Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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07/22/1993 | WO1993014090A1 Heterocyclic compounds and their preparation and use |
07/22/1993 | WO1993014089A1 Heterocyclic compounds and their preparation and use |
07/22/1993 | CA2127251A1 Heterocyclic compounds and their preparation and use |
07/21/1993 | EP0551963A2 Use of heterocyclic derivatives for the manufacture of medicaments |
07/20/1993 | US5229403 Enzyme inhibitors, antiinflammatory |
07/20/1993 | CA1320448C Method of enhancing memory or correcting memory deficiency with arylamido (and arylthioamido)-azabicycloalkanes |
07/14/1993 | EP0550587A1 Stereoselective preparation of acid sensitive amides and intermediates useful in said preparation |
07/13/1993 | US5227543 Facilitation of turnover in the ADH by additives which catalyze the hydrolysis of the OS(VI) glycolate esters |
07/13/1993 | US5227394 Muscarinic cholinergic agonists, cognition activators, analgesics |
07/13/1993 | US5227386 Indole derivatives |
07/08/1993 | WO1993013096A1 Quinuclidine derivatives as squalene synthase inhibitors |
07/08/1993 | WO1993013083A1 Oxadiazole derivatives having acetylcholinesterase-inhibitory and muscarinic agonist activity |
07/08/1993 | CA2126976A1 Oxadiazole derivatives having acetylcholinesterase-inhibitory and muscarinic agonist activity |
06/29/1993 | US5223511 Benzimidazoline-2-oxo-1-carboxylic acid compounds useful as 5-HT receptor antagonists |
06/24/1993 | CA2085913A1 Heterocyclic derivatives |
06/22/1993 | US5221593 Silver halide photographic materials containing novel nucleating agent |
06/16/1993 | EP0546181A1 Indole derivatives and their use as serotonin antagonists |
06/15/1993 | US5219849 Substituted pyrazines, pyrimidines and pyridazines for use in the treatment of glaucoma |
06/09/1993 | EP0544779A1 Heterocyclic compounds and their preparation and use |
06/08/1993 | US5217975 Azabicyclic compounds for treating dementia |
06/02/1993 | EP0543969A1 Heterocyclic chiral ligands and method for catalytic asymmetric dihydroxylation of olefins |
06/01/1993 | US5216163 Process for preparing azabicyclo[2.2.2]octan-3-imines |
06/01/1993 | US5215974 Antisecretory agents for gastrointestinal disorders; water solubility, chemical stability |
06/01/1993 | US5215918 Acid anhydride esterification; preferential enzymatic hydrolysis with a subtilisin protease |
06/01/1993 | CA1318595C 2-alkoxy-n-(1-azabicyclo[2.2.2]oct-3-yl) benzamides and thiobenzamides |
05/18/1993 | US5212185 Piperidinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension |
05/13/1993 | WO1993009116A1 Quinuclidine compound and medicinal use thereof |
05/13/1993 | WO1993009115A1 Biphenylylquinuclidines, useful as squalene synthetase inhibitors |
05/12/1993 | EP0541407A1 Nitrogen containing bicyclic derivatives, method for their preparation and pharmaceutical compositions containing them |
05/12/1993 | EP0540604A1 Substituted bicyclic bis-aryl compounds exhibiting selective leukotriene b 4? antagonist activity, their preparation and use in pharmaceutical compositions |
05/12/1993 | CN1071916A 2,3-phthalazine containing ether or sulfide group at 1-position and process for preparing same |
05/06/1993 | DE4234933A1 New phthalazine derivs. |
05/05/1993 | EP0539805A1 Phthalazines substituted on position 1 by an ether or a thioether group and process for their preparation |
05/05/1993 | CN1071667A Phenothiazine quaternary ammonium derivative and process for preparing their composition |
05/04/1993 | US5208036 Complexing a liposomal composition with a quaternary ammonium diether |
05/01/1993 | CA2081819A1 Phthalazines containing an ether or thioether group in the 1-position and a process for their preparation |
05/01/1993 | CA2081674A1 Heterocyclic compounds |
04/29/1993 | WO1993008192A1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment |
04/29/1993 | WO1993008186A1 Pyridine-3-carboxylic acid esters or amides useful as 5-ht3 antagonists |
04/29/1993 | WO1993007871A1 Methods for the treatment of hyperlipidemia using azaspiranes |
04/27/1993 | US5206246 Anxiolytic-R-n(1-azabicyclo[2.2.2]oct-3-yl) benzamides and thiobenzamides |
04/27/1993 | US5206235 Animal growth regulators; stimulants |
04/21/1993 | CN1071168A Fused tricycle nitrogen containing heterocycles |
04/15/1993 | WO1993007142A1 New ligands for asymmetric dihydroxylation: multiple cinchona alkaloid units attached to a central heterocyclic core |
04/14/1993 | EP0536817A1 Azabicyclic compounds as tachykinin antagonists |
04/14/1993 | CN1070911A Therapeutic compounds |
04/13/1993 | US5202333 Tricyclic 5-HT3 receptor antagonists |
04/13/1993 | US5202318 Tricyclic compounds acting at serotonin receptor subtypes |
04/06/1993 | US5200419 Substituted tetrazoles and derivatives thereof acting at muscarinic receptors |
04/01/1993 | WO1993006099A1 Fused tricyclic nitrogen containing heterocycles as substance p receptor antagonists |
04/01/1993 | WO1993006098A1 Quinuclidine esters process and intermediate for their preparation and pharmaceutical compositions containing them |
04/01/1993 | WO1993006092A1 Piperazinyl (sulfonyl)amide derivatives of camphor as oxytocin antagonists |
03/31/1993 | CN1070399A Substituted amide derivatives of piperizinylcamphorsulfonyl oxytocin antagonists |
03/30/1993 | US5198435 Antiinflammatory, antiallergen |
03/28/1993 | CA2079185A1 Dicyclic nitrogens derivatives, preparation process thereof and pharmaceutical compositions containing them |
03/24/1993 | EP0533516A2 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them |
03/24/1993 | EP0533280A1 Novel medical use for tachykinin antagonists |
03/24/1993 | EP0533242A2 Substituted derivatives of piperazinylcamphorsulfonyl oxytocin antagonists |
03/24/1993 | EP0533241A2 Substituted alkyl derivatives of piperazinylcamphorsulfonyl oxytocin antagonists |
03/24/1993 | EP0533240A2 Substituted amine derivatives of piperazinylcamphorsulfonyl oxytocin antagonists |
03/24/1993 | EP0533048A1 Process for the preparation of lactams |
03/17/1993 | EP0532097A1 Piperazinyl(sulfon)amide derivatives of camphor as oxytocin antagonists |
03/17/1993 | CN1069971A Novel sulfonamide fibrinogen receptor antagonists |
03/17/1993 | CN1020102C Preparation for bicyclic carboxylic ether and bicyclic carboxylic amide |
03/17/1993 | CA2078264A1 Substituted derivatives of piperizinylcamphorsulfonyl oxytocin antagonists |
03/17/1993 | CA2078263A1 Substituted alkyl derivatives of piperizinylcamphorsulfonyl oxytocin antagonists |
03/17/1993 | CA2078025A1 Substituted amine derivatives of piperizinylcamphorsulfonyl oxytocin antagonists |
03/16/1993 | US5194605 Cyclic renin inhibitors containing 2-substituted (3S,4S)-4-amino-5-cyclohexyl-3-hydroxy pentanoic acid, 2-substituted (3S,4S)-5-cyclohexyl-3,4-di-hydroxy pentanoic acid or 2-substituted (4S,5S)-5-amino-6-cyclohexyl-4-hydroxyhexanoic acid or its analogs |
03/14/1993 | CA2077922A1 Substituted amide derivatives of piperizinylcamphorsulfonyl oxytocin antagonists |
03/10/1993 | EP0530353A1 New imidazopyridines as serotonergic 5-ht 3? antagonists |
03/09/1993 | US5192770 Serotonergic alpha-oxoacetamides |
03/03/1993 | EP0529462A1 Benzodioxan derivatives |
02/23/1993 | US5189061 Fungicide |
02/23/1993 | CA2076573A1 Benzodioxane derivatives |
02/21/1993 | CA2076443A1 1-(alcoxybenzyl)piperazins amidic compounds, process for their preparation and pharmaceutical compositions containing same |
02/18/1993 | WO1993003029A1 (-) and (+) 10-(1-azabicyclo[2.2.2.]oct-3-yl-methyl)-10 h-phenothiazine quaternary ammonium derivatives, pharmaceutical compositions containing them and process for their preparation |
02/18/1993 | CA2114844A1 (-) and (+) 10-(1-azabicyclo[2.2.2.]oct-3-yl-methyl)-10 h-phenothiazine quaternary ammonium derivatives, pharmaceutical compositions containing them and process for their preparation |
02/16/1993 | US5187164 Psychological disorders, antiemetics |
02/10/1993 | EP0526582A1 Heterocyclic chiral ligands and method for catalytic asymmetric dihydroxylation of olefins |
02/10/1993 | EP0526545A1 Isoquinoline amides and esters as 5 ht3 receptor antagonists |
02/09/1993 | US5185333 Benzazine compounds and pharmaceutical uses thereof |
02/03/1993 | EP0525879A1 Pyrazole derivatives |
02/03/1993 | CN1068571A Substituted 3-aminoquinuclidines |
02/02/1993 | US5183893 Alzheimer's disease and learning enhancement |
02/02/1993 | US5183822 Substituted 3,4-annelated benzimidazol-2(1h)-ones |
01/27/1993 | CA2074601A1 Pyrazole derivatives |
01/26/1993 | US5182283 Alzheimer's disease |
01/19/1993 | US5180823 Intramolecular Cyclization |
01/13/1993 | EP0523013A2 Use of benzimidazoline-2-oxo-1-carboxylic acid derivatives in the treatment of organic mental diseases |
01/07/1993 | WO1993000331A1 Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles |
01/06/1993 | CN1067655A Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles |
01/06/1993 | CA2072676A1 Azabicyclic compounds, pharmaceutical compositions containing them and their use in therapy |
01/05/1993 | US5177084 1-Azabicycles, Treating Mental Disorders |
01/05/1993 | CA2072911A1 Use of benzimidazoline-2-oxo-1-carboxylic acid derivatives |
12/30/1992 | EP0520555A1 Azabicyclic compounds, pharmaceutical compositions containing them and their use in therapy |
12/30/1992 | CN1067428A 奎宁环衍生物 Quinuclidine derivatives |
12/25/1992 | CA2071800A1 Azabicyclic compounds, pharmaceutical compositions containing them and their use in therapy |
12/23/1992 | WO1992022294A1 Immunomodulatory azaspiranes |
12/23/1992 | CA2110577A1 Immunomodulatory azaspiranes |
12/16/1992 | EP0518676A2 Cyclic renin inhibitors |