| Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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| 08/24/1999 | US5942517 Antagonist of alpha(1c) receptors; treatment of benign prostatic hyperplasia |
| 08/19/1999 | WO1999041251A1 Antagonists of gonadotropin releasing hormone |
| 08/19/1999 | CA2317451A1 Antagonists of gonadotropin releasing hormone |
| 08/18/1999 | CN1226163A Formulation for treatment and/or prevention of dementia |
| 08/17/1999 | US5939449 Novel compounds having high affinity for the neurotensin receptors |
| 08/17/1999 | US5939434 Tetrazolyl-substituted quinuclidines as substance P antagonists |
| 08/17/1999 | US5939433 Quinuclidine derivatives |
| 08/11/1999 | EP0934316A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use |
| 08/10/1999 | US5936123 Compounds such as 3-isopropyl-4-hydrazinobenzoic acid and its salts |
| 08/10/1999 | US5936088 Nervous system disorders |
| 08/10/1999 | CA2178160C Hydroxymethyl quinuclidine catalyst compositions for making polyurethane foams |
| 08/05/1999 | WO1999038820A1 The use of compressed co2 in chemical reactions |
| 08/04/1999 | EP0854720B1 Nk-1 receptor antagonists for prevention of neurogenic inflammation in gene therapy |
| 08/03/1999 | US5932620 Administering to the patient for treating senile dementia of alzheimer type, huntington's chorea, riley-day syndrome, traumatic nerve injury and amyotrophic lateral sclerosis |
| 07/27/1999 | US5929247 Heterocyclic compounds and their preparation and use |
| 07/27/1999 | CA2164804C Nk-1 receptor antagonists for the treatment of neuronal injury and stroke |
| 07/20/1999 | US5925661 Nervous system disorders |
| 07/14/1999 | CN1222910A 1,2,4-benzothiadiazine derivatives, their preparation and use |
| 07/13/1999 | US5922723 Administering to the patient suffering with central nervous system disorder a 2-azabicyclo(2,2,1)hept-5-ene derivative |
| 07/13/1999 | US5922721 Use in treating alzheimer's disease, huntington's chorea, amyotrophic lateral sclerosis and trauamtic nerve injuries |
| 07/07/1999 | EP0927170A1 Piperazino derivatives as neurokinin antagonists |
| 07/07/1999 | CN1221608A Synergistic combination of AIDS antiviral compounds and HIV inhibitor |
| 07/06/1999 | US5919829 Gastrin and cck receptor ligands |
| 07/06/1999 | US5919793 Quinuclidine derivatives, squalene synthetase inhibitors, anticholesterol agents |
| 07/01/1999 | WO1999032468A1 Anilide derivative, production and use thereof |
| 07/01/1999 | CA2311428A1 Anilide derivative, production and use thereof |
| 06/30/1999 | CN1043884C New substituted azacylobutanone, preparation method and medicinal use thereof |
| 06/24/1999 | WO1999031097A1 Imidazol derivatives as muscarinic m3 receptor antagonists |
| 06/24/1999 | WO1999031088A1 Triazine angiogenesis inhibitors |
| 06/24/1999 | CA2313776A1 Triazine angiogenesis inhibitors |
| 06/23/1999 | EP0923579A1 Herbicidal s-substituted 1,2,4,6-thiatriazines |
| 06/23/1999 | EP0923536A1 Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation |
| 06/17/1999 | WO1999029692A1 Method for preparing mequitazine and novel synthesis intermediate |
| 06/15/1999 | US5912260 Gastrin and CCK antagonists |
| 06/09/1999 | CN1219172A Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists |
| 06/03/1999 | WO1999026932A1 By amidino group substituted heterocyclic derivatives and their use as anticoagulants |
| 06/02/1999 | EP0919245A2 NK-1 receptor antagonist and a systemic antiinflammatory corticosteroid for the treatment of emesis |
| 06/02/1999 | EP0918521A1 Formulation for the treatment and/or prophylaxis of dementia |
| 06/02/1999 | CN1218454A Preparation of 1-alkoxycarbonyl-3-phenylpropyl derivatives |
| 06/01/1999 | CA1340570C Process for synthesizing n-alkylated amino-acides and the esters thereof. their use for synthesizing carboxyalkyl dipeptides |
| 05/19/1999 | EP0916346A2 NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis |
| 05/11/1999 | US5902814 Treating psychotic disorder, intellectual disorders and anxiety, such as attention deficit hyperactivity disorder and schizophrenia |
| 05/06/1999 | WO1999021855A1 Pleuromutilin derivatives as antimicrobials |
| 05/06/1999 | WO1999021854A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants |
| 05/06/1999 | WO1999021553A1 Antagonists of gonadotropin releasing hormone |
| 05/06/1999 | EP0912563A1 Cinchonan based chiral selectors for separation of stereoisomers |
| 05/06/1999 | EP0912555A1 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders |
| 05/06/1999 | CA2308454A1 Antagonists of gonadotropin releasing hormone |
| 05/06/1999 | CA2306878A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants |
| 04/29/1999 | WO1999020633A1 Benzoxazine derivatives, preparation and application in therapy |
| 04/29/1999 | WO1998057931A3 Quinoline-indole antimicrobial agents, uses and compositions related thereto |
| 04/28/1999 | EP0910566A1 Heterocyclic compounds and their preparation and use |
| 04/28/1999 | CN1215401A 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives endothelin antagonists |
| 04/28/1999 | CN1215054A Bychclic fibrinogen antagonists |
| 04/22/1999 | WO1998050383A8 5-phenyl-1,3,4-oxadiazol-2(3h)-one derivatives and their use as 5-ht4 ligands |
| 04/21/1999 | CN1214685A Inhibitors of farnesyl protein transferase |
| 04/20/1999 | CA2124990C Pharmaceutical agents for treatment of emesis |
| 04/14/1999 | CN1214046A 4,5-dihydronaphth [1,2-C] isoxazoles and derivatives thereof having CNS activity |
| 04/14/1999 | CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials |
| 04/07/1999 | EP0906297A1 1,2,4-benzothiadiazine derivatives, their preparation and use |
| 04/06/1999 | US5892047 Process for the preparation of substituted 4-ethyl-piperidines and an intermediate for the preparation of same |
| 04/06/1999 | US5892039 Piperazino derivatives as neurokinin antagonists |
| 04/06/1999 | US5891887 Brain disorders |
| 03/30/1999 | US5889019 Heterocyclic compounds and their use |
| 03/30/1999 | US5888999 Using azacyclic and azabicyclic pyrazine compounds |
| 03/24/1999 | EP0903337A1 Process for the preparation of 1-alkoxycarbonyl-3-phenylpropyl derivatives |
| 03/24/1999 | CN1211983A Azabicyclic esters of carbamic acids useful in therapy |
| 03/23/1999 | US5886175 Tetracycline antibiotics |
| 03/23/1999 | US5886009 Quinuclidine derivative as a substance P antagonist |
| 03/18/1999 | WO1999012877A1 Enantioselective reduction of ketones with a silane agent/metal compound/chiral ligand system |
| 03/18/1999 | CA2298533A1 Reduction enantioselective de cetones avec un systeme agent silanique/compose metallique/ligand chiral |
| 03/17/1999 | EP0901489A1 Antagonists of gonadotropin releasing hormone |
| 03/17/1999 | EP0901471A1 Antagonists of gonadotropin releasing hormone |
| 03/17/1999 | CN1211251A 1,4-dihydropyridine compounds as bradykinin antagonists |
| 03/16/1999 | US5883254 Cyanation of pyrimidines by reacting with an alkali cyanide in the presence of 1-azabicyclo(2,2,2)octane or 1,4-diazabicyclo(2,2,2)octane |
| 03/16/1999 | CA2167198C Benzylaminoquinuclidines |
| 03/16/1999 | CA2164689C Nk-1 receptor antagonists and 5ht3 receptor antagonists for the treatment of emesis |
| 03/16/1999 | CA2058264C Dihydrobenzofuran carboxamides and process for their preparation |
| 03/10/1999 | EP0900218A1 Heterocyclic compounds |
| 03/09/1999 | US5880284 Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them |
| 03/09/1999 | US5880136 Sulfonamide fibrinogen receptor antagonists |
| 03/09/1999 | US5880121 Serotonin 5ht3 antagonist, useful for treating anxiety, phychiatric disorders, nausea, vomiting and drug dependency |
| 03/04/1999 | WO1999010339A1 2-aminopyridines containing fused ring substituents as nos inhibitors |
| 03/04/1999 | WO1999009987A1 Method for treating premenstrual or late luteal phase syndrome |
| 03/04/1999 | CA2298979A1 Method for treating premenstrual or late luteal phase syndrome |
| 03/03/1999 | EP0899261A1 Optical active 1,4-dihydropyridine compounds as bradykinin antagonists |
| 02/24/1999 | CN1042225C Substituted isoxazole derivatives prepn. method |
| 02/23/1999 | US5874428 N-substituted aza-heterocyclic carboxylic acids and esters thereof |
| 02/23/1999 | CA2146007C Substituted quinuclidines |
| 02/18/1999 | CA2245041A1 Optical active 1,4-dihydropyridine compounds as bradykinin antagonists |
| 02/17/1999 | CN1208348A Method for treating pain |
| 02/16/1999 | US5872117 Treating cerebrovascular dementia, senile dementia, alzheimer's dementia, sequelae of ischemic encephalopathy and cerebral apoplexy |
| 02/10/1999 | CN1207739A 1,2,3-thiadiazole carboxylic acid (thio) esters and use thereof as pest control agent or as microbicide |
| 02/09/1999 | US5869663 Intermediates for neurokinin receptor antagonists |
| 02/09/1999 | US5869499 Benzyloxyquinuclidines as substance P antagonists |
| 02/09/1999 | US5869488 Piperazino derivatives as neurokinin antagonists |
| 02/03/1999 | CN1041921C Bicyclic fibrinogen antagonists |
| 01/28/1999 | WO1999003472A1 Peripherally acting anti-pruritic opiates |
| 01/28/1999 | CA2288833A1 Peripherally acting anti-pruritic opiates |
| 01/27/1999 | EP0892797A1 Inhibitors of farnesyl protein transferase |