| Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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| 03/17/1994 | WO1994005660A1 Quinuclidine derivatives as squalene synthase inhibitors |
| 03/17/1994 | WO1994005634A1 Benzo-fused lactams promote release of growth hormone |
| 03/17/1994 | CA2143430A1 Quinuclidine derivatives as squalene synthase inhibitors |
| 03/16/1994 | EP0587194A1 2-(Heterocycloalkoxy)-1-(subst.-phenyl)-ethanol derivatives as cerebral function improving agents |
| 03/16/1994 | EP0587193A1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same |
| 03/16/1994 | EP0587134A2 Cyclic urea derivatives, medicaments containing them and process for their preparation |
| 03/15/1994 | CA1327800C Derivatives of aza-2-bicyclooctane-3-carboxylic acid, processes for their preparation and pharmaceutical compositions containing them |
| 03/15/1994 | CA1327750C Therapeutic use of serotonin-antagonists |
| 03/12/1994 | CA2105934A1 Cyclic urea derivatives |
| 03/09/1994 | EP0585328A1 Substituted 3-aminoquinuclidines |
| 03/08/1994 | US5292756 Novel sulfonamide fibrinogen receptor antagonists |
| 03/08/1994 | US5292749 Antimuscarinic bronchodilators |
| 03/03/1994 | WO1994004496A1 Substituted benzylamino nitrogen containing non-aromatic heterocycles |
| 03/03/1994 | WO1994004495A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension |
| 03/01/1994 | US5290938 Preparation of S-(-)- and R-(+)-N-(quinuclidinyl-3)-amide |
| 03/01/1994 | US5290795 Substituted urea compound and use |
| 03/01/1994 | CA2104981A1 Heterocyclic compounds |
| 02/22/1994 | US5288731 2,6-methano-2H-1-benzoxocincarboxylic acids, esters and amides |
| 02/22/1994 | US5288730 Azabicyclic compounds, pharmaceutical compositions containing them and their use in therapy |
| 02/17/1994 | WO1994003451A1 Quinuclidine derivatives as squalene synthase inhibitors |
| 02/17/1994 | WO1994003440A1 Benzoxazinones as inhibitors of hiv reverse transcriptase |
| 02/17/1994 | WO1994003437A1 Benzodiazepine derivatives |
| 02/17/1994 | WO1994003426A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists |
| 02/17/1994 | CA2141806A1 Quinuclidine derivatives as squalene synthase inhibitors |
| 02/17/1994 | CA2141791A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists |
| 02/17/1994 | CA2140009A1 Benzodiazepine derivatives |
| 02/16/1994 | EP0582810A1 Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxyetracyclines as antibiotic agents |
| 02/16/1994 | EP0409931B1 Quinuclidine therapeutic agents |
| 02/15/1994 | US5286864 Deprotonation and salt formation with sodium hydride; alkylation, deprotecting |
| 02/15/1994 | US5286732 Nitrogen-containing bicyclic compounds and pharmaceutical compositions thereof |
| 02/09/1994 | EP0582455A1 Benzoxazinones as inhibitors of HIV reverse transcriptase |
| 02/07/1994 | CA2101901A1 Therapeutic heterocyclic derivatives |
| 02/02/1994 | EP0581165A2 Acrylamide derivatives as antirussive agent |
| 02/01/1994 | US5283241 Animal growth regulators |
| 01/25/1994 | US5281626 Benzenesulfonamide derivatives |
| 01/25/1994 | US5281585 Fibrinogen receptor antagonists for inhibiting aggregation of blood platelets |
| 01/20/1994 | WO1994001402A1 Heterocyclic amide derivatives as tachykinin derivatives |
| 01/18/1994 | US5280032 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same |
| 01/11/1994 | US5278170 Azabicylo oxime compounds |
| 01/06/1994 | WO1994000449A1 Benzimidazole compounds |
| 01/06/1994 | WO1994000448A1 Azacyclic and azabicyclic hydroxylamines as muscarinic receptor agonists |
| 01/06/1994 | WO1994000119A1 Aminobutanoic acid compounds having metalloprotease inhibiting properties |
| 01/05/1994 | EP0577253A2 Enantiomeric enrichment of (R,S)-3-quinuclidinol |
| 01/05/1994 | EP0576974A1 Benzyliden-quinuclidinones as sunscreen agents |
| 12/29/1993 | EP0576357A1 Pyrazole derivatives, process for their preparation and pharmaceutical compositions containing them |
| 12/28/1993 | US5273972 [(2-diakylaminomethyl)-3-quinuclidinyl]-benzamides and benzoates |
| 12/28/1993 | US5273686 Using an organic solution for reaction with an alpha olefin, as a reducing agent or to prepare hydrides |
| 12/21/1993 | US5272154 3,7 substituted indole and indazole compounds and pharmaceutical compositions containing them |
| 12/20/1993 | CA2093890A1 Enantiomeric enrichment of (r,s)-3-quinuclidinol |
| 12/09/1993 | WO1993024486A1 Quinuclidine derivatives as squalene synthetase inhibitors |
| 12/05/1993 | CA2097671A1 Heterocyclic derivatives |
| 12/01/1993 | EP0422154B1 Therapeutic use of 5-ht3 receptor antagonists |
| 11/30/1993 | US5266576 N-myristoyl transferase inhibitors |
| 11/25/1993 | WO1993023395A1 Heteroaromatic quinuclidinenes, their use and preparation |
| 11/23/1993 | US5264577 Cyclic amino acids and derivatives thereof |
| 11/23/1993 | US5264435 Pyrimidines and their pharmaceutical acceptable salts, and their use as medicines |
| 11/18/1993 | EP0569564A1 Biphenylylquinuclidines, useful as squalene synthetase inhibitors |
| 11/16/1993 | US5262427 3-substituted and optionally 1-substituted azacyclic or azabicyclic compounds, pharmaceutical compositions, thereof and their use as stimulants of cognitive functions |
| 11/09/1993 | US5260461 Ligands for ADH: cinchona alkaloids and moderately sized organic substituents linked through a planar aromatic spacer group |
| 11/09/1993 | US5260320 Diaminotrifluoromethylpyridine compounds and phospholipase A2 inhibitor containing them |
| 11/09/1993 | US5260314 Certain 3-(1,2,5-oxa- or thiadiazol-4-yl)-1-azabicyclo [2.2.2]octanes having pharmaceutical properties |
| 11/09/1993 | US5260303 Imidazopyridines as serotonergic 5-HT3 antagonists |
| 11/09/1993 | US5260293 Simulate central muscarinic acetlycholine receptors |
| 11/02/1993 | US5258392 3-quinuclidine derivatives |
| 10/28/1993 | WO1993021184A1 Biphenylylquinuclidine derivatives as squalene synthase inhibitors |
| 10/28/1993 | WO1993021183A1 Quinuclidine derivatives as squalene synthase inhibitors |
| 10/28/1993 | WO1993021176A1 Novel cyclic amino acids and derivatives thereof |
| 10/28/1993 | WO1993021172A1 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists |
| 10/27/1993 | EP0566609A1 Azabicydic and azatricydic derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them |
| 10/27/1993 | EP0566589A1 N-alkyl quinuclidinium salts as substance p antagonists |
| 10/26/1993 | US5256671 A prodrug as tachykinin antagonists for treating headaches, pain or inflammation |
| 10/20/1993 | CN1022488C Antimuscainic bronchodilators |
| 10/19/1993 | US5254682 Cyclic renin inhibitors containing 3(S)-amino-4-cyclohexyl-2(R)-hydroxy-butanoic acid or 4-cyclo-hexyl-(2R, 3S)-dihydroxybutanoic acid or related analogs |
| 10/11/1993 | CA2093782A1 Heterocyclic derivatives |
| 10/11/1993 | CA2093778A1 Heterocyclic compounds |
| 10/06/1993 | EP0563087A1 Azabicyclic amides or esters of halogenated benzoic acids |
| 09/30/1993 | WO1993019064A1 Quinuclidine derivatives as substance p antagonists |
| 09/30/1993 | WO1993019046A1 Novel sulfonamide fibrinogen receptor antagonists |
| 09/29/1993 | EP0561910A1 Pharmaceuticals |
| 09/28/1993 | CA1322552C Anxiolytic-r-n(1-azabicyclo[2.2.2)oct-3-yl) benzamides and thiobenzamides |
| 09/21/1993 | US5246942 Pharmaceutically useful dibenzofurancarboxamides of specific stereo-configuration |
| 09/15/1993 | EP0560604A1 Cinnoline-3-carboxylic acid derivatives as 5-HT3 antagonists |
| 09/15/1993 | EP0559656A1 Process for preparing multicyclic oxy-containing ring components |
| 09/14/1993 | US5244899 Azabicycloalkyl and azatricycloalkyl amides used to treat inflammation, allergy, asthma and skin disorders |
| 09/13/1993 | CA2091375A1 Cinnoline-3-carboxylic acid derivatives |
| 09/08/1993 | EP0559297A1 Use of heterocyclic derivatives for the manufacture of medicaments |
| 09/07/1993 | US5242930 Tachykinin antagonists; nervous system disorders, anxiolytic agents |
| 09/07/1993 | US5242929 Derivatives of substituted imidazol-2-one and process for their preparation |
| 09/07/1993 | US5242927 Prodrugs for oxadiazole muscarinic agonists |
| 09/07/1993 | US5242925 Piperazinylbenzodioxane derivatives |
| 09/02/1993 | WO1993017018A1 Nitrosation process |
| 08/24/1993 | CA1321586C Bicyclic compounds, their use as pharmaceuticals, their preparation, and intermediates useful in their preparation |
| 08/19/1993 | WO1993016048A1 Substituted acetamide compound |
| 08/19/1993 | WO1993015735A1 (non descriptive)-a method for delaying hiv individual aids by administration of substituted azaspirane compounds |
| 08/19/1993 | CA2155320A1 Substituted acetamide compound |
| 08/18/1993 | EP0555478A1 Pyrimidine derivative and medicine |
| 08/17/1993 | US5237066 Reacting quinuclidone with (R)-alpha-methylbenzylamine; reduction with alkali metal borohydride; hydrogenolysis in acid |
| 08/17/1993 | US5236931 Treating anxiety, psychosis, cognitive dysfunction, migrane, cluster headache, trigeminal neuralgia emesis and impaired gastric motility |
| 08/05/1993 | WO1993015073A1 Azabricyclic compounds as calcium channel antagonists |
| 07/31/1993 | CA2088091A1 3-quinuclidinol catalyst compositions for making polyurethane foams |