Patents
Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273)
11/2012
11/01/2012WO2012146724A2 Novel rock inhibitors
11/01/2012US20120276050 Methods and compositions of treating a flaviviridae family viral infection
11/01/2012CA2834387A1 Novel rock inhibitors
10/2012
10/31/2012EP2518069A1 Cyclic amine compound and acaricide
10/31/2012EP2516428A1 Tropinone benzylamines as beta-tryptase inhibitors
10/31/2012EP2516427A1 Radioiodinated tropane derivatives
10/31/2012CN102267992B Preparation method of pleuromutilin antibiotic
10/30/2012CA2474874C Anticholinergic agents, method for producing the same and use thereof as medicaments
10/26/2012WO2012143526A1 1,4-disubstituted 1,2,3-triazoles, methods for preparing same, and diagnostic and therapeutic uses thereof
10/26/2012CA2833648A1 1,4-disubstituted 1,2,3-triazoles, methods for preparing same, and diagnostic and therapeutic uses thereof
10/25/2012US20120269828 Anti-drug vaccines
10/24/2012EP2513099A1 Preparation of n-monofluoroalkyl tropanes
10/23/2012CA2488635C Antagonists of melanin concentrating hormone receptor
10/18/2012US20120264779 Quinolinone-carboxamide compounds as 5-ht4 receptor agonists
10/17/2012CN102741226A 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators
10/17/2012CN102731494A Novel forms of tiotropium bromide and processes for preparation thereof
10/16/2012US8288368 inhibitors of the C5a induced chemotaxis; psoriasis, ulcerative cholitis, glomerular nephritis, acute respiratory insufficiency, idiopathic fibrosis, rheumatoid arthritis and in the prevention and the treatment of injury caused by ischemia and reperfusion
10/10/2012CN102718760A Trospium chloride synthesis process
10/04/2012US20120251447 Radioiodinated tropane derivatives
10/03/2012CN101687801B Ethers of naphtalene carboxylic acid amides as cancer cure
09/2012
09/27/2012US20120245195 Novel monohydrate of azaadamantane derivatives
09/27/2012US20120244072 Preparation of n-monofluoroalkyl tropanes
09/25/2012US8273889 Method for producing 2-azaadamantane
09/20/2012US20120238740 Non-polar and polar leaving groups
09/20/2012US20120238600 Tropinone benzylamines as beta-tryptase inhibitors
09/19/2012EP2500345A1 8-azabicyclo[3.2.1]octane-8-carboxamide derivative
09/18/2012CA2531832C Powdery formulations for inhalation, containing a novel anticholinergic agent
09/18/2012CA2519110C Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain
09/13/2012WO2012091628A3 Substituted hydrogenated thieno-pyrrolo[3,2-c]pyridine, ligands, a pharmaceutical composition and a method for using the above
09/13/2012US20120232109 3-substituted sulfonyl piperidine derivative
09/12/2012CN101277955B Cyclic amine compound and pest control agent
09/11/2012US8263617 Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
09/11/2012US8263611 Hydrochloride salt of an azabicyclo[3.2.1]octane derivative
09/11/2012US8263605 Modulators of muscarinic receptors
09/11/2012CA2533792C Medicaments for inhalation comprising steroids and fluorene carboxylic acid esters
09/07/2012WO2012118462A1 Anhydrous crystalline form of tiotropium bromide
09/07/2012WO2012118461A1 Crystalline compound comprising tiotropium bromide
09/07/2012WO2012118460A1 Crystalline compound comprising tiotropium bromide
09/06/2012US20120225890 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes and parkinson's disease
09/06/2012US20120225884 Bridged piperidine derivatives
09/05/2012EP2493852A1 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators
09/05/2012CN102656170A Cyclic amine compound and acaricide
09/05/2012CN102656169A Radioiodinated tropane derivatives
09/05/2012CN101790529B 8-azabicyclo[3.2.1]octyl-2-hydroxybenzamide compounds as mu opioid receptor antagonists
09/05/2012CN101563319B Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives
08/2012
08/28/2012CA2671744C Compounds and compositions as protein kinase inhibitors
08/23/2012US20120214805 Bridged bicyclic piperidine derivatives and methods of use thereof
08/22/2012EP1881980B1 Novel crystalline forms of tiotropium bromide
08/22/2012CN101765599B Tropane derivatives useful as pesticides
08/21/2012US8247559 Process for preparing an intermediate to mu opioid receptor antagonists
08/16/2012WO2012108490A1 Isoquinoline amide derivative
08/16/2012US20120208841 Modulators of Cystic Fibrosis Transmembrane Conductance Regulator
08/15/2012CN102639531A Anhydrate of triotropium bromide
08/09/2012WO2012103806A1 Bicyclic heteroaryl compounds as gpr119 receptor agonists
08/09/2012US20120203004 process for the synthesis of alkyl/aralkyl (2s)-2-(tert-butoxycarbonyl)-amino-2-[-8-azabicyclo[3.2.1]oct-3-yl]-exo-acetate and analogs thereof: key intermediates for the preparation of dppiv inhibitors
08/09/2012US20120202796 Method for combating adverse effects arising from antipsychotic treatment
08/09/2012CA2828988A1 Bicyclic heteroaryl compounds as gpr119 receptor agonists
08/08/2012EP1740177B1 Muscarinic acetylcholine receptor antagonists
07/2012
07/26/2012US20120190845 Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
07/25/2012EP2477984A1 A method for the n-demethylation of n-methyl heterocycles
07/25/2012EP2477983A1 (4-phenyl-piperidin-1-yl)-[5-1h-pyrazol-4yl)-thiophen-3-yl]-methanone compounds and their use
07/25/2012EP1989202B1 Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
07/19/2012WO2012095781A1 Indazole derivatives as sodium channel inhibitors
07/18/2012CN1443167B Azacyclic compounds for use in treatment of 5-serotonin related diseases
07/18/2012CN102596949A 8-azabicyclo[3.2.1]octane-8-carboxamide derivative
07/18/2012CN102584815A Method for preparing tropisetron hydrochloride on large scale
07/18/2012CN102584814A Preparation method for 8-benzyl-3-(3-isopropyl-5-methyl-4H-1,2,4-triazole-4-base)-8-azabicyclo[3.2.1]octane
07/12/2012US20120178920 Method for preparing [18f]fallypride with low base concentration
07/11/2012EP1682142B1 M3 muscarinic acetylcholine receptor antagonists
07/10/2012CA2542110C Method for producing n-substituted 3.beta.-aminonortropanes
07/10/2012CA2507110C Carbamic acid esters with an anticholinergic action
07/10/2012CA2479652C Crystalline micronisate of tiotropium bromide
07/05/2012US20120172393 (4-Phenyl-piperidin-1-yl)-[5-(1H-pyrazol-4-yl)-thiophen-3-yl]-methanone Compounds and Their Use
07/05/2012CA2845505A1 Substituted hydrogenated thieno-pyrrolo[3,2-c]pyridine, ligands, a pharmaceutical composition and a method for using the above
07/04/2012CN102532128A Synthetic method of tropisetron and prepare method of hydrochloric acid tropisetron
06/2012
06/28/2012WO2012087519A1 Compositions and methods for modulating fxr
06/28/2012CA2819825A1 Compositions and methods for modulating fxr
06/27/2012EP2185553B1 Amidoalkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
06/27/2012CN102516241A CNS active fused bicycloheterocycle substituted azabicyclic alkane derivatives
06/26/2012US8207191 Process, salts, composition and use
06/21/2012WO2012082381A1 Indeno- fused ring compounds having photochromic properties
06/21/2012CA2821392A1 Indeno-fused ring compounds having photochromic properties
06/20/2012EP2465850A1 Therapeutic compounds
06/20/2012EP1960347B1 17-beta-hydroxysteroid dehydrogenase type 3 (17beta-hsd3) inhibitors
06/14/2012WO2012050315A3 Azetidinium salt as fp-cit precursor, method for selectively preparing same, and fp-cit synthesis
06/13/2012EP2462140A2 Anhydrate of triotropium bromide
05/2012
05/31/2012WO2012069275A1 Glycine derivatives and their use as muscarinic receptor antagonists
05/31/2012US20120134934 Glycine derivatives and medicinal compositions thereof
05/31/2012CA2820600A1 Glycine derivatives and their use as muscarinic receptor antagonists
05/30/2012CN101863885B Method for preparing tiotropium bromide
05/29/2012US8188280 3-substituted sulfonyl piperidine derivative
05/22/2012US8183366 Chemokine receptor antagonists
05/16/2012CN102459248A 作为PI3K/mTOR抑制剂的苯并氧杂环庚三烯以及它们使用与制造方法 As the PI3K / mTOR inhibitor benzoxepin-triene and their method of use and manufacture
05/15/2012USRE43390 Pleuromutilin derivatives as antimicrobials
05/15/2012US8178668 2-aminopyridine kinase inhibitors
05/10/2012US20120115853 Aryl- and Heteroarylcarbonyl derivatives of substituted nortropanes, medicaments containing such compounds and their use
05/08/2012CA2531905C Specific glucocorticosteroid compound having anti-inflammatory activity
05/03/2012WO2012055018A1 Therapeutic compositions for diabetic symmetrical polyneuropathy
05/03/2012US20120108575 Heterocyclic-substituted piperidine compounds and the uses thereof
05/03/2012CA2804797A1 Therapeutic compositions for diabetic symmetrical polyneuropathy and/or tactile allodynia
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