Patents
Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704)
11/1994
11/10/1994CA2160795A1 Heterocyclic derivatives
11/09/1994EP0623592A1 Peptide analogs as irreversible interleukin-1beta protease inhibitors
11/09/1994EP0532527B1 3-amino-2-aryl quinuclidines, process for their preparation and pharmaceutical compositions containing them
11/09/1994CN1094718A Bicyclic fibrinogen antagonists
11/08/1994US5362740 Dihydrobenzofuran carboxamides and process for their preparation
11/08/1994US5362734 Certain benzo-quinolizine compounds and derivatives thereof
11/02/1994CN1094404A Heterocyclic compounds
11/01/1994US5360820 Medical use for tachykinin antagonists
11/01/1994CA1332834C Substituted basic 2-aminotetralins
10/1994
10/30/1994CA2122227A1 Peptide analogs as irreversible interleukin-1.beta. protease inhibitors
10/26/1994CN1094050A Novel heterocyclic compounds with antiasthmatic/anti-auergie, anti-inflammatory positive inotropic and blood pressure-reducing effect
10/26/1994CN1094035A Carboxylic acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
10/25/1994US5358954 Benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-HT receptor antagonists
10/19/1994EP0619814A1 Oxadiazole derivatives having acetylcholinesterase-inhibitory and muscarinic agonist activity
10/18/1994US5356912 3-(5-isoxazolyl)-1-methyl-1,2,3,6-tetrahydropyridine useful for treating Alzheimer's disease
10/13/1994WO1994022907A1 New urea derivates, their preparation and their use
10/11/1994US5354750 Phthalazines containing an aromatic ether or thioether group in the 1-position
10/05/1994EP0618193A1 Nitrogen containing bicyclic derivatives as prolyl-endopeptidase inhibitors
10/05/1994EP0618190A1 9-[(Substituted glycyl)amido]-6-(substituted)-5-hydroxy-6-deoxytetracyclines
10/05/1994CN1026111C Quinuclidine therapeutic agents
09/1994
09/29/1994DE4309213A1 Cyclic urea derivatives, medicaments containing these compounds and processes for their preparation
09/28/1994CN1092769A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
09/28/1994CN1092767A Spiro piperdines and homologs promote release of growth hormone
09/21/1994EP0615751A1 Use of tachykinin antagonists in the treatment of emesis
09/20/1994US5348967 Diaminotrifluoromethylpyridine derivatives, process for their production and phospholipase A2 inhibitor containing them
09/20/1994CA1332057C Bicycloalkyl, tricycloalkyl, azabicycloalkyl and azatricycloalkyl amides
09/15/1994WO1994020496A1 Heterocyclic compounds and their preparation and use
09/15/1994WO1994020465A1 Indole derivatives as antagonists of excitatory amino acids
09/13/1994US5346911 Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
09/13/1994US5346906 Substituted pyridines, their preparation, formulations and use in dementia
09/01/1994WO1994019348A1 Bicyclic nitrogenous compound
09/01/1994WO1994014776A3 Bicyclic fibrinogen antagonists
08/1994
08/31/1994EP0612746A1 Pyrimidines and their pharmaceutical acceptable salts and their use as medicines
08/30/1994US5342845 Indole derivatives and drugs
08/24/1994EP0611370A1 Pyridine-3-carboxylic acid esters or amides useful as 5-ht 3? antagonists
08/24/1994CN1091134A Quinuclidine derivative for treatment of inflammatory and gastrointestinal disorders
08/23/1994US5340809 New 1-(alkoxybenzyl)piperazine amide compounds
08/18/1994WO1994018201A1 Isoxazoleoxy derivative
08/10/1994EP0609335A1 Methods for the treatment of hyperlipidemia using azaspiranes
08/03/1994EP0608858A1 5-Membered heterocycles as aggregation inhibitors
08/03/1994EP0608336A1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment
08/03/1994EP0608307A1 New ligands for asymmetric dihydroxylation: multiple cinchona alkaloid units attached to a central heterocyclic core
08/03/1994CN1090277A Benzoxazinones as inhibitors of HIV reverse transcriptase
08/03/1994CN1090272A New substituted azetidinones as anti-inflammatory and antidegenerative agents
08/03/1994CN1090267A Novel 7-(substituted)-8-(substituted)-9-(substituted Amino)-6-demethyi-6-deoxytetracyclines
07/1994
07/28/1994DE4302052A1 Cyclic urea derivatives, medicaments containing these compounds and process for their preparation
07/27/1994EP0607164A1 Fused tricyclic nitrogen containing heterocycles as substance p receptor antagonists
07/27/1994CA2114178A1 5-membered heterocycles, processes for preparing them and pharmaceutical compositions containing these compounds
07/19/1994US5330990 Substituted urea compounds and their preparation and use
07/07/1994WO1994014805A1 Quinuclidine derivatives as squalene synthase inhibitors
07/07/1994WO1994014804A1 Quinuclidine derivatives as squalene synthase inhibitors
07/07/1994WO1994014776A2 Bicyclic fibrinogen antagonists
07/07/1994CA2152631A1 Bicyclic fibrinogen antagonists
07/06/1994EP0604800A1 4- 4- 4-(carboxyalkyl)-phenyl amino carbonyl -phenyl -piperedines as aggregation inhibitors
07/06/1994CN1088917A Substituted benzylamino nitrogen containing non-aromatic heterocycles
07/05/1994USRE34653 Heterocyclic spiro compounds and methods for preparing the same
07/05/1994US5326768 5-hydroxytryptamine antagonists
07/05/1994US5326760 Aminobutanoic acid compounds having metalloprotease inhibiting properties
06/1994
06/29/1994EP0603229A1 Quinuclidine esters process and intermediate for their preparation and pharmaceutical compositions containing them
06/29/1994CN1088582A Quaternary basic amides, method of preparing them and pharmaceutical compositions in which they are present
06/29/1994CN1088435A Anti-arrhythmic, analgesically acting phthalzinone derivatives that break through multi-drug-resistance
06/28/1994US5324724 Azabicyclic compounds; Alzheimer's disease treatment
06/28/1994US5324723 Oxazoles and thiazoles for the treatment of senile dementia
06/23/1994WO1994014803A1 Quinuclidine derivatives as squalene synthase inhibitors
06/22/1994CA2111895A1 Heterocyclic compounds
06/16/1994DE4241632A1 New (aza)aromatic or alicyclic carboxylic acid cpds. - used e.g. for treating thrombosis, inflammation, osteoporosis, cardiac infarct or tumour metastasis
06/14/1994US5321034 Fibrinogen receptor antagonists
06/12/1994CA2110672A1 Spiro peperidines and holologs which promote release of growth hormone
06/11/1994CA2111035A1 Carboxylic acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
06/08/1994EP0599896A1 (-) and (+) 10-(1-azabicyclo 2.2.2.]oct-3-yl-methyl)-10 h-phenothiazine quaternary ammonium derivatives, pharmaceutical compositions containing them and process for their preparation
06/01/1994EP0599152A1 Triazinones and Triazinophthalazinones possessing antiasthmatic/antiallergic, positive inotropic and antihypertensive activities
05/1994
05/26/1994WO1994011368A1 Quinuclidine derivative as substance p antagonist
05/26/1994CA2109900A1 Heterocyclic compounds with antiasthmatic/anti-allergic, anti-inflammatory, positive inotropic and blood pressure-reducing effect
05/25/1994EP0598093A1 Quinuclidine derivatives as squalene synthetase inhibitors
05/11/1994WO1994010170A1 Substituted quinuclidines as substance p antagonists
05/11/1994WO1994010167A1 Tachykinin antagonists
05/11/1994WO1994010142A1 New substituted azetidinones as anti-inflammatory and antidegenerative agents
05/11/1994EP0596058A1 Biphenylylquinuclidine derivatives as squalene synthase inhibitors
05/11/1994EP0596057A1 Quinuclidine derivatives as squalene synthase inhibitors
05/10/1994US5310737 Benzo-fused lactams that promote the release of growth hormone
05/04/1994EP0595557A1 New substituted azetidinones as anti-inflammatory and antidegenerative agents
05/04/1994EP0594605A1 1-azabicyclic compounds, processes and pharmaceutical compositons containing them
05/04/1994EP0594569A1 Preparation of s-(-)- and r-(+)-n-(quinuclidinyl-3)-amide
04/1994
04/28/1994WO1994008997A1 Substituted benzylaminoquinuclidines as substance p antagonists
04/26/1994US5306718 Analgesics, cognition activators
04/19/1994US5304552 Renin inhibitors
04/14/1994DE4230470A1 New cyclic urea derivs.
04/06/1994EP0591040A1 Quaternary basic amides as tachykinines antagonists
04/06/1994EP0590551A2 New therapeutic uses of phthalazinone-derivatives
04/05/1994US5300649 Reacting 1,3-dienes with sulfonyl cyanides
04/05/1994US5300512 Antiserotonine agents; antagonist or agonist
04/03/1994CA2107548A1 Anti-arrhythmic, analgesically acting phthalazinone derivatives that break through multi-drug resistance
03/1994
03/31/1994WO1994006792A1 Optically active hydroquinine (amino-3 phenyl)-1 ethanesulfonate, preparation and use thereof
03/31/1994CA2144158A1 Optically active hydroquinine 1-(3-aminophenyl)ethanesulfonate; preparation thereof and its use
03/30/1994EP0589484A1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
03/30/1994CN1084516A Azacyclic and azabicyclic alkyliden hydroxylamines
03/29/1994US5298513 Serotonin antagonist
03/29/1994CA1328107C2 Enantiomers of absolute configuration s and r of 3-aminoquinuclidine, and processes for preparing them
03/23/1994EP0587800A1 Immunomodulatory azaspiranes
03/23/1994CN1084169A Compounds
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