Patents
Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704)
08/1995
08/29/1995US5446050 Azabicyclo amides and esters as 5-HT3 receptor antagonists
08/22/1995CA2030077C Azabicyclo amides and esters as 5-ht _receptor antagonists
08/17/1995WO1995021820A1 Novel carbamate derivative and medicinal composition containing the same
08/17/1995CA2182568A1 Novel carbamate derivative and medicinal composition containing the same
08/15/1995US5442078 Intermediates for specific 5-HT3 antagonists
08/15/1995US5442068 Reducing imine to amine with sodium triacetoxyborohydride and acetic acid
08/09/1995EP0665844A1 Substituted benzylaminoquinuclidines as substance p antagonists
08/09/1995EP0665843A1 Substituted quinuclidines as substance p antagonists
08/09/1995EP0659179A4 Benzo-fused lactams promote release of growth hormone.
08/03/1995WO1995004720A3 Gastrin and cck receptor ligands
08/02/1995EP0546181B1 Indole derivatives and their use as serotonin antagonists
07/1995
07/25/1995CA1336435C Copper and nickel dihalide complexes, their preparation and the use thereof
07/25/1995CA1336434C Soluble magnesium hydrides, method of preparing them, and use thereof
07/20/1995WO1995019337A1 NOVEL HIGH ENANTIO-SELECTIVE PROCESS FOR PRODUCING PURE ENANTIOMERIC CYCLOPENTANE AND CYCLOPENTENE-β-AMINO ACIDS
07/20/1995DE4400749A1 Neues hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan- und -penten-beta-Aminosäuren New highly enantioselective process for the preparation of enantiomerically pure cyclopentane- and -pentene beta amino acids
07/18/1995US5434261 Benzo-fused lactams promote release of growth hormone
07/18/1995US5434161 Imidazopyridines as serotonergic 5-HT3 antagonists
07/13/1995WO1995018617A1 1-aminoindan derivatives and compositions thereof
07/12/1995EP0662481A1 Spiro piperidines and homologs promote release of growth hormone
07/06/1995WO1995018104A1 Novel benzamide derivative and medicinal composition containing the same
07/04/1995US5430162 7-(substituted)-8-(substituted)-9-substituted amino)-6-demethyl-6-deoxytetracyclines
06/1995
06/29/1995WO1995017180A1 A method of treating gastrointestinal motility disorders
06/29/1995CA2179492A1 A method of treating gastrointestinal motility disorders
06/28/1995EP0659184A1 Optically active hydroquinine (amino-3 phenyl)-1 ethanesulfonate, preparation and use thereof.
06/28/1995EP0659179A1 Benzo-fused lactams promote release of growth hormone
06/28/1995EP0521067B1 Azacyclic or azabicyclic compounds, their preparation and use
06/21/1995EP0658539A1 Excitatory amino acid receptor antagonists
06/21/1995EP0658532A1 Ligand-accelerated catalytic asymmetric dihydroxylation
06/14/1995EP0656897A1 Quinuclidine derivatives as squalene synthase inhibitors
06/07/1995EP0655996A1 Substituted benzylamino nitrogen containing non-aromatic heterocycles
06/06/1995US5422354 Quinuclidine derivatives
06/04/1995CA2136904A1 Excitatory amino acid receptor antagonists
05/1995
05/31/1995EP0655056A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
05/30/1995US5420279 Crystallised microporous gallium phosphate and its substituted derivatives and a method of preparing them
05/30/1995US5420141 Capable of binding to neurotensin receptor
05/24/1995EP0654023A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists
05/18/1995WO1995013069A1 Piperidines, pyrrolidines and hexahydro-1h-azepines promote release of growth hormone
05/18/1995CA2175218A1 Piperidines, pyrrolidines and hexahydro-1h-azepines promote release of growth hormone
05/17/1995EP0652871A1 Benzodiazepine derivatives
05/09/1995US5414009 Azabicyclo substituted oxa- or thia-diazole compounds
04/1995
04/11/1995US5405853 Thiadiazoles useful in the treatment of senile dementia
03/1995
03/28/1995US5401750 Derivatives of substituted imidazol-2-one and process for their preparation
03/23/1995WO1995007908A1 Heteroarylamino and heteroarylsulfonamido substituted 3-benzylaminomethyl piperidines and related compounds
03/22/1995EP0644198A1 Alpha-heteroaryloxymethyl ketones as interleukin-1beta converting enzyme inhibitors
03/21/1995US5399563 Benzylidenequinuclidinones
03/21/1995US5399562 Indolones useful as serotonergic agents
03/09/1995WO1995006635A1 Carbamate derivative and medicine containing the same
03/07/1995US5395766 Optically active trans-2-aryl-1-cyclohexanol derivatives and a process for producing the compounds
03/02/1995WO1995006035A1 Benzazepine derivative, pharmaceutical composition containing the same, and intermediate for the same
03/02/1995WO1995006029A1 Enantioselective synthesis of alpha - alkylated amino acid derivatives by phase - transfer catalysis
03/02/1995WO1995003303A3 Aza spiro compounds acting on the cholinergic system with muscarinic agonist activity
03/02/1995CA2170373A1 Benzazepine derivative, pharmaceutical composition thereof, and intermediate thereof
03/01/1995EP0640082A1 Heteroaromatic quinuclidinenes, their use and preparation
02/1995
02/28/1995US5393762 Pharmaceutical agents for treatment of emesis
02/23/1995WO1995005379A1 Antipsychotic method
02/21/1995US5391549 Cinnoline-3-carboxylic acid derivatives
02/16/1995WO1995004720A2 Gastrin and cck receptor ligands
02/16/1995CA2167154A1 Gastrin and cck receptor ligands
02/15/1995EP0638569A1 Bicyclic nitrogenous compound
02/15/1995EP0638553A1 Carboxylic acid amides having a terminal carboxylic acid group as aggregation inhibiting drugs
02/14/1995CA1334413C Amino-substituted bridged azabicyclic quinolone carboxylic acids and esters
02/08/1995EP0637305A1 Novel cyclic amino acids and derivatives thereof
02/08/1995CN1098413A Xanthene derivant
02/06/1995CA2129374A1 Carbonamides, pharmaceutical compositions containing these compounds and processes for their preparation
02/02/1995WO1995003306A1 Arthropodicidal azacyclic heterocycles
02/02/1995WO1995003303A2 Aza spiro compounds acting on the cholinergic system with muscarinic agonist activity
02/02/1995WO1995003301A1 Azalicyclooctane derivatives as anti-arrhythmic agents
02/02/1995WO1995003289A1 Benzo-fused lactams promote release of growth hormone
02/01/1995EP0636125A1 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists
01/1995
01/31/1995US5385912 Multicyclic tertiary amine polyaromatic squalene synthase inhibitors
01/31/1995US5385898 Hypertensive agents; cardiovascular disorders; renin inhibitors; glaucoma
01/26/1995WO1995002595A1 Benzyloxyquinuclidines as substance p antagonists
01/26/1995WO1995002587A1 Substituted piperazinylcamphor derivatives as oxytocin antagonists
01/26/1995CA2166974A1 Substituted amide derivatives of piperizinylcamphor sulfonyl and carbonyl oxytocin antagonists
01/25/1995CN1097753A 5-membered heterocycles, processes for preparing them and pharmaceutical compositions containing these compounds
01/24/1995US5384408 Nervous system disorders such as Alzheimer*s and senility
01/24/1995US5384322 Nitrogen-containing bicyclic compounds and pharmaceutical compositions thereof
01/24/1995CA1334095C Aroyl urea and carbamic acid derivatives
01/11/1995EP0632809A1 Quinuclidine derivatives as substance p antagonists
01/10/1995US5380925 Cyclic amino acids and derivatives thereof
01/03/1995US5378712 Antithrombosis
12/1994
12/28/1994EP0540526B1 Quinuclidine derivatives
12/14/1994EP0628041A1 Heterocyclic compounds and their preparation and use
12/14/1994EP0565558B1 Process and intermediates for preparing azabicyclo 2.2.2]octan-3-imines
12/07/1994EP0627221A2 Substance P antagonists for the treatment of emesis
12/07/1994EP0626961A1 Nitrosation process
12/07/1994EP0626960A1 Quinuclidine derivatives as squalene synthase inhibitors
12/06/1994US5371076 9-[(substituted glycyl)amido]-6-(substituted)-5-hydroxy-6-deoxytetracyclines
12/04/1994CA2125021A1 Alpha-heteroaryloxymethyl ketones as interleukin-1 beta converting enzyme inhibitors
11/1994
11/30/1994EP0626373A1 Quinazolinone derivatives
11/30/1994EP0625979A1 Azabricyclic compounds as calcium channel antagonists
11/29/1994US5368780 Quinine, sulfuric acid, iodine clathrate
11/24/1994WO1994026740A1 Heteroatom substituted alkyl benzylaminoquinuclidines as substance p antagonists
11/23/1994EP0625507A2 Urea derivatives and their use as acat inhibitors
11/22/1994US5366982 Substituted bicyclic bis-aryl compounds exhibiting selective leukotriene B4 antagonist activity, their preparation and use in pharmaceutical compositions
11/22/1994US5366737 Drug delivery, DNA transfection
11/22/1994CA2123728A1 Urea derivatives and their use as acat inhibitors
11/22/1994CA1333154C Memory enhancing-r-n-(1-azabicyclo[2.2.2]oct-3-yl) benzamides and thiobenzamides
11/15/1994US5364863 Treatment of migraine, emesis, schizophrenia, anxiety, gastrointestinal disorders
11/10/1994WO1994025459A1 Heterocyclic derivatives
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