Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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11/01/2012 | WO2012146724A2 Novel rock inhibitors |
11/01/2012 | US20120276050 Methods and compositions of treating a flaviviridae family viral infection |
11/01/2012 | CA2834387A1 Novel rock inhibitors |
10/31/2012 | EP2518069A1 Cyclic amine compound and acaricide |
10/31/2012 | EP2516428A1 Tropinone benzylamines as beta-tryptase inhibitors |
10/31/2012 | EP2516427A1 Radioiodinated tropane derivatives |
10/31/2012 | CN102267992B Preparation method of pleuromutilin antibiotic |
10/30/2012 | CA2474874C Anticholinergic agents, method for producing the same and use thereof as medicaments |
10/26/2012 | WO2012143526A1 1,4-disubstituted 1,2,3-triazoles, methods for preparing same, and diagnostic and therapeutic uses thereof |
10/26/2012 | CA2833648A1 1,4-disubstituted 1,2,3-triazoles, methods for preparing same, and diagnostic and therapeutic uses thereof |
10/25/2012 | US20120269828 Anti-drug vaccines |
10/24/2012 | EP2513099A1 Preparation of n-monofluoroalkyl tropanes |
10/23/2012 | CA2488635C Antagonists of melanin concentrating hormone receptor |
10/18/2012 | US20120264779 Quinolinone-carboxamide compounds as 5-ht4 receptor agonists |
10/17/2012 | CN102741226A 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators |
10/17/2012 | CN102731494A Novel forms of tiotropium bromide and processes for preparation thereof |
10/16/2012 | US8288368 inhibitors of the C5a induced chemotaxis; psoriasis, ulcerative cholitis, glomerular nephritis, acute respiratory insufficiency, idiopathic fibrosis, rheumatoid arthritis and in the prevention and the treatment of injury caused by ischemia and reperfusion |
10/10/2012 | CN102718760A Trospium chloride synthesis process |
10/04/2012 | US20120251447 Radioiodinated tropane derivatives |
10/03/2012 | CN101687801B Ethers of naphtalene carboxylic acid amides as cancer cure |
09/27/2012 | US20120245195 Novel monohydrate of azaadamantane derivatives |
09/27/2012 | US20120244072 Preparation of n-monofluoroalkyl tropanes |
09/25/2012 | US8273889 Method for producing 2-azaadamantane |
09/20/2012 | US20120238740 Non-polar and polar leaving groups |
09/20/2012 | US20120238600 Tropinone benzylamines as beta-tryptase inhibitors |
09/19/2012 | EP2500345A1 8-azabicyclo[3.2.1]octane-8-carboxamide derivative |
09/18/2012 | CA2531832C Powdery formulations for inhalation, containing a novel anticholinergic agent |
09/18/2012 | CA2519110C Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain |
09/13/2012 | WO2012091628A3 Substituted hydrogenated thieno-pyrrolo[3,2-c]pyridine, ligands, a pharmaceutical composition and a method for using the above |
09/13/2012 | US20120232109 3-substituted sulfonyl piperidine derivative |
09/12/2012 | CN101277955B Cyclic amine compound and pest control agent |
09/11/2012 | US8263617 Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
09/11/2012 | US8263611 Hydrochloride salt of an azabicyclo[3.2.1]octane derivative |
09/11/2012 | US8263605 Modulators of muscarinic receptors |
09/11/2012 | CA2533792C Medicaments for inhalation comprising steroids and fluorene carboxylic acid esters |
09/07/2012 | WO2012118462A1 Anhydrous crystalline form of tiotropium bromide |
09/07/2012 | WO2012118461A1 Crystalline compound comprising tiotropium bromide |
09/07/2012 | WO2012118460A1 Crystalline compound comprising tiotropium bromide |
09/06/2012 | US20120225890 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes and parkinson's disease |
09/06/2012 | US20120225884 Bridged piperidine derivatives |
09/05/2012 | EP2493852A1 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators |
09/05/2012 | CN102656170A Cyclic amine compound and acaricide |
09/05/2012 | CN102656169A Radioiodinated tropane derivatives |
09/05/2012 | CN101790529B 8-azabicyclo[3.2.1]octyl-2-hydroxybenzamide compounds as mu opioid receptor antagonists |
09/05/2012 | CN101563319B Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives |
08/28/2012 | CA2671744C Compounds and compositions as protein kinase inhibitors |
08/23/2012 | US20120214805 Bridged bicyclic piperidine derivatives and methods of use thereof |
08/22/2012 | EP1881980B1 Novel crystalline forms of tiotropium bromide |
08/22/2012 | CN101765599B Tropane derivatives useful as pesticides |
08/21/2012 | US8247559 Process for preparing an intermediate to mu opioid receptor antagonists |
08/16/2012 | WO2012108490A1 Isoquinoline amide derivative |
08/16/2012 | US20120208841 Modulators of Cystic Fibrosis Transmembrane Conductance Regulator |
08/15/2012 | CN102639531A Anhydrate of triotropium bromide |
08/09/2012 | WO2012103806A1 Bicyclic heteroaryl compounds as gpr119 receptor agonists |
08/09/2012 | US20120203004 process for the synthesis of alkyl/aralkyl (2s)-2-(tert-butoxycarbonyl)-amino-2-[-8-azabicyclo[3.2.1]oct-3-yl]-exo-acetate and analogs thereof: key intermediates for the preparation of dppiv inhibitors |
08/09/2012 | US20120202796 Method for combating adverse effects arising from antipsychotic treatment |
08/09/2012 | CA2828988A1 Bicyclic heteroaryl compounds as gpr119 receptor agonists |
08/08/2012 | EP1740177B1 Muscarinic acetylcholine receptor antagonists |
07/26/2012 | US20120190845 Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor |
07/25/2012 | EP2477984A1 A method for the n-demethylation of n-methyl heterocycles |
07/25/2012 | EP2477983A1 (4-phenyl-piperidin-1-yl)-[5-1h-pyrazol-4yl)-thiophen-3-yl]-methanone compounds and their use |
07/25/2012 | EP1989202B1 Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
07/19/2012 | WO2012095781A1 Indazole derivatives as sodium channel inhibitors |
07/18/2012 | CN1443167B Azacyclic compounds for use in treatment of 5-serotonin related diseases |
07/18/2012 | CN102596949A 8-azabicyclo[3.2.1]octane-8-carboxamide derivative |
07/18/2012 | CN102584815A Method for preparing tropisetron hydrochloride on large scale |
07/18/2012 | CN102584814A Preparation method for 8-benzyl-3-(3-isopropyl-5-methyl-4H-1,2,4-triazole-4-base)-8-azabicyclo[3.2.1]octane |
07/12/2012 | US20120178920 Method for preparing [18f]fallypride with low base concentration |
07/11/2012 | EP1682142B1 M3 muscarinic acetylcholine receptor antagonists |
07/10/2012 | CA2542110C Method for producing n-substituted 3.beta.-aminonortropanes |
07/10/2012 | CA2507110C Carbamic acid esters with an anticholinergic action |
07/10/2012 | CA2479652C Crystalline micronisate of tiotropium bromide |
07/05/2012 | US20120172393 (4-Phenyl-piperidin-1-yl)-[5-(1H-pyrazol-4-yl)-thiophen-3-yl]-methanone Compounds and Their Use |
07/05/2012 | CA2845505A1 Substituted hydrogenated thieno-pyrrolo[3,2-c]pyridine, ligands, a pharmaceutical composition and a method for using the above |
07/04/2012 | CN102532128A Synthetic method of tropisetron and prepare method of hydrochloric acid tropisetron |
06/28/2012 | WO2012087519A1 Compositions and methods for modulating fxr |
06/28/2012 | CA2819825A1 Compositions and methods for modulating fxr |
06/27/2012 | EP2185553B1 Amidoalkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists |
06/27/2012 | CN102516241A CNS active fused bicycloheterocycle substituted azabicyclic alkane derivatives |
06/26/2012 | US8207191 Process, salts, composition and use |
06/21/2012 | WO2012082381A1 Indeno- fused ring compounds having photochromic properties |
06/21/2012 | CA2821392A1 Indeno-fused ring compounds having photochromic properties |
06/20/2012 | EP2465850A1 Therapeutic compounds |
06/20/2012 | EP1960347B1 17-beta-hydroxysteroid dehydrogenase type 3 (17beta-hsd3) inhibitors |
06/14/2012 | WO2012050315A3 Azetidinium salt as fp-cit precursor, method for selectively preparing same, and fp-cit synthesis |
06/13/2012 | EP2462140A2 Anhydrate of triotropium bromide |
05/31/2012 | WO2012069275A1 Glycine derivatives and their use as muscarinic receptor antagonists |
05/31/2012 | US20120134934 Glycine derivatives and medicinal compositions thereof |
05/31/2012 | CA2820600A1 Glycine derivatives and their use as muscarinic receptor antagonists |
05/30/2012 | CN101863885B Method for preparing tiotropium bromide |
05/29/2012 | US8188280 3-substituted sulfonyl piperidine derivative |
05/22/2012 | US8183366 Chemokine receptor antagonists |
05/16/2012 | CN102459248A 作为PI3K/mTOR抑制剂的苯并氧杂环庚三烯以及它们使用与制造方法 As the PI3K / mTOR inhibitor benzoxepin-triene and their method of use and manufacture |
05/15/2012 | USRE43390 Pleuromutilin derivatives as antimicrobials |
05/15/2012 | US8178668 2-aminopyridine kinase inhibitors |
05/10/2012 | US20120115853 Aryl- and Heteroarylcarbonyl derivatives of substituted nortropanes, medicaments containing such compounds and their use |
05/08/2012 | CA2531905C Specific glucocorticosteroid compound having anti-inflammatory activity |
05/03/2012 | WO2012055018A1 Therapeutic compositions for diabetic symmetrical polyneuropathy |
05/03/2012 | US20120108575 Heterocyclic-substituted piperidine compounds and the uses thereof |
05/03/2012 | CA2804797A1 Therapeutic compositions for diabetic symmetrical polyneuropathy and/or tactile allodynia |