Patents
Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704)
03/2000
03/15/2000EP0984778A1 Neuropeptide-y ligands
03/15/2000EP0739204A4 Piperidines, pyrrolidines and hexahydro-1h-azepines promote release of growth hormone
03/08/2000EP0984008A2 Nitrosation process
03/07/2000US6034119 Agent for potentiating nerve growth factor activity containing 1,2-ethanediol derivative or salt thereof
03/02/2000WO1999064054A9 Multibinding inhibitors of topoisomerase
03/02/2000WO1999063937A3 Multivalent macrolide antibiotics
03/01/2000EP0981340A1 Pharmaceutical formulations in dry form for the oral administration of a cyclic quaternary ammonium compound
02/2000
02/29/2000US6030966 Heterocyclic compound and their use
02/23/2000EP0980370A1 5-phenyl-1,3,4-oxadiazol-2(3h)-one derivatives and their use as 5-ht4 ligands
02/15/2000CA2197739C 1,4-dihydropyridine compounds
02/09/2000EP0978280A1 2-azabicyclo compounds
02/09/2000EP0977755A1 Heterocyclic compounds and their preparation and use
02/09/2000EP0977567A1 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment
02/08/2000CA2014379C Compounds
02/03/2000WO2000005229A1 Phenylindole derivatives as 5-ht2a receptor ligands
02/03/2000WO1999063929A3 Multibinding inhibitors of microsomal triglyceride transferase protein
02/02/2000EP0976722A1 Benzamidine derivatives
02/02/2000CN1243505A Benzamidine derivatives
02/02/2000CN1048986C Heterocyclic compounds and their preparation and use
02/01/2000US6020368 Microbiocides
01/2000
01/26/2000CN1048727C Process for prepn. of 2-(1-azabicyclo (2,2,2) oct-3-yl)-2,4,5,6-tetrahydro-1H-benz
01/26/2000CN1048719C Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxytetracyclines, prepn. method, their compositions and use thereof
01/25/2000US6017944 Treating a variety of sex-hormone related and other conditions in both men and women; preventing pregnancy, treating lupus erythematosis, irritable bowel syndrome, premenstrual syndrome, hirsutism, sleep disorders
01/25/2000US6017927 Quinuclidine derivatives and medicinal composition thereof
01/19/2000CN1048492C Quinuclidine derivatives and its preparation
01/18/2000US6015813 Heterocyclic compounds and their preparation and use
01/12/2000CN1241187A Piperazino derivs as neurokinin antagonists
01/05/2000EP0711299B1 AZABICYCLOALKYL DERIVATIVES OF IMIDAZO(1,5-a)INDOL-3-ONE AS 5HT 3 ANTAGONISTS
01/05/2000CN1048013C Process for preparation of azabicyclic derivatives
01/04/2000US6011154 Substituted heterocyclic compounds, method of preparing them and pharmaceutical compositions in which they are present
01/04/2000US6011029 Benzodiazepine compounds
12/1999
12/28/1999US6008357 1 -azabicyclo(2.2.2)octan-3-amine, (2-diphenylmethyl)-n-((2-methoxy-5-(1-methylethyl)phenyl)methy l) is reacted with 1r-(-)-10-camphorsulfonic acid to obtain camphorsulfonic acid salt
12/21/1999CA2003422C Quinuclidines, their use as medicaments and processes for their preparation
12/16/1999WO1999064054A1 Multibinding inhibitors of topoisomerase
12/16/1999WO1999064051A1 Novel antibacterial compounds
12/16/1999WO1999064049A1 Novel antibacterial agents
12/16/1999WO1999064048A1 Inhibitors of hiv reverse transcriptase
12/16/1999WO1999064047A1 Novel antiviral compounds
12/16/1999WO1999064037A1 Novel therapeutic agents that modulate enzymatic processes
12/16/1999WO1999064033A1 Phosphodiesterase-v modulator drugs and their uses
12/16/1999WO1999063988A1 Inhibitors of nitric oxide synthase
12/16/1999WO1999063940A2 INHIBITORS OF H+K+-ATPase
12/16/1999WO1999063937A2 Multivalent macrolide antibiotics
12/16/1999WO1999063929A2 Multibinding inhibitors of microsomal triglyceride transferase protein
12/16/1999CA2321274A1 Novel antiviral compounds
12/16/1999CA2321190A1 Novel therapeutic agents that modulate enzymatic processes
12/16/1999CA2321166A1 Multibinding inhibitors of topoisomerase
12/16/1999CA2321162A1 Novel antibacterial compounds
12/16/1999CA2320241A1 Multivalent macrolide antibiotics
12/16/1999CA2319495A1 Multibinding inhibitors of microsomal triglyceride transferase protein
12/16/1999CA2319477A1 Inhibitors of h+k+-atpase
12/16/1999CA2319474A1 Inhibitors of nitric oxide synthase
12/16/1999CA2319120A1 Phosphodiesterase-v modulator drugs and their uses
12/16/1999CA2316999A1 Inhibitors of hiv reverse transcriptase
12/14/1999CA2135487C Heteroaromatic quinuclidinenes, their use and preparation
12/07/1999US5998434 Composition for treating pain
12/07/1999US5998429 Azabicyclic esters of carbamic acids useful in therapy
12/07/1999US5998404 Nervous system disorders
12/07/1999CA2198231C Dihydropyridine derivatives as bradykinin antagonists
12/07/1999CA2161886C Heteroatom substituted alkylbenzylaminoquinuclidines
12/01/1999EP0960108A1 Matrix metalloproteinase inhibitors
12/01/1999EP0655056B1 Azacyclyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
11/1999
11/25/1999WO1999059995A1 Heterocyclic compounds and their preparation and use
11/25/1999WO1999059957A1 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
11/24/1999EP0957916A1 Methods and compositions for treating urinary incontinence using enantiomerically enriched (r)-clidinium
11/24/1999CN1046722C Heterocyclic compounds and their preparation and use
11/23/1999US5990124 Neuromuscular relaxants
11/09/1999US5981545 N-linked azabicyclic heterocycles useful for treating dementia
11/09/1999US5981525 Indole derivatives useful in the treatment of osteoporosis
11/09/1999US5981520 Useful for treating asthma, bronchospasm, allergies, anxiety, coughing or pain
11/04/1999WO1999048894B1 Novel cephalotaxane derivatives and process for their preparation
11/03/1999CN1234026A Piperazino derivatives as neurokinin antagonists
11/02/1999US5977359 Substituted heterocyclic compounds, method of preparing them and pharmaceutical compositions in which they are present
11/02/1999US5977129 Alzheimer's disease
10/1999
10/27/1999CN1232825A Process for resolving (R,S(Z))-a-(methoximino)-a-(1-azabicyclo (2,2,2) oct-3 yl) acetonitrile
10/19/1999US5968935 Agent for potentiating nerve growth factor activity containing 1,2-ethanediol derivative or salt thereof
10/19/1999US5968929 Piperazino derivatives as neurokinin antagonists
10/19/1999US5968926 Schizophrenia treatment with 1,2,5-oxadiazole or 1,2,5-thiadiazole
10/19/1999US5968924 Benzo-fused lactams promote release of growth hormone
10/19/1999US5968867 Silica gel supported bis-cinchona alkaloid derivatives and a preparation method and use thereof
10/14/1999WO1999051234A1 Antagonists of gonadotropin releasing hormone
10/14/1999WO1999051232A1 Antagonists of gonadotropin releasing hormone
10/14/1999CA2326143A1 Antagonists of gonadotropin releasing hormone
10/14/1999CA2326139A1 Antagonists of gonadotropin releasing hormone
10/13/1999CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/13/1999CN1045601C Novel quinuclidine derivatives and medicinal composition thereof
10/12/1999US5965579 Antagonists of the neurotensin receptors; increasing affinity for human neurotensin receptors
10/12/1999US5965572 Methods for treating antibiotic-resistant infections
10/05/1999US5962724 High enantio-selective process for producing pure enantiomeric cyclopentane and cyclopentene-(β)-amino acids
09/1999
09/30/1999WO1999048894A1 Novel cephalotaxane derivatives and process for their preparation
09/30/1999CA2324895A1 Novel cephalotaxane derivatives and process for their preparation
09/15/1999EP0941228A1 PROCESS FOR PREPARING MeO-Peg-PROTECTED DIHYDROQUININE OR DIHYDROQUINIDINE DERIVATIVES, DIHYDROQUININE OR DIHYDROQUINIDINE DERIVATIVES AND THEIR USE
09/10/1999WO1999026932A8 By amidino group substituted heterocyclic derivatives and their use as anticoagulants
09/07/1999CA2098944C Novel pyrazole derivatives, method of preparing them and pharmaceutical compositions in which they are present
09/01/1999EP0938313A1 Methods and compositions for treating urinary incontinence using enantiomerically enriched (s)-clidinium
08/1999
08/26/1999WO1999042463A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/26/1999WO1999042461A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/25/1999EP0937069A1 Piperazino derivatives as neurokinin antagonists
08/25/1999EP0936866A1 Compounds, compositions and methods for treating antibiotic-resistant infections
08/25/1999CN1226886A Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation
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