Patents for C07D - Heterocyclic compounds (10,420) |
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06/02/2005 | CA2546093A1 5-substituted imidazoles |
06/01/2005 | EP1534730A2 Modified transferin-antibody fusion proteins |
06/01/2005 | EP1534717A1 Beta-lactamase inhibitor prodrug |
06/01/2005 | EP1534695A2 Tyrosine kinase inhibitors |
06/01/2005 | EP1534677A1 Piperidine derivatives and their use as selective inhibitors of mip-1alpha binding to its receptor ccr1 |
06/01/2005 | EP0991625B1 Inhibitors of factor xa with a neutral p1 specificity group |
06/01/2005 | CN1622946A Methods of treating p38 kinase-associated conditions and pyrrolotriazine compounds useful as kinase inhibitors |
06/01/2005 | CN1204138C Pyrazolo [4, 3-d] pyrimidine derivs. |
05/31/2005 | US6900327 Used as antidepressants, to treat obsessive compulsive disorder, panic disorders, bulimia, anorexia, pain, obesity, senile demential, migraines, and social phobias |
05/26/2005 | WO2004108664A3 Bicyclic heterocycles, drugs containing said compounds, the use thereof and method for preparing the same |
05/26/2005 | US20050113373 medicine to inhibit proliferative conditions, such as cancer and psoriasis; detecting or identifying a histone deactylase (HDAC) in a biological sample |
05/26/2005 | US20050113340 9-(Substituted aryl, heteroaryl, alicyclyl, or heterocyclyl)methyl-2-amino-6-halopurines, e.g., 6-chloro-9-(4-methoxy-3,5-dimethyl-pyridin-2-ylmethyl)-9H-purin-2-ylamine; used in the treatment and prevention of various Heat Shock Protein 90 mediated disorders, e.g., proliferative disorders |
05/26/2005 | US20050113339 inflammatory diseases, infections, autoimmune disorders, stroke, ischemia, cardiac disorder, neurological disorders, fibrogenetic disorders, proliferative disorders, tumors, leukemias, neoplasms, cancers, carcinomas, metabolic diseases, and malignant disease |
05/25/2005 | EP1533318A1 Prodrugs of thrombin inhibitors |
05/25/2005 | EP1532122A1 11-beta-hydroxysteroid dehydrogenase 1 inhibitors useful for the treatment of diabetes, obesity and dyslipidemia |
05/25/2005 | EP0946511B1 Novel compounds with analgesic effect |
05/25/2005 | CN1620438A 5, 6-diaryl-pyrazine-2-amide derivatives as CBI antagonists |
05/25/2005 | CN1620430A 3-phenyl-2-arylalkylthiopropionic acid derivatives as selective agonists of PPAR-alpha |
05/25/2005 | CN1620291A 3-(imidazolyl)-2-alkoxypropanoic acids as TAFIA inhibitors |
05/25/2005 | CN1203065C Non-yellowing para-tertiaryl-alkyl phenyl substituted triazine and pyrimidine ultraviolet light absorbers |
05/25/2005 | CN1203061C Substituted isoquinolines, its preparing process, medical composition and its use for preparing medicine |
05/24/2005 | US6897321 Process for preparing azacycloalkanoylaminothiazoles (LD 137e) |
05/24/2005 | US6897207 Kinase inhibitors; angiogenesis inhibitors, anticancer agents, antiinflammatory agents and chronic obstructive pulmonary disease inhibitors |
05/24/2005 | CA2157792C N-(3-piperidinyl-carbonyl)-beta-alanine derivatives as paf antagonists |
05/19/2005 | WO2005044794A2 Immunohistochemical methods |
05/19/2005 | WO2005044793A2 Nitrogen-containing fused heterocyclic compounds |
05/19/2005 | WO2005044792A2 Compositions and methods for detecting and treating diseases and conditions related to chemokine receptors |
05/19/2005 | WO2005044268A1 Preparation of pharmaceutical salts of [1, 4] - bipiperidine |
05/19/2005 | WO2005021496A3 Synthesis of derivatives of ginkgolide c |
05/19/2005 | WO2005016228A3 Compositions and methods for reducing the risk of epileptic occurrence and/or for treatment of seizure disorders |
05/19/2005 | WO2004092123A3 Inhibitors of fungal invasion |
05/19/2005 | WO2004035565A8 Method for the synthesis of a benzimidazole compound |
05/19/2005 | US20050107607 Processes for preparing novel methylene blue derivative |
05/19/2005 | US20050107458 used as diagnostic kits, bioassay and/or drugs for preventing cancers, Alzheimer's disease, amyotrophic lateral sclerosis, Parkinson's disease, stroke, ischaemia, Huntington's disease, epilepsy, multiple sclerosis, neuropathy, or injuries of the brain or spinal chord, or as tyrosine kinase inhibitors |
05/19/2005 | US20050107436 Compounds for inflammation and immune-related uses |
05/19/2005 | US20050107435 antibiotics such as (5S,5S')-N-(3-{4'-[5-(Acetylamino-methyl)-2-oxo-oxazolidin-3-yl]-2,2'-difluoro-biphenyl-4-yl}-2-oxo-oxazolidin-5-ylmethyl)-acetamide, used for treating a bacterial infections in mammals |
05/19/2005 | US20050107418 Macrolides |
05/19/2005 | US20050107399 Cytokine inhibitors |
05/19/2005 | US20050107369 Heteroaromatic selective inhibitors of neuronal nitric oxide synthase |
05/19/2005 | US20050107343 Pyrrolo[2,3-d]pyrimidin-2-ylamines substituted in the 7th position by a aryl, heteroaryl, alicyclic, or heterocyclic group connected by methyl, C(O) , C(S) , S(O) or SO2; used in the treatment and prevention of various Heat Shock Protein 90 mediated disorders, e.g., proliferative disorders |
05/19/2005 | CA2544855A1 Immunohistochemical methods |
05/19/2005 | CA2544845A1 Preparation of pharmaceutical salts of [1, 4] - bipiperidine |
05/19/2005 | CA2543707A1 Nitrogen-containing fused heterocyclic compounds |
05/19/2005 | CA2543115A1 Compositions and methods for detecting and treating diseases and conditions related to chemokine receptors |
05/18/2005 | EP1530430A2 Method for producing an avocado unsaponifiable rich in furan lipids |
05/18/2005 | CN1617869A 4-(piperidyl- and pyrrolidyl-alkyl-ureido) -quinolines as urotensin ii receptor antagonists |
05/18/2005 | CN1617712A Pharmaceutical nanoparticulate composition of a tachykinin receptor antagonist |
05/18/2005 | CN1202108C Spiro compounds, preparing method and intermediate |
05/18/2005 | CN1202087C Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments |
05/17/2005 | US6894064 Benzothiophenes, formulations containing same, and methods |
05/17/2005 | US6894041 Oxazolyl-acid amide derivatives useful as inhibitors of PDE4 isozymes |
05/17/2005 | CA2347757C Method for producing (+)-exo-6-phenyl-3-azabicyclo-[3.2.0]heptanes |
05/12/2005 | WO2005042481A2 COMPOUNDS AND RELATED METHODS FOR MUTANT p53 REACTIVATION |
05/12/2005 | WO2005014537A3 Tetrahydropyran heterocyclic cyclopentyl heteroaryl modulators of chemokine receptor activity |
05/12/2005 | WO2005009948A3 Peptide inhibitors of beta-lactamases |
05/12/2005 | WO2005000803A8 Asymmetric urea compound and process for producing asymmetric compound by asymmetric conjugate addition reaction with the same as catalyst |
05/12/2005 | WO2004106297A3 Nonionic surfactant compositions |
05/12/2005 | WO2004101510A3 Polymorphs of cabergoline |
05/12/2005 | WO2004089312A3 New piperidinylamino-thieno[2,3-d] pyrimidine compounds |
05/12/2005 | US20050101788 Method for manufacture of sertindole |
05/12/2005 | US20050101651 Viricides; protease inbhibitors; useful for inhibiting the activity of picornaviral 3C proteases; for example, 6-carbamoyl-4S-{2S-[(5-naphthalen-1-yl-1H-pyrrole-2-carbonyl)-amino-3-phenyl-propionylamino}-hex-2(trans)-enoic acid ethyl ester |
05/12/2005 | US20050101628 Useful in the prevention or treatment of certain inflammatory and immunoregulatory disorders and diseases, allergic diseases, atopic conditions including allergic rhinitis, dermatitis, conjunctivitis, and asthma, as well as autoimmune pathologies |
05/12/2005 | US20050101626 Imidazo-fused oxazolo[4,5-beta]pyridine and imidazo-fused thiazolo[4,5-beta]pyridine based tricyclic compounds and pharmaceutical compositions comprising same |
05/11/2005 | EP1363899B1 Quinazolone derivatives as alpha 1a/b adrenergic receptor antagonists |
05/11/2005 | EP0971898B1 Substituted isoquinolines as ultra short acting neuromuscular blockers |
05/11/2005 | CN1615306A C-5 modified indazolylpyrrolotriazines |
05/11/2005 | CN1615166A Device for mini-invasive ultrasound treatment of an object by a heat-isolated transducer |
05/11/2005 | CN1615133A Crystalline solids of carvedilol and processes for their preparation |
05/11/2005 | CN1200940C Triazole pyrimidine compounds |
05/11/2005 | CN1200939C Novel tetrahydropyridines, preparation method and pharmaceutical compositions containing same |
05/11/2005 | CN1200930C New crystalline polymorphic form of 1-methyl-5-P-toluoylpyrroel-2-ac-etamidoacetic acid guaiacyl ester (MED 15) |
05/10/2005 | US6890927 Tartrate salts of 5,8, 14-triazateracyclo[10.3.1.02,11 04.9]-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof |
05/10/2005 | US6890922 For treatment of erectile dysfunction as well as female sexual dysfunction, incontinence, and hypertrophy of the prostate; inhibitors of cGMP-metabolizing phosphodiesterases (cGMP= cyclic guanosine monophosphate) |
05/06/2005 | WO2005040107A2 Methods for making simvastatin and intermediates |
05/06/2005 | WO2005009949A3 17-acetamido-4-azasteroid derivatives as androgen receptor modulators |
05/06/2005 | WO2004080960A3 Methods and compositions for the enzymatic synthesis of gangliosides |
05/06/2005 | WO2004067505A3 Bismuth dithiocarbamate compounds and uses thereof |
05/06/2005 | WO2004065363A3 Computational design of a water-soluble analog of a protein, such as phospholamban and potassium channel kcsa |
05/06/2005 | CA2543348A1 Methods for making simvastatin and intermediates |
05/05/2005 | US20050096229 Biocidal compounds and their preparation |
05/04/2005 | EP1528061A1 Heterocyclic derivatives which inhibit factor Xa |
05/04/2005 | CN1612876A Derivatives of 5-(pyridin-3-yl)-1-azabicyclo[3.2.1] octane, the preparation thereof and the application of same in therapeutics |
05/03/2005 | US6887905 Treatment of depression or generalized anxiety disorder |
05/03/2005 | US6887893 Methods and compositions for treatment and prevention of tumors, tumor-related disorders and cachexia |
05/03/2005 | US6887881 For use as antiarrhythmic drug |
05/03/2005 | CA2149886C Process for preparing tetrazolyl-benzopyranones |
04/28/2005 | WO2005037834A1 NOVEL TETRAYDROSPIRO{PIPERIDINE-2,7’ -PYRROLO[3,2-b]PYRIDINE DERIVATIVES AND NOVEL INDOLE DERIVATIVES USEFUL IN THE TREATMENT OF 5-HT6 RECEPTOR -RELATED DISORDERS |
04/28/2005 | WO2005037814A1 Novel tricyclic spiroderivatives as modulators of chemokine receptor activity |
04/28/2005 | WO2005037784A2 Crystalline form of gamma-aminobutyric acid analog |
04/28/2005 | WO2005037052A2 Binding assay with labelled bispidine variant |
04/28/2005 | WO2005021495A3 Quaternary salt derivatives of 1,4-diphenylazetidin-2-ones |
04/28/2005 | WO2005016877A3 Pyrazole carboxamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1 |
04/28/2005 | WO2004092125A3 Using alkylmetal reagents for directed metalation of azaaromatics |
04/28/2005 | WO2004083170A3 Compounds, a process for their preparation and their use as dyes and pigments |
04/28/2005 | US20050090539 Intermediates for making 1(alpha-amino-1-(cyclopropyl-fused pyrrolidinylcarbonyl)methyl)-3-hydroxyadamantanes, e.g., methyl 3-hydroxy-<a-oxotricyclo[3.3.1.13,7]decane-1-acetate |
04/28/2005 | US20050090494 Such as N-[2-(3-{[1-(3,4-dichlorobenzylpiperidinyl]aminohydroxypropoxy)phenyl]acetamide; antiinflammatory agents, antiarthritic agents; chronic obstructive pulmonary disease, asthma, multiple sclerosis |
04/28/2005 | CA2540861A1 Novel tetraydrospiro{piperidine-2,7' -pyrrolo[3,2-b]pyridine derivatives and novel indole derivatives useful in the treatment of 5-ht6 receptor -related disorders |
04/27/2005 | EP1526134A2 Triazolyl tropane derivatives as ccr5 modulators |
04/27/2005 | EP1526130A1 Substituted isoquinolines as ultra short acting neuromuscular blockers |
04/27/2005 | EP1419150B1 Phenylsulfonyl-1,3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use |