Patents for C07D - Heterocyclic compounds (10,420) |
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08/11/2005 | US20050176964 Nicotinamide derivatives useful as p38 inhibitors |
08/11/2005 | US20050176718 Aza- and polyaza-naphthalenyl carboxamides useful as HIV integrase inhibitors |
08/11/2005 | US20050176700 (2-methoxyphenyl)acetic acid-7-{4-[3-(2-methoxybenzyloxy)-propoxy]phenyl}-3-(2-thiophen-2-ylacetyl)-3,9-diazabicyclo[3.3.1]non-6-en-6-yl-methyl ester; metabolically stable, orally bioavailable and sufficiently soluble; industrial scale; non-peptidic nature, low molecular weight |
08/11/2005 | US20050176683 Hexa-/Tetra-hydro-pyrrolo[1,2-a]imidazole-2,5-dione derivatives; solid phase synthesis |
08/10/2005 | EP1561752A1 Heterocyclic compounds that are inhibitors of the enzyme DPP-IV |
08/10/2005 | EP1086093B1 Tetrahydroquinoline derivatives as glycine antagonists |
08/10/2005 | EP0968158B1 Method of preparing substituted indanones, the substituted indanones and metallocenes prepared therefrom |
08/10/2005 | CN1653064A Oxazolidinone derivatives, processes for their preparation, and pharmaceutical compositions containing them |
08/10/2005 | CN1652771A Annelated pyrrole compounds as proton pump inhibitors for treating ulcer |
08/10/2005 | CN1214029C 4-amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4-tetrahydroi-soquinol-2-yl)-5-(2-pyridyl) quinazo line mesylat and polymorphs |
08/10/2005 | CN1214013C HIV replication inhibiting pyrimidines |
08/09/2005 | CA2327029C Method for making 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinoline |
08/09/2005 | CA2310627C Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance p antagonists |
08/04/2005 | WO2005035489A3 Improved synthesis of discodermolide and variants thereof |
08/04/2005 | WO2005000804A3 Substituted indoles and a process for preparing substituted indoles |
08/04/2005 | US20050171354 Heterocyclic amines such as (2S,3S)-3-((1R)-6-methoxy-1-methyl -1-trifluoromethylisochroman-7-yl)methylamino-2-phenyl piperidine, used as analgesics, antiinflammatory agents, or for prophylaxis of cardiovascular disorders |
08/04/2005 | US20050171118 Central nervous system, gastrointestinal and psycological disorders; such as 3-(4-chlorobenzenesulfonyl)-2-methyl-7-piperazin-1-yl-1H-indole; synthesis |
08/04/2005 | US20050171061 Phenylsulfanylphenyl and phenyloxyphenyl substituted piperazine compounds; glycine transport inhibitors; for the treatment of psychoses and convulsive disorders: epilepsy, spasticity, and myoclonus |
08/03/2005 | EP1559717A2 Oxabispidine compounds useful in the treatment of cardiac arrythmias |
08/03/2005 | EP1558599A2 Heteroarylpiperidine modulators of chemokine receptor activity |
08/03/2005 | CN1649870A 7-aryl-3, 9-diazabicyclo(3.3.1)non-6-ene derivatives and their use as renin inhibitors in the treatment of hypertension, cardiovascular or renal diseases |
08/03/2005 | CN1649868A Process for preparing acid salts of gemifloxacin |
08/03/2005 | CN1649867A Novel 1, 2, 3-substituted indolizine derivatives, inhibitors of FGFs, method for making same and pharmaceutical compositions containing same |
08/03/2005 | CN1649842A 2, 6-quinolinyl and 2, 6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors |
08/02/2005 | CA2362339C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives |
08/02/2005 | CA2362337C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives |
08/02/2005 | CA2170020C Retroviral protease inhibiting compounds |
07/28/2005 | WO2005033073A3 Spirocyclic heterocyclic derivatives and methods of their use |
07/28/2005 | WO2005016875A3 Geometrically restricted 3-cyclopentylidene-1,3-dihydroindol-2-ones as potent protein kinase inhibitors |
07/28/2005 | US20050165244 precipitating the citalopram base in crystalline form, and transforming the base into a pharmaceutically acceptable citalopram salt; useful for removing intermediates which are structurally closely related to citalopram |
07/28/2005 | US20050165092 Crystalline base of citalopram |
07/28/2005 | US20050165051 Taxanes having a C7 carbonate substituent |
07/28/2005 | US20050165022 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
07/28/2005 | US20050163698 Novel graphite nanocatalysts |
07/27/2005 | EP1556382A1 3-phenyl substituted pyridoindolone, preparation and therapeutic use thereof |
07/27/2005 | EP1556370A1 Method for the synthesis of a benzimidazole compound |
07/27/2005 | EP1309555B1 Process for making amlodipine maleate |
07/27/2005 | EP1287004B1 Synthetic process for the manufacture of an ecteinascidin compound |
07/27/2005 | CN1646531A Thioxanthine derivatives as myeloperoxidase inhibitors |
07/27/2005 | CN1646528A Polycyclic compounds as potent alpha2-adrenoceptor antagonists |
07/27/2005 | CN1646165A Combinations of peroxisome proliferator-activated receptor (PPAR) activator(s) and sterol absorption inhibitor(s) and treatments for vascular indications |
07/26/2005 | US6921760 Psychotherapeutic agents. |
07/26/2005 | US6921759 For therapy, prophylaxis or delaying the onset of AIDS and infection by HIV |
07/26/2005 | CA2253948C Carboline derivatives |
07/21/2005 | WO2005066148A1 Diarylmethyl piperazine derivatives, preparations thereof and uses thereof |
07/21/2005 | WO2005035490A3 PROCESS FOR SYNTHESIZING d-TOCOTRIENOLS |
07/21/2005 | US20050159466 Production method of isoxazolidinedione compound |
07/21/2005 | US20050159450 Derivative of n-[phenyl(piperidin-2-yl)methyl]benzamide, the preparation method thereof and application of same in therapeutics |
07/21/2005 | US20050159438 Spirocyclic heterocyclic derivatives and methods of their use |
07/21/2005 | US20050159424 pharmaceutically-acceptable salts, prodrugs, solvates, isomers, and/or hydrates thereof, wherein Q is an optionally-substituted phenyl, pyridyl, pyridazinyl, pyrimidinyl, or pyrazinyl ring; R2 is alkyl or an amino group as defined herein; and Z is optionally-substituted oxadiazolyl or C( .dbd. O)NR6, |
07/21/2005 | CA2552851A1 Diarylmethyl piperazine derivatives, preparations thereof and uses thereof |
07/20/2005 | EP1303514B1 Process for preparing azacycloalkanoylaminothiazoles |
07/20/2005 | CN1642954A Tricyclic 2-pyrimidone compounds useful as HIV reverse transcriptase inhibitors |
07/20/2005 | CN1642942A Method for manufacture of sertindole |
07/20/2005 | CN1642931A Sulfonylamino-derivatives as novel inhibitors of histone deacetylase |
07/20/2005 | CN1640877A Novel spiro compounds |
07/20/2005 | CN1211386C Antitumoral analogue of Et-743 |
07/20/2005 | CN1211368C Amorphous torasemide modification |
07/20/2005 | CN1211367C Prostaglandin agonists and their use to treat bone disorders |
07/20/2005 | CN1211365C Novel salt of perindopril and pharmacetuical composition contg. same |
07/19/2005 | US6919087 And an excipient wherein the pH is within the range of 5.5-7.0; stability; dosage forms |
07/14/2005 | WO2005023761A3 Cytokine inhibitors |
07/14/2005 | WO2004098528A3 Pyrazole-amine compounds useful as kinase inhibitors |
07/14/2005 | US20050154199 Bridged macrocyclic module compositions |
07/14/2005 | US20050154057 Crystalline form of y-aminobutyric acid analog |
07/14/2005 | US20050154051 Method for the preparation of escitalopram |
07/14/2005 | US20050153952 Methods for inhibiting sterol absorption |
07/14/2005 | US20050153942 Heterocyclic inhibitors of MEK and methods of use thereof |
07/14/2005 | US20050151467 Electrochromic salts, solutions, and devices |
07/13/2005 | EP1551802A1 Indole-3-sulphur derivatives |
07/13/2005 | EP1427711B1 Oxazolidinone and/or isoxazoline derivatives as antibacterial agents |
07/13/2005 | CN1639136A Oxazolidinone and/or isoxazoline as antibacterial agents |
07/13/2005 | CN1639115A Semicarbazide derivatives and their use as antithrombotics |
07/13/2005 | CN1638768A Thiazole and oxazole derivatives that modulate PPAR activity |
07/13/2005 | CN1636991A Sodium-hydrogen exchanger type 1 inhibitor crystals |
07/13/2005 | CN1210279C Thiazolo (4,5-D) pyrimidine compounds |
07/13/2005 | CN1210274C Piperazine and piperidine derivatives |
07/12/2005 | US6916815 C-6 modified indazolylpyrrolotriazines |
07/12/2005 | CA2146047C 13-substituted milbemycin derivatives, their preparation and use |
07/07/2005 | WO2005061484A1 1,2,3,4-tetrahydroisoquinoline derivatives, preparations thereof and uses thereof |
07/07/2005 | WO2005037052A3 Binding assay with labelled bispidine variant |
07/07/2005 | WO2005033071A3 Toluene methylation process |
07/07/2005 | WO2005009954A3 Method for modulating calcium ion-release-activated calcium ion channels |
07/07/2005 | US20050148777 (2R)-6-chloro-7-isobutyl-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid; cyclooxygenase-2 mediated disorders |
07/07/2005 | US20050148633 Method for modulating calcium ion-release-activated calcium ion channels |
07/07/2005 | US20050148622 Process for preparing acid salts of gemifloxacin |
07/07/2005 | US20050148591 Tartrate salts of 5,8,14-triazatetracyclo [10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaen and pharmaceutical compositions thereof |
07/07/2005 | US20050148546 Solid phase acid hydrolysis on cation exchange resin; high yield, stability and purity with fewer clean up steps; reduced acid use and recycle; low cost, industrial scale production of glucosamine and salts |
07/07/2005 | CA2550643A1 1,2,3,4-tetrahydroisoquinoline derivatives, preparations thereof and uses thereof |
07/06/2005 | EP1549143A2 Antibacterial pyrazole carboxylic acid hydrazides |
07/06/2005 | EP1549141A2 Methods and compositions for the treatment of autoimmune disorders using clofarabine |
07/06/2005 | EP1212320B1 Phenylpiperazines as serotonin reuptake inhibitors |
07/06/2005 | CN1636005A Benzothiazinone and benzoxazinone compounds |
07/05/2005 | US6913740 Graphite nanocatalysts |
06/30/2005 | WO2005058895A1 Novel crystalline forms of 2, 3 dimethyl-8- (2, 6-dimethylbenzylamino) -n-hydroxyethyl-imidazo [1, 2-a] pyridine-6-carboxamide mesylate salt. |
06/30/2005 | WO2005058815A2 Ip-10 antibodies and their uses |
06/30/2005 | WO2005058814A2 Biocidal siloxane coating material containing n-halogenated amine and amide functional groups |
06/30/2005 | WO2005058321A1 USE OF METABOTROPIC GLUTAMATE RECEPTOR 5 (mGLuR5) ANTAGONISTS FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS. |
06/30/2005 | WO2004089890A3 Process and intermediates for preparing benzazepines |
06/30/2005 | WO2004087649A3 Benodiazepine spirohydantoin cgrp receptor antagonists |