Patents for C07D - Heterocyclic compounds (10,420) |
---|
02/03/2005 | WO2005009948A2 Peptide inhibitors of beta-lactamases |
02/03/2005 | WO2005009539A2 Compounds for inflammation and immune-related uses |
02/03/2005 | WO2004094369A3 Stabilized derivatives of ascorbic acid |
02/03/2005 | WO2004083175A3 Methods for identifying enzyme inhibitors and protein kinases |
02/03/2005 | WO2004074242A3 Halogenated oxime derivatives and the use thereof as latent acids |
02/03/2005 | US20050027129 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them |
02/03/2005 | US20050026968 Heterocyclic amides with anti-tuberculosis activity |
02/03/2005 | US20050026922 For treating CNS or other disorders, including concurrent treatment of disorders such as schizophrenia and depression; side effect reduction; for example, (7R,9aS)-trans-7-[6-(2,6-Dimethyl-piperidin-1-ylmethyl)-pyridin-2-yloxymethyl]-2-(5-fluoro-benzo[d]isoxazol-3-yl)-octahydro-pyrido[1,2-a]pyrazine |
02/03/2005 | CA2533594A1 Compounds for inflammation and immune-related uses |
02/03/2005 | CA2533392A1 Diphenyl substituted cycloalkanes, compositions containing such compounds and methods of use |
02/03/2005 | CA2532808A1 Piperidine derivatives as melanocortin-4 receptor agonists |
02/03/2005 | CA2531492A1 Compositions for purifying and crystallizing molecules of interest |
02/03/2005 | CA2530047A1 17-acetamido-4-azasteroid derivatives as androgen receptor modulators |
02/02/2005 | EP1501830A1 7-aryl-3,9-diazabicyclo[3.3.1]non-6-ene derivatives and their use as renin inhibitors in the treatment of hypertension, cardiovascular or renal diseases |
02/02/2005 | EP1501801A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors |
02/02/2005 | CN1572792A Pyrazolo [4, 3-d] pyrimidine derivatives |
02/02/2005 | CN1187351C Bispidine compounds, their use and preparation method, intermediate and pharmaceutical compositions containing same |
02/02/2005 | CN1187350C Bispidine compounds, their use and preparation method, intermediate and pharmaceutical compositions containing same |
02/01/2005 | US6849629 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders |
01/27/2005 | WO2005007625A2 Heterocyclic amides with anti-tuberculosis activity |
01/27/2005 | WO2005007624A2 Compositions of orthogonal glutamyl-trna and aminoacyl trna synthetase pairs and uses thereof |
01/27/2005 | WO2005007623A2 Inhibition of syk kinase expression |
01/27/2005 | WO2005007622A2 OPTICALLY ACTIVE QUATERNARY AMMONIUM SALT, PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING OPTICALLY ACTIVE α-AMINO ACID DERIVATIVE WITH THE SAME |
01/27/2005 | WO2005006899A1 Treatment of male sexual dysfunction |
01/27/2005 | WO2004101512A3 Naphthyridine integrase inhibitors |
01/27/2005 | WO2004099130A3 1,2-diarylimidazoles useful as inhibitors of cox |
01/27/2005 | WO2004098518A3 Pyrazole-amide compounds useful as kinase inhibitors |
01/27/2005 | WO2004087654A3 Phospholipase c inhibitors for use in treating inflammatory disorders |
01/27/2005 | WO2004069794B1 New arylpiperazinyl compounds |
01/27/2005 | US20050020670 Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)-1,3-dihydroisobenzofuran |
01/27/2005 | US20050020635 C7 carbamoyloxy substituted taxane compositions |
01/27/2005 | US20050020568 Derivatives of 5-(pyridin-3-yl)-1-azabicyclo[3.2.1] octane, the preparation thereof and the application of same in therapeutics |
01/27/2005 | US20050020481 Ion channel modulating compounds and uses thereof |
01/27/2005 | CA2533177A1 Treatment of male sexual dysfunction |
01/27/2005 | CA2531069A1 Inhibition of syk kinase expression |
01/26/2005 | EP1499613A1 Thioxanthine derivatives as myeloperoxidase inhibitors |
01/26/2005 | EP1499607A1 4-(piperidyl- and pyrrolidyl-alkyl-ureido)-quinolines as urotensin ii receptor antagonists |
01/26/2005 | EP1499589A1 Derivatives of n-phenyl(piperidin-2-yl)methyl benzamide, the preparation method thereof and application of same in therapeutics |
01/26/2005 | EP1499312A1 The use of hydroxypyridone-derivatives in wound healing |
01/26/2005 | EP1084109B1 2-aminopyridines containing fused ring substituents as nitric oxide synthase inhibitors |
01/26/2005 | EP0975637B1 Amidino-camptothecin derivatives |
01/26/2005 | CN1571770A Aralkyl-tetrahydro-pyridines, their preparation and pharmaceutical compositions containing same |
01/26/2005 | CN1571670A Treating sexual desire disorders with flibanserin |
01/26/2005 | CN1186340C C10 carbonate substituted taxanes as antitumor agents |
01/25/2005 | CA2159478C (s)-alpha-phenyl-2-pyridineethanamine (s)-malate and its use as a medicament |
01/20/2005 | WO2005005382A2 Compounds, compositions and methods |
01/20/2005 | WO2005005381A2 Multi-mode internal imaging |
01/20/2005 | WO2005005380A2 17-acetamido-4-azasteroid derivatives as androgen receptor modulators |
01/20/2005 | WO2005005378A2 Indolinone hydrazides as c-met inhibitors |
01/20/2005 | WO2004100865A3 New benzimidazole derivatives |
01/20/2005 | WO2004083177A3 Linear chain substituted monocyclic and bicyclic derivatives as factor xa inhibitors |
01/20/2005 | WO2004069793A3 Novel 2-substituted cyclic amines as calcium sensing receptor modulators |
01/20/2005 | US20050014814 Methods and compositions for the treatment and prevention of tumors, tumor-related disorders and cachexia |
01/20/2005 | US20050014795 Aralkyl-tetrahydro-pyridines, their preparation and pharmaceutical compositions containing same |
01/20/2005 | US20050014788 Piperidine derivatives and their use as modulators of chemokine receptor activity (especially ccr5) |
01/20/2005 | US20050014772 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for preparing them |
01/20/2005 | US20050014766 Use of n-(indolecarbonyl-)piperazine derivatives |
01/20/2005 | DE10329860A1 Sulfonamidderivate polycyclischer Farbstoffe für analytische Anwendungen Sulfonamide derivatives of polycyclic dyes for analytical applications |
01/20/2005 | CA2530536A1 Multi-mode internal imaging |
01/20/2005 | CA2530025A1 17-acetamido-4-azasteroid derivatives as androgen receptor modulators |
01/20/2005 | CA2529622A1 Indolinone hydrazides as c-met inhibitors |
01/19/2005 | EP1497450A2 Methods for identifying compounds that modulate enzymatic activity |
01/19/2005 | EP1497290A1 Process for preparing acid salts of gemifloxacin |
01/19/2005 | EP1497266A2 Quinoline derivatives and their use as 5-ht6 ligands |
01/19/2005 | EP0994880B1 Crystalline macrolides and process for their preparation |
01/19/2005 | CN1568207A 2-amino-6-(2, 4, 5-substituted-phenyl)-pyridines |
01/19/2005 | CN1568189A [[2-(amino-3, 4-dioxo-1-cyclobuten-1-yl)amino]alkyl]-acid derivatives for the treatment of pain |
01/19/2005 | CN1568184A Nicontinic acetylcholine receptor antagonists in the treatment of restless legs syndrome |
01/19/2005 | CN1566096A Prostaglandin agonists and their use to treat bonedisorders |
01/19/2005 | CN1185234C Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives |
01/19/2005 | CN1185227C Novel compounds |
01/18/2005 | US6844349 Salt forms of E-2-methoxy-N-(3-{4-[3 methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide and method of production |
01/18/2005 | US6844340 Tricyclic 2-pyrimidone compounds useful as HIV reverse transcriptase inhibitors |
01/13/2005 | WO2005003089A2 7-ethynyl-2,4,9-trithiaadamantane and related methods |
01/13/2005 | WO2005003088A2 Esters with antimicrobial, bioresistant and fungal resistant properties |
01/13/2005 | WO2005003087A2 Oxazole derivatives as antibacterial agents |
01/13/2005 | WO2005003086A2 Sulfonic acid derivatives of polycyclic dyes used for analytical applications |
01/13/2005 | WO2004087650A3 Process and intermediates for the preparation of beta-amino acid amide dipeptidyl peptidase-iv inhibitors |
01/13/2005 | WO2004076406A3 Losartan potassium polymorphs and process for the preparation thereof |
01/13/2005 | US20050009889 Synergistic fungicide compositions containing at least one n-(2-pyridinyl) 1-3-pyridinecarboxamide derivative and one or more further fungicides useful for controlling fungal plant diseases |
01/13/2005 | US20050009840 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer |
01/13/2005 | US20050009054 Compounds having a fused, bicyclic moiety for binding to the minor groove of dsDNA |
01/12/2005 | EP1496060A1 Antitumoral analogs of ET-743 |
01/12/2005 | EP1495023A1 Novel 1,2,3-substituted indolizine derivatives, inhibitors of fgfs, method for making same and pharmaceutical compositions containing same |
01/12/2005 | EP1305314B1 Crystalline therapeutic agent |
01/12/2005 | EP0991628B1 QUINOLINE AND QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR P56lck TYROSINE KINASES |
01/12/2005 | CN1184220C Process for preparation of 5-carboxy-phthalide and its use for production of CITALOPRAM |
01/12/2005 | CN1184208C Substituted benzimidazoles and their prepn. and use |
01/11/2005 | CA2100924C Oxadiazine derivatives |
01/06/2005 | WO2005000807A2 Benzodiazepine cgrp receptor antagonists |
01/06/2005 | WO2005000806A2 Ligands for nicotinic acetylcholine receptors, and methods of making and using them |
01/06/2005 | WO2005000804A2 Substituted indoles and a process for preparing substituted indoles |
01/06/2005 | WO2005000803A2 Asymmetric urea compound and process for producing asymmetric compound by asymmetric conjugate addition reaction with the same as catalyst |
01/06/2005 | WO2004087646A3 Pyrrolidino-1,2-dicarboxy-1-(phenylamide)-2-(4-(3-oxo-morpholino-4-yl)-phenylamide) derivatives and related compounds for use as inhibitors of coagulation factor xa in the treatment of thrombo-embolic diseases |
01/06/2005 | WO2003042177A8 Piperidine derivatives and their use as modulators of chemokine receptor activity (especially ccr5) |
01/06/2005 | US20050004204 2-Iminopyrrolidine derivatives |
01/06/2005 | US20050004197 Thrombin receptors antagonists; oral efficacy |
01/06/2005 | US20050004176 Pyrazole-amide compounds useful as kinase inhibitors |
01/06/2005 | US20050004151 Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators |
01/06/2005 | US20050004148 Human immunodeficiency and hepatitis B infections; high activity, low toxicity |