro radioactive material [18F]Fluorohaloalkanes radiotracer through halogenation, or solid phase synthesis; use in positron emission tomography (PET) studies |
05/17/2006 | EP1657239A2 Chromene compound |
05/16/2006 | US7045522 8-Azabicyclo[3.2.1]oct-2-ene and -octane derivatives technical field |
05/16/2006 | CA2237752C Novel substituted aryl compounds useful as modulators of acetylcholine receptors |
05/11/2006 | WO2005099706A3 Muscarinic acetylcholine receptor antagonists |
05/11/2006 | US20060100426 Containing a nortropane ring, e.g., 1-isopropyl-2-oxo-1,2-dihydroquinoline-3-carboxylic acid {(1S,3R,5R)-8-[2-hydroxy-3-(4-methanesulfonylpiperazin-1-yl)propyl]-8-azabicyclo[3.2.1]oct-3-yl}amide; 5-HT4 receptor agonists |
05/11/2006 | US20060100211 2-(3,4-dichlorophenylamino)-4-thiocyanato-5-nitro-pyrimidine; 2-chloro-4-(2-acetylamino-ethylamino)-5-trifluoromethyl-pyrimidine; lung cancer |
05/10/2006 | EP1655294A2 Chromene compound |
05/10/2006 | EP1655293A2 Chromene compound |
05/09/2006 | US7041674 nortropane or nortropene derivatives; antagonists of the M3 receptor for treating asthma, COPD, vagally induced sinus bradycardia, arrhythmia, gastrointestinal and urinary tract spasms, and menstrual pain |
05/09/2006 | US7041667 CCR5 modulators |
05/09/2006 | CA2418908C 1,4-dihydropyridines as bradykinin antagonists |
05/09/2006 | CA2395653C New inhalable powder containing tiotropium |
05/03/2006 | EP1651230A1 Medicaments for inhalation comprising steroids and a novel anticholinergic |
05/03/2006 | EP1651223A1 2-methoxymethyl-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octane tartrate salts |
05/03/2006 | EP0937069B1 Piperazino derivatives as neurokinin antagonists |
05/03/2006 | CN1768051A Substituted pyrazoles |
05/03/2006 | CN1767859A Improved radiometal complex compositions |
04/27/2006 | WO2006044174A2 Aryl substituted 8-azabicyclo[3.2.1]octane compounds as ligands of the melanin concentrating hormone receptor |
04/27/2006 | CA2581745A1 Aryl substituted 8-azabicyclo[3.2.1]octane compounds as ligands of the melanin concentrating hormone receptor |
04/26/2006 | EP1648888A1 N-(heterobicycloalkanes)-substituted indoles or heteroderivatives thereof |
04/26/2006 | EP1648462A1 Muscarinic acetylcholine receptor antagonists |
04/26/2006 | EP1648461A2 Muscarinic acetylcholine receptor antagonists |
04/26/2006 | EP1648460A1 Muscarinic acetylcholine receptor antagonists |
04/26/2006 | EP1379520B1 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists |
04/26/2006 | CN1764661A Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain. |
04/26/2006 | CN1764458A Bicyclic piperidine derivatives as melanocortin-4 receptor agonists |
04/20/2006 | WO2006021655A3 Oxopiperidine derivatives, preparation and therapeutic use thereof |
04/20/2006 | WO2006018609A3 Anti-inflammatory agents |
04/20/2006 | US20060083692 Combination of formoterol and a tiotropium salt |
04/19/2006 | EP1646365A1 Powdery formulations for inhalation, containing a novel anticholinergic agent |
04/19/2006 | CN1252068C Heteroaryl derivatives as superior ligands for nociceptin receptor ORL-1 |
04/18/2006 | US7030138 Benzamidine derivatives |
04/13/2006 | WO2006038989A1 Substituted arylamides |
04/13/2006 | US20060079503 Thiazolidinones and the use therof as polo-like kinase inhibitors |
04/12/2006 | EP1644398A1 Specific glucocorticosteroid compound having anti- inflammatory activity |
04/12/2006 | EP1644397A1 Specific glucocorticosteroid compound having anti- inflammatory activity |
04/12/2006 | EP1644343A1 5-substituted quinazolinone derivatives |
04/12/2006 | EP1643998A1 Dual nk1/nk3 antagonists for treating schizophrenia |